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Molecular Features of the YAP Inhibitor Verteporfin: Synthesis of Hexasubstituted Dipyrrins as Potential Inhibitors of YAP/TAZ, the Downstream Effectors of the Hippo Pathway
Floriane Gibault
,
Fabrice Bailly
,
Mathieu Corvaisier
,
Mathilde Coevoet
,
Guillemette Huet
,
et al.
Article dans une revue
hal-02060557v1
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Antagonists of the adenosine A 2A receptor based on a 2-arylbenzoxazole scaffold: Investigation of the C5- and C7-positions to enhance affinity
Romain Duroux
,
Laurence Agouridas
,
Nicolas Renault
,
Jamal El Bakali
,
Christophe Furman
,
et al.
Article dans une revue
hal-02060715v1
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MUC4-ErbB2 Oncogenic Complex: Binding studies using Microscale Thermophoresis
Maxime Liberelle
,
Romain Magnez
,
Xavier Thuru
,
Yamina Bencheikh
,
Séverine Ravez
,
et al.
Article dans une revue
hal-02407901v1
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Synthesis and pharmacological evaluation of benzannulated derivatives as potent and selective sigma-1 protein ligands
Marion Donnier-Marechal
,
Pascal Carato
,
Delphine Le Broc
,
Christophe Furman
,
Patricia Melnyk
Article dans une revue
hal-02060851v1
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Design, Synthesis and Evaluation of a Series of 1,5‐Diaryl‐1,2,3‐triazole‐4‐carbohydrazones as Inhibitors of the YAP‐TAZ/TEAD Complex
Floriane Gibault
,
Manon Sturbaut
,
Mathilde Coevoet
,
Martine Pugnière
,
Ashley Burtscher
,
et al.
Article dans une revue
hal-04481612v1
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6-Sulfonylbenzothiazolones as potential scaffolds for the design of 5-HT6 ligands
Paul-Emmanuel Larchanche
,
Vincent Ultré
,
Delphine Le Broc
,
Céline Ballandonne
,
Christophe Furman
,
et al.
Article dans une revue
hal-01116521v1
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(Hetero)aryl substituted thiazol-2,4-yl scaffold as human carbonic anhydrase I, II, VII and XIV activators
Marouan Rami
,
Jean-Yves Winum
,
Claudiu T Supuran
,
Patricia Melnyk
,
Saïd Yous
Article dans une revue
hal-02060639v1
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Melatonergic ligands: Design, synthesis and pharmacological evaluation of novel series of naphthofuranic derivatives
Elodie Landagaray
,
Mohamed Ettaoussi
,
Romain Duroux
,
J.A. Boutin
,
Daniel-Henri Caignard
,
et al.
Article dans une revue
hal-02060776v1
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Design, synthesis and evaluation of 2-aryl benzoxazoles as promising hit for the A2A receptor
Romain Duroux
,
Nicolas Renault
,
Joana Esteves
,
Laurence Agouridas
,
David Blum
,
et al.
Article dans une revue
hal-02060508v1
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Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline
Sandrine Delarue-Cochin
,
Philippe Grellier
,
L Maes
,
Elisabeth Mouray
,
Christian Sergheraert
,
et al.
Article dans une revue
istex
mnhn-02070092v1
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A β-secretase modulator decreases Tau pathology and preserves short-term memory in a mouse model of neurofibrillary degeneration
Marie Tautou
,
Sabiha Eddarkaoui
,
Florian Descamps
,
Paul-Emmanuel Larchanché
,
Mélanie Dumoulin
,
et al.
2021
Pré-publication, Document de travail
hal-03203349v1
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The EGF Domains of MUC4 Oncomucin Mediate HER2 Binding Affinity and Promote Pancreatic Cancer Cell Tumorigenesis
Nicolas Stoup
,
Maxime Liberelle
,
Céline Schulz
,
Sumeyye Cavdarli
,
Romain Vasseur
,
et al.
Article dans une revue
hal-03641795v1
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Quinazoline and phthalazine derivatives as novel melatonin receptor ligands analogues of agomelatine
Raphaël Bolteau
,
Florian Descamps
,
Mohamed Ettaoussi
,
Daniel H. Caignard
,
Philippe Delagrange
,
et al.
Article dans une revue
hal-03489716v1
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Identification of a New Benzimidazole Derivative as an Antiviral against Hepatitis C Virus
Thibaut Vausselin
,
Karin Séron
,
Muriel Lavie
,
Ahmed Atef Mesalam
,
Matthieu Lemasson
,
et al.
Article dans une revue
hal-02060744v1
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Design, synthesis and antimalarial activity of a glyoxylylhydrazone library
Adina Ryckebusch
,
J-S Fruchart
,
L Cattiaux
,
P Rousselot-Paillet
,
V Leroux
,
et al.
