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Vinyl nosylates as partner in copper and silver co-catalyzed Sonogashira cross-coupling reactions

Nicolas Cheval , Barbara Hoffmann , Anna Dikova , Fatih Sirindil , Philippe Bertus , et al.
Tetrahedron, 2018, 74 (50), pp.7111-7119. ⟨10.1016/j.tet.2018.10.017⟩
Article dans une revue hal-02312575v1
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Convenient and easy access to 2-hydroxycyclopent-2-enones from acylcyanohydrins

Mathilde Pantin , Florent Bodinier , Jordan Saillour , Yassine Youssouf , Fabien Boeda , et al.
Tetrahedron, 2019, 75 (33), pp.4657-4662. ⟨10.1016/j.tet.2019.07.010⟩
Article dans une revue hal-02312591v1

Simple and convenient access to α,α,α-trisubstituted amides by double addition of Grignard reagents to acyl cyanohydrins

Fatma Boukattaya , Andrii Stanovych , Paul Setzer , Souhir Abid , Houcine Ammar , et al.
Chemical Communications, 2012, 48 (69), pp.8655-8657. ⟨10.1039/c2cc34841a⟩
Article dans une revue hal-00752112v1

Synthesis of New Cyclopropanated Tryptamine Analogues

Claude Szalata , Janos Sapi , Jan Szymoniak , Philippe Bertus , Stéphane Gérard
SYNLETT, 2008, 10, pp.1479-1482. ⟨10.1055/s-2008-1078426⟩
Article dans une revue hal-00330476v1

Titanium-Mediated Synthesis of 1,4-Diketones from Grignard Reagents and Acyl Cyanohydrins

Paul Setzer , Alice Beauseigneur , Morwenna S.M. Pearson-Long , Philippe Bertus
Angewandte Chemie International Edition, 2010, 49, pp.8691-8694. ⟨10.1002/anie.201003923⟩
Article dans une revue istex hal-00532800v1

Successive addition of two different Grignard reagents to nitriles: access to α,α-disubstituted propargylamine derivatives

Julien Caillé , Fatma Boukattaya , Fabien Boeda , Morwenna Pearson-Long , Houcine Ammar , et al.
Organic & Biomolecular Chemistry, 2018, 16 (9), pp.1519 - 1526. ⟨10.1039/c7ob03047a⟩
Article dans une revue hal-01914744v1

Cyclopropyl-tryptamine Analogues: Synthesis and Biological Evaluation as 5-HT6 Receptor Ligands

Claude Szalata , Jan Szymoniak , Frédéric Fabis , Sabrina Butt-Gueulle , Sylvain Rault , et al.
ChemMedChem, 2012, 8 (1), pp.70-73. ⟨10.1002/cmdc.201200396⟩
Article dans une revue istex hal-00764886v1

The combination of Prolinoamino Acids and Cyclopropylamino Acids Leads to Fully Functionalized, Stable β-Turns in Water

Karine Guitot , Maud Larregola , Tarun K. Pradhan , Jean-Luc Vasse , Solange Lavielle , et al.
ChemBioChem, 2011, 12, pp.1039-1042. ⟨10.1002/cbic.201000707⟩
Article dans une revue istex hal-00593499v1

Synthesis and biological evaluation of 3-cyano-4H-chromene derivatives bearing carbamate functionality

Fatma Boukattaya , Amal Daoud , Fabien Boeda , Morwenna Pearson-Long , Neji Gharsallah , et al.
Medicinal Chemistry, 2018, 14, ⟨10.2174/1573406414666181009124449⟩
Article dans une revue hal-01921815v1

Synthesis of a C-glucosylated cyclopropylamide and evaluation as a glycogen phosphorylase inhibitor

Philippe Bertus , Jan Szymoniak , Erwann Jeanneau , Tibor Docsa , Pal Gergely , et al.
Bioorganic and Medicinal Chemistry Letters, 2008, 18 (17), pp.4774-4778. ⟨10.1016/j.bmcl.2008.07.098⟩
Article dans une revue istex hal-00330492v1

