Recherche - Archive ouverte HAL Accéder directement au contenu

Filtrer vos résultats

53 résultats
Image document

2-Aminophenones, a common precursor to N-aryl isatins and acridines endowed with bioactivities

Nahida Mokhtari Brikci-Nigassa , Ghenia Bentabed-Ababsa , William Erb , Floris Chevallier , Laurent Picot , et al.
Tetrahedron, 2018, 74 (15), pp.1785-1801. ⟨10.1016/j.tet.2018.02.038⟩
Article dans une revue hal-01774406v1
Image document

Bisphosphonylallenes as Suitable Scaffolds for Unprecedented 4,5-Diphosphonyldihydropyridazines and 3,4-Diphosphonylpyrroles Displaying Antimelanoma Activity

Kmar Abaid , William Erb , David Virieux , Laurent Picot , Benjamin Musnier , et al.
ACS Omega, 2022, 7 (43), pp.38894-38901. ⟨10.1021/acsomega.2c04619⟩
Article dans une revue hal-03884897v1
Image document

Could Fucoxanthin Interaction with Lipid Rafts Mediate its Cytotoxicity in Cancer Cells?

Raimundo Gonçalves Oliveira-Junior , Valérie Thiéry , Odile Sergent , Martine Chevanne , Laurent Picot
Journal of Oceanography and Marine Research, 2016, 4 (1), pp.1000144. ⟨10.4172/jomr.1000144⟩
Article dans une revue hal-01391001v1
Image document

Sensitization of tumor cells to chemotherapy by natural products: a systematic review of preclinical data and molecular mechanisms

Raimundo Gonçalves de Oliveira Júnior , Christiane Adrielly Alves Ferraz , Jackson Roberto Guedes da Silva Almeida , Raphäel Grougnet , Valérie Thiéry , et al.
Fitoterapia, 2018, 129, pp.383-400. ⟨10.1016/j.fitote.2018.02.025⟩
Article dans une revue hal-01807405v1
Image document

Synthesis of azafluorenones and related compounds using deprotocupration-aroylation followed by intramolecular direct arylation

Nada Marquise , Philip J. Harford , Floris Chevallier , Thierry Roisnel , Vincent Dorcet , et al.
Tetrahedron, 2013, 69 (47), pp.10123-10133. ⟨10.1016/j.tet.2013.09.030⟩
Article dans une revue hal-00869376v1

Eco-Friendly Microwave-Assisted Scaleable Synthesis of 2-Cyanobenzothiazoles via N -Arylimino-1,2,3-dithiazoles

Stéphane Frère , Valérie Thiéry , Thierry Besson
Synthetic Communications, 2003, 33 (21), pp.3795-3804. ⟨10.1081/SCC-120025190⟩
Article dans une revue hal-02357713v1
Image document

2-Aminobenzaldehyde, a common precursor to acridines and acridones endowed with bioactivities

Sarah Zeghada , Ghenia Bentabed-Ababsa , Olivier Mongin , William Erb , Laurent Picot , et al.
Tetrahedron, 2020, 76 (38), pp.131435. ⟨10.1016/j.tet.2020.131435⟩
Article dans une revue hal-03302141v1
Image document

Crystal Structure of 6,7-Dihydro-5a,7a,13,14-tetraaza-pentaphene-5,8-dione

Jean Guillon , Maria de Fatima Pereira-Rosenfeld , Noël Pinaud , Thierry Besson , Valérie Thiéry , et al.
X-Ray Structure Analysis Online, 2019, 35 (10), pp.57-59. ⟨10.2116/xraystruct.35.57⟩
Article dans une revue hal-02330806v1

Microwave-assisted Synthesis of Novel Thiazolocarbazoles and Evaluation as Potential Anticancer Agents. Part III

Alexandra Testard , Laurent Picot , Ingrid Fruitier-Arnaudin , Jean-Marie Piot , Hadjila Chabane , et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2008, 19 (6), pp.467-473. ⟨10.1080/14756360412331280491⟩
Article dans une revue hal-01967795v1
Image document

From benzofuro-, benzothieno- and 10-methylindolo-[2,3-b]-fused benzothiopyrano[4,3,2-de]quinolines to the corresponding benzothiopyrano[4,3,2-de]1,8-naphthyridines: synthesis and properties of these hexacyclic heteroaromatic compounds

