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Synthesis of new piperazinyl-pyrrolo[1,2- a ]quinoxaline derivatives as inhibitors of Candida albicans multidrug transporters by a Buchwald–Hartwig cross-coupling reaction

Jean Guillon , Shweta Nim , Stéphane Moreau , Luisa Ronga , Solène Savrimoutou , et al.
RSC Advances, 2020, 10 (5), pp.2915-2931. ⟨10.1039/C9RA09348F⟩
Article dans une revue hal-02449065v1

Synthesis and antiproliferative effect of ethyl 4-[4-(4-substituted piperidin-1-yl)]benzylpyrrolo[1,2-a]quinoxalinecarboxylate derivatives on human leukemia cells

Vanessa Desplat , Marian Vincenzi , Romain Lucas , Stéphane Moreau , Solène Savrimoutou , et al.
ChemMedChem, 2017, 12 (12), pp.940-953. ⟨10.1002/cmdc.201700049⟩
Article dans une revue hal-01560237v1

Crystal structure of a fluoro analogue of 3,4-(methylenedioxy)

Jean Guillon , Noël Pinaud , Mathieu Marchivie , Luisa Ronga , Abdelhamid Benazzouz , et al.
X-Ray Structure Analysis Online, 2015, 31 (4), pp.23-24. ⟨10.2116/xraystruct.31.23⟩
Article dans une revue hal-01166909v1
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Synthesis and Antimalarial Evaluation of New 1,3,5-tris[(4-(Substituted-aminomethyl)phenyl)methyl]benzene Derivatives: A Novel Alternative Antiparasitic Scaffold

Sandra Albenque-Rubio , Jean Guillon , Anita Cohen , Patrice Agnamey , Solène Savrimoutou , et al.
Drugs and Drug Candidates, 2023, 2 (3), pp.653-672. ⟨10.3390/ddc2030033⟩
Article dans une revue hal-04441752v1

Oxyfold: A simple and efficient solid-supported reagent for disulfide bond formation

P. Verdié , Luisa Ronga , M. Cristau , M. Amblard , S. Cantel , et al.
Chemistry - An Asian Journal, 2011, 6 (9), pp.2382-2389. ⟨10.1002/asia.201100202⟩
Article dans une revue istex hal-01563744v1

Aptasensors for the detection of emerging contaminants : development of an electrochemical platform

Quentin Palas , Adama Drabo , Mohamed Amine Berkal , Corinne Nardin , Christine Lartigau-Dagron , et al.
Les journées de la Société Chimique de France dans le Grand Sud-Ouest 2022, Jul 2022, Toulouse, France
Communication dans un congrès hal-03812406v1

Design, synthesis and antimalarial activity of novel bis\N-[(pyrrolo[1,2-a]quinoxalin-4-yl)benzyl]-3-aminopropyl\amine derivatives

J. Guillon , Anita Cohen , N.M. Gueddouda , R.N. Das , S. Moreau , et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2017, 32 (1), pp.547-563. ⟨10.1080/14756366.2016.1268608⟩
Article dans une revue hal-01535439v1

Peptide fragment approach to prion misfolding: The alpha-2 domain

P. Palladino , Luisa Ronga , E. Benedetti , F. Rossi , R. Ragone
International Journal of Peptide Research and Therapeutics, 2009, 15 (3), pp.165-176. ⟨10.1007/s10989-009-9171-6⟩
Article dans une revue istex hal-01563748v1

Crystal Structure of (E)-1-(3,4-Methylenedioxy-6-fluorophenyl)-2-nitropropene

Jean Guillon , Luisa Ronga , Mathieu Marchivie , Stéphane Moreau
X-Ray Structure Analysis Online, 2016, 32, pp.23-24. ⟨10.2116/xraystruct.32.23⟩
Article dans une revue hal-01432378v1

Gold‐promoted biocompatible selenium arylation of small molecules, peptides and proteins

Douglas Nakahata , Ioannis Kanavos , Maria Zubiria-Ulacia , Alex Inague , Luca Salassa , et al.
Chemistry - A European Journal, 2024, pp.e202304050. ⟨10.1002/chem.202304050⟩
Article dans une revue hal-04425725v1

Conformational diseases and structure-toxicity relationships: Lessons from prion-derived peptides

