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Ligand-free Pd/Cu-catalyzed microwave-assisted C-H arylation of quinazolin-4(3H)-ones with aryl iodides

Marine Harari , Corinne Fruit , Thierry Besson
Semaine d'études en chimie organique (SECO, 52, 2015), May 2015, Morzine, France
Communication dans un congrès hal-02378695v1

Nouvelle dioxygénases alpha-cetoglutarate dépendantes pour la synthèse de plateformes chirales

Anne Zaparucha , Damien Baud , Pierre-Loic Saaidi , Marine Harari , Julien Cuccaro , et al.
CBSO, Jun 2014, Carry Le Rouet, France
Communication dans un congrès hal-04303652v1

Rational multistep synthesis of a novel polyfunctionalized benzo[d]thiazole and its thiazolo[5,4-b]pyridine analogue

Damien Hédou , Emmanuel Deau , Marine Harari , Morgane Sanselme , Corinne Fruit , et al.
Tetrahedron, 2014, 70 (5541-5549), pp.5541-5549. ⟨10.1016/j.tet.2014.06.103⟩
Article dans une revue hal-01141181v1

Microwave-assisted C-H arylation of Quinazolin-4-one-type Precursors of Bioactive Heterocycles

Corinne Fruit , Julien Godeau , Marine Harari , Vincent Levacher , Thierry Besson
International Electronic Conference on Medicinal Chemistry (ECMC, 1, 2015), Jean-Jacques Vanden Eynde (coord.), Nov 2015, [online], Belgium. ⟨10.3390/ecmc-1-A004⟩
Communication dans un congrès hal-02383839v1

Synthesis of polyfunctionalized benzo[d]thiazoles as novel anthranilic acid derivatives

Damien Hédou , Marine Harari , Julien Godeau , Carole Dubouilh-Benard , Corinne Fruit , et al.
Tetrahedron Letters, 2015, 56 (27), pp.4088-4092. ⟨10.1016/j.tetlet.2015.05.018⟩
Article dans une revue hal-01160622v1

Ligand-Free Pd-Catalyzed and Copper-Assisted C−H Arylation ofQuinazolin-4-ones with Aryl Iodides under Microwave Heating

Sylvain Laclef , Marine Harari , Julien Godeau , Isabelle Schmitz-Afonso , Laurent Bischoff , et al.
Organic Letters, 2015, organic letters, 17 (7), pp.1700-1713. ⟨10.1021/acs.orglett.5b00467⟩
Article dans une revue hal-01141150v1

Pd-Catalyzed and Copper Assisted Regioselective Sequential C2 and C7 Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one with Aryl Halides

Marine Harari , Florence Couly , Corinne Fruit , Thierry Besson
Organic Letters, 2016, 18 (13), pp.3282-3285. ⟨10.1021/acs.orglett.6b01552⟩
Article dans une revue hal-02046211v1

Late-Stage Sequential C-H Functionalization of Thiazolo[5,4-f]quina-zolin-9(8H)-one: Synthesis of a Library of Potential Kinase Inhibitors

Corinne Fruit , Florence Couly , Marine Harari , Vincent Levacher , Thierry Besson
International Electronic Conference on Synthetic Organic Chemistry (ECSOC, 20, 2016), Julio A. Seijas Vázquez (coord.), Nov 2016, [online], Spain
Communication dans un congrès hal-02383920v1
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Development of Kinase Inhibitors via Metal-Catalyzed C–H Arylation of 8-Alkyl-thiazolo[5,4-f]-quinazolin-9-ones Designed by Fragment-Growing Studies

Florence Couly , Marine Harari , Carole Dubouilh-Benard , Laëtitia Bailly , Emilie Petit , et al.
Molecules, 2018, 23 (9), pp.2181. ⟨10.3390/molecules23092181⟩
Article dans une revue hal-02024491v1
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Synthesis of Mono- and Dihydroxylated Amino Acids with New $\alpha$-Ketoglutarate-Dependent Dioxygenases: Biocatalytic Oxidation of C$-$H Bonds

Damien Baud , Pierre-Loïc Saaidi , Adam Monfleur , Marine Harari , Julien Cuccaro , et al.
ChemCatChem, 2014, 6, pp.3012 - 3017. ⟨10.1002/cctc.201402498⟩
Article dans une revue istex cea-01591870v1