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	Pour les 53 documents Envoyer sur ORCID RSS ATOM Exporter BibTeX XML-TEI CSV RTF EndNote PDF HTML Export avancé	Page : Page précédente 1 2 Page suivante	triés par Pertinence Auteur A→Z Auteur Z→A Titre A→Z Titre Z→A Date de publication croissante Date de publication décroissante Date de dépôt croissante Date de dépôt décroissante

		A facile consensus ranking approach enhances virtual screening robustness and identifies a cell-active DYRK1α inhibitor Maria Mavrogeni , Filippos Pronios , Danae Zareifi , Sofia Vasilakaki , Olivier Lozach , et al. Future Medicinal Chemistry, 2018, 10 (20), pp.2411 - 2430. ⟨10.4155/fmc-2018-0198⟩ Article dans une revue hal-01906403v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis of new pyridazino[4,5-b]indol-4-ones and pyridazin-3(2H)-one analogs as DYRK1A inhibitors Amélie Bruel , Romain Bénéteau , Mylène Chabanne , Olivier Lozach , Rémy Le Guevel , et al. Bioorganic and Medicinal Chemistry Letters, 2014, 24 (21), pp.5037 - 5040. ⟨10.1016/j.bmcl.2014.09.017⟩ Article dans une revue hal-01086026v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Novel 9-oxo-thiazolo[5,4-f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: Synthesis, biological evaluation and molecular modeling studies Cédric Logé , Alexandra Testard , Valérie Thiéry , Olivier Lozach , Mélina Blairvacq , et al. European Journal of Medicinal Chemistry, 2008, 43 (7), pp.1469-1477. ⟨10.1016/j.ejmech.2007.09.020⟩ Article dans une revue istex hal-02357774v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and optimization of an original V-shaped collection of 4-7-disubstituted Pyrido[3,2-d]pyrimidines as CDK5 and DYRK1A inhibitors Oussama Dehbi , Abdellatif Tikad , Stéphane Bourg , Pascal Bonnet , Olivier Lozach , et al. European Journal of Medicinal Chemistry, 2014, 80, pp.352-363. ⟨10.1016/j.ejmech.2014.04.055⟩ Article dans une revue hal-02904758v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Advances in tetrahydropyrido[1,2-a]isoindolone (valmerins) series: Potent glycogen synthase kinase 3 and cyclin dependent kinase 5 inhibitors. Rajâa Boulahjar , Aziz Ouach , Stéphane Bourg , Pascal Bonnet , Olivier Lozach , et al. European Journal of Medicinal Chemistry, 2015, 101, pp.274-287. ⟨10.1016/j.ejmech.2015.06.046⟩ Article dans une revue hal-01212495v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Acridone Alkaloids from Glycosmis chlorosperma as DYRK1A Inhibitors Mehdi A. Beniddir , Erell Le Borgne , Bogdan I. Iorga , Nadège Loaëc , Olivier Lozach , et al. Journal of Natural Products, 2014, 77 (5), pp.1117-1122. ⟨10.1021/np400856h⟩ Article dans une revue hal-01162685v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and biological evaluation of bolaamphiphilic sophorolipids Elisabeth Delbeke , Jonas Everaert , Olivier Lozach , Tony Le Gall , Mathieu Berchel , et al. ACS Sustainable Chemistry & Engineering, 2018, 6 (7), pp.8992-9005. ⟨10.1021/acssuschemeng.8b01354⟩ Article dans une revue hal-01806695v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Dérivés d'imidazolones, procédé de préparation et applications biologiques. J.P. Bazureau , François Carreaux , Stéven Renault , Laurent Meijer , Olivier Lozach Patent n° : FR 291 9608 (A1). 2009 Brevet hal-00411458v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Identification of potential cellular targets of aloisine A by affinity chromatography. Caroline Corbel , Rose Haddoub , Damien Guiffant , Olivier Lozach , David Gueyrard , et al. Bioorganic and Medicinal Chemistry, 2009, 17 (15), pp.5572-82. ⟨10.1016/j.bmc.2009.06.024⟩ Article dans une revue istex hal-00416033v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and preliminary biological evaluation of new derivatives of the marine alkaloid leucettamine B as kinase inhibitors. Mansour Debdab , Stéven Renault , Olivier Lozach , Laurent Meijer , Ludovic Paquin , et al. European Journal