Luisa Ronga , P. Palladino , S. Costantini , A. Facchiano , M. Ruvo , et al.
Current Protein and Peptide Science, 2007, 8 (1), pp.83-90. ⟨10.2174/138920307779941505⟩
Article dans une revue hal-01563750v1

The prion protein: Structural features and related toxic peptides

E. Benedetti , F. Rossi , Luisa Ronga , B. Tizzano , P. Palladino , et al.
Chemical Biology and Drug Design, 2006, 68 (3), pp.139-147. ⟨10.1111/j.1747-0285.2006.00427.x⟩
Article dans une revue istex hal-01563753v1
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Characterization and Quantification of Selenoprotein P: Challenges to Mass Spectrometry

Jérémy Lamarche , Luisa Ronga , Joanna Szpunar , Ryszard Lobinski
International Journal of Molecular Sciences, 2021, 22 (12), pp.6283. ⟨10.3390/ijms22126283⟩
Article dans une revue hal-03265397v1
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Design, synthesis, and antiprotozoal evaluation of new 2,4-bis[(substituted-aminomethyl)phenyl]quinoline, 1,3-bis[(substituted-aminomethyl)phenyl]isoquinoline and 2,4-bis[(substituted-aminomethyl)phenyl]quinazoline derivatives

Jean Guillon , Anita Cohen , Clotilde Boudot , Alessandra Valle , Vittoria Milano , et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2020, 35 (1), pp.432-459. ⟨10.1080/14756366.2019.1706502⟩
Article dans une revue hal-02428661v1
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Synthesis and crystal structure of 3-{4-[(4-(2-Oxo-2,3-dihydro-1H-benzimidazol-1-yl)piperidin-1-yl)benzyl]}-2-phenylindole

Jean Guillon , Marian Vincenzi , Noël Pinaud , Luisa Ronga , Filomena Rossi , et al.
Structural Chemistry & Crystallography Communication, 2016, 2 (1), pp.18. ⟨10.21767/2470-9905.100018⟩
Article dans une revue hal-01432803v1

Crystal Structure of 7-Amino-4-iodo-3-propyl-1H-isochromen-1-one

Jean Guillon , Luisa Ronga , Mathieu Marchivie , Vincent Lisowki
X-Ray Structure Analysis Online, 2016, 32, pp.45-46. ⟨10.2116/xraystruct.32.45⟩
Article dans une revue hal-01432492v1

Design, synthesis, and antiprotozoal evaluation of new 2,9-bis[(substituted-aminomethyl)phenyl]-1,10-phenanthroline derivatives

Jean Guillon , Anita Cohen , Rabindra Nath Das , Clotilde Boudot , Nassima Meriem Gueddouda , et al.
Chemical Biology & Drug Design, 2018, ⟨10.1111/cbdd.13164⟩
Article dans une revue hal-01690455v1

A thermodynamic approach to the conformational preferences of the 180-195 segment derived from the human prion protein α2-helix

Luisa Ronga , P. Palladino , R. Ragone , E. Benedetti , F. Rossi
Journal of Peptide Science, 2009, 15 (1), pp.30-35. ⟨10.1002/psc.1086⟩
Article dans une revue istex hal-01563746v1

Spectroscopic analysis of synthetic PrP helix2-binding peptide constructs.

Luisa Ronga , P. Palladino , R. Ragone , J. Martinez , E. Benedetti , et al.
Advances in experimental medicine and biology, 2009, 611, pp.75-76. ⟨10.1007/978-0-387-73657-0_33⟩
Article dans une revue istex hal-01563747v1

Structural characterization of a neurotoxic threonine-rich peptide corresponding to the human prion protein α2-helical 180-195 segment and comparison with full-length α2-helix-derived peptides

Luisa Ronga , P. Palladino , G. Saviano , T. Tancredi , E. Benedetti , et al.
Journal of Peptide Science, 2008, 14 (10), pp.1096-1102. ⟨10.1002/psc.1046⟩
Article dans une revue istex hal-01563749v1
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Mechanistic Evaluations of the Effects of Auranofin Triethylphosphine Replacement with a Trimethylphosphite Moiety

Luisa Ronga , Iogann Tolbatov , Ester Giorgi , Paulina Pisarek , Christine Enjalbal , et al.
Inorganic Chemistry, 2023, 62, pp.10389 - 10396. ⟨10.1021/acs.inorgchem.3c01280⟩
Article dans une revue hal-04170599v1

