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	Pour les 58 documents Envoyer sur ORCID RSS ATOM Exporter BibTeX XML-TEI CSV RTF EndNote PDF HTML Export avancé	Page : Page précédente 1 2 Page suivante	triés par Pertinence Auteur A→Z Auteur Z→A Titre A→Z Titre Z→A Date de publication croissante Date de publication décroissante Date de dépôt croissante Date de dépôt décroissante

		4-Substituted Thieno[3,2-d]pyrimidines as Dual-Stage Antiplasmodial Derivatives Prisca Lagardère , Romain Mustière , Nadia Amanzougaghene , Sébastien Hutter , Jean-François Franetich , et al. Pharmaceuticals, 2022, 15 (7), pp.820. ⟨10.3390/ph15070820⟩ Article dans une revue hal-03725749v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Safety Review: Squalene and Thimerosal in Vaccines Marc Montana , Pierre Verhaeghe , Caroline Ducros , Thierry Terme , Patrice Vanelle , et al. Thérapie, 2010, 65 (6), pp.533--541. ⟨10.2515/therapie/2010069⟩ Article dans une revue istex hal-01460254v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium Anita Cohen , Peggy Suzanne , Jean-Charles Lancelot , Pierre Verhaeghe , Aurélien Lesnard , et al. European Journal of Medicinal Chemistry, 2015, 95, pp.16-28. ⟨10.1016/j.ejmech.2015.03.011⟩ Article dans une revue hal-01460555v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Anticancer and anti-inflammatory activities of some new pyrazolo[3,4-b]pyrazines Hussein El-Kashef , Talaat El-Emary , Pierre Verhaeghe , P. Vanelle , Maha Samy Molecules, 2018, 23 (10), pp.2657. ⟨10.3390/molecules23102657⟩ Article dans une revue hal-01954194v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthetic Polypeptide Polymers as Simplified Analogues of Antimicrobial Peptides Pedro Salas-Ambrosio , Antoine Tronnet , Pierre Verhaeghe , Colin Bonduelle Biomacromolecules, 2021, 22 (1), pp.57-75. ⟨10.1021/acs.biomac.0c00797⟩ Article dans une revue hal-02931945v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthèse et évaluations biologiques de nouvelles 8-nitroquinoléin-2(1H)-ones antiparisitaires. Julien Pedron , Clotilde Boudot , Sebastien Hutter , Sandra Bourgeade-Delmas , Lucie Paloque , et al. 8èmes Journées du Consortium anti-Parasitaires et anti-Fongique (CaPF), Mar 2018, Lyon, France Communication dans un congrès hal-01939612v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Albumin-Bound Paclitaxel: The Benefit of This New Formulation in the Treatment of Various Cancers M. Montana , C. Ducros , P. Verhaeghe , T. Terme , P. Vanelle , et al. Journal of Chemotherapy, 2011, 23 (2), pp.59--66 Article dans une revue hal-01460327v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		New nitroaromatic candidats for trypanosomiasis therapeutics. Clotilde Boudot , Cyril Fersing , Julien Pedron , Valere Belle Mbou , Caroline Castera-Ducros , et al. Congress ICOPA (14th International Congress of Parasitology), Aug 2018, Daegu, South Korea Poster de conférence hal-01936829v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Highly efficient microwave assisted α-trichlorination reaction of α-methylated nitrogen containing heterocycles P. Verhaeghe , P. Rathelot , A. Gellis , S. Rault , P. Vanelle Tetrahedron, 2006, 62, pp.8173-8176 Article dans une revue hal-00096229v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		A new DMAP-catalyzed and microwave-assisted approach for introducing heteroarylamino substituents at position 4 of the quinazoline ring. Armand Gellis , Charline Kieffer , Nicolas Primas , Gilles Lanzada , Michel Giorgi , et al. Tetrahedron, 2014, 78 (44), pp.8257-8266. ⟨10.1016/j.tet.2014.09.024⟩ Article dans une revue hal-01417081v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Antiplasmodial 2-thiophenoxy-3-trichloromethyl quinoxalines target the apicoplast of Plasmodium falciparum Dyhia Amrane , Nicolas Primas , Christophe-Sébastien Arnold , Sébastien Hutter , Béatrice Louis , et al. European Journal of Medicinal Chemistry, 