Number of documents

28

Sylvie Radix


Maitre de Conférences - HDR

EA4446 B2MC

ISPB - Faculté de Pharmacie de Lyon


Journal articles28 documents

  • Anthony Prandina, Sylvie Radix, Marc Le Borgne, Lars Petter Jordheim, Zineb Bousfiha, et al.. Synthesis and biological evaluation of new dipicolylamine zinc chelators as metallo-β-lactamase inhibitors. Tetrahedron, Elsevier, 2019, 75 (11), pp.1525-1540. ⟨hal-02054167⟩
  • Geir Kildahl-Andersen, Christian Schnaars, Anthony Prandina, Sylvie Radix, Marc Le Borgne, et al.. Synthesis and biological evaluation of zinc chelating compounds as metallo-β-lactamase inhibitors. MedChemComm, Royal Society of Chemistry, In press, ⟨10.1039/C8MD00578H⟩. ⟨hal-02077900⟩
  • Christian Schnaars, Geir Kildahl-Andersen, Anthony Prandina, Roya Popal, Sylvie Large Radix, et al.. Synthesis and preclinical evaluation of TPA-based zinc chelators as metallo-β-lactamase inhibitors. ACS Infectious Diseases, American Chemical Society, 2018, ⟨10.1021/acsinfecdis.8b00137⟩. ⟨hal-01844562⟩
  • Sylvie Radix, Anne Doléans Jordheim, Luc Rocheblave, Serge N'Digo, Anne-Laure Prignon, et al.. N,N′-disubstituted cinnamamide derivatives potentiate ciprofloxacin activity against overexpressing NorA efflux pump Staphylococcus aureus 1199B strains. European Journal of Medicinal Chemistry, Elsevier, 2018, 150, pp.900-907. ⟨10.1016/j.ejmech.2018.03.028⟩. ⟨hal-02149739⟩
  • Sylvie Radix, Anne Doléans Jordheim, Luc Rocheblave, Serge N'Digo, Anne-Laure Prignon, et al.. N,N′-disubstituted cinnamamide derivatives potentiate ciprofloxacin activity against overexpressing NorA efflux pump Staphylococcus aureus 1199B strains. European Journal of Medicinal Chemistry, Elsevier, 2018, 150, pp.900 - 907. ⟨10.1016/j.ejmech.2018.03.028⟩. ⟨hal-01763023⟩
  • Anthony Prandina, Lars Herfindal, Sylvie Radix, Pal Rongved, Stein Døskeland, et al.. Enhancement of iodinin solubility by encapsulation into cyclodextrin nanoparticles. Journal of Enzyme Inhibition and Medicinal Chemistry, Informa Healthcare, 2018, 33 (1), pp.370 - 375. ⟨10.1080/14756366.2017.1421638⟩. ⟨hal-01688994⟩
  • Anthony Prandina, Lars Herfindal, Sylvie Radix, Pal Rongved, Stein Døskeland, et al.. Enhancement of iodinin solubility by encapsulation into cyclodextrin nanoparticles. Journal of Enzyme Inhibition and Medicinal Chemistry, Informa Healthcare, 2018, 33 (1), pp.370-375. ⟨10.1080/14756366.2017.1421638⟩. ⟨hal-02149736⟩
  • Luc Rocheblave, Marc Rolland Ravel, Elodie Monniot, Jeremy Tavenard, Claude-Yves Cuilleron, et al.. Deoxycholic acid derivatives as inhibitors of P-glycoprotein-mediated multidrug efflux. Steroids, 2016, 116 (1878-5867 (Electronic)), pp.5-12. ⟨10.1016/j.steroids.2016.09.017⟩. ⟨hal-01800021⟩