Total chemical synthesis, refolding, and crystallographic structure of fully active immunophilin calstabin 2 (FKBP12.6): Chemical Synthesis of Catalytically Active Calstabin and Mutants

Marine Bacchi , Magali Jullian , Serena Sirigu , Benjamin Fould , Tiphaine Huet , et al.
Protein Science, 2016, 25 (12), pp.2225-2242. ⟨10.1002/pro.3051⟩
Article dans une revue hal-01498750v1

Selenol (-SeH) as a target for mercury and gold in biological systems: Contributions of mass spectrometry and atomic spectroscopy

Mikel Bernabeu de Maria , Jérémy Lamarche , Luisa Ronga , Luigi Messori , Joanna Szpunar , et al.
Coordination Chemistry Reviews, 2023, 474, pp.214836. ⟨10.1016/j.ccr.2022.214836⟩
Article dans une revue hal-03842066v1
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Study of metalation of thioredoxin by gold(I) therapeutic compounds using combined liquid chromatography/capillary electrophoresis with inductively coupled plasma/electrospray MS/MS detection

Mikel Bernabeu de Maria , Magdalena Matczuk , Diego Tesauro , Michele Saviano , Jacek Sikorski , et al.
Analytical and Bioanalytical Chemistry, 2024, ⟨10.1007/s00216-024-05140-z⟩
Article dans une revue hal-04425803v1

Conformational ensembles explored dynamically from disordered peptides targeting chemokine receptor CXCR4

M. Vincenzi , S. Costantini , S. Scala , D. Tesauro , A. Accardo , et al.
International Journal of Molecular Sciences, 2015, 16 (6), pp.12159-12173. ⟨10.3390/ijms160612159⟩
Article dans une revue hal-01563738v1

Crystal structure of a fluoro analogue of 3,4-(methylenedioxy)amphetamine

J. Guillon , N. Pinaud , M. Marchivie , Luisa Ronga , A. Benazzouz , et al.
X-Ray Structure Analysis Online, 2015, 31 (4), pp.23-24
Article dans une revue hal-01563739v1

Synthesis and evaluation of the cytotoxic activity of novel ethyl 4-[4-(4-substitutedpiperidin-1-yl)]benzyl-phenylpyrrolo[1,2-a]quinoxaline-carboxylate derivatives in myeloid and lymphoid leukemia cell lines

Vanessa Desplat , Marian Vincenzi , Romain Lucas , Stéphane Moreau , Solène Savrimoutou , et al.
European Journal of Medicinal Chemistry, 2016, 113, pp.214-227. ⟨10.1016/j.ejmech.2016.02.047⟩
Article dans une revue hal-01307573v1

Design, synthesis and biological evaluation of novel 4- alkapolyenylpyrrolo[1,2-a]quinoxalines as antileishmanial agents - Part III

Luisa Ronga , M. del Favero , A. Cohen , C. Soum , P. Le Pape , et al.
European Journal of Medicinal Chemistry, 2014, 81, pp.378-393. ⟨10.1016/j.ejmech.2014.05.037⟩
Article dans une revue hal-01563740v1
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Design, Synthesis, and Antiprotozoal Evaluation of New Promising 2,9-Bis[(substituted-aminomethyl)]-4,7-phenyl-1,10phenanthroline Derivatives, a Potential Alternative Scaffold to Drug Efflux

Jean Guillon , Anita Cohen , Clotilde Boudot , Sarah Monic , Solène Savrimoutou , et al.
Pathogens, 2022, 11 (11), pp.1339. ⟨10.3390/pathogens11111339⟩
Article dans une revue inserm-03850360v1
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New 2,4-bis[(substituted-aminomethyl)phenyl]phenylquinazoline and 2,4-bis[(substituted-aminomethyl)phenyl]phenylquinoline derivatives: synthesis and biological evaluation as novel anticancer agents by targeting G-quadruplex

Jean Guillon , Marc Le Borgne , Vittoria Milano , Aurore Guédin-Beaurepaire , Stéphane Moreau , et al.
Pharmaceuticals, 2024, 17 (1), pp.30. ⟨10.3390/ph17010030⟩
Article dans une revue hal-04390485v1