Recherche - Archive ouverte HAL Accéder directement au contenu

Filtrer vos résultats

40 résultats
Image document

Mixed Polymeric Micelles for Rapamycin Skin Delivery

Guillaume Le Guyader , Bernard Do , Ivo Rietveld , Pascale Coric , Serge Bouaziz , et al.
Pharmaceutics, 2022, 14 (3), pp.569. ⟨10.3390/pharmaceutics14030569⟩
Article dans une revue hal-03843621v1

Potent and systemically active aminopeptidase N inhibitors designed from active-site investigation

Marie Claude Fournie-Zaluski , Pascale Coric , Serge Turcaud , Luce Bruetschy , Evelyne Lucas , et al.
Journal of Medicinal Chemistry, 1992, 35 (7), pp.1259-1266. ⟨10.1021/jm00085a013⟩
Article dans une revue istex hal-02461529v1
Image document

Nuclear Magnetic Resonance Structure of the Human Polyoma JC Virus Agnoprotein

Pascale Coric , A. Sami Saribas , Magid Abou-Gharbia , Wayne Childers , Jon Condra , et al.
Journal of Cellular Biochemistry, 2017, 118 (10), pp.3268-3280. ⟨10.1002/jcb.25977⟩
Article dans une revue hal-02122339v1

Investigation of the Active Site of Aminopeptidase A Using a Series of New Thiol-Containing Inhibitors

Eric Chauvel , Pascale Coric , Catherine Llorens-Cortès , Sherwin Wilk , Bernard P. Roques , et al.
Journal of Medicinal Chemistry, 1994, 37 (9), pp.1339-1346. ⟨10.1021/jm00035a014⟩
Article dans une revue istex hal-02461480v1

Differential Inhibition of Aminopeptidase A and Aminopeptidase N by New .beta.-Amino Thiols

Eric Chauvel , Catherine Llorens-Cortès , Pascale Coric , Sherwin Wilk , Bernard P. Roques , et al.
Journal of Medicinal Chemistry, 1994, 37 (18), pp.2950-2957. ⟨10.1021/jm00044a016⟩
Article dans une revue istex hal-02461510v1
Image document

Characterization of a Novel Type of HIV-1 Particle Assembly Inhibitor Using a Quantitative Luciferase-Vpr Packaging-Based Assay

Gaëlle Gonzalez , Sandrina Dafonseca , Elisabeth Errazuriz , Pascale Coric , Florence Souquet , et al.
PLoS ONE, 2011, 6 (11), pp.e27234. ⟨10.1371/journal.pone.0027234⟩
Article dans une revue hal-02122413v1

Guttiferone A Aggregates Modulate Silent Information Regulator 1 (SIRT1) Activity

Kévin Cottet , Bin Xu , Pascale Coric , Serge Bouaziz , Michel Michel , et al.
Journal of Medicinal Chemistry, 2016, 59 (20), pp.9560-9566. ⟨10.1021/acs.jmedchem.6b01182⟩
Article dans une revue hal-02122343v1

Design of Orally Active Dual Inhibitors of Neutral Endopeptidase and Angiotensin-Converting Enzyme with Long Duration of Action

Marie-Claude Fournie-Zaluski , Pascale Coric , Vincent Théry , Walter D Gonzalez , Hervé Meudal , et al.
Journal of Medicinal Chemistry, 1996, 39 (13), pp.2594-2608. ⟨10.1021/jm950783c⟩
Article dans une revue istex hal-02122108v1

New Dual Inhibitors of Neutral Endopeptidase and Angiotensin-Converting Enzyme: Rational Design, Bioavailability, and Pharmacological Responses in Experimental Hypertension

Marie-Claude Fournie-Zaluski , Pascale Coric , Serge Turcaud , Nathalie Rousselet , Walter D Gonzalez , et al.
Journal of Medicinal Chemistry, 1994, 37 (8), pp.1070-1083. ⟨10.1021/jm00034a005⟩
Article dans une revue istex hal-02461485v1
Image document

Structural studies of the binding of an antagonistic cyclic peptide to the VEGFR1 domain 2