2021, 224, pp.113722. ⟨10.1016/j.ejmech.2021.113722⟩ Article dans une revue hal-03323972v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Discovery of a new antileishmanial hit in 8-nitroquinoline series Lucie Paloque , Pierre Verhaeghe , Magali Casanova , Caroline Castera-Ducros , Aurélien Dumètre , et al. European Journal of Medicinal Chemistry, 2012, 54, pp.75-86 Article dans une revue hal-02049707v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis of antiplasmodial 2-aminothieno[3,2-d]pyrimidin-4(3H)-one analogues using the scaffold hopping strategy Romain Mustière , Prisca Lagardère , Sébastien Hutter , Viviana Dell’orco , Nadia Amanzougaghene , et al. European Journal of Medicinal Chemistry, 2022, 241, pp.114619. ⟨10.1016/j.ejmech.2022.114619⟩ Article dans une revue hal-03737417v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Multicenter prospective randomized study comparing the technique of using a bovine pericardium biological prosthesis reinforcement in parietal herniorrhaphy (Tutomesh TUTOGEN) with simple parietal herniorrhaphy, in a potentially contaminated setting Marius Nedelcu , Pierre Verhaeghe , Mehdi Skalli , Gerard Champault , Christophe Barrat , et al. Wound Repair and Regeneration: Official Publication of the Wound Healing Society [and] the European Tissue Repair Society, 2016, 24 (2), p. 427-433. ⟨10.1111/wrr.12386⟩ Article dans une revue istex hal-01474696v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and in vitro evaluation of 4-trichloromethylpyrrolo[1,2-a]quinoxalines as new antiplasmodial agents Nicolas Primas , Peggy Suzanne , Pierre Verhaeghe , Sébastien Hutter , Charline Kieffer , et al. European Journal of Medicinal Chemistry, 2014, 83, pp.26-35. ⟨10.1016/j.ejmech.2014.06.014⟩ Article dans une revue hal-01417058v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Discovery of new hit-molecules targeting Plasmodium falciparum through a global SAR study of the 4-substituted-2-trichloromethylquinazoline antiplasmodial scaffold Justine Desroches , Charline Kieffer , Nicolas Primas , Sébastien Hutter , Armand Gellis , et al. European Journal of Medicinal Chemistry, 2017, 125 (128), pp.68-86. ⟨10.1016/j.ejmech.2016.09.029⟩ Article dans une revue hal-01416990v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Preventing the contamination of hospital personnel by cytotoxic agents: evaluation and training of the para-professional healthcare workers in oncology units C. Kieffer , Pierre Verhaeghe , S. Lagrassa , R. Gregoire , Z. Moussaoui , et al. European Journal of Cancer Care, 2015, 24 (3), pp.404-410. ⟨10.1111/ecc.12249⟩ Article dans une revue istex hal-01460563v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis of New 5- or 7-Substituted 3-Nitroimidazo[1,2-a]pyridine Derivatives Using SNAr and Palladium-Catalyzed Reactions To Explore Antiparasitic Structure–Activity Relationships Romain Paoli-Lombardo , Nicolas Primas , Sandra Bourgeade-Delmas , Alix Sournia-Saquet , Caroline Castera-Ducros , et al. Synthesis: Journal of Synthetic Organic Chemistry, 2023, 56 (8), pp.1297-1308. ⟨10.1055/a-2232-8113⟩ Article dans une revue hal-04503326v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Looking for new antiplasmodial quinazolines: DMAP-catalyzed synthesis of 4-benzyloxy- and 4-aryloxy-2-trichloromethylquinazolines and their in vitro evaluation toward Plasmodium falciparum Armand Gellis , Nicolas Primas , Sébastien Hutter , Gilles Lanzada , Vincent Remusat , et al. European Journal of Medicinal Chemistry, 2016, 119, pp.34-44. ⟨10.1016/j.ejmech.2016.04.059⟩ Article dans une revue hal-01417007v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Tandem synthesis and in vitro antiplasmodial evaluation of new naphtho[2,1-d] thiazole derivatives Anita D Cohen , Pierre Verhaeghe , Maxime D. Crozet , Sébastien Hutter , Pascal Rathelot , et al. European Journal of Medicinal Chemistry, 2012, 