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From natural to artificial antitumor lipidic alkynylcarbinols: Asymmetric synthesis, enzymatic resolution, and refined SARs

 Dymytrii Listunov , Etienne Joly , Pauline Rullière , Hafida Gaspard , Vania Bernardes-Génisson , et al.
Synthesis: Journal of Synthetic Organic Chemistry, 2018, 50 (16), pp.3114-3130. ⟨10.1055/s-0037-1610006⟩
Article dans une revue hal-01952874v1

Séparation chirale par chromatographie liquide et par fluide supercritique des analogues cliquables de Jaspine B

 Cécile Santos , Isabelle Fabing , Stéphanie Ballereau , Yves Génisson , A. Rozie , et al.
33e journée Chimie-Biologie-Santé, Apr 2019, Toulouse, France
Poster de conférence hal-02338505v1
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Fragment-Based Ligand Discovery Applied to the Mycolic Acid Methyltransferase Hma (MmaA4) from Mycobacterium tuberculosis

 Romain Galy , Stéphanie Ballereau , Yves Génisson , Lionel Mourey , Jean-Christophe Plaquevent , et al.
Pharmaceuticals, 2021, 14 (12), pp.1282. ⟨10.3390/ph14121282⟩
Article dans une revue hal-03683937v1

The integrated screening platform of Toulouse (PICT) : A tool for accelerated molecular discovery

 Isabelle Fabing , Michel Baltas , Stéphanie Ballereau , Yves Génisson , Brigitte Guidetti , et al.
Congress SFC 2018 Chemistry and Life Symposium, Jun 2018, Montpellier, France
Poster de conférence hal-02337455v1

Alkyne-tagged analogue of jaspine B: new tool for identifying jaspine B mode of action

 Cécile Santos , Isabelle Fabing , Stéphanie Ballereau , Yves Génisson
Congrès JCO 2019, Oct 2019, Palaiseau, France
Poster de conférence hal-02893206v1

C-branched iminosugars: synthesis and biological relevance

 Cécile Baudoin-Dehoux , Yves Génisson
European Journal of Organic Chemistry, 2019, pp.6386-6397. ⟨10.1002/ejoc.201900605⟩
Article dans une revue hal-02328842v1

The integrated screening platform of Toulouse (PICT) : A tool for accelerated molecular discovery

 Brigitte Guidetti , Isabelle Fabing , Michel Baltas , Stéphanie Ballereau , Tessa Castellan , et al.
33e journée Chimie-Biologie-Santé, Apr 2019, Toulouse, France
Poster de conférence hal-02338497v1
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Pharmacological Chaperone Therapy for Pompe Disease

 Marc Borie-Guichot , My Lan Tran , Stéphanie Ballereau , Cécile Dehoux , Yves Génisson
Molecules, 2021, 26 (23), pp.7223. ⟨10.3390/molecules26237223⟩
Article dans une revue hal-03758482v1

Extended structural modulation of bio-inspired chiral lipidic alkynylcarbinols as antitumor pharmacophores

 Dymytrii Listunov , C. Billot , Etienne Joly , Isabelle Fabing , Yulian Volovenko , et al.
Tetrahedron, 2015, 71 (41), pp.7920-7930. ⟨10.1016/j.tet.2015.08.003⟩
Article dans une revue hal-01916644v1

Bioinspired lipidic alkynylcarbinols as anticancer agents

 Margaux Bossuat , Stéphanie Ballereau , Antonio Peixoto , Valérie Maraval , Vania Bernades-Génisson , et al.
Journées de Chimie Organique 2022 (JCO 2022), Nov 2022, Palaiseau, France
Communication dans un congrès hal-04402220v1

Mechanism-guided development of covalent prodrugs for targeted anticancer therapy.

 Margaux Bossuat , Nadège Preuilh , Stéphanie Ballereau , Antonio Peixoto , V. Bernades-Génisson , et al.
Journée du GDR ChemBio, Jun 2023, Strasbourg, France
Poster de conférence hal-04198409v1

Development of Bioinspired Lipidic Alcynylcarbinol Prodrugs for Targeted Anticancer Therapy.

 Margaux Bossuat , Nadège Preuilh , Stéphanie Ballereau , V. Bernades-Génisson , Valérie Maraval , et al.
Congrès SCF23, Jun 2023, Nantes, France
Poster de conférence hal-04198468v1

Methinylogation approach in chiral pharmacophore design: from alkynyl- to allenyl-carbinol warheads against tumor cells

 Dymytrii Listunov , Etienne Joly , Carine Guyard-Duhayon , N. Saffon-Merceron , Isabelle Fabing , et al.
ChemMedChem, 2018, 13 (16), pp.1711-1722. ⟨10.1002/cmdc.201800284⟩
Article dans une revue hal-01952875v1

Synthesis of Cytotoxic Aza Analogues of Jaspine B.

 Arnaud Rives , Sonia Ladeira , Thierry Levade , Nathalie Andrieu-Abadie , Yves Génisson
Journal of Organic Chemistry, 2010, epub ahead of print. ⟨10.1021/jo1014239⟩
Article dans une revue inserm-00550705v1

Bio-inspired antitumor acetylenic lipids bearing alkynylcarbinol pharmacophores

 Pauline Rullière , Maroua Bourkhis , Dymytrii Listunov , Hafida Gaspard , Valérie Maraval , et al.
10th International Chemistry Conference Toulouse-Kiev (ICTK-10), Jun 2019, Toulouse, France
Poster de conférence hal-02335633v1
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The natural marine anhydrophytosphingosine, Jaspine B, induces apoptosis in melanoma cells by interfering with ceramide metabolism

 Yahya Salma , Elodie Lafont , Nicole Therville , Stéphane Carpentier , Marie-José Bonnafé , et al.
Biochemical Pharmacology, 2009, 78 (5), pp.477. ⟨10.1016/j.bcp.2009.05.002⟩
Article dans une revue istex hal-00497269v1

The Integrated Screening Platform of Toulouse (PICT): a tool for accelerated molecular discovery

 Brigitte Guidetti , Isabelle Fabing , Michel Baltas , Stéphanie Ballereau , Tessa Castellan , et al.
Congrès JCO 2019, Oct 2019, Palaiseau, France
Poster de conférence hal-02893197v1
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Synthesis of novel room temperature chiral ionic liquids. application as reaction media for the heck arylation of aza-endocyclic acrylates.

