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Transcription-associated topoisomerase 2α (TOP2A) activity is a major effector of cytotoxicity induced by G-quadruplex ligands
Madeleine Bossaert
,
Angélique Pipier
,
Jean-Francois Riou
,
Céline Noirot
,
Linh-Trang Nguyên
,
et al.
Article dans une revue
hal-04478256v1
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Phenyl dialkynylcarbinols, a Bioinspired Series of Synthetic Antitumor Acetylenic Lipids
Margaux Bossuat
,
Pauline Rullière
,
Nadège Preuilh
,
Antonio Peixoto
,
Etienne Joly
,
et al.
Article dans une revue
hal-04274040v1
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Dual Processing of R-Loops and Topoisomerase I Induces Transcription-Dependent DNA Double-Strand Breaks
Agnese Cristini
,
Giulia Ricci
,
Sébastien Britton
,
Simona Salimbeni
,
Shar-Yin Naomi Huang
,
et al.
Article dans une revue
hal-02378250v1
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Séparation chirale par chromatographie liquide et par fluide supercritique des analogues cliquables de Jaspine B
Cécile Santos
,
Isabelle Fabing
,
Stéphanie Ballereau
,
Yves Génisson
,
A. Rozie
,
et al.
33e journée Chimie-Biologie-Santé, Apr 2019, Toulouse, France
Poster de conférence
hal-02338505v1
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TRF2 and Apollo Cooperate with Topoisomerase 2α to Protect Human Telomeres from Replicative Damage
Jing Ye
,
Christelle Lenain
,
Serge Bauwens
,
Angela Rizzo
,
Adelaïde Saint-Léger
,
et al.
Article dans une revue
ensl-00817706v1
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Alkyne-Tagged Analogue of Jaspine B: New Tool for Identifying Jaspine B Mode of Action
Alexandrine Rozié
,
Cécile Santos
,
Isabelle Fabing
,
Patrick Calsou
,
Sébastien Britton
,
et al.
Article dans une revue
hal-02059233v1
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Human HDAC1 and HDAC2 function in the DNA-damage response to promote DNA nonhomologous end-joining
Kyle Miller
,
Jorrit Tjeertes
,
Julia Coates
,
Gaëlle Legube
,
Sophie Polo
,
et al.
Article dans une revue
hal-03082153v1
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DNA damage triggers SAF-A and RNA biogenesis factors exclusion from chromatin coupled to R-loops removal
Sébastien Britton
,
Emma Dernoncourt
,
Christine Delteil
,
Carine Froment
,
Odile Schiltz
,
et al.
Article dans une revue
hal-01191434v1
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Bio-inspired antitumor acetylenic lipids bearing alkynylcarbinol pharmacophores
Pauline Rullière
,
Maroua Bourkhis
,
Dymytrii Listunov
,
Hafida Gaspard
,
Valérie Maraval
,
et al.
Flash communication, Congrès SCF18, Jul 2018, Montpellier, France
Communication dans un congrès
hal-02335955v1
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New tool for identification of jaspine B pharmacological target
Stéphanie Ballereau
,
Yves Génisson
,
P. Calsou
,
S. Britton
9ème Ecole Thématique de Criblage, Oct 2018, Carry-Le-Rouet, France
Poster de conférence
hal-02337302v1
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Constrained G4 structures unveil topology specificity of known and new G4 binding proteins
A. Pipier
,
A. Devaux
,
T. Lavergne
,
A. Adrait
,
Y. Couté
,
et al.
Article dans une revue
hal-03369749v1
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Structural and functional basis of inositol hexaphosphate stimulation of NHEJ through stabilization of Ku-XLF interaction
Antonia Kefala Stavridi
,
Amandine Gontier
,
Vincent Morin
,
Philippe Frit
,
Virginie Ropars
,
et al.
Article dans une revue
hal-04284601v1
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ATM antagonizes NHEJ proteins assembly and DNA-ends synapsis at single-ended DNA double strand breaks
Sébastien Britton
,
Pauline Chanut
,
Christine Delteil
,
Nadia Barboule
,
Philippe Frit
,
et al.
Article dans une revue
hal-02989041v1
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SDR enzymes oxidize specific lipidic alkynylcarbinols into cytotoxic protein-reactive species
Pascal Demange
,
Etienne Joly
,
Julien Marcoux
,
Patrick Ra Zanon
,
Dymytrii Listunov
,
et al.
Article dans une revue
hal-03719267v2
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Development of Bioinspired Lipidic Alcynylcarbinol Prodrugs for Targeted Anticancer Therapy.
Margaux Bossuat
,
Nadège Preuilh
,
Stéphanie Ballereau
,
V. Bernades-Génisson
,
Valérie Maraval
,
et al.