55, pp.315--324. ⟨10.1016/j.ejmech.2012.07.034⟩ Article dans une revue istex hal-01460344v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Antileishmanial pharmacomodulation in 8-nitroquinolin-2(1H)-one series Charline Kieffer , Anita Cohen , Pierre Verhaeghe , Lucie Paloque , Sébastien Hutter , et al. Bioorganic and Medicinal Chemistry, 2015, 23 (10), pp.2377-2386. ⟨10.1016/j.bmc.2015.03.064⟩ Article dans une revue hal-01460646v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		The Renewal of Interest in Nitroaromatic Drugs: Towards New Anti-Kinetoplastid Agents Nicolas Primas , Caroline Ducros , Patrice Vanelle , Pierre Verhaeghe Venkatesan Jayaprakash; Daniele Castagnolo; Yusuf Özkay. Medicinal Chemistry of Neglected and Tropical Diseases. Advances in the Design and Synthesis of Antimicrobial Agents, CRC Press, pp.250-280, 2019, 978-1-138-54124-5. ⟨10.1201/9781351011655-12⟩ Chapitre d'ouvrage hal-02923853v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Using the Sonogashira Reaction for Preparing a New Fragment Library based on the 3-alkynylimidazo[1,2-alpha] pyridine Scaffold Caroline Castera-Ducros , Hussein El-Kashef , Melanie Piednoel , Vincent Remusat , Jean-Claude Teulade , et al. Letters in Organic Chemistry, 2016, 13 (7), pp.519-525. ⟨10.2174/1570178613666160919124456⟩ Article dans une revue hal-01460673v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Antitrypanosomatid Pharmacomodulation at Position 3 of the 8-Nitroquinolin-2(1 H)-one Scaffold Using Palladium-Catalysed Cross-Coupling Reactions Julien Pedron , Clotilde Boudot , Sandra Bourgeade-Delmas , Alix Sournia-Saquet , Lucie Paloque , et al. ChemMedChem, 2018, 13 (20), pp.2217-2228. ⟨10.1002/cmdc.201800456⟩ Article dans une revue hal-01888530v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Access to Original Vinylic Chlorides in the Quinazoline Series via a Monoelectronic Transfer Reaction Approach Martine Maillard-Boyer , Caroline Castera-Ducros , Pierre Verhaeghe , France Sifredi , Pascal Rathelot , et al. Molecules, 2010, 15 (4), pp.2719--2729. ⟨10.3390/molecules15042719⟩ Article dans une revue hal-01460257v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and Antiplasmodial Evaluation of 4-Carboxamido- and 4-Alkoxy-2-trichloromethyl Quinazolines Dyhia Amrane , Armand Gellis , Sebastien Hutter , Marion Prieri , Pierre Verhaeghe , et al. Molecules, 2020, 25 (17), pp.3929. ⟨10.3390/molecules25173929⟩ Article dans une revue hal-02924455v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		New 8-Nitroquinolinone Derivative Displaying Submicromolar in Vitro Activities against Both Trypanosoma brucei and cruzi Julien Pedron , Clotilde Boudot , Jean-Yves Brossas , Emilie Pinault , Sandra Bourgeade-Delmas , et al. ACS Medicinal Chemistry Letters, 2020, 11 (4), pp.464-472. ⟨10.1021/acsmedchemlett.9b00566⟩ Article dans une revue hal-02476867v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Effect of N-alkylation in N-carboxyanhydride (NCA) ring-opening polymerization kinetics Pedro Salas-Ambrosio , Antoine Tronnet , Mostafa Badreldin , Sifan Ji , Sébastien Lecommandoux , et al. Polymer Chemistry, 2022, 13, pp.6149-6161. ⟨10.1039/D2PY00985D⟩ Article dans une revue hal-03813069v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Ionic polypeptide polymers with unusual β-sheet stability Michel Nguyen , Jean-Luc Stigliani , Christian Bijani , Pierre Verhaeghe , G. Pratviel , et al. Biomacromolecules, 2018, 19 (10), pp.4068-4074. ⟨10.1021/acs.biomac.8b01084⟩ Article dans une revue hal-01954190v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Regioselective Suzuki-Miyaura Reaction: Application to the Microwave-promoted Synthesis of 4,7-Diarylquinazolines Youssef Kabri , Pierre Verhaeghe , Armand Gellis , Patrice Vanelle Molecules, 2010, 15 (5), pp.2949--2961. ⟨10.3390/molecules15052949⟩ Article dans une revue hal-01460231v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More