 Julio C. Pastre , Yves Génisson , Nathalie Saffon , Jany Dandurand , Carlos R. D. Correia
Journal of the Brazilian Chemical Society, 2010, 21 (5), pp.0. ⟨10.1590/S0103-50532010000500009⟩
Article dans une revue hal-03550343v1
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Alkyne-Tagged Analogue of Jaspine B: New Tool for Identifying Jaspine B Mode of Action

 Alexandrine Rozié , Cécile Santos , Isabelle Fabing , Patrick Calsou , Sébastien Britton , et al.
ChemBioChem, 2018, 19 (23), pp.2438-2442. ⟨10.1002/cbic.201800496⟩
Article dans une revue hal-02059233v1
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Enantioselective Stereodivergent Synthesis of Jaspine B and 4-epi-Jaspine B from Axially Chiral Allenols

 Heba Alnazer , Tessa Castellan , Yahya Salma , Yves Génisson , Stéphanie Ballereau
SYNLETT, 2019, 30 (02), pp.185-188. ⟨10.1055/s-0037-1610344⟩
Article dans une revue hal-02059333v1

Fluorophore-tagged pharmacophores for antitumor cytotoxicity: Modified chiral lipidic dialkynylcarbinols for cell imaging

 Dymytrii Listunov , S. Mazeres , Yulian Volovenko , Etienne Joly , Yves Génisson , et al.
Bioorganic and Medicinal Chemistry Letters, 2015, 25 (20), pp.4652-4656. ⟨10.1016/j.bmcl.2015.08.029⟩
Article dans une revue hal-01915503v1

Multivalent pharmacological chaperones based on dendrimers against Gaucher disease

 My Lan Tran , Marc Borie-Guichot , Yves Génisson , C.O. Turrin , Abdelouahd Oukhrib , et al.
JCO 2022, Nov 2022, Palaiseau, France
Poster de conférence hal-03857556v1

Origin of the Enantioselectivity in Organocatalytic Michael Additions of beta-Ketoamides to alpha,beta-Unsaturated Carbonyls: A Combined Experimental, Spectroscopic and Theoretical Study

 Adrien Quintard , Diana Cheshmedzhieva , Maria del Mar Sanchez Duque , Anouk Gaudel-Siri , Jean-Valère Naubron , et al.
Chemistry - A European Journal, 2015, 21, pp.778-790. ⟨10.1002/chem.201404481⟩
Article dans une revue istex hal-01133609v1

Transalpinecine and Analogues: First Total Synthesis, Stereochemical Revision and Biological Evaluation

 Cécile Baudoin-Dehoux , Tessa Castellan , Morgane Enel , Christiane André-Barrès , Sandra Mirval , et al.
European Journal of Organic Chemistry, 2019, 19, pp.1830-1834. ⟨10.1002/ejoc.201900071⟩
Article dans une revue hal-02330547v1
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Phosphorus Dendrimers for Metal‐Free Ligation: Design of Multivalent Pharmacological Chaperones against Gaucher Disease

 My Lan Tran , Marc Borie-Guichot , Virginie Garcia , Abdelouahd Oukhrib , Yves Génisson , et al.
Chemistry - A European Journal, 2023, 29 (53), pp.e202301210. ⟨10.1002/chem.202301210⟩
Article dans une revue hal-04175496v1

Identification of Novel CERT Ligands as Potential Ceramide Trafficking Inhibitors

 Cécile Santos , Frédéric Rodriguez , Virginie Garcia , Daniela Moravčíková , Dušan Berkeš , et al.
ChemBioChem, 2014, 15 (17), pp.2522-2528. ⟨10.1002/cbic.201402366⟩
Article dans une revue istex hal-02063974v1

Première synthèse totale et révision structurale de la Transalpinécine

 Christiane André-Barrès , Cécile Baudoin-Dehoux , Morgane Enel , Stéphanie Ballereau , Tessa Castellan , et al.
Congress SFC 2018 Chemistry and Life Symposium, Jun 2018, Montpellier, France
Poster de conférence hal-02337494v1

Alkyne-tagged analogue of jaspine B: new tool for identifying jaspine B mode of action

 Stéphanie Ballereau , Yves Génisson , Patrick Calsou , Sébastien Britton
10th International Chemistry Conference Toulouse-Kiev (ICTK-10), Jun 2019, TOULOUSE, France
Communication dans un congrès hal-02333441v1
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1-Ethyl-3-methylimidazolium tartrate chiral ionic liquids: preparation, characterization and opportunities thereof

 Tessa Castellan , Claire Cuyamendous , Juliette Fitremann , Jean-Marie Galano , Camille Oger , et al.
New Journal of Chemistry, 2018, 42 (23), pp.18739-18748. ⟨10.1039/C8NJ03175D⟩
Article dans une revue hal-02059223v1

Première synthèse totale et révision structurale de la Transalpinécine

 Stéphanie Ballereau , Tessa Castellan , Morgane Enel , Christiane André-Barrès , Yves Génisson , et al.
8ème Symposium Francophone de Synthèse Totale, May 2018, Bordeaux, France
Poster de conférence hal-02337257v1
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