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Structural modeling of RND family efflux pumps : From antibioresistance to chemotherapyresistance

Méliné Simsir
Molecular biology. Université Côte d'Azur, 2020. English. ⟨NNT : 2020COAZ6040⟩
Thèse tel-03171909v1
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Studying dynamics without explicit dynamics: a structure-based study of the export mechanism by AcrB

Méliné Simsir , Isabelle Broutin , Isabelle Mus-Veteau , Frédéric Cazals
2020
Pré-publication, Document de travail hal-02532366v2
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Studying dynamics without explicit dynamics: A structure‐based study of the export mechanism by AcrB

Méliné Simsir , Isabelle Broutin , Isabelle Mus‐veteau , Frédéric Cazals
Proteins - Structure, Function and Bioinformatics, 2020, ⟨10.1002/prot.26012⟩
Article dans une revue hal-03011350v1
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Inhibition of the drug efflux activity of Ptch1 as a promising strategy to overcome chemotherapy resistance in cancer cells

Sandra Kovachka , Giuliano Malloci , Méliné Simsir , Paolo Ruggerone , Stéphane Azoulay , et al.
European Journal of Medicinal Chemistry, 2022, 236, pp.114306. ⟨10.1016/j.ejmech.2022.114306⟩
Article dans une revue hal-03845877v1
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Astemizole Sensitizes Adrenocortical Carcinoma Cells to Doxorubicin by Inhibiting Patched Drug Efflux Activity.

Anida Hasanovic , Méliné Simsir , Choveau Fs , Enzo Lalli , Isabelle Mus-Veteau
Biomedicines, 2020, 8, ⟨10.3390/biomedicines8080251⟩
Article dans une revue hal-02917455v1
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Inhibition of patched drug efflux increases vemurafenib effectiveness against resistant braf(V600E) melanoma

Laurie Signetti , Nelli Elizarov , Méliné Simsir , Agnès Paquet , Dominique Douguet , et al.
Cancers, 2020, 12 (6), pp.1500. ⟨10.3390/cancers12061500⟩
Article dans une revue hal-02884136v1