Lei Wang , Pascale Coric , Sylvain Broussy , Rossella Di Stasi , Lingyu Zhou , et al.
European Journal of Medicinal Chemistry, 2019, 169, pp.65-75. ⟨10.1016/j.ejmech.2019.02.069⟩
Article dans une revue hal-02122310v1
Image document

Genuine selective caspase-2 inhibition with new irreversible small peptidomimetics

Elodie Bosc , Julie Anastasie , Feryel Soualmia , Pascale Coric , Ju Youn Kim , et al.
Cell Death and Disease, 2022, 13 (11), pp.959. ⟨10.1038/s41419-022-05396-2⟩
Article dans une revue hal-04275435v1

Extensive biochemical and pharmacological studies of the first systemically-active, mixed inhibitors of enkephalin-degrading enzymes

B.R. Roques , P. Coric , F. Noble , R. Maldonado , P. Delay-Goyet , et al.
European Journal of Pharmacology, 1990, 183 (6), pp.2315-2316. ⟨10.1016/0014-2999(90)93871-M⟩
Article dans une revue istex hal-02461556v1

Optimal Recognition of Neutral Endopeptidase and Angiotensin-Converting Enzyme Active Sites by Mercaptoacyldipeptides as a Means To Design Potent Dual Inhibitors

Pascale Coric , Serge Turcaud , Hervé Meudal , Bernard Pierre Roques , Marie-Claude Fournie-Zaluski
Journal of Medicinal Chemistry, 1996, 39 (6), pp.1210-1219. ⟨10.1021/jm950590p⟩
Article dans une revue istex hal-02122055v1

Toward an optimal joint recognition of the S1' subsites of endothelin converting enzyme-1 (ECE-1), angiotensin converting enzyme (ACE), and neutral endopeptidase (NEP).

Nicolas Inguimbert , Pascale Coric , Hervé Poras , Hervé Meudal , Franck Teffot , et al.
Journal of Medicinal Chemistry, 2002, 45 (7), pp.1477-86
Article dans une revue hal-02122182v1
Image document

Expression of novel proteins by polyomaviruses and recent advances in the structural and functional features of agnoprotein of JC virus, BK virus, and simian virus 40

A. Sami Saribas , Pascale Coric , Serge Bouaziz , Mahmut Safak
Journal of Cellular Physiology, 2019, 234 (6), pp.8295-8315. ⟨10.1002/jcp.27715⟩
Article dans une revue hal-02122318v1

β-Amino-thiols Inhibit the Zinc Metallopeptidase Activity of Tetanus Toxin Light Chain

Loïc M Martin , Fabrice Cornille , Pascale Coric , Bernard P. Roques , Marie-Claude Fournie-Zaluski
Journal of Medicinal Chemistry, 1998, 41 (18), pp.3450-3460. ⟨10.1021/jm981015z⟩
Article dans une revue istex hal-02461413v1

Novel approaches in the development of new analgesics

Bp Roques , G Gacel , V. Daugé , A Baamonde , G Calenco , et al.
Neurophysiologie Clinique = Clinical Neurophysiology, 1990, 20 (5), pp.369-387. ⟨10.1016/s0987-7053(05)80205-9⟩
Article dans une revue istex hal-02461566v1

Synthesis and in vitro activities of new non-peptidic APA Inhibitors

N. Inguimbert , P. Coric , H. Dhotel , E. Bonnard , C. Llorens-Cortes , et al.
The Journal of Peptide Research, 2005, 65 (2), pp.175-188. ⟨10.1111/j.1399-3011.2004.00211.x⟩
Article dans une revue istex hal-02461342v1

Targeting the Proangiogenic VEGF-VEGFR Protein-Protein Interface with Drug-like Compounds by In Silico and In Vitro Screening

Benoit Gautier , Maria A. Miteva , Victor Goncalves , Florent Huguenot , Pascale Coric , et al.
Chemistry and Biology, 2011, 18 (12), pp.1631-1639. ⟨10.1016/j.chembiol.2011.10.016⟩
Article dans une revue hal-01061760v1

Synthesis and separation of tritiated inhibitors of aminopeptidase A and their prodrugs