  • Wael Zeinyeh, Sylvie Radix, Raphael Terreux, Julie-Anne Chemelle, Nadia Walchshofer. Unsymmetrical α,ω-end-functionalized oligo(cyclohexylidenes): efficient synthesis and conformational analysis. Tetrahedron, Elsevier, 2016, 72 (27-28), pp.4032 - 4038. ⟨10.1016/j.tet.2016.05.040⟩. ⟨hal-01800196⟩
  • Wael Zeinyeh, Zahia Mahiout, Sylvie Radix, Thierry Lomberget, Axel Dumoulin, et al.. Progesterone–adenine hybrids as bivalent inhibitors of P-glycoprotein-mediated multidrug efflux: Design, synthesis, characterization and biological evaluation. Steroids, Elsevier, 2012, 77 (12), pp.1177 - 1191. ⟨10.1016/j.steroids.2012.07.010⟩. ⟨hal-01800194⟩
  • Wael Zeinyeh, Ghina Alameh, Sylvie Radix, Catherine Grenot, Charles Dumontet, et al.. Design, synthesis and evaluation of progesterone–adenine hybrids as bivalent inhibitors of P-glycoprotein-mediated multidrug efflux. Bioorganic and Medicinal Chemistry Letters, Elsevier, 2010, 20 (10), pp.3165 - 3168. ⟨10.1016/j.bmcl.2010.03.085⟩. ⟨hal-01800193⟩
  • Wael Zeinyeh, Hexue Xia, Philippe Lawton, Sylvie Radix, Christelle Marminon, et al.. Synthesis and modulation properties of imidazo[4,5-b]pyridin-7-one and indazole-4,7-dione derivatives towards the Cryptosporidium parvum CpABC3 transporter. European Journal of Medicinal Chemistry, Elsevier, 2010, 45 (6), pp.2480 - 2488. ⟨10.1016/j.ejmech.2010.02.033⟩. ⟨hal-01800190⟩
  • Wael Zeinyeh, Julien Pilmé, Sylvie Radix, Nadia Walchshofer. Regioselective N-alkylation of imidazo[4,5-b]pyridine-4-oxide derivatives: an experimental and DFT study. Tetrahedron Letters, Elsevier, 2009, 50 (16), pp.1828 - 1833. ⟨10.1016/j.tetlet.2009.02.006⟩. ⟨hal-01800189⟩
  • Marie-Emmanuelle Million, Sylvie Radix, Sébastien Marrot, Magali Imbert, Joëlle Paris. A Simple and High-Yield Route to N-9-purinyl-acetic Acid Derivatives Coupled with Amino Acids. Letters in Organic Chemistry, Bentham Science Publishers, 2008, 5 (6), pp.484 - 489. ⟨10.2174/157017808785740408⟩. ⟨hal-01800186⟩
  • Sylvie Radix, Roland Barret. Total synthesis of two natural phenanthrenes: confusarin and a regioisomer. Tetrahedron, Elsevier, 2007, 63 (50), pp.12379 - 12387. ⟨10.1016/j.tet.2007.09.052⟩. ⟨hal-01800184⟩
  • E. Peter Kündig, Alejandro Bellido, Krishna Kaliappan, Andrew Pape, Sylvie Radix. Synthesis of [6,n] cis-fused ring compounds via Cr-mediated dearomatisation–ring-closing metathesis. Organic and Biomolecular Chemistry, Royal Society of Chemistry, 2006, 4 (2), pp.342 - 351. ⟨10.1039/b513261d⟩. ⟨hal-01800180⟩
  • R. Terreux, P. Iawton, S. Radix, D. Deruaz, M. Lussignol, et al.. Rational design of inhibitors of the cryptosporidium parvum ATP-binding cassette 3 protein.. Abstracts of Papers of the American Chemical Society, American Chemical Society, 2005, 229, pp.U179-U179. ⟨hal-00314914⟩
  • Thierry Lomberget, Sylvie Radix, Roland Barret. A Regioselective Route to 5- and 6-Azaindoles. SYNLETT, Georg Thieme Verlag, 2005, pp.2080 - 2082. ⟨10.1055/s-2005-871946⟩. ⟨hal-01800182⟩
