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C5-DNA methyltransferase inhibitors: from screening to effects on zebrafish embryo development.

 Alexandre Ceccaldi , Arumugam Rajavelu , Christine Champion , Christine Rampon , Renata Z. Jurkowska , et al.
ChemBioChem, 2011, (12) (9), pp.1337-45. ⟨10.1002/cbic.201100130⟩
Article dans une revue istex hal-00632453v1
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New insights into the role of DNA methylation in Biomphalaria glabrata infection susceptibility

 Nelia Luviano , Marie Lopez , Fleur Gawehns , Cristian Chaparro , Paola B Arimondo , et al.
XVI Symposium on Schistosomiasis, FIOCRUZ, Nov 2022, Ouro Preto, Brazil
Communication dans un congrès hal-03963335v1

Synthesis and biological study of a new series of 4'-O-Demethyl-epipodophyllotoxin derivatives.

 M. Duca , D. Guianvarc'H , P. Meresse , E. Bertounesque , Daniel Dauzonne , et al.
Journal of Medicinal Chemistry, 2005, 48(2), pp.593-603
Article dans une revue hal-00017177v1
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Hemisynthetic alkaloids derived from trilobine are antimalarials with sustained activity in multidrug-resistant Plasmodium falciparum

 Flore Nardella , Irina Dobrescu , Haitham Hassan , Fabien Rodrigues , Sabine Thiberge , et al.
iScience, 2023, 26 (2), pp.105940. ⟨10.1016/j.isci.2023.105940⟩
Article dans une revue pasteur-04099097v1

Triplex Formation on DNA Targets: How To Choose the Oligonucleotide

 Pierre Vekhoff , Alexandre Ceccaldi , David Polverari , Jean Pylouster , Claudio Pisano , et al.
Biochemistry, 2008, 47 (47), pp.12277-12289
Article dans une revue hal-01991319v1
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Targeting DNA Methylation with Small Molecules: What’s Next?

 Alexandre Erdmann , Ludovic Halby , Jacques Fahy , Paola B Arimondo
Journal of Medicinal Chemistry, 2015, 58 (6), pp.2569-2583. ⟨10.1021/jm500843d⟩
Article dans une revue hal-03043209v1

Identification of novel quinazoline derivatives as potent antiplasmodial agents

 Anne Bouchut , Dante Rotili , Christine Pierrot , Sergio Valente , Sophia Lafitte , et al.
European Journal of Medicinal Chemistry, 2019, 161, pp.277-291. ⟨10.1016/j.ejmech.2018.10.041⟩
Article dans une revue pasteur-03036828v1

DNA Methylation Analysis of ChIP Products at Single Nucleotide Resolution by Pyrosequencing®

 Céline Moison , Fanny Assemat , Antoine Daunay , Paola B Arimondo , Jörg Tost
Pyrosequencing, 1315, Springer, pp.315 - 333, 2015, Methods in Molecular Biology, 978-1-4939-2715-9. ⟨10.1007/978-1-4939-2715-9_22⟩
Chapitre d'ouvrage pasteur-03046253v1
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The Many Faces of Epigenetics Oxford, December 2017

 Paola Arimondo , Anouk Barberousse , Gaëlle Pontarotti
Epigenetics, 2019, 14 (6), pp.623-631. ⟨10.1080/15592294.2019.1595298⟩
Article dans une revue pasteur-03026588v1
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Malaria Parasite Stress Tolerance Is Regulated by DNMT2-Mediated tRNA Cytosine Methylation

 Elie Hammam , Ameya Sinha , Sebastian Baumgarten , Flore Nardella , Jiaqi Liang , et al.
mBio, 2021, 12, pp.e02558-21. ⟨10.1128/mBio.02558-21⟩
Article dans une revue pasteur-03427780v1

Combined analysis of DNA methylation and cell cycle in cancer cells

 Cecile Desjobert , Mounir El Mai , Tom Gerard-Hirne , Dominique Guianvarc'H , Arnaud Carrier , et al.
Epigenetics, 2015, 10 (1), pp.82-91. ⟨10.1080/15592294.2014.995542⟩
Article dans une revue hal-01365337v1
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Targeting DOT1L for mixed-lineage rearranged leukemia

 Corentin Bon , Yang Si , Paola B Arimondo
Histone Modifications in Therapy, 20, Elsevier, pp.81-99, 2020, Translational Epigenetics, 978-0-12-816422-8. ⟨10.1016/B978-0-12-816422-8.00005-2⟩
Chapitre d'ouvrage pasteur-03414682v1
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Non-canonical functions of UHRF1 maintain DNA methylation homeostasis in cancer cells

 Kosuke Yamaguchi , Xiaoying Chen , Brianna Rodgers , Fumihito Miura , Pavel Bashtrykov , et al.
2023
Pré-publication, Document de travail hal-04295168v1
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The methylome of Biomphalaria glabrata and other mollusks: enduring modification of epigenetic landscape and phenotypic traits by a new DNA methylation inhibitor

 Nelia Luviano , Marie Lopez , Fleur Gawehns , Cristian Chaparro , Paola B Arimondo , et al.
Epigenetics & Chromatin, 2021, 14 (1), pp.48. ⟨10.1186/s13072-021-00422-7⟩
Article dans une revue pasteur-03427775v2

The DNMT3A R882H mutant displays altered flanking sequence preferences

 Max Emperle , Arumugam Rajavelu , Stefan Kunert , Paola Arimondo , Richard Reinhardt , et al.
Nucleic Acids Research, 2018, 46 (6), pp.3130-3139. ⟨10.1093/nar/gky168⟩
Article dans une revue hal-02383683v1

