Recherche - Archive ouverte HAL Accéder directement au contenu

Filtrer vos résultats

39 résultats

Cinnamides Target Leishmania amazonensis Arginase Selectively

Edson Roberto da Silva , Júlio Abel Alfredo dos Santos Simone Come , Simone Brogi , Vincenzo Calderone , Giulia Chemi , et al.
Molecules, 2020, 25 (22), pp.5271. ⟨10.3390/molecules25225271⟩
Article dans une revue hal-03409117v1

Carbon nanotubes as gene carriers: Focus on internalization pathways related to functionalization and properties

Cécile Caoduro , Eric Hervouet , Corine Girard-Thernier , Tijani Gharbi , Hatem Boulahdour , et al.
Acta Biomaterialia, 2017, 49, pp.36-44. ⟨10.1016/j.actbio.2016.11.013⟩
Article dans une revue hal-03407824v1

In Vitro Mammalian Arginase Inhibitory and Antioxidant Effects of Amide Derivatives Isolated from the Hempseed Cakes (Cannabis sativa)

Mélanie Bourjot , Andy Zedet , Belinda Demange , M. Pudlo , Corine Girard-Thernier
Planta Medica International Open, 2016, 3 (03), pp.e64-e67. ⟨10.1055/s-0042-119400⟩
Article dans une revue hal-03409030v1

First domino radical cyclisation/Smiles rearrangement combination

M. Pudlo , Ingrid Allart-Simon , Bernard Tinant , Stéphane Gérard , Janos Sapi
Chemical Communications, 2012, 48 (18), pp.2442. ⟨10.1039/C2CC15670A⟩
Article dans une revue hal-03407875v1

Carbon nanotube – Protamine hybrid: Evaluation of DNA cell penetration

Cécile Caoduro , Raoudha Kacem , Khaoula Boukari , Fabien Picaud , Claire-Hélène Brachais , et al.
Carbon, 2016, 96, pp.742 - 752. ⟨10.1016/j.carbon.2015.09.098⟩
Article dans une revue hal-01399272v1

Nanovectorization of DNA Through Cells Using Protamine Complexation

Khaoula Boukari , Cécile Caoduro , Raoudha Kacem , Nadia Skandrani , Christophe Borg , et al.
Journal of Membrane Biology, 2016, 249 (4), pp.493-501. ⟨10.1007/s00232-016-9890-5⟩
Article dans une revue hal-03407844v1

Human-based evidence for the therapeutic potential of arginase inhibitors in cardiovascular diseases

Johnny Moretto , M. Pudlo , Céline Demougeot
Drug Discovery Today, 2021, 26 (1), pp.138-147. ⟨10.1016/j.drudis.2020.11.005⟩
Article dans une revue hal-03407776v1

Carbon nanotube – Protamine hybrid: Evaluation of DNA cell penetration

Cécile Caoduro , Raoudha Kacem , Khaoula Boukari , Fabien Picaud , Claire-Hélène Brachais , et al.
Carbon, 2016, 96, pp.742-752. ⟨10.1016/j.carbon.2015.09.098⟩
Article dans une revue hal-03407855v1

Cinnamide Derivatives as Mammalian Arginase Inhibitors: Synthesis, Biological Evaluation and Molecular Docking

Thanh-Nhat Pham , Simon Bordage , M. Pudlo , Céline Demougeot , Khac-Minh Thai , et al.
International Journal of Molecular Sciences, 2016, 17 (10), pp.1656. ⟨10.3390/ijms17101656⟩
Article dans une revue hal-03409018v1

Cinnamide Derivatives as Mammalian Arginase Inhibitors: Synthesis, Biological Evaluation and Molecular Docking

Thanh-Nhat Pham , Simon Bordage , M. Pudlo , Céline Demougeot , Khac-Minh Thai , et al.
International Journal of Molecular Sciences, 2016, 17 (10), pp.1656. ⟨10.3390/ijms17101656⟩
Article dans une revue hal-03409019v1

