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Enhanced copper-mediated 18 F-fluorination of aryl boronic esters provides eight radiotracers for PET applications
Sean Preshlock
,
Samuel Calderwood
,
Stefan Verhoog
,
Matthew Tredwell
,
Mickael Huiban
,
et al.
Article dans une revue
hal-02011096v1
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Functionalisation Methods and Reagents Used in Such Methods Using an Azaisatoic Anhydride or One of the Derivatives of Same, Biological Molecules Thereby Treated, and Kits
Thomas Cailly
,
Frédéric Fabis
,
Ali Laayoun
,
Alain Laurent
,
Sylvain Ursuegui
France, Patent n° : WO2014019966 (A1). 2014
Brevet
hal-02042938v1
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Design of a serotonin 4 receptor radiotracer with decreased lipophilicity for single photon emission computed tomography
Nathalie Fresneau
,
Noé Dumas
,
Benjamin B. Tournier
,
Christine Fossey
,
Céline Ballandonne
,
et al.
Article dans une revue
hal-02011103v1
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Small-animal single-photon emission computed tomographic imaging of the brain serotoninergic systems in wild-type and mdr1a knockout rats.
Noé Dumas
,
M. Moulin-Sallanon,
,
N. Ginovart,
,
B. Tournier,
,
Peggy Suzanne
,
et al.
Molecular Imaging, 2014, 13, pp.1-12
Article dans une revue
hal-00997602v1
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TSPO and amyloid deposits in sub-regions of the hippocampus in the 3xTgAD mouse model of Alzheimer’s disease
Benjamin B. Tournier
,
Stergios Tsartsalis
,
Daphney Rigaud
,
Christine Fossey
,
Thomas Cailly
,
et al.
Article dans une revue
hal-02011091v1
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General method for the synthesis of substituted phenanthridin-6(5H)-ones using a KOH-mediated anionic ring closure as the key step
Emmanuelle Dubost
,
Rosa Magnelli
,
Thomas Cailly
,
Rémi Legay
,
Frédéric Fabis
,
et al.
Tetrahedron, 2010, 66 (27-28), pp.5008-5016
Article dans une revue
hal-02045912v1
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Selective ortho-bromination of substituted benzaldoximes using Pd-catalyzed C-H activation : Application to the synthesis of substituted 2-bromobenzaldehydes.
Emmanuelle Dubost
,
Christine Fossey
,
Thomas Cailly
,
Sylvain Rault
,
Frédéric Fabis
Journal of Organic Chemistry, 2011, 76 (15), pp.6414-6420
Article dans une revue
hal-01061746v1
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Improvements of C–H Radio-Iodination of N-Acylsulfonamides toward Implementation in Clinics
Emmanuelle Dubost
,
Victor Babin
,
Florian Benoist
,
Alexandra Hébert
,
Gilbert Pigrée
,
et al.
Article dans une revue
hal-02400013v1
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Room-Temperature ortho -Alkoxylation and -Halogenation of N -Tosylbenzamides by Using Palladium(II)-Catalyzed CH Activation
Florent Péron
,
Christine Fossey
,
Jana Sopkova-de Oliveira Santos
,
Thomas Cailly
,
Frédéric Fabis
Article dans une revue
istex
hal-02011110v1
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Boron reagents for divergent radiochemistry
Thomas L. Wilson
,
Thomas Cailly
,
Veronique Gouverneur
Article dans une revue
hal-02010669v1
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Synthesis of the calcilytic ligand NPS 2143.
Henrik Johansson
,
Thomas Cailly
,
Alex Rojas Bie Thomsen
,
Hans Bräuner-Osborne
,
Daniel Pedersen Sejer
Journal of Organic Chemistry, 2013, 9, pp.1383-1387
Article dans une revue
hal-00918393v1
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A general synthesis of diversely substituted indazoles and hetero-aromatic derivatives from o-halo-(het)arylaldehydes or -phenones
Emmanuelle Dubost
,
Silvia Stiebing
,
Thibault Ferrary
,
Thomas Cailly
,
Frédéric Fabis
,
et al.
Article dans une revue
hal-02011108v1
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Design of fluorinated 5-HT4R antagonists: Influence of the basicity and lipophilicity toward the 5-HT4R binding affinities.
Clément Fontenelle
,
Zhong Wang
,
Christine Fossey
,
Bruno Linclau
,
Thomas Cailly
,
et al.
Bioorganic and Medicinal Chemistry, 2013, 21, pp.7529 - 7538
Article dans une revue
hal-00918408v1
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Biotin-conjugated N-methylisatoic anhydride: a chemical tool for nucleic acid separation by selective 2'-hydroxyl acylation of RNA.
Sylvain Ursuegui
,
N. Chivot
,
S. Moutin
,
A. Burr
,
Christine Fossey
,
et al.
