Recherche - Archive ouverte HAL Accéder directement au contenu

Filtrer vos résultats

50 résultats
Page :
triés par

Synthesis and evaluation of antiviral cyclopeptides isolated from a tropical plant

 Clément Grisel , Prisca Lagardère , Cécile Apel , Marc Litaudon , Charline Herrscher , et al.
23ème reunion du Groupement Français des Peptides et Protéines (GFPP), Sep 2023, Fournols, France
Poster de conférence hal-04401150v1

Specialized metabolites with antiviral properties from a Vietnamese plant: isolation & synthesis

 Linh Phan , Bastien Petit , Juliano Haddad , Chaker El Kalamouni , Karine Seron , et al.
6ème symposium international de l’AFERP, Jul 2023, Orsay, France
Poster de conférence hal-04401116v1

From biodiversity to the synthesis of anti-apoptotic proteins inhibitors

 Sandy Desrat , Shelly Gapil Tiamas , Khalijah Awang , Alma Abou Samra , Camille Remeur , et al.
8ème Rencontres de Chimie Organique et Bioorganique (RECOB), Mar 2022, Aussois, France.
Poster de conférence hal-04400541v1

Design of chemical probes derived from schweinfurthins to hijack OSBP, implicated in cholesterol homeostasis

 Clément Grisel , Ophélie Bento , Isabel Ramon Martinez , Laurie Azkenatzis , Jérôme Bignon , et al.
27th EFMC International Symposium on Medicinal Chemistry, Sep 2022, Nice, France.
Poster de conférence hal-04400602v1
Image document

Pro-apoptotic carboxamide analogues of natural fislatifolic acid targeting Mcl-1 and Bcl-2

 Shelly Gapil Tiamas , Florian Daressy , Alma Abou Samra , Jérôme Bignon , Vincent Steinmetz , et al.
Bioorganic and Medicinal Chemistry Letters, 2020, 30, pp.127003. ⟨10.1016/j.bmcl.2020.127003⟩
Article dans une revue hal-02483122v1

New dual molecules as an innovative strategy against glioblastoma: synthesis and biological evaluation

 Gwenaëlle Jézéquel , Tiphaine Péresse , Thierry Virolle , Jérome Bignon , Sandy Desrat , et al.
8th EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry, Sep 2019, Athènes, Greece
Poster de conférence hal-04400486v1
Image document

Characterization, Diversity, and Structure-Activity Relationship Study of Lipoamino Acids from Pantoea sp. and Synthetic Analogues

 Seindé Touré , Sandy Desrat , Léonie Pellissier , Pierre-Marie Allard , Jean-Luc Wolfender , et al.
International Journal of Molecular Sciences, 2019, 20 (5), pp.1083. ⟨10.3390/ijms20051083⟩
Article dans une revue hal-02095583v1

Fast & easy preparation of original dispatchers: toward the chemical space exploration

 Dominique Petit , Sandy Desrat , Pascal Retailleau , Vincent Dumontet , Philippe Breton , et al.
17ème Rencontres de Chimie Organique et Bioorganique(RECOB), Mar 2018, Aussois, France
Poster de conférence hal-04394434v1

Les métabolites spécialisés : pour quoi faire ?

 Sandy Desrat
2018
Autre publication scientifique hal-04410215v1

Process for the biobased synthesis of schweinfurthins G, K and R

 Marc Litaudon , Fanny Roussi , Sandy Desrat , Gwenaëlle Jézéquel , Celine Rampal , et al.
France, Patent n° : WO2023/275324. 2023
Brevet hal-04258372v1

Asymmetric Synthesis of Two Analogues of Meiogynin A

 J. Dardenne , S. Desrat , F. Roussi
European Journal of Organic Chemistry, 2013, 11, pp.2116-2122. ⟨10.1002/ejoc.201201628⟩
Article dans une revue istex hal-00912836v1
Image document

NA1—115—7, from Zygogynum pancheri, is a new selective MCL-1 inhibitor inducing the apoptosis of hematological cancer cells but non-toxic to normal blood cells or cardiomyocytes

 Florian Daressy , Line Séguy , Loëtitia Favre , Sophie Corvaisier , Cécile Apel , et al.
Biomedicine and Pharmacotherapy, 2022, 154, pp.113546. ⟨10.1016/j.biopha.2022.113546⟩
Article dans une revue hal-03777709v1

Dual inhibitors of the pro-survival proteins Bcl-2 and Mcl-1 derived from natural compound meiogynin A

 Alma Abou Samra , Aude Robert , Crystal Gov , Loëtitia Favre , Laure Eloy , et al.
European Journal of Medicinal Chemistry, 2018, 148, pp.26-38. ⟨10.1016/j.ejmech.2018.01.100⟩
Article dans une revue hal-02343193v1

Fast & easy preparation of 3D scaffolds from methyl benzoate by a diversity oriented synthesis strategy based on Diels–Alder and ene-reactions

 Dominique Brossard , Pascal Retailleau , Vincent Dumontet , Philippe Breton , Sandy Desrat , et al.
Organic & Biomolecular Chemistry, 2017, 15 (26), pp.5585-5592. ⟨10.1039/C7OB01236E⟩
Article dans une revue hal-02355151v1
Image document

Synthesis and Anti-Leishmanial Properties of Quinolones Derived from Zanthosimuline

 Gwenaëlle Jézéquel , Laura Nogueira de Faria Cardoso , Florent Olivon , Indi Dennemont , Cécile Apel , et al.
Molecules, 2022, 27 (22), pp.7892. ⟨10.3390/molecules27227892⟩
Article dans une revue hal-03853782v1