Carbon nanotubes as gene carriers: Focus on internalization pathways related to functionalization and properties

Cécile Caoduro , Eric Hervouet , Corine Girard-Thernier , Tijani Gharbi , Hatem Boulahdour , et al.
Acta Biomaterialia, 2017, 49, pp.36-44. ⟨10.1016/j.actbio.2016.11.013⟩
Article dans une revue hal-03409033v1

Arginase Inhibitors: A Rational Approach Over One Century

M. Pudlo , Céline Demougeot , Corine Girard-Thernier
Medicinal Research Reviews, 2017, 37 (3), pp.475-513. ⟨10.1002/med.21419⟩
Article dans une revue hal-03409036v1

Arginase inhibitory properties of flavonoid compounds from the leaves of Mulberry ( Morus alba , Moraceae)

Kamel Arraki , Perle Totoson , Rym Attia , Andy Zedet , M. Pudlo , et al.
Journal of Pharmacy and Pharmacology, 2020, 72 (9), pp.1269-1277. ⟨10.1111/jphp.13297⟩
Article dans une revue hal-03409113v1

Donepezil–ferulic acid hybrids as anti-Alzheimer drugs

Mohamed Benchekroun , Lhassane Ismaili , M. Pudlo , Vincent Luzet , Tijani Gharbi , et al.
Future Medicinal Chemistry, 2015, 7 (1), pp.15-21. ⟨10.4155/fmc.14.148⟩
Article dans une revue hal-03407863v1

Novel aminotetrazole derivatives as selective STAT3 non-peptide inhibitors

Jean-René Pallandre , Christophe Borg , Didier Rognan , Thibault Boibessot , Vincent Luzet , et al.
European Journal of Medicinal Chemistry, 2015, 103, pp.163-174. ⟨10.1016/j.ejmech.2015.08.054⟩
Article dans une revue hal-03407857v1

Nanovectorization of TRAIL with Single Wall Carbon Nanotubes Enhances Tumor Cell Killing

Al Batoul Zakaria , Fabien Picaud , Thibault Rattier , M. Pudlo , Lucien Saviot , et al.
Nano Letters, 2015, 15 (2), pp.891-895. ⟨10.1021/nl503565t⟩
Article dans une revue hal-03407860v1

Cyperaceae Species Are Potential Sources of Natural Mammalian Arginase Inhibitors with Positive Effects on Vascular Function

Kamel Arraki , Perle Totoson , Alain Decendit , Alain Badoc , Andy Zedet , et al.
Journal of Natural Products, 2017, 80 (9), pp.2432-2438. ⟨10.1021/acs.jnatprod.7b00197⟩
Article dans une revue hal-03407791v1

Cinnamide Derivatives as Mammalian Arginase Inhibitors: Synthesis, Biological Evaluation and Molecular Docking

Thanh-Nhat Pham , Simon Bordage , M. Pudlo , Céline Demougeot , Khac-Minh Thai , et al.
International Journal of Molecular Sciences, 2016, 17 (10), pp.1656. ⟨10.3390/ijms17101656⟩
Article dans une revue hal-03407831v1
Image document

Nanovectorization of TRAIL with single wall carbon nanotubes enhances tumor cell killing

Al Batoul Zakaria , Fabien Picaud , Thibault Rattier , M. Pudlo , Lucien Saviot , et al.
Nano Letters, 2015, 15 (2), [Epub ahead of print]. ⟨10.1021/nl503565t⟩
Article dans une revue inserm-01113419v1

A tandem radical cyclization approach to 3-(2-oxopyrrolidin-3-yl)indolin-2-ones, potential intermediates toward complex indole-heterocycles

M. Pudlo , Stéphane Gérard , Catherine Mirand , Janos Sapi
Tetrahedron Letters, 2008, 49 (6), pp.1066-1070. ⟨10.1016/j.tetlet.2007.11.194⟩
Article dans une revue istex hal-03407879v1

