Comparison of 2 strategies to enhance pyridoclax solubility: Nanoemulsion delivery system versus salt synthesis
A.-C. Groo
,
M. de Pascale
,
A.-S. Voisin-Chiret
,
S. Corvaisier
,
M. Since
,
et al.
European Journal of Pharmaceutical Sciences , 2017, 97, pp.218-226
Article dans une revue
hal-02053808v1
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Inhibiting Acetylcholinesterase to Activate Pleiotropic Prodrugs with Therapeutic Interest in Alzheimer’s Disease
François-Xavier Toublet
,
Cédric Lecoutey
,
Julien Lalut
,
Bérénice Hatat
,
Audrey Davis
,
et al.
Article dans une revue
hal-02399906v1
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Development of a nasal drug delivery composite nanosystem for Alzheimer’s desease treatment
Adnet Thomas
,
Anne-Claire Groo
,
Loïc Le Pluart
,
Celine Picard
,
A. Davis
,
et al.
Journée normande de recherche biomédicale , Nov 2017, caen, France
Poster de conférence
hal-02295929v1
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Pleiotropic prodrugs: Design of a dual butyrylcholinesterase inhibitor and 5-HT6 receptor antagonist with therapeutic interest in Alzheimer’s disease
François-Xavier Toublet
,
Julien Lalut
,
Bérénice Hatat
,
Cédric Lecoutey
,
Audrey Davis
,
et al.
Article dans une revue
hal-03082877v1
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New 8-Nitroquinolinone Derivative Displaying Submicromolar in Vitro Activities against Both Trypanosoma brucei and cruzi
Julien Pedron
,
Clotilde Boudot
,
Jean-Yves Brossas
,
Emilie Pinault
,
Sandra Bourgeade-Delmas
,
et al.
Article dans une revue
hal-02476867v1
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Design, synthesis and biological evaluation of novel indano- and thiaindano-pyrazoles with potential interest for Alzheimer's disease.
David Genest
,
Christophe Rochais
,
Cédric Lecoutey
,
Jana Sopkova-de Oliveira Santos
,
Céline Ballandonne
,
et al.
MedChemComm , 2013, 4, pp.925-931
Article dans une revue
hal-00840942v1
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Comparison of 2 strategies to enhance pyridoclax solubility: Nanoemulsion delivery system versus salt synthesis
A.-C. Groo
,
M. de Pascale
,
A.-S. Voisin-Chiret
,
S. Corvaisier
,
M. Since
,
et al.
European Journal of Pharmaceutical Sciences , 2017, 97, pp.218-226
Article dans une revue
hal-02043745v1
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Pyridoclax-loaded nanoemulsion for enhanced anticancer effect on ovarian cancer
A.C. Groo
,
S. Hedir
,
M. Since
,
E. Brotin
,
L.-B. Weiswald
,
et al.
Article dans une revue
hal-03492393v1
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A functional m 6 A‐RNA methylation pathway in the oyster Crassostrea gigas assumes epitranscriptomic regulation of lophotrochozoan development
Lorane Le Franc
,
Benoit Bernay
,
Bruno Petton
,
Marc Since
,
Pascal Favrel
,
et al.
Article dans une revue
hal-02952460v1
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Evaluation of the versatile character of a nanoemulsion formulation
Emilie Gué
,
Marc Since
,
S. Ropars
,
R. Herbinet
,
L. Le Pluart
,
et al.
Article dans une revue
hal-01847973v1
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A biomimetic multiparametric assay to characterise anti-amyloid drugs
Willy Smeralda
,
Marc Since
,
Sophie Corvaisier
,
Dimitri Fayoll
,
Julien Cardin
,
et al.
Article dans une revue
hal-04315267v1
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Evaluation préclinique de nanoémulsions polyvalentes comme vecteurs d’un nouvel inhibiteur de Mcl-1, le Pyridoclax : application au traitement des cancers de l’ovaire (PYRINANO)
Aurélie Malzert-Fréon
,
Anne-Claire Groo
,
Siham Hedir
,
Marc Since
,
Martina de Pascale
,
et al.
10émes journées scientifiques du cancéropole nord-ouest , May 2017, Deauville, France
Communication dans un congrès
hal-02295794v1
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Design of donecopride, a dual serotonin subtype 4 receptor agonist/acetylcholinesterase inhibitor with potential interest for Alzheimer's disease treatment
Cédric Lecoutey
,
Damien Hedou
,
Thomas Freret
,
Patrizia Giannoni
,
Florence Gaven
,
et al.
Proceedings of the National Academy of Sciences of the United States of America , 2014, 111 (36), pp.E3825--30.
⟨10.1073/pnas.1410315111⟩
Article dans une revue
hal-01800439v2
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Benzylphenylpyrrolizinones with Anti-amyloid and Radical Scavenging Effects, Potentially Useful in Alzheimer's Disease Treatment
Jean-Pierre Jourdan
,
Marc Since
,
Laïla El kihel
,
Cédric Lecoutey
,
Sophie Corvaisier
,
et al.
Article dans une revue
hal-02043731v1
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Synthesis of antiplasmodial 2-aminothieno[3,2-d]pyrimidin-4(3H)-one analogues using the scaffold hopping strategy
Romain Mustière
,
Prisca Lagardère
,
Sébastien Hutter
,
Viviana Dell’orco
,
Nadia Amanzougaghene
,
et al.