Filtrer vos résultats

4-Substituted Thieno[3,2-d]pyrimidines as Dual-Stage Antiplasmodial Derivatives

Safety Review: Squalene and Thimerosal in Vaccines

Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium

Anticancer and anti-inflammatory activities of some new pyrazolo[3,4-b]pyrazines

Synthetic Polypeptide Polymers as Simplified Analogues of Antimicrobial Peptides

Synthèse et évaluations biologiques de nouvelles 8-nitroquinoléin-2(1H)-ones antiparisitaires.

Albumin-Bound Paclitaxel: The Benefit of This New Formulation in the Treatment of Various Cancers

New nitroaromatic candidats for trypanosomiasis therapeutics.

Highly efficient microwave assisted α-trichlorination reaction of α-methylated nitrogen containing heterocycles

A new DMAP-catalyzed and microwave-assisted approach for introducing heteroarylamino substituents at position 4 of the quinazoline ring.

Antiplasmodial 2-thiophenoxy-3-trichloromethyl quinoxalines target the apicoplast of Plasmodium falciparum

Discovery of a new antileishmanial hit in 8-nitroquinoline series

Synthesis of antiplasmodial 2-aminothieno[3,2-d]pyrimidin-4(3H)-one analogues using the scaffold hopping strategy

Multicenter prospective randomized study comparing the technique of using a bovine pericardium biological prosthesis reinforcement in parietal herniorrhaphy (Tutomesh TUTOGEN) with simple parietal herniorrhaphy, in a potentially contaminated setting

Synthesis and in vitro evaluation of 4-trichloromethylpyrrolo[1,2-a]quinoxalines as new antiplasmodial agents

Discovery of new hit-molecules targeting Plasmodium falciparum through a global SAR study of the 4-substituted-2-trichloromethylquinazoline antiplasmodial scaffold

Preventing the contamination of hospital personnel by cytotoxic agents: evaluation and training of the para-professional healthcare workers in oncology units

Synthesis of New 5- or 7-Substituted 3-Nitroimidazo[1,2-a]pyridine Derivatives Using SNAr and Palladium-Catalyzed Reactions To Explore Antiparasitic Structure–Activity Relationships

Looking for new antiplasmodial quinazolines: DMAP-catalyzed synthesis of 4-benzyloxy- and 4-aryloxy-2-trichloromethylquinazolines and their in vitro evaluation toward Plasmodium falciparum

Tandem synthesis and in vitro antiplasmodial evaluation of new naphtho[2,1-d] thiazole derivatives

Antileishmanial pharmacomodulation in 8-nitroquinolin-2(1H)-one series

The Renewal of Interest in Nitroaromatic Drugs: Towards New Anti-Kinetoplastid Agents

Using the Sonogashira Reaction for Preparing a New Fragment Library based on the 3-alkynylimidazo[1,2-alpha] pyridine Scaffold

Antitrypanosomatid Pharmacomodulation at Position 3 of the 8-Nitroquinolin-2(1 H)-one Scaffold Using Palladium-Catalysed Cross-Coupling Reactions

Access to Original Vinylic Chlorides in the Quinazoline Series via a Monoelectronic Transfer Reaction Approach

Synthesis and Antiplasmodial Evaluation of 4-Carboxamido- and 4-Alkoxy-2-trichloromethyl Quinazolines

New 8-Nitroquinolinone Derivative Displaying Submicromolar in Vitro Activities against Both Trypanosoma brucei and cruzi

Effect of N-alkylation in N-carboxyanhydride (NCA) ring-opening polymerization kinetics

Ionic polypeptide polymers with unusual β-sheet stability

Regioselective Suzuki-Miyaura Reaction: Application to the Microwave-promoted Synthesis of 4,7-Diarylquinazolines