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Vinyl nosylates as partner in copper and silver co-catalyzed Sonogashira cross-coupling reactions
Nicolas Cheval
,
Barbara Hoffmann
,
Anna Dikova
,
Fatih Sirindil
,
Philippe Bertus
,
et al.
Article dans une revue
hal-02312575v1
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Convenient and easy access to 2-hydroxycyclopent-2-enones from acylcyanohydrins
Mathilde Pantin
,
Florent Bodinier
,
Jordan Saillour
,
Yassine Youssouf
,
Fabien Boeda
,
et al.
Article dans une revue
hal-02312591v1
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Simple and convenient access to α,α,α-trisubstituted amides by double addition of Grignard reagents to acyl cyanohydrins
Fatma Boukattaya
,
Andrii Stanovych
,
Paul Setzer
,
Souhir Abid
,
Houcine Ammar
,
et al.
Article dans une revue
hal-00752112v1
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Synthesis of New Cyclopropanated Tryptamine Analogues
Claude Szalata
,
Janos Sapi
,
Jan Szymoniak
,
Philippe Bertus
,
Stéphane Gérard
Article dans une revue
hal-00330476v1
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Titanium-Mediated Synthesis of 1,4-Diketones from Grignard Reagents and Acyl Cyanohydrins
Paul Setzer
,
Alice Beauseigneur
,
Morwenna S.M. Pearson-Long
,
Philippe Bertus
Article dans une revue
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hal-00532800v1
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Successive addition of two different Grignard reagents to nitriles: access to α,α-disubstituted propargylamine derivatives
Julien Caillé
,
Fatma Boukattaya
,
Fabien Boeda
,
Morwenna Pearson-Long
,
Houcine Ammar
,
et al.
Article dans une revue
hal-01914744v1
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Cyclopropyl-tryptamine Analogues: Synthesis and Biological Evaluation as 5-HT6 Receptor Ligands
Claude Szalata
,
Jan Szymoniak
,
Frédéric Fabis
,
Sabrina Butt-Gueulle
,
Sylvain Rault
,
et al.
Article dans une revue
istex
hal-00764886v1
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The combination of Prolinoamino Acids and Cyclopropylamino Acids Leads to Fully Functionalized, Stable β-Turns in Water
Karine Guitot
,
Maud Larregola
,
Tarun K. Pradhan
,
Jean-Luc Vasse
,
Solange Lavielle
,
et al.
Article dans une revue
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hal-00593499v1
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Synthesis and biological evaluation of 3-cyano-4H-chromene derivatives bearing carbamate functionality
Fatma Boukattaya
,
Amal Daoud
,
Fabien Boeda
,
Morwenna Pearson-Long
,
Neji Gharsallah
,
et al.
Article dans une revue
hal-01921815v1
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Synthesis of a C-glucosylated cyclopropylamide and evaluation as a glycogen phosphorylase inhibitor
Philippe Bertus
,
Jan Szymoniak
,
Erwann Jeanneau
,
Tibor Docsa
,
Pal Gergely
,
et al.
Article dans une revue
istex
hal-00330492v1
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The spirocyclopropyl moiety as a methyl surrogate in the structure of L-fucosidase and L-rhamnosidase inhibitors
Morwenna Pearson
,
Nicolas Floquet
,
Claudia Bello
,
Pierre Vogel
,
Richard Plantier-Royon
,
et al.
Article dans une revue
istex
hal-00439568v1
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Enantiomerically Pure Cyclopropenylcarbinols as a Source of Chiral Alkylidenecyclopropane Derivatives
Samah Simaan
,
Ahmad Masarwa
,
Philippe Bertus
,
Ilan Marek
Article dans une revue
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hal-02132561v1
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New and easy route to primary cyclopropylamines from nitriles
Philippe Bertus
,
Jan Szymoniak
Article dans une revue
istex
hal-02132524v1
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A concise Stereoselective Synthesis of 2-substituted 1-Aminocyclopropanecarboxylic Acids
Tarun K. Pradhan
,
Antoine Joosten
,
Jean-Luc Vasse
,
Philippe Bertus
,
Philippe Karoyan
,
et al.