Synthesis, biological assessment and molecular modeling of new dihydroquinoline-3-carboxamides and dihydroquinoline-3-carbohydrazide derivatives as cholinesterase inhibitors, and Ca channel antagonists

Isabelle Tomassoli , Lhassane Ismaili , M. Pudlo , Cristóbal de Los Ríos , Elena Soriano , et al.
European Journal of Medicinal Chemistry, 2011, 46 (1), pp.1-10. ⟨10.1016/j.ejmech.2010.08.054⟩
Article dans une revue istex hal-03407876v1

Novel aminotetrazole derivatives as selective STAT3 non-peptide inhibitors

Jean-René Pallandre , Christophe Borg , Didier Rognan , Thibault Boibessot , Vincent Luzet , et al.
European Journal of Medicinal Chemistry, 2015, 103, pp.163-174. ⟨10.1016/j.ejmech.2015.08.054⟩
Article dans une revue hal-04227818v1

Arginase inhibitory properties of flavonoid compounds from the leaves of Mulberry ( Morus alba , Moraceae)

Kamel Arraki , Perle Totoson , Rym Attia , Andy Zedet , M. Pudlo , et al.
Journal of Pharmacy and Pharmacology, 2020, 72 (9), pp.1269-1277. ⟨10.1111/jphp.13297⟩
Article dans une revue hal-03407767v1

Arginase Inhibitors: A Rational Approach Over One Century

M. Pudlo , Céline Demougeot , Corine Girard-Thernier
Medicinal Research Reviews, 2017, 37 (3), pp.475-513. ⟨10.1002/med.21419⟩
Article dans une revue hal-03407805v1

Synthesis, evaluation and molecular modelling of piceatannol analogues as arginase inhibitors

J. Muller , B. Cardey , A. Zedet , C. Desingle , M. Grzybowski , et al.
RSC Medicinal Chemistry, 2020, 11 (5), pp.559-568. ⟨10.1039/D0MD00011F⟩
Article dans une revue hal-02900460v1

An Update on Arginase Inhibitors and Inhibitory Assays

Jason Muller , Rym Attia , Andy Zedet , Corine Girard , M. Pudlo
Mini-Reviews in Medicinal Chemistry, 2021, 22, ⟨10.2174/1389557522666211229105703⟩
Article dans une revue hal-03581420v1

First Suzuki–Miyaura type cross-coupling of ortho-azidobromobenzene with arylboronic acids and its application to the synthesis of fused aromatic indole-heterocycles

M. Pudlo , Dorottya Csányi , Fabien Moreau , György Hajós , Zsuzsanna Riedl , et al.
Tetrahedron, 2007, 63 (41), pp.10320-10329. ⟨10.1016/j.tet.2007.07.068⟩
Article dans une revue istex hal-03407883v1

Selective Inhibition of STAT3 with Respect to STAT1: Insights from Molecular Dynamics and Ensemble Docking Simulations

Semen Yesylevskyy , Christophe Ramseyer , M. Pudlo , Jean-René Pallandre , Christophe Borg
Journal of Chemical Information and Modeling, 2016, 56 (8), pp.1588-1596. ⟨10.1021/acs.jcim.6b00198⟩
Article dans une revue hal-03407835v1

In Vitro Mammalian Arginase Inhibitory and Antioxidant Effects of Amide Derivatives Isolated from the Hempseed Cakes (Cannabis sativa)

Mélanie Bourjot , Andy Zedet , Belinda Demange , M. Pudlo , Corine Girard-Thernier
Planta Medica International Open, 2016, 3 (03), pp.e64-e67. ⟨10.1055/s-0042-119400⟩
Article dans une revue hal-03407799v1

Cinnamide Derivatives as Mammalian Arginase Inhibitors: Synthesis, Biological Evaluation and Molecular Docking

Thanh-Nhat Pham , Simon Bordage , M. Pudlo , Céline Demougeot , Khac-Minh Thai , et al.
International Journal of Molecular Sciences, 2016, 17 (10), pp.1656. ⟨10.3390/ijms17101656⟩
Article dans une revue hal-03409024v1