  • Sylvie Radix-Large, Stéphanie Kucharski, Bernard Langlois. Trifluoromethylated Vinylic and Aromatic Compounds from α-(Trifluoro­methyl)allyl Alcohols. SYNTHESIS, Georg Thieme Verlag, 2004, pp.456 - 465. ⟨10.1055/s-2004-815928⟩. ⟨hal-01800179⟩
  • E. Peter Kündig, Alejandro Bellido, Krishna Kaliappan, Andrew Pape, Sylvie Radix. Efficient Access to Fused Ring Compounds via Dearomatization/Ring-Closing Metathesis. SYNLETT, Georg Thieme Verlag, 2003, pp.2407 - 2409. ⟨10.1055/s-2003-43330⟩. ⟨hal-01800173⟩
  • Sylvie Large-Radix, Thierry Billard, Bernard Langlois. Fluoride-assisted trifluoromethylation of aromatic thiones with (trifluoromethyl)trimethylsilane. Journal of Fluorine Chemistry, Elsevier, 2003, 124 (2), pp.147 - 149. ⟨10.1016/S0022-1139(03)00203-3⟩. ⟨hal-01800170⟩
  • Sylvie Large, Nicolas Roques, Bernard Langlois. Nucleophilic Trifluoromethylation of Carbonyl Compounds and Disulfides with Trifluoromethane and Silicon-Containing Bases. Journal of Organic Chemistry, American Chemical Society, 2000, 65 (26), pp.8848 - 8856. ⟨10.1021/jo000150s⟩. ⟨hal-01800146⟩
  • Bouyssi Didier, Marcello Cavicchioli, Sylvie Large, Monteiro Nuno, Geneviève Balme. Rearrangement of Oxasphiroheptanes to Cyclohexanones Mediated by Lithium Iodide. SYNLETT, Georg Thieme Verlag, 2000, 2000 (05), pp.0749 - 0751. ⟨10.1055/s-2000-6606⟩. ⟨hal-01800154⟩
  • Bernard Langlois, Thierry Billard, Sophie Guérin, Sylvie Large, Nathalie Roidot-Perol. Electrophilic Trifluoromethylation of Vinyl Sulfides. Phosphorus, Sulfur, and Silicon and the Related Elements, Taylor & Francis, 1999, 153 (1), pp.323 - 324. ⟨10.1080/10426509908546452⟩. ⟨hal-01800163⟩
  • Thierry Billard, Bernard Langlois, Sylvie Large. Synthesis of Trifluoromethyl Selenides. Phosphorus, Sulfur, and Silicon and the Related Elements, Taylor & Francis, 1998, 136 (1), pp.521 - 524. ⟨10.1080/10426509808545987⟩. ⟨hal-01800167⟩
  • Marie-Noëlle Bouchu, Sylvie Large, Michaela Steng, Bernard Langlois, Jean-Pierre Praly. An unprecedented access to trifluoromethylthiosugar derivatives from thiocyanate precursors upon treatment with trifluoromethyltrimethylsilane. Carbohydrate Research, Elsevier, 1998, 314 (1-2), pp.37 - 45. ⟨10.1016/S0008-6215(98)00289-4⟩. ⟨hal-01800131⟩
  • Thierry Billard, Sylvie Large, Bernard Langlois. Preparation of trifluoromethyl sulfides or selenides from trifluoromethyl trimethylsilane and thiocyanates or selenocyanates. Tetrahedron Letters, Elsevier, 1997, 38 (1), pp.65 - 68. ⟨10.1016/S0040-4039(96)02216-2⟩. ⟨hal-01800102⟩
  • Thierry Billard, Bernard Langlois, Sylvie Large, Daniel Anker, Nathalie Roidot, et al.. A New Route to Thio- and Selenosulfonates from Disulfides and Diselenides. Application to the Synthesis of New Thio- and Selenoesters of Triflic Acid. Journal of Organic Chemistry, American Chemical Society, 1996, 61 (21), pp.7545 - 7550. ⟨10.1021/jo960619c⟩. ⟨hal-01800094⟩