Journée Chimie et Cancer du Cancéropole Grand Sud-Ouest, Jun 2023, Toulouse, France
Poster de conférence
hal-04198422v1
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Identification of Three-Way DNA Junction Ligands through Screening of Chemical Libraries and Validation by Complementary in Vitro Assays
Katerina Duskova
,
Jérémy Lamarche
,
Souheila Amor
,
Coralie Caron
,
Nicolas Queyriaux
,
et al.
Article dans une revue
hal-02121543v3
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Biased and unbiased strategies to identify biologically active small molecules.
Valentina Abet
,
Angelica Mariani
,
Fiona R Truscott
,
Sébastien Britton
,
Raphaël Rodriguez
Article dans une revue
hal-01067769v1
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Bioinspired lipidic alkynylcarbinols as anticancer agents
Margaux Bossuat
,
Stéphanie Ballereau
,
Antonio Peixoto
,
Valérie Maraval
,
Vania Bernades-Génisson
,
et al.
Journées de Chimie Organique 2022 (JCO 2022), Nov 2022, Palaiseau, France
Communication dans un congrès
hal-04402220v1
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Mechanism-guided development of covalent prodrugs for targeted anticancer therapy.
Margaux Bossuat
,
Nadège Preuilh
,
Stéphanie Ballereau
,
Antonio Peixoto
,
V. Bernades-Génisson
,
et al.
Journée du GDR ChemBio, Jun 2023, Strasbourg, France
Poster de conférence
hal-04198409v1
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Development of Bioinspired Lipidic Alcynylcarbinol Prodrugs for Targeted Anticancer Therapy.
Margaux Bossuat
,
Nadège Preuilh
,
Stéphanie Ballereau
,
V. Bernades-Génisson
,
Valérie Maraval
,
et al.
Congrès SCF23, Jun 2023, Nantes, France
Poster de conférence
hal-04198468v1
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PAXX binding to the NHEJ machinery explains functional redundancy with XLF
Murielle Seif-El-Dahan
,
Antonia Kefala-Stavridi
,
Philippe Frit
,
Steven Hardwick
,
Dima Chirgadze
,
et al.
Article dans une revue
hal-04234621v1
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Bio-inspired antitumor acetylenic lipids bearing alkynylcarbinol pharmacophores
Pauline Rullière
,
Maroua Bourkhis
,
Dymytrii Listunov
,
Hafida Gaspard
,
Valérie Maraval
,
et al.
10th International Chemistry Conference Toulouse-Kiev (ICTK-10), Jun 2019, Toulouse, France
Poster de conférence
hal-02335633v1
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Chemical inhibition of NAT10 corrects defects of laminopathic cells.
Delphine Larrieu
,
Sébastien Britton
,
Mukerrem Demir
,
Raphaël Rodriguez
,
Stephen P Jackson
Article dans une revue
hal-00988813v1
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Dual targeting of higher-order DNA structures by azacryptands induces DNA junction-mediated DNA damage in cancer cells
Joanna Zell
,
Katerina Duskova
,
Leïla Chouh
,
Madeleine Bossaert
,
Nicolas Chéron
,
et al.
Article dans une revue
hal-03372655v1
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Bioinspired lipidic alkynylcarbinols as anticancer agents
Margaux Bossuat
,
Sébastien Britton
,
Remi Chauvin
,
Yves Génisson
Journées Jeunes Chercheurs SCT, Feb 2023, Paris, France
Poster de conférence
hal-04402496v1
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Transcription-associated topoisomerase activities control DNA-breaks production by G-quadruplex ligands
A Pipier
,
M Bossaert
,
J F Riou
,
C Noirot
,
L-T Nguyễn
,
et al.
2020
Pré-publication, Document de travail
hal-02989065v1
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Alkyne-tagged analogue of jaspine B: new tool for identifying jaspine B mode of action
Stéphanie Ballereau
,
Yves Génisson
,
Patrick Calsou
,
Sébastien Britton
10th International Chemistry Conference Toulouse-Kiev (ICTK-10), Jun 2019, TOULOUSE, France
Communication dans un congrès
hal-02333441v1
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DNA junction ligands trigger DNA damage and are synthetic lethal with DNA repair inhibitors in cancer cells
Katerina Duskova
,
Pauline Lejault
,
Élie Benchimol
,
Régis Guillot
,
Sébastien Britton
,
et al.
Article dans une revue
hal-02412757v1
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XAB2 promotes Ku eviction from single-ended DNA double-strand breaks independently of the ATM kinase
Abhishek Bharadwaj Sharma
,
Hélène Erasimus
,
Lia Pinto
,
Marie-Christine Caron
,
Diyavarshini Gopaul
,
et al.
Article dans une revue
hal-03371180v1
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BRCA1 prevents R-loop-associated centromeric instability
Carine Racca
,
Sébastien Britton
,
Sabrine Hédouin
,
Claire Francastel
,
Patrick Calsou
,
et al.
Article dans une revue
hal-03371200v1
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