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Synthesis of Novel G Factor or Chloroquine-Artemisinin Hybrids and Conjugates with Potent Antiplasmodial Activity

 Christophe Menendez , Dionissia A Pepe , Dimitra Toumpa , Christiane André-Barrès , Christophe Me- Nendez , et al.
ACS Medicinal Chemistry Letters, 2020, 11 (5), pp.921-927. ⟨10.1021/acsmedchemlett.9b00669⟩
Article dans une revue hal-03006874v1

Effect of Zearalenone gestational exposure: modulation of placenta cell differentiation and transport function

 Caroline Prouillac , Farah Koraichi , Bernadette Videmann , Michelle Mazallon , Frédéric Rodriguez , et al.
49. Congress of the European Societies of Toxicology (EUROTOX), Sep 2013, Interlaken, Switzerland. ⟨10.1016/j.toxlet.2013.05.506⟩
Communication dans un congrès hal-02748356v1

Cinnamic Acid Derivatives as Anticancer Agents-A Review

 P. De , Michel Baltas , Florence Bedos-Belval
Current Medicinal Chemistry, 2011, 18 (11), pp.1672-1703. ⟨10.2174/092986711795471347⟩
Article dans une revue hal-03102550v1

The Integrated Screening Platform of Toulouse (PICT): a tool for accelerated molecular discovery

 Brigitte Guidetti , Isabelle Fabing , Michel Baltas , Stéphanie Ballereau , Tessa Castellan , et al.
Congrès JCO 2019, Oct 2019, Palaiseau, France
Poster de conférence hal-02893197v1
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Design of Anti-infectious Agents from Lawsone in a Three-Component Reaction with Aldehydes and Isocyanides

 Christina L Koumpoura , Michel Nguyen , Christian Bijani , Laure Vendier , Elena G Salina , et al.
ACS Omega, 2022, 7 (40), pp.35635-35655. ⟨10.1021/acsomega.2c03421⟩
Article dans une revue hal-03818601v1
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Crystal structure of the enoyl-ACP reductase of Mycobacterium tuberculosis (InhA) in the apo-form and in complex with the active metabolite of isoniazid pre-formed by a biomimetic approach

 Aurélien Chollet , Lionel Mourey , Christian Lherbet , Alexandra Delbot , Sylviane Julien , et al.
Journal of Structural Biology, 2015, 190, pp.328 - 337. ⟨10.1016/j.jsb.2015.04.008⟩
Article dans une revue hal-03002973v1

Synthesis of Fosmidomycin Analogues, Hybrids and Conjugates with 7-chloroquinoline and Artemisinin as promising Antimalarial Agents

 Despina Palla , Michel Baltas , Christophe Menendez , Philippe Grellier , Elisabeth Mouray , et al.
12th AIMECS 2019, AFMC International Medicinal Chemistrty Symposium, Sep 2019, Istanbul, Turkey
Poster de conférence hal-02338884v1

Small molecules inhibitors of plasminogen activator inhibitor-1 – An overview

 Anne Rouch , Corinne Vanucci-Bacqué , Florence Bedos-Belval , Michel Baltas
European Journal of Medicinal Chemistry, 2015, 92, pp.619-636. ⟨10.1016/j.ejmech.2015.01.010⟩
Article dans une revue hal-03102594v1
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Mechanochemical Studies on Coupling of Hydrazines and Hydrazine Amides with Phenolic and Furanyl Aldehydes—Hydrazones with Antileishmanial and Antibacterial Activities

 Anna Kapusterynska , Christian Bijani , Damian Paliwoda , Laure Vendier , Valérie Bourdon , et al.
Molecules, 2023, 28 (13), pp.5284. ⟨10.3390/molecules28135284⟩
Article dans une revue hal-04157067v1

Distinct CCK-2 Receptor Conformations Associated with β-Arrestin-2 Recruitment or Phospholipase-C Activation Revealed by a Biased Antagonist

 Remi Magnan , Chantal Escrieut , Véronique Gigoux , Kavita De , Fan Niu , et al.
Journal of the American Chemical Society, 2013, 135 (7), pp.2560-2573. ⟨10.1021/ja308784w⟩
Article dans une revue hal-02393278v1
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Synthesis, In Silico, and In Vitro Evaluation of Anti-Leishmanial Activity of Oxadiazoles and Indolizine Containing Compounds Flagged against Anti-Targets