of Medicinal Chemistry, 2010, 45 (2), pp.805-10. ⟨10.1016/j.ejmech.2009.10.009⟩ Article dans une revue istex hal-00869769v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		An efficient method for the preparation of new analogs of Leucettamine B under solvent-free microwave irradiation. Mansour Debdab , Stéven Renault , Samar Eid , Olivier Lozach , Laurent Meijer , et al. Heterocycles, 2009, pp.1191-1203 Article dans une revue hal-00411456v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthetic phospholipids and phospho-bola-amphiphiles for nucleic acid delivery Mathieu Berchel , Olivier Lozach , Wilfried Berthe , Sylvie Hernot , Hélène Couthon , et al. Phosphorus, Sulfur, and Silicon and the Related Elements, 2016, 191 (11-12), pp.1485 - 1487. ⟨10.1080/10426507.2016.1212049⟩ Article dans une revue hal-01539538v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and evaluation of the antiproliferative activity of novel thiazoloquinazolinone kinases inhibitors. Alexandra Testard , Laurent Picot , Olivier Lozach , Melina Blairvacq , Laurent Meijer , et al. Journal of Enzyme Inhibition and Medicinal Chemistry, 2005, 20 (6), pp.557-568. ⟨10.1080/14756360500212399⟩ Article dans une revue hal-01443570v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Antimalarial potential of xestoquinone, a protein kinase inhibitor isolated from a Vanuatu marine sponge Xestospongia sp. Dominique Laurent , Valérie Jullian , Arnaud Parenty , Martine Knibiehler , Dominique Dorin , et al. Bioorganic and Medicinal Chemistry, 2006, 14(13), pp.4477-4482 Article dans une revue hal-00090890v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Thiazolo[5,4-f]quinazolin-9-ones, inhibitors of glycogen synthase kinase-3 Alexandra Testard , Cédric Logé , Benoît Léger , Jean-Michel Robert , Olivier Lozach , et al. Bioorganic and Medicinal Chemistry Letters, 2006, 16 (13), pp.3419-3423. ⟨10.1016/j.bmcl.2006.04.006⟩ Article dans une revue istex hal-02357746v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Novel Tetrahydropyrido[1,2- a ]isoindolone Derivatives (Valmerins): Potent Cyclin-Dependent Kinase/Glycogen Synthase Kinase 3 Inhibitors with Antiproliferative Activities and Antitumor Effects in Human Tumor Xenografts Rajâa Boulahjar , Aziz Ouach , Chiurato Matteo , Stéphane Bourg , Myriam Ravache , et al. Journal of Medicinal Chemistry, 2012, 55 (22), pp.9589-9606. ⟨10.1021/jm3008536⟩ Article dans une revue hal-02904751v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Novel optimization of valmerins (tetrahydropyrido[1,2-a]isoindolones) as potent dual CDK5/GSK3 inhibitors Aziz Ouach , Rajâa Boulahjar , Christine Vala , Stéphane Bourg , Pascal Bonnet , et al. European Journal of Medicinal Chemistry, 2016, 115, pp.311--325. ⟨10.1016/j.ejmech.2016.02.072⟩ Article dans une revue hal-01295635v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Lipophosphoramidate-based bipolar amphiphiles: their syntheses and transfection properties Mathieu Berchel , Tony Le Gall , Olivier Lozach , Jean-Pierre Haelters , Tristan Montier , et al. Organic & Biomolecular Chemistry, 2016, 14 (10), pp.2846 - 2853. ⟨10.1039/C5OB02512E⟩ Article dans une revue hal-01539654v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Substitution of unsaturated lipid chains by thioether-containing lipid chains in cationic amphiphiles: physicochemical consequences and application for gene delivery Amal Bouraoui , Mathieu Berchel , Rosy Ghanem , Véronique Vie , Gilles Paboeuf , et al. Organic & Biomolecular Chemistry, 2019, 17 (14), pp.3609-3616. ⟨10.1039/c9ob00473d⟩ Article dans une revue hal-02088106v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Rebeccamycin derivatives as dual DNA damaging agents and potent checkpoint kinase 1 inhibitors. Christelle Marminon , Fabrice Anizon , Pascale Moreau , Bruno Pfeiffer , Alain Pierre , et al. Molecular Pharmacology, 2008, 74 (6), pp.1620-1629. ⟨10.1124/mol.108.049346⟩ Article dans une revue hal-00319800v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		An expeditious, environment-friendly, and microwave-assisted synthesis of 5-isatinylidenerhodanine derivatives Abdelmounaim Safer , Mustapha Rahmouni , François Carreaux , Ludovic Paquin , Olivier Lozach , et al. Chemical Papers, 2011, 65 (3), pp.332-337. ⟨10.2478/s11696-010-0104-9⟩ Article dans une revue hal-00869920v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Further investigation of Paprotrain: Towards the conception of selective and multi-targeted CNS kinase inhibitors Christophe Labrière , Olivier Lozach , Mélina Blairvacq , Laurent Meijer , Catherine Guillou European Journal of Medicinal Chemistry, 2016, 124, pp.920 - 934. ⟨10.1016/j.ejmech.2016.08.069⟩ Article dans une revue hal-01517780v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and biological evaluation of new 3-(6-hydroxyindol-2-yl)-5-(Phenyl) pyridine or pyrazine V-Shaped molecules as kinase inhibitors and cytotoxic agents. Pamela Kassis , Joanna Brzeszcz , Valérie Bénéteau , Olivier Lozach , Laurent Meijer , et al. European Journal of Medicinal Chemistry, 2011, 46 (11), pp.5416-34. ⟨10.1016/j.ejmech.2011.08.048⟩ Article dans une revue istex hal-00720615v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis, biological evaluation, and molecular modeling of natural and unnatural flavonoidal alkaloids, inhibitors of kinases. T .B. Nguyen , Olivier Lozach , Georgiana Surpateanu , Qian Wang , Pascal Retailleau , et al. Journal of Medicinal Chemistry, 2012, 55 (6), pp.2811-9. ⟨10.1021/jm201727w⟩ Article dans une revue hal-00692489v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Azine and Diazine Functionalization Using 2,2,6,6-Tetramethylpiperidino-Based Lithium–Metal Combinations: Application to the Synthesis of 5,9-Disubstituted Pyrido[3′,2′:4,5]pyrrolo[1,2-c] pyrimidines Nada Marquise , Tan Tai Nguyen , Floris Chevallier , Laurent Picot , Valérie Thiéry , et al. SYNLETT, 2015, 26 (20), pp.2811-2816. ⟨10.1055/s-0035-1560496⟩ Article dans une revue hal-01248092v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Novel Tetrahydropyrido[1,2-a]isoindolone Derivatives (Valmerins): Potent Cyclin-Dependent Kinase/Glycogen Synthase Kinase 3 Inhibitors with Antiproliferative Activities and Antitumor Effects in Human Tumor Xenografts Rajâa Boulahjar , Aziz Ouach , Chiurato Matteo , Stéphane Bourg , Myriam Ravache , et al. Journal of Medicinal Chemistry, 2012, 55, pp.9589-9606 Article dans une revue hal-00785213v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Design and Microwave Synthesis of New (5Z) 5-Arylidene-2-thioxo-1,3-thiazolinidin-4-one and (5Z) 2-Amino-5-arylidene-1,3-thiazol-4(5H)-one as New Inhibitors of Protein Kinase DYRK1A Khadidja Bourahla , Solène Guihéneuf , Emmanuelle Limanton , Ludovic Paquin , Rémy Le Guével , et al. Pharmaceuticals, 2021, 14 (11), pp.1086-1117. ⟨10.3390/ph14111086⟩ Article dans une revue hal-03467664v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Anticancer alkaloid lamellarins inhibit protein kinases. Dianne Baunbaek , Nolwenn Trinkler , Yoan Ferandin , Olivier Lozach , Poonsakdi Ploypradith , et al. Marine drugs, 2008, 6 (4), pp.514-27. ⟨10.3390/md20080026⟩ Article dans une revue hal-00416040v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Dérivés d'imidazolones, procédé de préparation et applications biologiques Olivier Lozach , L. Meijer , F. Bazureau , Renault J.P Patent n° : FR07/05632. 2007 Brevet hal-00169570v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis, protein kinase inhibitory potencies and in vitro antiproliferative activities of meridianin derivatives Pascale Moreau , Francis Giraud , Elisabeth Pereira , Fabrice Anizon , Georges Alves , et al. 17th European Symposium on Organic Chemistry, Jul 2011, Hersonissos, Greece Communication dans un congrès hal-00609975v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More