Nicolas Inguimbert , Pascale Coric , Hélène Dhotel , Catherine Llorens-Cortès , Marie-Claude Fournie-Zaluski , et al.
Journal of Labelled Compounds and Radiopharmaceuticals, 2004, 47 (13), pp.997-1005. ⟨10.1002/jlcr.888⟩
Article dans une revue istex hal-02461363v1
Image document

Insight into the mechanism of action of EP-39, a bevirimat derivative that inhibits HIV-1 maturation

Aymeric Neyret , Bernard Gay , Anaïs Cransac , Laurence Briant , Pascale Coric , et al.
Antiviral Research, 2019, 164, pp.162-175. ⟨10.1016/j.antiviral.2019.02.014⟩
Article dans une revue hal-02147099v1

Pain-suppressive effects on various nociceptive stimuli (thermal, chemical, electrical and inflammatory) of the first orally active enkephalin-metabolizing enzyme inhibitor RB 120

Florence Noble , Claire Smadja , Olga Valverde , Rafael Maldonado , Pascale Coric , et al.
Pain, 1997, 73 (3), pp.383-391. ⟨10.1016/S0304-3959(97)00125-5⟩
Article dans une revue istex hal-02461424v1

Synthesis and characterization of water-soluble macrocyclic peptides stabilizing protein α-turn

Lei Wang , Pascale Coric , Kexin Zhu , Wang-Qing Liu , Michel Vidal , et al.
Organic & Biomolecular Chemistry, 2018, 16 (3), pp.459-471. ⟨10.1039/c7ob02852k⟩
Article dans une revue hal-02122321v1
Image document

Emerging From the Unknown: Structural and Functional Features of Agnoprotein of Polyomaviruses

A. Sami Saribas , Pascale Coric , Anahit Hamazaspyan , William Davis , Rachael Axman , et al.
Journal of Cellular Physiology, 2016, 231 (10), pp.2115-2127. ⟨10.1002/jcp.25329⟩
Article dans une revue hal-02460685v1

Aminophosphinic inhibitors as transition state analogues of enkephalin-degrading enzymes: A class of central analgesics

H. Chen , F. Noble , P. Coric , M.-C. Fournie-Zaluski , B. Roques
Proceedings of the National Academy of Sciences of the United States of America, 1998, 95 (20), pp.12028-12033. ⟨10.1073/pnas.95.20.12028⟩
Article dans une revue hal-03456417v1

Unexpected formation of new chiral 3-amino-5-alkyl-2,5-dihydro-1H-pyrrolin-2-ones from N-Boc-α-amino esters

Nicolas Inguimbert , Hélène Dhotel , Pascale Coric , Bernard P. Roques
Tetrahedron Letters, 2005, 46 (20), pp.3517-3520. ⟨10.1016/j.tetlet.2005.03.067⟩
Article dans une revue istex hal-02461306v1

The 3-O-(3',3'-dimethylsuccinyl) derivative of betulinic acid (DSB) inhibits the assembly of virus-like particles in HIV-1 Gag precursor-expressing cells.

Sandrina Dafonseca , Armand Blommaert , Pascale Coric , Saw See Hong , Serge Bouaziz , et al.
Antiviral Therapy, 2019, 12 (8), pp.1185-203
Article dans une revue hal-02122515v1

CCK-B receptors in the limbic system modulate the antidepressant-like effects induced by endogenous enkephalins

Claire Smadja , Fernando Ruiz , Pascale Coric , Marie Claude Fournié-Zaluski , Bernard P. Roques , et al.
Psychopharmacology, 1997, 132 (3), pp.227-236. ⟨10.1007/s002130050340⟩
Article dans une revue istex hal-02461428v1

Phosphinic derivatives as new dual enkephalin-degrading enzyme inhibitors: synthesis, biological properties, and antinociceptive activities.

H Chen , F Noble , A Mothé , H Meudal , P Coric , et al.
Journal of Medicinal Chemistry, 2000, 43 (7), pp.1398-408
Article dans une revue hal-02122153v1

Antinociception induced by exogenous and endogenous opioids: Role of different brain structures

O. Valverde , P. Coric , B.P. Roques , R. Maldonado
Regulatory Peptides, 1994, 54 (1), pp.309-310. ⟨10.1016/0167-0115(94)90513-4⟩
Article dans une revue istex hal-02461434v1