 Strahinja Stevanovic , Milan Sencanski , Mathieu Danel , Christophe Menendez , Roumaissa Belguedj , et al.
Molecules, 2019, 24 (7), pp.1282. ⟨10.3390/molecules24071282⟩
Article dans une revue hal-02169888v1

Synthesis, antioxidant and cytoprotective evaluation of potential antiatherogenic phenolic hydrazones. A structure–activity relationship insight

 Corinne Vanucci-Bacqué , Chantal Carayon , Corinne Bernis , Caroline Camaré , Anne Nègre-Salvayre , et al.
Bioorganic and Medicinal Chemistry, 2014, 22 (15), pp.4269-4276. ⟨10.1016/j.bmc.2014.05.034⟩
Article dans une revue hal-02063985v1

Synthesis and application of pure and (B and/or N) doped carbon nanomaterials

 Flavien Valensi , Djamel Eddine Gourari , Manitra Razafinimanana , R. Arenal , M. Monthioux , et al.
EMN Metamaterials Meeting (Energy materials Nanotechnology) May 8-12, 2016, Dubrovnik (CROATIA), 2016, Dubrovnik, Croatia
Communication dans un congrès hal-03965672v1

Effect of the Nature of Surfactant on the Reactivity of C,N-diphenylnitrone towards Acrylonitrile in Different Microemulsions Systems

 Kahina Hamza , Abdelkader Touati , Ahmed Ait-Yahia , Michel Baltas , Christiane André-Barrès , et al.
Chemistry Journal of Moldova, 2018, 13 (2), pp.82-88. ⟨10.19261/cjm.2018.522⟩
Article dans une revue hal-02169807v1

Synthesis and evaluation of antioxidant phenolic diaryl hydrazones as potent antiangiogenic agents in atherosclerosis

 Corinne Vanucci-Bacqué , Caroline Camaré , Chantal Carayon , Corinne Bernis , Michel Baltas , et al.
Bioorganic and Medicinal Chemistry, 2016, 24 (16), pp.3571-3578. ⟨10.1016/j.bmc.2016.05.067⟩
Article dans une revue hal-02060616v1

The integrated screening platform of Toulouse (PICT) : A tool for accelerated molecular discovery

 Isabelle Fabing , Michel Baltas , Stéphanie Ballereau , Yves Génisson , Brigitte Guidetti , et al.
Congress SFC 2018 Chemistry and Life Symposium, Jun 2018, Montpellier, France
Poster de conférence hal-02337455v1
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Synthesis and biological evaluation of diarylheptanoids as potential antioxidant and anti-inflammatory agents

 Kelly Maurent , Corinne Vanucci-Bacqué , Michel Baltas , Anne Nègre-Salvayre , Nathalie Augé , et al.
European Journal of Medicinal Chemistry, 2018, 144 (7), pp.289-299. ⟨10.1016/j.ejmech.2017.12.033⟩
Article dans une revue hal-03118254v1
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Synthesis of Novel Artemisinin, Ciprofloxacin, and Norfloxacin Hybrids with Potent Antiplasmodial Activity

 Georgia Vamvoukaki , Antonia I Antoniou , Michel Baltas , Elisabeth Mouray , Sebastien Charneau , et al.
Antibiotics, 2024, 13 (2), pp.142. ⟨10.3390/antibiotics13020142⟩
Article dans une revue hal-04509679v1

Kinetic and inhibition studies of cinnamoyl-CoA reductase 1 from Arabidopsis thaliana

 Michel Baltas , Corentin J Lapeyre , F. Bedos-Belval , M. Maturano , P. Saint-Aguet , et al.
Plant Physiology and Biochemistry, 2005, 43 (8), pp.746-753. ⟨10.1016/j.plaphy.2005.06.003⟩
Article dans une revue istex hal-02444219v1

Antiproliferative and apoptotic activity of new indazole derivatives as potential anticancer agents