The spirocyclopropyl moiety as a methyl surrogate in the structure of L-fucosidase and L-rhamnosidase inhibitors

Morwenna Pearson , Nicolas Floquet , Claudia Bello , Pierre Vogel , Richard Plantier-Royon , et al.
Bioorganic and Medicinal Chemistry, 2009, 17 (23), pp.8020-8026. ⟨10.1016/j.bmc.2009.10.010⟩
Article dans une revue istex hal-00439568v1

Enantiomerically Pure Cyclopropenylcarbinols as a Source of Chiral Alkylidenecyclopropane Derivatives

Samah Simaan , Ahmad Masarwa , Philippe Bertus , Ilan Marek
Angewandte Chemie International Edition, 2006, 45 (24), pp.3963-3965. ⟨10.1002/ANIE.200600556⟩
Article dans une revue istex hal-02132561v1

New and easy route to primary cyclopropylamines from nitriles

Philippe Bertus , Jan Szymoniak
Chemical Communications, 2001, 18, pp.1792-1793. ⟨10.1039/B105293B⟩
Article dans une revue istex hal-02132524v1

A concise Stereoselective Synthesis of 2-substituted 1-Aminocyclopropanecarboxylic Acids

Tarun K. Pradhan , Antoine Joosten , Jean-Luc Vasse , Philippe Bertus , Philippe Karoyan , et al.
European Journal of Organic Chemistry, 2009, 2009 (29), pp.5072-5078. ⟨10.1002/ejoc.200900656⟩
Article dans une revue hal-00420475v1

Titanium-Catalyzed Cyclopropanation of Boc-Protected Cyanohydrins: A Short Access to Aminocyclopropanecarboxylic Acid Derivatives

Morwenna S.M. Pearson-Long , Alice Beauseigneur , Philippe Karoyan , Jan Szymoniak , Philippe Bertus
Synthesis: Journal of Synthetic Organic Chemistry, 2010, 20, pp.3410-3414. ⟨10.1055/s-0030-1258260⟩
Article dans une revue hal-00525607v1

A Short Access to Symmetrically α,α-Disubstituted α-Amino Acids from Acyl Cyanohydrins

Fatma Boukattaya , Julien Caillé , Houcine Ammar , Florian Rouzier , Fabien Boeda , et al.
Synthesis: Journal of Synthetic Organic Chemistry, 2016, 48 (06), pp.906-916. ⟨10.1055/s-0035-1560404⟩
Article dans une revue hal-02132492v1

Synthesis of 2-(1-aminocyclopropyl)pyrrolidine-3,4-diol derivatives applying titanium-mediated reaction conditions

Delphine Declerck , Albert Nguyen van Nhien , Solen Josse , Jan Szymoniak , Philippe Bertus , et al.
Tetrahedron, 2012, 68 (6), pp.1802-1809. ⟨10.1016/j.tet.2011.12.024⟩
Article dans une revue istex hal-00711775v1

Titanium-Mediated Cyclopropanation of Nitriles with Unsaturated Grignard Reagents: Application to the Synthesis of Constrained Lysine Derivatives

Gwénaël Forcher , Nathalie Clousier , Alice Beauseigneur , Paul Setzer , Fabien Boeda , et al.
Synthesis: Journal of Synthetic Organic Chemistry, 2015, 47 (07), pp.992-1006. ⟨10.1055/s-0034-1379978⟩
Article dans une revue hal-02132648v1

Zinc-Mediated Double Addition on Functionalized Nitriles

Julien Caillé , Mathilde Pantin , Fabien Boeda , Morwenna Pearson-Long , Philippe Bertus
Synthesis: Journal of Synthetic Organic Chemistry, 2019, 51 (06), pp.1329-1341. ⟨10.1055/s-0037-1611704⟩
Article dans une revue hal-02132643v1