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A facile consensus ranking approach enhances virtual screening robustness and identifies a cell-active DYRK1α inhibitor

Synthesis of new pyridazino[4,5-b]indol-4-ones and pyridazin-3(2H)-one analogs as DYRK1A inhibitors

Novel 9-oxo-thiazolo[5,4-f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: Synthesis, biological evaluation and molecular modeling studies

Synthesis and optimization of an original V-shaped collection of 4-7-disubstituted Pyrido[3,2-d]pyrimidines as CDK5 and DYRK1A inhibitors

Advances in tetrahydropyrido[1,2-a]isoindolone (valmerins) series: Potent glycogen synthase kinase 3 and cyclin dependent kinase 5 inhibitors.

Acridone Alkaloids from Glycosmis chlorosperma as DYRK1A Inhibitors

Synthesis and biological evaluation of bolaamphiphilic sophorolipids

Dérivés d'imidazolones, procédé de préparation et applications biologiques.

Identification of potential cellular targets of aloisine A by affinity chromatography.

Synthesis and preliminary biological evaluation of new derivatives of the marine alkaloid leucettamine B as kinase inhibitors.

An efficient method for the preparation of new analogs of Leucettamine B under solvent-free microwave irradiation.

Synthetic phospholipids and phospho-bola-amphiphiles for nucleic acid delivery

Synthesis and evaluation of the antiproliferative activity of novel thiazoloquinazolinone kinases inhibitors.

Antimalarial potential of xestoquinone, a protein kinase inhibitor isolated from a Vanuatu marine sponge Xestospongia sp.

Thiazolo[5,4-f]quinazolin-9-ones, inhibitors of glycogen synthase kinase-3

Novel Tetrahydropyrido[1,2- a ]isoindolone Derivatives (Valmerins): Potent Cyclin-Dependent Kinase/Glycogen Synthase Kinase 3 Inhibitors with Antiproliferative Activities and Antitumor Effects in Human Tumor Xenografts

Novel optimization of valmerins (tetrahydropyrido[1,2-a]isoindolones) as potent dual CDK5/GSK3 inhibitors

Lipophosphoramidate-based bipolar amphiphiles: their syntheses and transfection properties

Substitution of unsaturated lipid chains by thioether-containing lipid chains in cationic amphiphiles: physicochemical consequences and application for gene delivery

Rebeccamycin derivatives as dual DNA damaging agents and potent checkpoint kinase 1 inhibitors.

An expeditious, environment-friendly, and microwave-assisted synthesis of 5-isatinylidenerhodanine derivatives

Further investigation of Paprotrain: Towards the conception of selective and multi-targeted CNS kinase inhibitors

Synthesis and biological evaluation of new 3-(6-hydroxyindol-2-yl)-5-(Phenyl) pyridine or pyrazine V-Shaped molecules as kinase inhibitors and cytotoxic agents.

Synthesis, biological evaluation, and molecular modeling of natural and unnatural flavonoidal alkaloids, inhibitors of kinases.

Azine and Diazine Functionalization Using 2,2,6,6-Tetramethylpiperidino-Based Lithium–Metal Combinations: Application to the Synthesis of 5,9-Disubstituted Pyrido[3′,2′:4,5]pyrrolo[1,2-c] pyrimidines

Novel Tetrahydropyrido[1,2-a]isoindolone Derivatives (Valmerins): Potent Cyclin-Dependent Kinase/Glycogen Synthase Kinase 3 Inhibitors with Antiproliferative Activities and Antitumor Effects in Human Tumor Xenografts

Design and Microwave Synthesis of New (5Z) 5-Arylidene-2-thioxo-1,3-thiazolinidin-4-one and (5Z) 2-Amino-5-arylidene-1,3-thiazol-4(5H)-one as New Inhibitors of Protein Kinase DYRK1A

Anticancer alkaloid lamellarins inhibit protein kinases.

Dérivés d'imidazolones, procédé de préparation et applications biologiques

Synthesis, protein kinase inhibitory potencies and in vitro antiproliferative activities of meridianin derivatives