Nicolas Mast , William Erb , Lionel Nauton , Pascale Moreau , Olivier Mongin , et al.
New Journal of Chemistry, 2023, 47 (1), pp.258-283. ⟨10.1039/D2NJ04567B⟩
Article dans une revue hal-03904365v1

Contribution of Professor Charles W. Rees to the development of the chemistry of disulfur dichloride

Thierry Besson , Lidia Konstantinova , Panayiotis Koutentis , Oleg Rakitin , Sivaprasad Sivadasan , et al.
ARKIVOC - Online Journal of Organic Chemistry, 2024, 2024 (1), ⟨10.24820/ark.5550190.p012.136⟩
Article dans une revue hal-04435494v1

Synthesis and kinase inhibitory activity of novel substituted indigoids

Anne Beauchard , Helene Laborie , Hervé Rouillard , Olivier Lozach , Yoan Ferandin , et al.
Bioorganic and Medicinal Chemistry Letters, 2009, 17 (17), pp.6257-6263. ⟨10.1016/j.bmc.2009.07.051⟩
Article dans une revue istex hal-02357759v1

Efficient solvent-free microwave phosphorylation of microcrystalline cellulose

Natalia Gospodinova , Axelle Grelard , Marc Jeannin , Gabrielle Chitanu , Adrian Carpov , et al.
Green Chemistry, 2002, 4 (3), pp.220-222. ⟨10.1039/b200295g⟩
Article dans une revue istex hal-02357733v1
Image document

Antiproliferative Activity of Cyanophora paradoxa Pigments in Melanoma, Breast and Lung Cancer Cells

Paul-Hubert Baudelet , Anne-Laure Gagez , Jean-Baptiste Bérard , Camille Juin , Nicolas Bridiau , et al.
Marine drugs, 2013, 11 (11), pp.4390-4406
Article dans une revue hal-01247728v1
Image document

Zeaxanthin from Porphyridium purpureum induces apoptosis in human melanoma cells expressing the oncogenic BRAF V600E mutation and sensitizes them to the BRAF inhibitor vemurafenib

Camille Juin , Raimundo Gonçalves de Oliveira Junior , Audrey Fleury , Chloé Oudinet , Lior Pytowski , et al.
Revista Brasileira de Farmacognosia, 2018, 28 (4), pp.457-467. ⟨10.1016/j.bjp.2018.05.009⟩
Article dans une revue hal-01868622v1
Image document

Synthesis of C,N'-linked bis-heterocycles using a deprotometalation-iodination-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells

Madani Hedidi , Ghenia Bentabed-Ababsa , Aicha Derdour , Thierry Roisnel , Vincent Dorcet , et al.
Bioorganic and Medicinal Chemistry, 2014, 22 (13), pp.3498-3507. ⟨10.1016/j.bmc.2014.04.028⟩
Article dans une revue hal-00990052v1

Synthesis and evaluation of the antimicrobial activity of novel quinazolinones

Maria de Fatima Pereira , Romain Chevrot , Eric Rosenfeld , Valérie Thiéry , Thierry Besson
Journal of Enzyme Inhibition and Medicinal Chemistry, 2008, 22 (5), pp.577-583. ⟨10.1080/14756360701425345⟩
Article dans une revue hal-01960717v1

Novel 9-oxo-thiazolo[5,4-f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: Synthesis, biological evaluation and molecular modeling studies

Cédric Logé , Alexandra Testard , Valérie Thiéry , Olivier Lozach , Mélina Blairvacq , et al.
European Journal of Medicinal Chemistry, 2008, 43 (7), pp.1469-1477. ⟨10.1016/j.ejmech.2007.09.020⟩
Article dans une revue istex hal-02357774v1

Synthesis of novel 2,3-condensed thieno[2,3- d ]pyrimidin-4-ones via Appel's salt chemistry

Maria de Fatima Pereira , Valérie Thiéry , Thierry Besson
Journal of Sulfur Chemistry, 2006, 27 (1), pp.49-55. ⟨10.1080/17415990500493213⟩
Article dans une revue hal-02357738v1
Image document

Azine and Diazine Functionalization Using 2,2,6,6-Tetramethylpiperidino-Based Lithium–Metal Combinations: Application to the Synthesis of 5,9-Disubstituted Pyrido[3′,2′:4,5]pyrrolo[1,2-c] pyrimidines

Nada Marquise , Tan Tai Nguyen , Floris Chevallier , Laurent Picot , Valérie Thiéry , et al.
SYNLETT, 2015, 26 (20), pp.2811-2816. ⟨10.1055/s-0035-1560496⟩
Article dans une revue hal-01248092v1

Synthesis and kinase inhibitory activity of novel substituted indigoids.

