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Identification of a trafficking motif involved in the stabilization and polarization of P2X receptors.
Séverine Chaumont-Dubel
,
Lin-Hua Jiang
,
Aubin Penna
,
R Alan North
,
A. Baranski
Article dans une revue
inserm-00320759v1
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Novel non-sulfonamide 5-HT 6 receptor partial inverse agonist in a group of imidazo[4,5- b ]pyridines with cognition enhancing properties
David Vanda
,
Miroslav Soural
,
Vittorio Canale
,
Séverine Chaumont-Dubel
,
Grzegorz Satała
,
et al.
Article dans une revue
hal-02366387v1
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Amelioration of Tau pathology and memory deficits by targeting 5-HT7 receptor
Josephine Labus
,
Kian-Fritz Röhrs
,
Jana Ackmann
,
Hristo Varbanov
,
Franziska Müller
,
et al.
Article dans une revue
hal-02940990v1
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Novel 1H-Pyrrolo[3,2-c]quinoline Based 5-HT6 Receptor Antagonists with Potential Application for the Treatment of Cognitive Disorders Associated with Alzheimer's Disease
Katarzyna Grychowska
,
Grzegorz Satala
,
Tomasz Kos
,
Anna Partyka
,
Evelina Colacino
,
et al.
Article dans une revue
hal-01941175v1
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International Union of Basic and Clinical Pharmacology. CX. Classification of Receptors for 5-hydroxytryptamine; Pharmacology and Function
Nicholas M Barnes
,
Gerard P Ahern
,
Carine Becamel
,
Joël Bockaert
,
Michael Camilleri
,
et al.
Article dans une revue
hal-03099832v1
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The 5-HT6 receptor interactome: New insight in receptor signaling and its impact on brain physiology and pathologies
Séverine Chaumont-Dubel
,
Vincent Dupuy
,
Joël Bockaert
,
Carine Becamel
,
Philippe Marin
Article dans une revue
hal-02364282v1
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A dual-acting 5-HT 6 receptor inverse agonist/MAO-B inhibitor displays glioprotective and pro-cognitive properties
Vittorio Canale
,
Katarzyna Grychowska
,
Rafał Kurczab
,
Mateusz Ryng
,
Abdul Raheem Keeri
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et al.
Article dans une revue
hal-03029988v1
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2-Phenyl-1 H -pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT 6 Receptor Inverse Agonists with Cognition-Enhancing Activity
Marcin Drop
,
Vittorio Canale
,
Séverine Chaumont-Dubel
,
Rafał Kurczab
,
Grzegorz Satała
,
et al.
Article dans une revue
hal-03192567v1
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Impact of the Substitution Pattern at the Basic Center and Geometry of the Amine Fragment on 5-HT6 and D3R Affinity in the 1H-pyrrolo[3,2-c]quinoline Series
Katarzyna Grychowska
,
Wojciech Pietruś
,
Ludmiła Kulawik
,
Ophélie Bento
,
Grzegorz Satała
,
et al.
Article dans une revue
hal-03956220v1
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Neuropathic pain-alleviating activity of novel 5-HT6 receptor inverse agonists derived from 2-aryl-1H-pyrrole-3-carboxamide
Marcin Drop
,
Florian Jacquot
,
Vittorio Canale
,
Séverine Chaumont-Dubel
,
Maria Walczak
,
et al.
Article dans une revue
hal-03324439v1
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Agonist-dependent Endocytosis of γ-Aminobutyric Acid Type A (GABAA) Receptors Revealed by a γ2(R43Q) Epilepsy Mutation.
Severine Chaumont
,
Caroline André
,
David Perrais
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Eric Boué-Grabot
,
Antoine Taly
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et al.
Article dans une revue
hal-01146637v1
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Dual 5-HT 6 and D 3 Receptor Antagonists in a Group of 1 H -Pyrrolo[3,2- c ]quinolines with Neuroprotective and Procognitive Activity
Katarzyna Grychowska
,
Séverine Chaumont-Dubel
,
Rafał Kurczab
,
Paulina Koczurkiewicz
,
Caroline Deville
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et al.
Article dans une revue
hal-02364291v1
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The atypical chemokine receptor 3 interacts with Connexin 43 inhibiting astrocytic gap junctional intercellular communication
Amos Fumagalli
,
Joyce Heuninck
,
Anne Pizzoccaro
,
Enora Moutin
,
Joyce Koenen
,
et al.
Article dans une revue
hal-02952514v1
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Classification and Signaling Characteristics of 5-HT Receptors: Towards the Concept of 5-HT Receptosomes
Philippe Marin
,
Carine Becamel
,
Séverine Chaumont-Dubel
,
Franck Vandermoere
,
Joël Bockaert
,
et al.
