|
|
Synthesis of pyrazolo[4,3-a]phenanthridines, a new scaffold for Pim kinase inhibition
Virginie Suchaud
,
Laurent Gavara
,
Francis Giraud
,
Lionel Nauton
,
Vincent Théry
,
et al.
Article dans une revue
hal-01077451v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Water-Soluble Gold–N-Heterocyclic Carbene Complexes for the Catalytic Homogeneous Acid- and Silver-Free Hydration of Hydrophilic Alkynes.
Houssein Ibrahim
,
Pierre De frémont
,
Pierre Braunstein
,
Vincent Théry
,
Lionel Nauton
,
et al.
Article dans une revue
istex
hal-01264762v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
12-Helix folding of cyclobutane beta-amino acid oligomers
Carlos Fernandes
,
Sophie Faure
,
Elisabeth Pereira
,
Vincent Thery
,
Valérie Declerck
,
et al.
Article dans une revue
hal-00530671v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Identification of pyrrolo[2,3-g]indazoles as new Pim kinase inhibitors.
Laurent Gavara
,
Virginie Suchaud
,
Lionel Nauton
,
Vincent Théry
,
Fabrice Anizon
,
et al.
Article dans une revue
istex
hal-01089114v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Synthesis, Pim kinase inhibitory potencies and in vitro antiproliferative activities of diversely substituted pyrrolo[2,3-a]carbazoles
Rufine Akué-Gédu
,
Lionel Nauton
,
Vincent Thery
,
Jenny Bain
,
Philip Cohen
,
et al.
Bioorganic and Medicinal Chemistry, 2010, 18, pp.6865-6873
Article dans une revue
hal-00530591v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Study of Bruylants' reaction
Elisabeth Pereira
,
David J Aitken
,
Virginie Beaufort
,
Vincent Thery
Journées de Chimie Organique, Sep 2004, Palaiseau, France
Communication dans un congrès
hal-00138706v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Synthesis and Solution Conformation of Homo-β-peptides Consisting of N-Mannofuranosyl-3-ulosonic acids
Manuel Andreini
,
Claude Taillefumier
,
Francoise Chrétien
,
Vincent Thery
,
Yves Chapleur
Journal of Organic Chemistry, 2009, 74, pp.7651-7659
Article dans une revue
hal-00435712v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Synthesis and molecular modelling study of new trimeric quinoline derivatives
Emmanuelle Saugues
,
Lionel Nauton
,
Vincent Thery
,
Fabrice Anizon
,
Pascale Moreau
Bioorganic Chemistry, 2011, 39, pp.143-150
Article dans une revue
hal-00625030v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Palladium catalyzed intramolecular allylic amination: diastereoselective synthesis of 2,6-disubstituted 1,2,3,6-tetrahydropyridines.
A. Visseq
,
T. Boibessot
,
L. Nauton
,
V. Théry
,
F. Anizon
,
et al.
Congrès des jeunes Chercheurs de la Société de Chimie Thérapeutique, Feb 2019, Paris, France
Poster de conférence
hal-02295647v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co–crystal structure.
Yannick J. Esvan
,
Wael Zeinyeh
,
Thibaut Boibessot
,
Lionel Nauton
,
Vincent Théry
,
et al.
Article dans une revue
hal-01308803v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Synthesis and preliminary in vitro kinase inhibition evaluation of new diversely substituted pyrido[3,4-g]quinazoline derivatives.
Wael Zeinyeh
,
Yannick J. Esvan
,
Lionel Nauton
,
Nadège Loaëc
,
Laurent Meijer
,
et al.
Article dans une revue
hal-01367659v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Synthesis, Pim kinase inhibitory potencies and in vitro antiproliferative activities of diversely substituted pyrrolo[2,3-a]carbazoles
Fabrice Anizon
,
Rufine Akué-Gédu
,
Lionel Nauton
,
Vincent Thery
,
J. Bain
,
et al.
17th European Symposium on Organic Chemistry, Hersonissos (Grèce), 10-15 juillet 2011, Jul 2011, Hersonissos, Greece
Communication dans un congrès
hal-00609939v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Synthesis, protein kinase inhibitory potencies and in vitro antiproliferative activities of meridianin derivatives
Pascale Moreau
,
Francis Giraud
,
Elisabeth Pereira
,
Fabrice Anizon
,
Georges Alves
,
et al.
17th European Symposium on Organic Chemistry, Jul 2011, Hersonissos, Greece
Communication dans un congrès
hal-00609975v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Fructose-1,6-bisphosphate aldolase-mediated synthesis of aminocyclitols (analogues of valiolamine) and their evaluation as glycosidase inhibitors
Lahssen El Blidi
,
Zeinab Assaf
,
Flora Camps Bres
,
Henri Veschambre
,
Vincent Thery
,
et al.
ChemCatChem, 2009, 1, pp.463-471
Article dans une revue
hal-00438420v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Pyridin-2(1H)one derivatives: A possible new class of therapeutics for mechanical allodynia
Alexia Visseq
,
Amélie Descheemaeker
,
Nicolas Pinto-Pardo
,
Lionel Nauton
,
Vincent Thery
,
et al.