DNA Methyltransferase Inhibitors: Development and Applications

 Marie Lopez , Ludovic Halby , Paola Arimondo
DNA Methyltransferases - Role and Function, pp.431-473, 2016, ⟨10.1007/978-3-319-43624-1_16⟩
Chapitre d'ouvrage hal-02399858v1
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Wandering along the epigenetic timeline

 Clémence Topart , Emilie Werner , Paola B Arimondo
Clinical Epigenetics, 2020, 12 (1), pp.97. ⟨10.1186/s13148-020-00893-7⟩
Article dans une revue pasteur-03043377v1
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DNA Methylation Targeting: The DNMT/HMT Crosstalk Challenge

 Omar Castillo-Aguilera , Patrick Depreux , Ludovic Halby , Paola B. Arimondo , Laurence Goossens
Biomolecules, 2017, 7 (1), pp.3. ⟨10.3390/biom7010003⟩
Article dans une revue pasteur-03043584v1
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Identification of Chemical Probes Targeting MBD2

 Diane Erdmann , Jean Contreras , Rémy Le Meur , Bruno Vitorge , Vincent Saverat , et al.
ACS Chemical Biology, 2022, Published as part of the ACS Chemical Biology special issue “Epigenetics 2022”., 17 (6), pp.1415-1426. ⟨10.1021/acschembio.1c00959⟩
Article dans une revue pasteur-03688129v1

Rapid synthesis of new DNMT inhibitors derivatives of procainamide.

 Ludovic Halby , Christine Champion , Catherine Sénamaud-Beaufort , Sophie Ajjan , Thierry Drujon , et al.
ChemBioChem, 2012, 13 ((1)), pp.157-65. ⟨10.1002/cbic.201100522⟩
Article dans une revue istex hal-00680950v1
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Procainamide-SAHA fused inhibitors of hHDAC6 tackle multi-drug resistant malaria parasites

 Flore Nardella , Ludovic Halby , Irina Dobrescu , Johanna Viluma , Corentin Bon , et al.
Journal of Medicinal Chemistry, 2021, 64 (14), pp.10403-10417. ⟨10.1021/acs.jmedchem.1c00821⟩
Article dans une revue hal-03264653v1
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Natural Products and Chemical Biology Tools: Alternatives to Target Epigenetic Mechanisms in Cancers

 Santiago Lascano , Marie Lopez , Paola B Arimondo
Chemical Record, 2018, 18 (12), pp.1854-1876. ⟨10.1002/tcr.201800133⟩
Article dans une revue hal-03082748v1

Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells

 Sergio Valente , Yiwei Liu , Michael Schnekenburger , Clemens Zwergel , Sandro Cosconati , et al.
Journal of Medicinal Chemistry, 2014, 57 (3), pp.701-713. ⟨10.1021/jm4012627⟩
Article dans une revue hal-01494552v1
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Properly Substituted Analogues of BIX-01294 Lose Inhibition of G9a Histone Methyltransferase and Gain Selective Anti-DNA Methyltransferase 3A Activity

 Dante Rotili , Domenico Tarantino , Biagina Marrocco , Christina Gros , Véronique Masson , et al.
PLoS ONE, 2014, 9 (5), pp.e96941. ⟨10.1371/journal.pone.0096941⟩
Article dans une revue pasteur-03182293v1
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Consequences of combining siRNA-mediated DNA methyltransferase 1 depletion with 5-aza-2′-deoxycytidine in human leukemic KG1 cells

 Stéphane Vispé , Arthur Deroide , Emeline Davoine , Cécile Desjobert , Fabrice Lestienne , et al.
Oncotarget, 2015, 6 (17), pp.15265-15282. ⟨10.18632/oncotarget.3317⟩
Article dans une revue pasteur-03043762v1
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Demethylation by low-dose 5-aza-2′-deoxycytidine impairs 3D melanoma invasion partially through miR-199a-3p expression revealing the role of this miR in melanoma

 Cécile Desjobert , Arnaud Carrier , Audrey Delmas , Diego Marzese , Antoine Daunay , et al.
Clinical Epigenetics, 2019, 11 (1), pp.9. ⟨10.1186/s13148-018-0600-2⟩
Article dans une revue hal-02332300v1

Identification of Novel Inhibitors of DNA Methylation by Screening of a Chemical Library.

 Alexandre Ceccaldi , Arumugam Rajavelu , Sergey Ragozin , Catherine Sénamaud-Beaufort , Pavel Bashtrykov , et al.
ACS Chemical Biology, 2013, 8 (3), pp.543-548. ⟨10.1021/cb300565z⟩
Article dans une revue hal-00777786v1

Hijacking DNA methyltransferase transition state analogues to produce chemical scaffolds for PRMT inhibitors

 Ludovic Halby , Nils Marechal , Dany Pechalrieu , Vincent Cura , Don-Marc Franchini , et al.
Philosophical Transactions of the Royal Society B: Biological Sciences, 2018, 373 (1748), pp.20170072. ⟨10.1098/rstb.2017.0072⟩
Article dans une revue hal-02094589v1
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The timeline of epigenetic drug discovery: from reality to dreams

 A. Ganesan , Paola Arimondo , Marianne Rots , Carmen Jeronimo , María Berdasco
Clinical Epigenetics, 2019, 11 (1), pp.174. ⟨10.1186/s13148-019-0776-0⟩
Article dans une revue pasteur-03036836v1

Espoirs et promesses de la méthylation de l’ADN et des histones comme cibles anticancéreuses

 Corentin Bon , Diane Erdmann , Ludovic Halby , Paola B Arimondo
Bulletin du Cancer, 2019, 106 (10), pp.823-833. ⟨10.1016/j.bulcan.2019.08.001⟩
Article dans une revue hal-02383686v1
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