Anne Beauchard , Hélène Laborie , Hervé Rouillard , Olivier Lozach , Yoan Ferandin , et al.
Bioorganic and Medicinal Chemistry, 2009, 17 (17), pp.6257-63. ⟨10.1016/j.bmc.2009.07.051⟩
Article dans une revue istex hal-00416031v1

Characterisation of the anti-migratory activity of the 6-bromoindirubin-3’oxime (BIO) derivative VTIND42 in patient-derived GBM subpopulations

Samuel Peat , Anke Bruning-Richardson , Laurent Meijer , Sean Lawler , Valérie Thiéry , et al.
Neuro-Oncology, 2019, 21 (Supplement_4), pp.iv6-iv7. ⟨10.1093/neuonc/noz167.026⟩
Article dans une revue hal-02550773v1

Complete Genome Sequence of the Polymyxin E (Colistin)-Producing Paenibacillus sp. Strain B-LR

Caroline Salsano , Sandrine Didelot , Fatoumata Tambadou , Thibault Caradec , Valérie Sopena , et al.
Microbiology Resource Announcements, 2018, 7 (23), ⟨10.1128/MRA.01013-18⟩
Article dans une revue hal-02383554v1
Image document

Functionalization of 9-thioxanthone at the 1-position: From arylamino derivatives to [1]benzo(thio)pyrano[4,3,2-de]benzothieno[2,3-b]quinolines of biological interest

Nahida Mokhtari Brikci-Nigassa , Lionel Nauton , Pascale Moreau , Olivier Mongin , Raphael E Duval , et al.
Bioorganic Chemistry, 2020, 94, pp.103347. ⟨10.1016/j.bioorg.2019.103347⟩
Article dans une revue hal-02404054v1

Imidazoquinolinethiones from 8-aminoquinolines by a novel peri-participation

Thierry Besson , Charles Rees , David Roe , Valérie Thiéry
Journal of the Chemical Society, Perkin Transactions 1, 2000, 4, pp.555-561. ⟨10.1039/a908952g⟩
Article dans une revue hal-02357793v1

Eco-Friendly Microwave-Assisted Scaleable Synthesis of 2-Cyanobenzothiazoles via N -Arylimino-1,2,3-dithiazoles

Valérie Thiéry , Thierry Besson
Synthetic Communications, 2003, 33 (21), pp.3795-3804. ⟨10.1081/SCC-120025190⟩
Article dans une revue hal-02357727v1
Image document

Improved racemate resolution of pentan-2-ol and trans-(Z)-cyclooct-5-ene-1,2-diol by lipase catalysis

Marianne Graber , Hervé Rouillard , Régis Delatouche , Najla Fniter , Belsem Belkhiria , et al.
Journal of Biotechnology, 2016, 238, pp.60-68. ⟨10.1016/j.jbiotec.2016.09.010⟩
Article dans une revue hal-01432549v1

Novel nonribosomal peptide synthetase (NRPS) genes sequenced from intertidal mudflat bacteria

Fatoumata Tambadou , Isabelle Lanneluc , Sophie Sablé , Géraldine Klein , Ibtissem Doghri , et al.
FEMS Microbiology Letters, 2014, pp.n/a-n/a. ⟨10.1111/1574-6968.12532⟩
Article dans une revue hal-01960564v1

Antimelanoma activity of Heterocapsa triquetra pigments

Quentin Haguet , Antoine Bonnet , Jean-Baptiste Bérard , Joelle Goldberg , Nicolas Joguet , et al.
Algal Research - Biomass, Biofuels and Bioproducts, 2017, 25, pp.207 - 215. ⟨10.1016/j.algal.2017.04.034⟩
Article dans une revue hal-01656289v1
Image document

Antiproliferative Activity of Violaxanthin Isolated from Bioguided Fractionation of Dunaliella tertiolecta Extracts

Virginie Pasquet , Perrine Morisset , Saïd Ihammouine , Amandine Chepied , Lucie Aumailley , et al.
Marine drugs, 2011, 9, pp.819-831. ⟨10.3390/md9050819⟩
Article dans une revue hal-01247755v1