Article dans une revue
hal-03737417v1
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Introduction to the versatility of biomimetic membranes to characterize modulators of Aβ1-42 fibrillization with potential interest in Alzheimer's disease treatment
Willy Smeralda
,
Marc Since
,
Michael Boisserie
,
Sophie Corvaisier
,
Julien Cardin
,
et al.
32ème Journées Franco-Belges de Chimie Thérapeutique et 26ème Rencontres Internationales des Pharmacochimistes de l'Arc Atlantique, , Jun 2018, Asnelles sur Mer, France. 2018
Poster de conférence
hal-01844495v1
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Star-like poly(peptoid)s with selective antibacterial activity
Pedro Salas-Ambrosio
,
Antoine Tronnet
,
Mostafa Badreldin
,
Luzangel Reyes
,
Marc Since
,
et al.
Article dans une revue
hal-03559890v1
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Comparison of 2 strategies to enhance pyridoclax solubility: Nanoemulsion delivery system versus salt synthesis
Anne-Claire Groo
,
Martina de Pascale
,
Anne-Sophie Voisin-Chiret
,
Sophie Corvaisier
,
Marc Since
,
et al.
Article dans une revue
hal-02160866v1
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β-Amyloid peptide interactions with biomimetic membranes: A multiparametric characterization
Willy Smeralda
,
Marc Since
,
Julien Cardin
,
Sophie Corvaisier
,
Sophie Lecomte
,
et al.
Article dans une revue
hal-03187852v1
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Pharmacotechnical Development of a Nasal Drug Delivery Composite Nanosystem Intended for Alzheimer’s Disease Treatment
Thomas Adnet
,
Anne-Claire Groo
,
Céline Picard
,
Audrey Davis
,
Sophie Corvaisier
,
et al.
Article dans une revue
hal-03969997v1
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New orally effective 3-(2-nitro)phenylpropanamide analgesic derivatives: Synthesis and antinociceptive evaluation
Marc Since
,
Thomas Freret
,
Gerald Nee
,
Thierry Terme
,
Patrice Vanelle
,
et al.
Article dans une revue
istex
hal-01460473v1
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Novel benzylidenephenylpyrrolizinones with pleiotropic activities potentially useful in Alzheimer's disease treatment
Jean-Pierre Jourdan
,
Marc Since
,
Laïla El Kihel
,
Cédric Lecoutey
,
Sophie Corvaisier
,
et al.
Article dans une revue
hal-02043765v1
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8-Alkynyl-3-nitroimidazopyridines display potent antitrypanosomal activity against both T. b. brucei and cruzi
Cyril Fersing
,
Clotilde Boudot
,
Caroline Castera-Ducros
,
Émilie Pinault
,
Sébastien Hutter
,
et al.
Article dans une revue
hal-02899751v1
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Synthesis of Pyridoclax Analogues: Insight into Their Druggability by Investigating Their Physicochemical Properties and Interactions with Membranes
Martina de Pascale
,
Domenico Iacopetta
,
Marc Since
,
Sophie Corvaisier
,
V. Vié
,
et al.
Article dans une revue
hal-02434628v1
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Nongenotoxic 3-Nitroimidazo[1,2- a ]pyridines Are NTR1 Substrates That Display Potent in Vitro Antileishmanial Activity
Cyril Fersing
,
Louise Basmaciyan
,
Clotilde Boudot
,
Julien Pedron
,
Sébastien Hutter
,
et al.
Article dans une revue
hal-02478935v1
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Microplate assay for lipophilicity determination using intrinsic fluorescence of drugs: Application to a promising anticancer lead, pyridoclax
Willy Smeralda
,
Marc Since
,
Sophie Corvaisier
,
Rémi Legay
,
Anne-Sophie Voisin-Chiret
,
et al.
Article dans une revue
hal-02168030v1
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Cyclic Poly(α-peptoid)s by Lithium bis(trimethylsilyl)amide (LiHMDS)-Mediated Ring-Expansion Polymerization
Pedro Salas-Ambrosio
,
Antoine Tronnet
,
Marc Since
,
Sandra Bourgeade-Delmas
,
Jean-Luc Stigliani
,
et al.
Article dans une revue
hal-03173586v1
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Improving Aqueous Solubility and In Vitro Pharmacokinetic Properties of the 3-Nitroimidazo[1,2-a]pyridine Antileishmanial Pharmacophore
Romain Paoli-Lombardo
,
Nicolas Primas
,
Sandra Bourgeade-Delmas
,
Sébastien Hutter
,
Alix Sournia-Saquet
,
et al.
Article dans une revue
hal-03755519v1
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First SNAr reaction using TDAE-initiated carbanions in quinazoline series
Marc Since
,
Omar Khoumeri
,
Pierre Verhaeghe
,
Martine Maillard-Boyer
,
Thierry Terme
,
et al.
Article dans une revue
istex
hal-01460328v1
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Antikinetoplastid SAR study in 3-nitroimidazopyridine series
Cyril Fersing
,
Clotilde Boudot
,
Romain Paoli-Lombardo
,
Nicolas Primas
,
Emilie Pinault
,
et al.
Article dans une revue
hal-02920293v1
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