Article dans une revue
hal-02444268v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Micelle dynamic simulation and physicochemical characterization of biorelevant media to reflect gastrointestinal environment in fasted and fed states
Xiaoyu Xie
,
Jean-Michel Cardot
,
Ghislain Garrait
,
Vincent Thery
,
Mohamed El-Hajji
,
et al.
Article dans une revue
hal-01082838v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Structure-Based Design of PDZ Ligands as Inhibitors of 5-HT2A Receptor/PSD-95 PDZ1 Domain Interaction Possessing Anti-hyperalgesic Activity
Alexandre Vogrig
,
Liam Dorr
,
Naoual Bouzidi
,
Benjamin Boucherle
,
Anne-Sophie Wattiez
,
et al.
Article dans une revue
hal-00948867v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Synthesis and biological activity of pyrazole analogues of the staurosporine aglycon K252c.
Yannick J. Esvan
,
Francis Giraud
,
Elisabeth Pereira
,
Virginie Suchaud
,
Lionel Nauton
,
et al.
Article dans une revue
hal-01367761v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
New potent and selective inhibitor of Pim-1/3 protein kinases sensitizes human colon carcinoma cells to doxorubicin.
Pascale Moreau
,
Lyubov G. Dezhenkova
,
Fabrice Anizon
,
Lionel Nauton
,
Vincent Thery
,
et al.
Article dans une revue
hal-01077420v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Access to functionalised silver(I) and gold(I) N-heterocyclic carbenes by [2+3] dipolar cycloadditions.
Audrey Hospital
,
Clémentine Gibard
,
Christelle Gaulier
,
Lionel Nauton
,
Vincent Thery
,
et al.
Dalton Transactions, 2012, 41, pp.6803-6812
Article dans une revue
hal-00711788v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Identification of 1,6-dihydropyrazolo[4,3-c]carbazoles and 3,6-dihydropyrazolo[3,4-c]carbazoles as new Pim kinase inhibitors.
Virginie Suchaud
,
Laurent Gavara
,
Emmanuelle Saugues
,
Lionel Nauton
,
Vincent Théry
,
et al.
Article dans une revue
istex
hal-01089084v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Présentation du projet Criblage Virtuel
Vincent Thery
Conférence LifeGrid, Nov 2008, CLERMONT-FERRAND, France
Communication dans un congrès
hal-00345623v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Design of Orally Active Dual Inhibitors of Neutral Endopeptidase and Angiotensin-Converting Enzyme with Long Duration of Action
Marie-Claude Fournie-Zaluski
,
Pascale Coric
,
Vincent Théry
,
Walter D Gonzalez
,
Hervé Meudal
,
et al.
Article dans une revue
istex
hal-02122108v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Kinase inhibitions in pyrido[4,3-h] and [3,4-g]quinazolines: Synthesis, SAR and molecular modeling studies
Waël Zeinyeh
,
Yannick Esvan
,
Béatrice Josselin
,
Blandine Baratte
,
Stéphane Bach
,
et al.
Article dans une revue
hal-02164744v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Evolved Thermostable Transketolase for Stereoselective Two-Carbon Elongation of Non-Phosphorylated Aldoses to Naturally Rare Ketoses
Marion Lorillière
,
Romain Dumoulin
,
Mélanie L’enfant
,
Agnès Rambourdin
,
Vincent Thery
,
et al.
Article dans une revue
hal-02195534v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Diastereoselective Synthesis of 2,6-Disubstituted-1,2,3,6-Tetrahydropyridines through a Palladium-Catalyzed Intramolecular Allylic Amination
Alexia Visseq
,
Thibaut Boibessot
,
Lionel Nauton
,
Vincent Thery
,
Fabrice Anizon
,
et al.
Article dans une revue
hal-02444228v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Palladium catalyzed intramolecular allylic amination: diastereoselective synthesis of 2,6-disubstituted 1,2,3,6-tetrahydropyridines.
A. Visseq
,
T. Boibessot
,
L. Nauton
,
V. Théry
,
F. Anizon
,
et al.
SCT 26th Young Research Fellows meeting, Feb 2019, Paris, France
Communication dans un congrès
hal-02288930v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Design and synthesis of new nitrogen-containing heterocycles for the treatment of mechanical allodynia.
A. Visseq
,
A. Descheemaeker
,
L. Nauton
,
V. Théry
,
F. Giraud
,
et al.
Bioheterocycle 2019, XVIII International Conference on Heterocycles in Bioorganic Chemistry, Jun 2019, Gand, Belgium
Communication dans un congrès
hal-02288758v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
FSAB: A new fructose-6-phosphate aldolase from Escherichia coli. Cloning, over-expression and comparative kinetic characterization with FSAA
Israel Sanchez-Moreno
,
Lionel Nauton
,
Vincent Théry
,
Agnès Pinet
,
Jean-Louis Petit
,
et al.
Journal of Molecular Catalysis B: Enzymatic, 2012, 84, pp.9-14
Article dans une revue
hal-00786230v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
QM/MM Study of Human Transketolase: Thiamine Diphosphate Activation Mechanism and Complete Catalytic Cycle
Lionel Nauton
,
Laurence Hecquet
,
Vincent Théry
Article dans une revue
hal-03286397v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|