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	Pour les 61 documents Envoyer sur ORCID RSS ATOM Exporter BibTeX XML-TEI CSV RTF EndNote PDF HTML Export avancé	Page : Page précédente 1 2 3 Page suivante	triés par Pertinence Auteur A→Z Auteur Z→A Titre A→Z Titre Z→A Date de publication croissante Date de publication décroissante Date de dépôt croissante Date de dépôt décroissante

		Molecular Features of the YAP Inhibitor Verteporfin: Synthesis of Hexasubstituted Dipyrrins as Potential Inhibitors of YAP/TAZ, the Downstream Effectors of the Hippo Pathway Floriane Gibault , Fabrice Bailly , Mathieu Corvaisier , Mathilde Coevoet , Guillemette Huet , et al. ChemMedChem, 2017, 52nd International Conference on Medicinal Chemistry, 12 (12), pp.954-961. ⟨10.1002/cmdc.201700063⟩ Article dans une revue hal-02060557v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Antagonists of the adenosine A 2A receptor based on a 2-arylbenzoxazole scaffold: Investigation of the C5- and C7-positions to enhance affinity Romain Duroux , Laurence Agouridas , Nicolas Renault , Jamal El Bakali , Christophe Furman , et al. European Journal of Medicinal Chemistry, 2018, 144, pp.151-163. ⟨10.1016/j.ejmech.2017.12.007⟩ Article dans une revue hal-02060715v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		The EGF Domains of MUC4 Oncomucin Mediate HER2 Binding Affinity and Promote Pancreatic Cancer Cell Tumorigenesis Nicolas Stoup , Maxime Liberelle , Céline Schulz , Sumeyye Cavdarli , Romain Vasseur , et al. Cancers, 2021, 13 (22), pp.5746. ⟨10.3390/cancers13225746⟩ Article dans une revue hal-03641795v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		A β-secretase modulator decreases Tau pathology and preserves short-term memory in a mouse model of neurofibrillary degeneration Marie Tautou , Sabiha Eddarkaoui , Florian Descamps , Paul-Emmanuel Larchanché , Mélanie Dumoulin , et al. 2021 Pré-publication, Document de travail hal-03203349v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Identification of a New Benzimidazole Derivative as an Antiviral against Hepatitis C Virus Thibaut Vausselin , Karin Séron , Muriel Lavie , Ahmed Atef Mesalam , Matthieu Lemasson , et al. Journal of Virology, 2016, 90 (19), pp.8422-8434. ⟨10.1128/JVI.00404-16⟩ Article dans une revue hal-02060744v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Design, synthesis and evaluation of 2-aryl benzoxazoles as promising hit for the A2A receptor Romain Duroux , Nicolas Renault , Joana Esteves , Laurence Agouridas , David Blum , et al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2017, 32 (1), pp.850-864. ⟨10.1080/14756366.2017.1334648⟩ Article dans une revue hal-02060508v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Design, synthesis and antimalarial activity of a glyoxylylhydrazone library Adina Ryckebusch , J-S Fruchart , L Cattiaux , P Rousselot-Paillet , V Leroux , et al. Bioorganic and Medicinal Chemistry Letters, 2004, 14 (17), pp.4439-4443. ⟨10.1016/j.bmcl.2004.06.056⟩ Article dans une revue istex mnhn-02070128v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Pharmacomodulations around an anti-Alzheimer drug-candidate Sylvain Marc , Christophe Mésangeau , Mathilde Coevoet , Amélie Barczyk , Stéphane Burlet , et al. European Journal of Medicinal Chemistry Reports, 2022, 4, pp.100020. ⟨10.1016/j.ejmcr.2021.100020⟩ Article dans une revue hal-04403572v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Quinazoline and phthalazine derivatives as novel melatonin receptor ligands analogues of agomelatine Raphaël Bolteau , Florian Descamps , Mohamed Ettaoussi , Daniel H. Caignard , Philippe Delagrange , et al. European Journal of Medicinal Chemistry, 2020, 189, pp.112078. ⟨10.1016/j.ejmech.2020.112078⟩ Article dans une revue hal-03489716v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline Sandrine Delarue-Cochin , Philippe Grellier , L Maes , Elisabeth Mouray , Christian Sergheraert , et al. European Journal of Medicinal Chemistry, 2008, 43 (10), pp.2045-2055. ⟨10.1016/j.ejmech.2007.11.003⟩ Article dans une revue istex mnhn-02070092v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Design, Synthesis and Evaluation of a Series of 1,5‐Diaryl‐1,2,3‐triazole‐4‐carbohydrazones as Inhibitors of the YAP‐TAZ/TEAD Complex Floriane Gibault , Manon Sturbaut , Mathilde Coevoet , Martine Pugnière , Ashley Burtscher , et al. ChemMedChem, 2021, 16 (18), pp.2823-2844. ⟨10.1002/cmdc.202100153⟩ Article dans une revue hal-04481612v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		MUC4-ErbB2 Oncogenic Complex: Binding studies using Microscale Thermophoresis Maxime Liberelle , Romain Magnez , Xavier Thuru , Yamina Bencheikh , Séverine Ravez , et al. Scientific Reports, 2019, 9 (1), ⟨10.1038/s41598-019-53099-0⟩ Article dans une revue hal-02407901v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		(Hetero)aryl substituted thiazol-2,4-yl scaffold as human carbonic anhydrase I, II, VII and XIV activators Marouan Rami , Jean-Yves Winum , Claudiu T Supuran , Patricia Melnyk , Saïd Yous Journal of Enzyme Inhibition and Medicinal Chemistry, 2019, 34 (1), pp.224-229. ⟨10.1080/14756366.2018.1543292⟩ Article dans une revue hal-02060639v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and pharmacological evaluation of benzannulated derivatives as potent and selective sigma-1 protein ligands Marion Donnier-Marechal , Pascal Carato , Delphine Le Broc , Christophe Furman , Patricia Melnyk European Journal of Medicinal Chemistry, 2014, ⟨10.1016/j.ejmech.2014.01.013⟩ Article dans une revue hal-02060851v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		6-Sulfonylbenzothiazolones as potential scaffolds for the design of 5-HT6 ligands Paul-Emmanuel Larchanche , Vincent Ultré , Delphine Le Broc , Céline Ballandonne , Christophe Furman , et al. European Journal of Medicinal Chemistry, 2015, 92, pp.807-817. ⟨10.1016/j.ejmech.2015.01.052⟩ Article dans une revue hal-01116521v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives Elodie Landagaray , Mohamed Ettaoussi , Romain Duroux , J.A. Boutin , Daniel-Henri Caignard , et al. European Journal of Medicinal Chemistry, 2016, 109, pp.360-370. ⟨10.1016/j.ejmech.2015.12.047⟩ Article dans une revue hal-02060776v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Chloroquine and Chloroquinoline Derivatives as Models for the Design of Modulators of Amyloid Peptide Precursor Metabolism Patricia Melnyk , Valérie Vingtdeux , Stéphane Burlet , Sabiha Eddarkaoui , Marie-Eve Grosjean , et al. ACS Chemical Neuroscience, 2015, 6 (4), pp.559-569. ⟨10.1021/cn5003013⟩ Article dans une revue hal-02060814v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and Biological Evaluation of N -[2-(4-Hydroxyphenylamino)-pyridin-3-yl]-4-methoxy-benzenesulfonamide (ABT-751) Tricyclic Analogues as Antimitotic and Antivascular Agents with Potent in Vivo Antitumor Activity Zacharie Segaoula , Julien Leclercq , Valérie Verones , Nathalie Flouquet , Marie Lecoeur , et al. Journal of Medicinal Chemistry, 2016, 59 (18), pp.8422-8440. ⟨10.1021/acs.jmedchem.6b00847⟩ Article dans une revue hal-02060584v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Toward the Discovery of a Novel Class of YAP–TEAD Interaction Inhibitors by Virtual Screening Approach Targeting YAP–TEAD Protein–Protein Interface Floriane Gibault , Mathilde Coevoet , Manon Sturbaut , Amaury Farce , Nicolas Renault , et al. Cancers, 2018, 10 (5), pp.140. ⟨10.3390/cancers10050140⟩ Article dans une revue hal-02060686v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		30th Franco-Belgian conference of pharmacochemistry Charlotte Bouckaert , Eric Goffin , Sebastien Dilly , Julien Hanson , Lionel Pochet , et al. Pharmaceuticals, 2016, 9 (4), pp.73. ⟨10.3390/ph9040073⟩ Article dans une revue hal-02141338v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		EGF-Containing Membrane-Bound Mucins: A Hidden ErbB2 Targeting Pathway? Maxime Liberelle , Nicolas Jonckheere , Patricia Melnyk , Isabelle van Seuningen , Nicolas Lebègue Journal of Medicinal Chemistry, 2020, 63 (10), pp.5074-5088. ⟨10.1021/acs.jmedchem.9b02001⟩ Article dans une revue hal-02955348v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Conception, synthèse et évaluation de composés à visée antipaludique, analogues de l'amodiaquine Emilia Paunescu , Philippe Grellier , Patricia Melnyk 20èmes Journées Franco-Belges de Pharmacochimie, 2006, Lille, France Communication dans un congrès hal-00101274v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and antimalarial activity of new amino analogues of amodiaquine. E Paunescu , Sophie Susplugas , E Boll , R A Varga , Elisabeth Mouray , et al. Medicinal Chemistry, 2008, 4 (5), pp.405-427. ⟨10.2174/157340608785700153⟩ Article dans une revue mnhn-02070086v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Discovery of the first peptide ligand targeting the EGF2 domain of MUC4 that rescues accessibility and sensitivity of pancreatic cancer cells to Herceptin targeted therapy Isabelle Van Seuningen , Nicolas Stoup , Maxime Liberelle , Leila Moum , Nicolas Renault , et al. XXXVIIèmes Journées Scientifiques Annuelles du Club Français du Pancréas (CFP), Club Français du Pancréas; La Cité des Échanges, Marcq-en-Barœul, Sep 2023, Lille, France Communication dans un congrès hal-04547238v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Discovery of a cryptic site at the interface 2 of TEAD – Towards a new family of YAP/TAZ-TEAD inhibitors Manon Sturbaut , Fabrice Bailly , Mathilde Coevoet , Pasquale Sileo , Martine Pugniere , et al. European Journal of Medicinal Chemistry, 2021, 226, pp.113835. ⟨10.1016/j.ejmech.2021.113835⟩ Article dans une revue hal-03429462v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthèse et évaluation biologique de nouveaux antipaludiques de la famille des 4-aminoquinolines Patricia Melnyk Conférence sur invitation à l'IRCOF, 2006, Rouen, France Communication dans un congrès hal-00101295v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Design, synthesis and in vitro antimalarial activity of an acylhydrazone library Patricia Melnyk , Virginie A. Leroux , Christian Sergheraert , Philippe Grellier Bioorganic and Medicinal Chemistry Letters, 2006, 16, pp.31-35 Article dans une revue hal-00097328v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Safe and Efficient Sigma1 Ligand: A Potential Drug Candidate for Multiple Sclerosis. Bénédicte Oxombre , Farima Madouri , Anne-Sophie Journe , Severine Ravez , Eloise Woitrain , et al. International Journal of Molecular Sciences, 2022, International Journal of Molecular Sciences, 23 (19), pp.11893. ⟨10.3390/ijms231911893⟩ Article dans une revue hal-04144548v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		High-affinity σ1 protein agonist reduces clinical and pathological signs of experimental autoimmune encephalomyelitis Bénédicte Oxombre , Catalina Lee Chang , Alain Duhamel , Marion Toussaint , Mariane Giroux , et al. British Journal of Pharmacology, 2015, 172 (7), pp.1769-1782. ⟨10.1111/bph.13037⟩ Article dans une revue hal-02060823v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Replacement of the 4′-Hydroxy Group of Amodiaquine and Amopyroquine by Aromatic and Aliphatic Substituents: Synthesis and Antimalarial Activity E Paunescu , Sophie Susplugas , E Boll , R Varga , Elisabeth Mouray , et al. ChemMedChem, 2009, 4 (4), pp.549-561. ⟨10.1002/cmdc.200800318⟩ Article dans une revue istex mnhn-02070078v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More