 Fatima E. Laghchioua , Assoman Kouakou , Mohammed Eddahmi , Maurizio Viale , Massimiliano Monticone , et al.
Archiv der Pharmazie / Arch Pharm Pharm Med Chem; Arch Pharm Chem Life Sci; Arch Pharm (Weinheim), 2020, 353 (12), pp.2000173. ⟨10.1002/ardp.202000173⟩
Article dans une revue hal-02899347v1
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Cinnamic Acid Derivatives in Tuberculosis, Malaria and Cardiovascular Diseases - A Review

 Prithwiraj De , Florence Bedos-Belval , Corinne Vanucci-Bacqué , Michel Baltas
Current Organic Chemistry, 2012, 16 (6), pp.747-768. ⟨10.2174/138527212799958020⟩
Article dans une revue hal-02444262v1

Investigation on the kinetic of a Diels-Alder reaction carried out in a vibratory ball mill

 Lori Gonnet , Alain Chamayou , Brigitte Guidetti , Christiane André-Barrès , Michel Baron , et al.
16th European Symposium on Comminution & Classification (ESCC 2019), Sep 2019, Leed, United Kingdom
Poster de conférence hal-03690215v1
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Unprecedented linear products by a mechanochemically activated Biginelli reaction using lawsone

 Christina L Koumpoura , Laure Vendier , Christian Bijani , Anne Robert , Philippe Carbonnière , et al.
RSC Mechanochemistry, In press, ⟨10.1039/d3mr00032j⟩
Article dans une revue hal-04550806v1

Structure of adducts of isoindolo[2,1-a]benzimidazole derivatives with maleimides

 Korolev Oleksandr , Tatyana Yegorova , Igor Levkov , Volodymyr Malytskyi , Oleg V. Shishkin , et al.
Journal of Molecular Structure, 2015, 1084, pp.177-181. ⟨10.1016/j.molstruc.2014.11.056⟩
Article dans une revue hal-01965764v1

In vitro toxicological effects of estrogenic mycotoxins on human placental cells: Structure activity relationships

 Caroline Prouillac , Farah Koraichi , Bernadette Videmann , Michelle Mazallon , Frédéric Rodriguez , et al.
Toxicology and Applied Pharmacology, 2012, 259 (3), pp.366 - 375. ⟨10.1016/j.taap.2012.01.016⟩
Article dans une revue hal-02643248v1

New chiral imidazolinic derivatives

 Yves Génisson , Nancy Lauth de Viguerie , C. Andre , Michel Baltas , L. Gorrichon
Tetrahedron: Asymmetry, 2005, 16 (5), pp.1017
Article dans une revue hal-00149078v1

Synthesis and evaluation of β-hydroxytriazoles and related compounds as antitubercular agents

 Christophe Menendez , Giorgia Mori , Mathilde Maillot , Isabelle Fabing , Chantal Carayon , et al.
8th International Chemistry Conference Toulouse-Kiev (ICTK-8), ., Jun 2015, Toulouse, France. 3 (1), pp.82-96, 2015, ⟨10.17721/fujcv3i1p82-96⟩
Poster de conférence hal-03969265v1
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Synthesis and biological evaluation against Leishmania donovani of novel hybrid molecules containing indazole-based 2-pyrone scaffolds

 M. El Ghozlani , L. Bouissane , M. Berkani , S. Mojahidi , A. Allam , et al.
MedChemComm, 2019, 10 (1), pp.120-127. ⟨10.1039/c8md00475g⟩
Article dans une revue hal-02059320v1
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Synthesis of Biologically Relevant 1,2,3-and 1,3,4-Triazoles: From Classical Pathway to Green Chemistry

 Lori Gonnet , Michel Baron , Michel Baltas
Molecules, 2021, 26 (18), pp.5667. ⟨10.3390/molecules26185667⟩
Article dans une revue hal-03360993v1
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Antimalarial Inhibitors Targeting Epigenetics or Mitochondria in Plasmodium falciparum: Recent Survey upon Synthesis and Biological Evaluation of Potential Drugs against Malaria

 Christina L Koumpoura , Anne Robert , Constantinos M Athanassopoulos , Michel Baltas
Molecules, 2021, 26 (18), pp.5711. ⟨10.3390/molecules26185711⟩
Article dans une revue hal-03366266v1
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