Article dans une revue
istex
mnhn-02070128v1
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Pharmacomodulations around an anti-Alzheimer drug-candidate
Sylvain Marc
,
Christophe Mésangeau
,
Mathilde Coevoet
,
Amélie Barczyk
,
Stéphane Burlet
,
et al.
Article dans une revue
hal-04403572v1
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High-affinity σ1 protein agonist reduces clinical and pathological signs of experimental autoimmune encephalomyelitis
Bénédicte Oxombre
,
Catalina Lee Chang
,
Alain Duhamel
,
Marion Toussaint
,
Mariane Giroux
,
et al.
Article dans une revue
hal-02060823v1
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Carboline- and phenothiazine-derivated heterocycles as potent SIGMA-1 protein ligands
Marion Donnier-Marechal
,
Paul-Emmanuel Larchanché
,
Delphine Le Broc
,
Christophe Furman
,
Pascal Carato
,
et al.
Article dans une revue
hal-02060843v1
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High ligand efficiency quinazoline compounds as novel A2A adenosine receptor antagonists
Raphaël Bolteau
,
Romain Duroux
,
Amelie Laversin
,
Brandon Vreulz
,
Anna Shiriaeva
,
et al.
Article dans une revue
hal-04402301v1
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Safe and Efficient Sigma1 Ligand: A Potential Drug Candidate for Multiple Sclerosis.
Bénédicte Oxombre
,
Farima Madouri
,
Anne-Sophie Journe
,
Severine Ravez
,
Eloise Woitrain
,
et al.
International Journal of Molecular Sciences, 2022, International Journal of Molecular Sciences, 23 (19), pp.11893. ⟨10.3390/ijms231911893⟩
Article dans une revue
hal-04144548v1
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Synthèse et évaluation biologique de nouveaux antipaludiques de la famille des 4-aminoquinolines
Patricia Melnyk
Conférence sur invitation à l'IRCOF, 2006, Rouen, France
Communication dans un congrès
hal-00101295v1
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Replacement of the 4′-Hydroxy Group of Amodiaquine and Amopyroquine by Aromatic and Aliphatic Substituents: Synthesis and Antimalarial Activity
E Paunescu
,
Sophie Susplugas
,
E Boll
,
R Varga
,
Elisabeth Mouray
,
et al.
Article dans une revue
istex
mnhn-02070078v1
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Design, synthesis and in vitro antimalarial activity of an acylhydrazone library
Patricia Melnyk
,
Virginie A. Leroux
,
Christian Sergheraert
,
Philippe Grellier
Bioorganic and Medicinal Chemistry Letters, 2006, 16, pp.31-35
Article dans une revue
hal-00097328v1
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Synthesis and biological evaluation of new naphtho- and quinolinocyclopentane derivatives as potent melatoninergic (MT 1 /MT 2 ) and serotoninergic (5-HT 2C ) dual ligands
Romain Duroux
,
Marouan Rami
,
Elodie Landagaray
,
Mohamed Ettaoussi
,
Daniel-Henri Caignard
,
et al.
Article dans une revue
hal-02011786v1
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New phenylaniline derivatives as modulators of amyloid protein precursor metabolism
Marion Gay
,
Pascal Carato
,
Mathilde Coevoet
,
Nicolas Renault
,
Paul-Emmanuel Larchanché
,
et al.
Article dans une revue
hal-02060708v1
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Direct and Regioselective C(sp3)–H Bond Fluorination of 2-Alkylazaarenes with Selectfluor
Clothilde Le Guen
,
Ahmed Mazzah
,
Maël Penhoat
,
Patricia Melnyk
,
Christian Rolando
,
et al.
Article dans une revue
hal-03061701v1
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New quinolinic derivatives as melatonergic ligands: Synthesis and pharmacological evaluation
Elodie Landagaray
,
Mohamed Ettaoussi
,
Marouan Rami
,
J.A. Boutin
,
Daniel Henri Caignard
,
et al.
Article dans une revue
hal-02060568v1
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Synthesis and pharmacological evaluation of dual ligands for melatonin (MT1/MT2) and serotonin 5-HT2C receptor subtypes (II)
Mohamed Ettaoussi
,
Basile Peres
,
A Errazani
,
J.A. Boutin
,
Daniel-Henri Caignard
,
et al.
Article dans une revue
hal-02060835v1
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Synthesis and pharmacological evaluation of benzamide derivatives as potent and selective sigma-1 protein ligands
Marion Donnier-Marechal
,
Pascal Carato
,
Paul-Emmanuel Larchanché
,
Séverine Ravez
,
Rajâa Boulahjar
,
et al.
Article dans une revue
hal-02011792v1
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Probing the role of the covalent linkage of ferrocene into a chloroquine template
Christophe Biot
,
Wassim Daher
,
Cheikh M. Ndiaye
,
Patricia Melnyk
,
Bruno Pradines
,
et al.
Article dans une revue
istex
hal-00097346v1
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