Chemical Communications, 2014, 50, pp.5748-5751
Article dans une revue
hal-00997629v1
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N-Tosylcarboxamide as a Transformable Directing Group for Pd-Catalyzed C-H Ortho-Arylation
Florent Péron
,
Christine Fossey
,
Thomas Cailly
,
Frédéric Fabis
Article dans une revue
hal-00821457v1
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Synthesis and Physicochemical Properties of Cryptophazane—A Soluble and Functionalizable C 1 ‐Symmetrical Cryptophane
Clément Vigier
,
Dimitri Fayolle
,
Hussein El Siblani
,
Jana Sopkova - de Oliveira Santos
,
Frederic Fabis
,
et al.
Article dans une revue
hal-03854418v1
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Radiotracers for the Central Serotoninergic System
Reynald Mangeant
,
Emmanuelle Dubost
,
Thomas Cailly
,
Valérie Collot
Article dans une revue
hal-03776739v1
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Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5-HT 4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers
Emmanuelle Dubost
,
Noé Dumas
,
Christine Fossey
,
Rosa Magnelli
,
Sabrina Butt-Gueulle
,
et al.
Article dans une revue
hal-01949598v1
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Synthesis and evaluation of novel serotonin 4 receptor radiotracers for single photon emission computed tomography
Julien Lalut
,
Benjamin B. Tournier
,
Thomas Cailly
,
Cédric Lecoutey
,
Sophie Corvaisier
,
et al.
Article dans une revue
hal-02011098v1
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Design and synthesis of new iodinated diazaphenanthridines as potent 5-HT4R SPECT radiotracers
Victor Babin
,
Tournier B.
,
Davis A.
,
Millet P.
,
Thomas Cailly
,
et al.
Young research fellow meeting (24, 2017), Feb 2017, Châtenay-Malabry, France
Communication dans un congrès
hal-02380919v1
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Site-selective palladium-catalysed C-H radio-iodination: a new access to radiotracers
Victor Babin
,
Dubost E.
,
Benoist F
,
Hébert A.
,
Barbey P.
,
et al.
Journées Nord-Ouest Européennes des Jeunes Chercheurs (JNOEJC, 2018), Jun 2018, Lille, France
Communication dans un congrès
hal-02389257v1
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Two-Step Synthesis of Substituted 3-Aminoindazoles from 2-Bromobenzonitriles
Valérie Lefebvre
,
Thomas Cailly
,
Frédéric Fabis
,
Sylvain Rault
Article dans une revue
hal-02045916v1
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Design of iodinated radioligands for SPECT imaging of central human 5-HT4R using a ligand lipophilicity efficiency approach
Victor Babin
,
Benjamin B. Tournier
,
Audrey Davis
,
Emmanuelle Dubost
,
Gilbert Pigrée
,
et al.
Article dans une revue
hal-02466870v1
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Synthesis of substituted diazino[c]quinolin-5(6H)-ones, diazino[c]isoquinolin-6(5H)-ones, diazino[c]naphthyridin-6(5H)-ones and diazino[c]naphthyridin-5(6H)-ones
Nathalie Fresneau
,
Thomas Cailly
,
Frédéric Fabis
,
J.-P. Bouillon
Article dans une revue
istex
hal-01015241v1
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Radiosynthesis of SPECT tracers via a copper mediated 123 I iodination of (hetero)aryl boron reagents
Thomas L. Wilson
,
Greg Mcsweeney
,
Sean Preshlock
,
Stefan Verhoog
,
Matthew Tredwell
,
et al.
Article dans une revue
hal-02011093v1
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Palladium-Mediated Site-Selective C–H Radio-iodination
Emmanuelle Dubost
,
Victor Babin
,
Florian Benoist
,
Alexandra Hébert
,
Pierre Barbey
,
et al.
Article dans une revue
hal-01950004v1
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Investigation by mass spectrometry and 32P post-labelling of DNA adducts formation from 1,2-naphthoquinone, an oxydated metabolite of naphthalene
Adeline Clergé
,
Jérémie Le Goff
,
Claire Lopez-Piffet
,
Sonnich Meier
,
Stéphanie Lagadu
,
et al.
Article dans une revue
hal-03022040v1
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Synthesis and characterization of a iodine-125-labeled pyrrolo[1,2-a]thieno[3,2-e]pyrazine and evaluation as a potential 5-HT4R SPECT tracer
Thomas Cailly
,
Noé Dumas
,
Philippe Millet
,
Stéphane Lemaître
,
Frédéric Fabis
,
et al.
European Journal of Medicinal Chemistry, 2010, 45 (11), pp.5465-5467
Article dans une revue
hal-02045910v1
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Iodoindazoles with Selective Magnesiation at Position 3: A Route to Highly Functionalized Indazoles
Bao Vy Lam
,
Yohann Berhault
,
Silvia Stiebing
,
Christine Fossey
,
Thomas Cailly
,
et al.
Article dans une revue
istex
hal-02043771v1
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One-pot synthesis of new aza- and diaza-aminopenanthrenes
Christophe Rochais
,
Rodrigue Yougnia
,
Thomas Cailly
,
Jana Sopkova-de Oliveira Santos
,
Sylvain Rault
,
et al.
Article dans une revue
istex
hal-01061754v1
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