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Successful Prediction of Substrate-binding Pocket in SLC17 Transporter Sialin
Nicolas Pietrancosta
,
Christine Anne
,
Horst Prescher
,
Raquel Ruivo
,
Corinne Sagné
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et al.
Article dans une revue
hal-02351288v1
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CADPS functional mutations in patients with bipolar disorder increase the sensitivity to stress
Jeremy Sitbon
,
Dennis Nestvogel
,
Caroline Kappeler
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Aude Nicolas
,
Stephanie Maciuba
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et al.
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inserm-03709071v1
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CYP2U1 activity is altered by missense mutations in hereditary spastic paraplegia 56
Christelle Durand
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Laura Dhers
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Christelle Tesson
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Alessandra Tessa
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Laetitia Fouillen
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et al.
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hal-01796579v1
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New 2-bromomethyl-8-substituted-benzo[c]chromen-6-ones. Synthesis and biological properties
Cédrik Garino
,
Frédéric Bihel
,
Nicolas Pietrancosta
,
Younes Laras
,
Gilles Quéléver
,
et al.
Article dans une revue
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hal-02351737v1
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Reverse Immunology Approach to Define a New HIV-gp41-Neutralizing Epitope
Karim Dorgham
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Nicolas Pietrancosta
,
Amel Affoune
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Olivier Lucar
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Tahar Bouceba
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et al.
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hal-02162037v1
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Identification of Privileged Scaffolds from a Diversified Chemical Library forβ-Secretase Inhibition
Nicolas Pietrancosta
,
Gilles Quéléver
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Cedrik Garino
,
Younes Laras
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Stéphane Burlet
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et al.
Article dans une revue
hal-02351752v1
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Enhanced delivery of γ-secretase inhibitor DAPT into the brain via an ascorbic acid mediated strategy
Gilles Quéléver
,
Philippe Kachidian
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Christophe Melon
,
Cédrik Garino
,
Younes Laras
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et al.
Article dans une revue
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hal-02351723v1
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Simple Coupling Reaction between Amino Acids and Weakly Nucleophilic Heteroaromatic Amines
Gilles Quéléver
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Stéphane Burlet
,
Cédrik Garino
,
Nicolas Pietrancosta
,
Younes Laras
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et al.
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BACE-1 inhibitory activities of new substituted phenyl-piperazine coupled to various heterocycles: Chromene, coumarin and quinoline
Cédrik Garino
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Nicolas Pietrancosta
,
Younes Laras
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Vincent Moret
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Amandine Rolland
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et al.
Article dans une revue
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hal-02351707v1
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Human Orphan Cytochrome P450 2U1 Catalyzes the ω-Hydroxylation of Leukotriene B4
Khawla Nouri
,
Nicolas Pietrancosta
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Laurent Le Corre
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Patrick Dansette
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Daniel Mansuy
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et al.
Article dans une revue
hal-03957648v1
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Pseudomonas aeruginosa Lipoxygenase LoxA Contributes to Lung Infection by Altering the Host Immune Lipid Signaling
Eric Morello
,
Teresa Pérez-Berezo
,
Chloé Boisseau
,
Thomas Baranek
,
Antoine Guillon
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et al.
Article dans une revue
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Amino Acids Bearing Aromatic or Heteroaromatic Substituents as a New Class of Ligands for the Lysosomal Sialic Acid Transporter Sialin
Lilian Dubois
,
Nicolas Pietrancosta
,
Alexandre Cabaye
,
Isabelle Fanget
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Cécile Debacker
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et al.
Article dans une revue
hal-02989894v1
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Thiazolamide - Ascorbic Acid Conjugate: a γ-Secretase Inhibitor with Enhanced Blood - Brain Barrier Permeation
Younes Laras
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Mahmoud Sheha
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Nicolas Pietrancosta
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Jean-Louis Kraus
Article dans une revue
hal-02351686v1
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Design of β-Secretase Inhibitors by Introduction of a Mandelyl Moiety in DAPT Analogues
Nicolas Pietrancosta
,
Gilles Quéléver
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Younes Laras
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Cédrik Garino
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Stéphane Burlet
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et al.
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hal-02351745v1
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Novel cyclized Pifithrin-α p53 inactivators: synthesis and biological studies
Nicolas Pietrancosta
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Flavio Maina
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Rosanna Dono
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Anice Moumen
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Cédrik Garino
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et al.
Article dans une revue
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Synthesis of Quinoline Dicarboxylic Esters as Biocompatible Fluorescent Tags
Franck-Cyril Favre-Besse
,
Odile Poirel
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Tiphaine Bersot
,
Elodie Kim-Grellier
,
Stéphanie Daumas
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et al.