Filtrer vos résultats

Molecular Features of the YAP Inhibitor Verteporfin: Synthesis of Hexasubstituted Dipyrrins as Potential Inhibitors of YAP/TAZ, the Downstream Effectors of the Hippo Pathway

Antagonists of the adenosine A 2A receptor based on a 2-arylbenzoxazole scaffold: Investigation of the C5- and C7-positions to enhance affinity

The EGF Domains of MUC4 Oncomucin Mediate HER2 Binding Affinity and Promote Pancreatic Cancer Cell Tumorigenesis

A β-secretase modulator decreases Tau pathology and preserves short-term memory in a mouse model of neurofibrillary degeneration

Identification of a New Benzimidazole Derivative as an Antiviral against Hepatitis C Virus

Design, synthesis and evaluation of 2-aryl benzoxazoles as promising hit for the A2A receptor

Design, synthesis and antimalarial activity of a glyoxylylhydrazone library

Pharmacomodulations around an anti-Alzheimer drug-candidate

Quinazoline and phthalazine derivatives as novel melatonin receptor ligands analogues of agomelatine

Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline

Design, Synthesis and Evaluation of a Series of 1,5‐Diaryl‐1,2,3‐triazole‐4‐carbohydrazones as Inhibitors of the YAP‐TAZ/TEAD Complex

MUC4-ErbB2 Oncogenic Complex: Binding studies using Microscale Thermophoresis

(Hetero)aryl substituted thiazol-2,4-yl scaffold as human carbonic anhydrase I, II, VII and XIV activators

Synthesis and pharmacological evaluation of benzannulated derivatives as potent and selective sigma-1 protein ligands

6-Sulfonylbenzothiazolones as potential scaffolds for the design of 5-HT6 ligands

Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives

Chloroquine and Chloroquinoline Derivatives as Models for the Design of Modulators of Amyloid Peptide Precursor Metabolism

Synthesis and Biological Evaluation of N -[2-(4-Hydroxyphenylamino)-pyridin-3-yl]-4-methoxy-benzenesulfonamide (ABT-751) Tricyclic Analogues as Antimitotic and Antivascular Agents with Potent in Vivo Antitumor Activity

Toward the Discovery of a Novel Class of YAP–TEAD Interaction Inhibitors by Virtual Screening Approach Targeting YAP–TEAD Protein–Protein Interface

30th Franco-Belgian conference of pharmacochemistry

EGF-Containing Membrane-Bound Mucins: A Hidden ErbB2 Targeting Pathway?

Conception, synthèse et évaluation de composés à visée antipaludique, analogues de l'amodiaquine

Synthesis and antimalarial activity of new amino analogues of amodiaquine.

Discovery of the first peptide ligand targeting the EGF2 domain of MUC4 that rescues accessibility and sensitivity of pancreatic cancer cells to Herceptin targeted therapy

Discovery of a cryptic site at the interface 2 of TEAD – Towards a new family of YAP/TAZ-TEAD inhibitors

Synthèse et évaluation biologique de nouveaux antipaludiques de la famille des 4-aminoquinolines

Design, synthesis and in vitro antimalarial activity of an acylhydrazone library

Safe and Efficient Sigma1 Ligand: A Potential Drug Candidate for Multiple Sclerosis.

High-affinity σ1 protein agonist reduces clinical and pathological signs of experimental autoimmune encephalomyelitis

Replacement of the 4′-Hydroxy Group of Amodiaquine and Amopyroquine by Aromatic and Aliphatic Substituents: Synthesis and Antimalarial Activity