Cyclopropenylcarbinol Derivatives as new versatile intermediates in organic synthesis : Application to the formation of enantiomerically pure alkylidenecyclopropane derivatives

Samah Simaan , Ahmad Masarwa , Elinor Zohar , Amnon Stanger , Philippe Bertus , et al.
Chemistry - A European Journal, 2009, 15 (34), pp.8449-8464. ⟨10.1002/chem.200901074⟩
Article dans une revue hal-00414338v1

From Dialkyltitanium Species to Titanacyclopropanes: An Ab Initio Study

Philippe Bertus
Organometallics, 2019, 38 (21), pp.4171-4182. ⟨10.1021/acs.organomet.9b00509⟩
Article dans une revue hal-02359376v1

Double Addition of Organometallics to Nitriles: Toward an Access to Tertiary Carbinamines

Morwenna Pearson-Long , Fabien Boeda , Philippe Bertus
Advanced Synthesis and Catalysis, 2017, 359 (2), pp.179-201. ⟨10.1002/adsc.201600727⟩
Article dans une revue hal-01914752v1

Heteromultifunctional Oxazolones as Versatile Linkers for Click Chemistry Reactions

Mathilde Pantin , Julien Caillé , Fabien Boeda , Laurent Fontaine , Morwenna Pearson-Long , et al.
European Journal of Organic Chemistry, 2019, 2019 (44), pp.7359-7366. ⟨10.1002/ejoc.201901350⟩
Article dans une revue hal-02380743v1

Asymmetric Titanium-Catalyzed Cyclopropanation of Nitriles with Grignard Reagents

Julien Caillé , Paul Setzer , Fabien Boeda , Morwenna Pearson-Long , Philippe Bertus
SynOpen, 2018, 02 (01), pp.0041-0049. ⟨10.1055/s-0036-1591933⟩
Article dans une revue hal-02132515v1

Reactivity of sugar α-aminonitrile derivatives under titanium-mediated cyclopropanation conditions

Delphine Declerck , Solen Josse , Albert Nguyen van Nhien , Jan Szymoniak , Philippe Bertus , et al.
Tetrahedron, 2012, 68 (4), pp.1145-1152. ⟨10.1016/j.tet.2011.11.067⟩
Article dans une revue istex hal-00711787v1

A stereoselective access to a ferrocene-based planar chiral triazolium salt

Gwénaël Forcher , Andrew Silvanus , Pierre de Frémont , Béatrice Jacques , Morwenna S.M. Pearson-Long , et al.
Journal of Organometallic Chemistry, 2015, 797, pp.1-7. ⟨10.1016/j.jorganchem.2015.07.038⟩
Article dans une revue hal-02132646v1

Titanium-Mediated Addition of Grignard Reagents to Acyl Cyanohydrins: Aminocyclopropane versus 1,4-Diketone Formation

Paul Setzer , Gwénaël Forcher , Fabien Boeda , Morwenna Pearson-Long , Philippe Bertus
European Journal of Organic Chemistry, 2014, 2014 (1), pp.171-180. ⟨10.1002/ejoc.201301251⟩
Article dans une revue istex hal-02132649v1

Preparation and Some Synthetic Applications of 2-Hydroxyethyl-Substituted Cyclopropylamines

Antoine Joosten , Jean-Luc Vasse , Philippe Bertus , Jan Szymoniak
SYNLETT, 2008, 16, pp.2455-2458. ⟨10.1055/s-2008-1078180⟩
Article dans une revue hal-00330480v1

Solvent-free direct reductive amination by catalytic use of an organotin reagent incorporated on an ionic liquid

Phuoc Dien Pham , Philippe Bertus , Stéphanie Legoupy
Chemical Communications, 2009, 41, pp.6207-6209. ⟨10.1039/b912697j⟩
Article dans une revue istex hal-00441088v1