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Regulation of IRE1 RNase activity by the Ribonuclease inhibitor 1 (RNH1)
Quentin Tavernier
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Evangeline Bennana
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Virginie Poindessous
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Céline Schaeffer
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Luca Rampoldi
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et al.
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Pseudoxanthoma Elasticum overlaps Hereditary Spastic Paraplegia Type 56
Anne Legrand
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Claire Pujol
,
Christelle M Durand
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Aurélie Mesnil
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Isabelle Rubera
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et al.
Article dans une revue
pasteur-03099934v1
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Imino-tetrahydro-benzothiazole Derivatives as p53 Inhibitors: Discovery of a Highly Potent in Vivo Inhibitor and Its Action Mechanism
Nicolas Pietrancosta
,
Anice Moumen
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Rosanna Dono
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Paul Lingor
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Veronique Planchamp
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et al.
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Synthesis of New Substituted 4,5-Dihydro-3H-spiro[1,5]-benzoxazepine-2,4′-piperidine and Biological Properties
Younes Laras
,
Nicolas Pietrancosta
,
Vincent Moret
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Sylvain Marc
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Cédrik Garino
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et al.
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hal-02351717v1
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Spectral and 3D model studies of the interaction of orphan human cytochrome P450 2U1 with substrates and ligands
Laura Dhers
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Nicolas Pietrancosta
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Lionel Ducassou
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Booma Ramassamy
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Julien Dairou
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et al.
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hal-02191703v1
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Bacterial Transferase MraY, a Source of Inspiration towards New Antibiotics
Mickaël Fer
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Laurent Le Corre
,
Nicolas Pietrancosta
,
Nathalie Evrard-Todeschi
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Samir Olatunji
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et al.
Article dans une revue
hal-02364241v1
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Fluorogenic Protein Probes with Red and Near‐Infrared Emission for Genetically Targeted Imaging
Sylvestre Bachollet
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Cyril Addi
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Nicolas Pietrancosta
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Jean‐maurice Mallet
,
Blaise Dumat
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hal-02974827v1
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Cerpegin-derived furo[3,4-c]pyridine-3,4(1H,5H)-diones enhance cellular response to interferons by de novo pyrimidine biosynthesis inhibition
Simon Hayek
,
Nicolas Pietrancosta
,
Anna Hovhannisyan
,
Rodolphe Alves de Sousa
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Nassima Bekaddour
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et al.
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hal-02372490v1
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Destabilization of the human RED–SMU1 splicing complex as a basis for host-directed antiinfluenza strategy
Usama Ashraf
,
Laura Tengo
,
Laurent Le Corre
,
Guillaume Fournier
,
Patricia Busca
,
et al.
Proceedings of the National Academy of Sciences of the United States of America, 2019, 116 (22), pp.10968-10977. ⟨10.1073/pnas.1901214116⟩
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hal-02160991v1
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Molecular, Structural, Functional, and Pharmacological Sites for Vesicular Glutamate Transporter Regulation
Nicolas Pietrancosta
,
Mahamadou Djibo
,
Stephanie Daumas
,
Salah El Mestikawy
,
Jeffrey D. Erickson
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hal-03007881v1
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Ctr9, a Protein in the Transcription Complex Paf1, Regulates Dopamine Transporter Activity at the Plasma Membrane
Stephanie de Gois
,
Patrick Slama
,
Nicolas Pietrancosta
,
Amaia M. Erdozain
,
Franck Louis
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et al.
Article dans une revue
hal-01542313v1
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Are p53 inhibitors potentially useful therapeutics?
Nicolas Pietrancosta
,
Cedrik Garino
,
Younes Laras
,
Gilles Quéléver
,
Philippe Pierre
,
et al.
Article dans une revue
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hal-02351741v1
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Structure of human glycolate oxidase in complex with the inhibitor 4-carboxy-5-[(4-chlorophenyl)sulfanyl]-1,2,3-thiadiazole.
Jean Marie Bourhis
,
Caroline Vignaud
,
Nicolas Pietrancosta
,
Françoise Guéritte
,
Daniel Guénard
,
et al.
Acta Crystallographica Section F: Structural Biology and Crystallization Communications, 2009, 65 (Pt 12), pp.1246-53. ⟨10.1107/S1744309109041670⟩
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hal-00769815v1
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5'-Methylene-triazole-substituted-aminoribosyl uridines as MraY inhibitors: synthesis, biological evaluation and molecular modeling.
Mickaël J Fer
,
Ahmed Bouhss
,
Mariana Patrão
,
Laurent Le Corre
,
Nicolas Pietrancosta
,
et al.
Article dans une revue
hal-01433063v1
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