Chapitre d'ouvrage
hal-02491823v1
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A serotonergic axon-cilium synapse drives nuclear signaling to alter chromatin accessibility
Shu-Hsien Sheu
,
Srigokul Upadhyayula
,
Vincent Dupuy
,
Song Pang
,
Fei Deng
,
et al.
Article dans une revue
hal-03796396v1
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Physical interaction between neurofibromin and serotonin 5-HT 6 receptor promotes receptor constitutive activity
Wissem Deraredj Nadim
,
Séverine Chaumont-Dubel
,
Fahima Madouri
,
Laetitia Cobret
,
Marie-Ludivine de Tauzia
,
et al.
Proceedings of the National Academy of Sciences of the United States of America, 2016, 113 (43), pp.12310 - 12315. ⟨10.1073/pnas.1600914113⟩
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Superiority of the Triple-Acting 5-HT 6 R/5-HT 3 R Antagonist and MAO-B Reversible Inhibitor PZ-1922 over 5-HT 6 R Antagonist Intepirdine in Alleviation of Cognitive Deficits in Rats
Katarzyna Grychowska
,
Uriel López-Sánchez
,
Mathieu Vitalis
,
Geoffrey Canet
,
Grzegorz Satała
,
et al.
Article dans une revue
hal-04235140v1
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The serotonin 6 receptor controls neuronal migration during corticogenesis via a ligand-independent Cdk5-dependent mechanism
M. Jacobshagen
,
M. Niquille
,
Séverine Chaumont-Dubel
,
Philippe Marin
,
A. Dayer
Article dans une revue
hal-01950135v1
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Impact of 5-HT6 Receptor Subcellular Localization on Its Signaling and Its Pathophysiological Roles
Séverine Chaumont-Dubel
,
Sonya Galant
,
Matthieu Prieur
,
Tristan Bouschet
,
Joël Bockaert
,
et al.
Article dans une revue
hal-04236957v1
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Early 5‐ HT 6 receptor blockade prevents symptom onset in a model of adolescent cannabis abuse
Coralie Berthoux
,
Al Mahdy Hamieh
,
Angelina Rogliardo
,
Emilie Doucet
,
Camille Coudert
,
et al.
Article dans une revue
hal-02863763v1
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Dynamic interactions of the 5-HT 6 receptor with protein partners control dendritic tree morphogenesis
Camille Pujol
,
Vincent Dupuy
,
Martial Séveno
,
Léonie Runtz
,
Joël Bockaert
,
et al.
Article dans une revue
hal-02485360v1
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1-(Arylsulfonyl-isoindol-2-yl)piperazines as 5-HT6R Antagonists: Mechanochemical Synthesis, In Vitro Pharmacological Properties and Glioprotective Activity
Vittorio Canale
,
Wojciech Trybała
,
Séverine Chaumont-Dubel
,
Paulina Koczurkiewicz-Adamczyk
,
Grzegorz Satała
,
et al.
Article dans une revue
hal-03933561v1
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mTOR activation by constitutively active serotonin6 receptors as new paradigm in neuropathic pain and its treatment
Pierre-Yves Martin
,
Stéphane Doly
,
Al Mahdy Hamieh
,
Eric Chapuy
,
Vittorio Canale
,
et al.
Article dans une revue
hal-02906397v1
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Structure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT 3 and 5-HT 6 Receptor Antagonist with Antipsychotic and Procognitive Properties
Paweł Zajdel
,
Katarzyna Grychowska
,
Szczepan Mogilski
,
Rafał Kurczab
,
Grzegorz Satała
,
et al.
Article dans une revue
hal-03357806v1
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Cdk5 induces constitutive activation of 5-HT6 receptors to promote neurite growth
Fanny Duhr
,
Paul Déléris
,
F. Raynaud
,
Martial Séveno
,
Séverine Morisset-Lopez
,
et al.
Article dans une revue
hal-01178901v1
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Spatiotemporal dynamics of 5-HT6 receptor ciliary localization during mouse brain development
Vincent Dupuy
,
Matthieu Prieur
,
Anne Pizzoccaro
,
Clara Margarido
,
Emmanuel Valjent
,
et al.
Article dans une revue
hal-03900095v1
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Novel and atypical pathways for serotonin signaling
Joël Bockaert
,
Carine Becamel
,
Séverine Chaumont-Dubel
,
Sylvie Claeysen
,
Franck Vandermoere
,
et al.
Article dans une revue
hal-03256253v1
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