Ring-rearrangement metathesis of substituted dihydropyrans and dihydrofurans

 Morgan Donnard , Théophile Tschamber , Didier Le Nouen , Sandy Desrat , Karen Hinsinger , et al.
Tetrahedron, 2011, 67 (2), pp.339-357. ⟨10.1016/j.tet.2010.11.036⟩
Article dans une revue istex hal-02319563v1

Synthesis and evaluation of a natural cyclopeptide

 Clément Grisel , Prisca Lagardère , Cécile Apel , Marc Litaudon , Charline Herrscher , et al.
Journée de l’école doctorale Innovation Thérapeutique : du Fondamental à l'Appliqué 2023, Jun 2023, Orsay, France
Poster de conférence hal-04401087v1

Design of chemical probes derived from schweinfurthins to hijack OSBP, implicated in cholesterol homeostasis

 Clément Grisel , Ophélie Bento , Isabel Ramon Martinez , Laurie Azkenatzis , Jérome Bignon , et al.
Journées de Chimie Organique (JCO) 2022, Nov 2022, Palaiseau, France.
Poster de conférence hal-04400652v1

Targeting OSBP degradation by PROTACs derived from schweinfurthin for cancer therapy

 Carole Guimard , Gwenaëlle Jézéquel , Laurie Askenatzis , Jérome Bignon , Sandy Desrat , et al.
27th EFMC International Symposium on Medicinal Chemistry, Sep 2022, Nice, France.
Poster de conférence hal-04400614v1

Toward natural inhibitors of carbapenemases

 Isabel Ramon Martinez , Saoussen Oueslati , Cécile Apel , Thierry Naas , Marc Litaudon , et al.
International Conference TRR261, May 2023, Bad Boll, Germany
Poster de conférence hal-04401004v1

Research of novel organocatalysts for reactions in water from plant extracts

 Sandy Desrat , Laura Nogueira Faria Cardoso , Adrien Vitrai , Cécile Apel , Fanny Roussi
Journées de Chimie Organique (JCO) 2022, Nov 2022, Palaiseau, France
Poster de conférence hal-04400631v1

Toward natural inhibitors of carbapenemases

 Isabel Ramon Martinez , Saoussen Oueslati , Cécile Apel , Thierry Naas , Marc Litaudon , et al.
Journée de l’école doctorale Innovation Thérapeutique : du Fondamental à l'Appliqué 2023, Jun 2023, Orsay, France
Poster de conférence hal-04401075v1

Intramolecular Imino Diels−Alder Reaction: Progress toward the Synthesis of Uncialamycin

 Sandy Desrat , Pierre van de Weghe
Journal of Organic Chemistry, 2009, 74 (17), pp.6728-6734. ⟨10.1021/jo901291t⟩
Article dans une revue hal-02355118v1

Setbacks and Hopes: En Route to the Synthesis of Uncialamycin

 Sandy Desrat , Mickaël Jean , Pierre van de Weghe
Tetrahedron, 2011, 67 (39), pp.7510-7516. ⟨10.1016/j.tet.2011.07.090⟩
Article dans une revue istex hal-00843821v1

Efficient synthetic strategy to access analogues of an original natural bioactive flavone

 Carole Guimard , Gwenaëlle Jézéquel , Laurie Askenatzis , Bruno Mesmin , Jérome Bignon , et al.
Journées de Chimie Organique (JCO) 2022, Nov 2022, Palaiseau, France
Poster de conférence hal-04400644v1

Specialized metabolites with antiviral properties from a Vietnamese plant: isolation & synthesis

 Linh Phan , Bastien Petit , Juliano Haddad , Chaker El Kalamouni , Karine Seron , et al.
Journée de l’école doctorale Innovation Thérapeutique : du Fondamentale à l'Appliqué, Jun 2023, Orsay, France
Poster de conférence hal-04401065v1

From plants to the synthesis of anti-apoptotic proteins inhibitors

 Sandy Desrat , Shelly Gapil Tiamas , Khalijah Awang , Alma Abou Samra , Camille Remeur , et al.
Symposium des metabolites spécialisés du Labex Saclay Plant Science, Jul 2019, Orsay, France
Poster de conférence hal-04400452v1

Methylaluminoxane (MAO)-Assisted Direct Amidation of Esters

 Sandy Desrat , Aline Ducousso , Shelly Gapil , Camille Remeur , Fanny Roussi
SYNLETT, 2015, 26 (03), pp.385-387. ⟨10.1055/s-0034-1378927⟩
Article dans une revue hal-01142881v1

Asymmetric Total Synthesis and Biological Evaluation of Proapoptotic Natural Myrcene-Derived Cyclohexenyl Chalcones

 Shelly Gapil Tiamas , Florian Audet , Alma Abou Samra , Jerome Bignon , Marc Litaudon , et al.
European Journal of Organic Chemistry, 2018, 2018 (42), pp.5830-5835. ⟨10.1002/ejoc.201800262⟩
Article dans une revue hal-02355166v1
Image document

Molecular and cellular dissection of the oxysterol-binding protein cycle through a fluorescent inhibitor

 Tiphaine Peresse , Davidi Kovacs , Mélody Subra , Joelle Bigay , Meng-Chen Tsai , et al.
Journal of Biological Chemistry, 2020, ⟨10.1074/jbc.RA119.012012⟩
Article dans une revue hal-02733227v1
Page :