Article dans une revue
hal-00420475v1
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Titanium-Catalyzed Cyclopropanation of Boc-Protected Cyanohydrins: A Short Access to Aminocyclopropanecarboxylic Acid Derivatives
Morwenna S.M. Pearson-Long
,
Alice Beauseigneur
,
Philippe Karoyan
,
Jan Szymoniak
,
Philippe Bertus
Article dans une revue
hal-00525607v1
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A Short Access to Symmetrically α,α-Disubstituted α-Amino Acids from Acyl Cyanohydrins
Fatma Boukattaya
,
Julien Caillé
,
Houcine Ammar
,
Florian Rouzier
,
Fabien Boeda
,
et al.
Article dans une revue
hal-02132492v1
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Synthesis of 2-(1-aminocyclopropyl)pyrrolidine-3,4-diol derivatives applying titanium-mediated reaction conditions
Delphine Declerck
,
Albert Nguyen van Nhien
,
Solen Josse
,
Jan Szymoniak
,
Philippe Bertus
,
et al.
Article dans une revue
istex
hal-00711775v1
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Titanium-Mediated Cyclopropanation of Nitriles with Unsaturated Grignard Reagents: Application to the Synthesis of Constrained Lysine Derivatives
Gwénaël Forcher
,
Nathalie Clousier
,
Alice Beauseigneur
,
Paul Setzer
,
Fabien Boeda
,
et al.
Article dans une revue
hal-02132648v1
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Zinc-Mediated Double Addition on Functionalized Nitriles
Julien Caillé
,
Mathilde Pantin
,
Fabien Boeda
,
Morwenna Pearson-Long
,
Philippe Bertus
Article dans une revue
hal-02132643v1
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Cyclopropenylcarbinol Derivatives as new versatile intermediates in organic synthesis : Application to the formation of enantiomerically pure alkylidenecyclopropane derivatives
Samah Simaan
,
Ahmad Masarwa
,
Elinor Zohar
,
Amnon Stanger
,
Philippe Bertus
,
et al.
Article dans une revue
hal-00414338v1
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From Dialkyltitanium Species to Titanacyclopropanes: An Ab Initio Study
Philippe Bertus
Article dans une revue
hal-02359376v1
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Double Addition of Organometallics to Nitriles: Toward an Access to Tertiary Carbinamines
Morwenna Pearson-Long
,
Fabien Boeda
,
Philippe Bertus
Article dans une revue
hal-01914752v1
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Heteromultifunctional Oxazolones as Versatile Linkers for Click Chemistry Reactions
Mathilde Pantin
,
Julien Caillé
,
Fabien Boeda
,
Laurent Fontaine
,
Morwenna Pearson-Long
,
et al.
Article dans une revue
hal-02380743v1
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Asymmetric Titanium-Catalyzed Cyclopropanation of Nitriles with Grignard Reagents
Julien Caillé
,
Paul Setzer
,
Fabien Boeda
,
Morwenna Pearson-Long
,
Philippe Bertus
Article dans une revue
hal-02132515v1
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Reactivity of sugar α-aminonitrile derivatives under titanium-mediated cyclopropanation conditions
Delphine Declerck
,
Solen Josse
,
Albert Nguyen van Nhien
,
Jan Szymoniak
,
Philippe Bertus
,
et al.
Article dans une revue
istex
hal-00711787v1
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A stereoselective access to a ferrocene-based planar chiral triazolium salt
Gwénaël Forcher
,
Andrew Silvanus
,
Pierre de Frémont
,
Béatrice Jacques
,
Morwenna S.M. Pearson-Long
,
et al.
Article dans une revue
hal-02132646v1
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Titanium-Mediated Addition of Grignard Reagents to Acyl Cyanohydrins: Aminocyclopropane versus 1,4-Diketone Formation
Paul Setzer
,
Gwénaël Forcher
,
Fabien Boeda
,
Morwenna Pearson-Long
,
Philippe Bertus
Article dans une revue
istex
hal-02132649v1
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Preparation and Some Synthetic Applications of 2-Hydroxyethyl-Substituted Cyclopropylamines
Antoine Joosten
,
Jean-Luc Vasse
,
Philippe Bertus
,
Jan Szymoniak
Article dans une revue
hal-00330480v1
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Solvent-free direct reductive amination by catalytic use of an organotin reagent incorporated on an ionic liquid
Phuoc Dien Pham
,
Philippe Bertus
,
Stéphanie Legoupy
Article dans une revue
istex
hal-00441088v1
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