|
|
Epidrugs as Promising Tools to Eliminate Plasmodium falciparum Artemisinin-Resistant and Quiescent Parasites
Thibaud Reyser
,
Lucie Paloque
,
Michel Nguyen
,
Jean-Michel Augereau
,
Matthew John Fuchter
,
et al.
Article dans une revue
hal-04269105v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Mutation in the Plasmodium falciparum BTB/POZ Domain of K13 Protein Confers Artemisinin Resistance
Lucie Paloque
,
Romain Coppée
,
Barbara Stokes
,
Nina Gnädig
,
Karamoko Niaré
,
et al.
Article dans une revue
hal-03561782v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Discovery of a new antileishmanial hit in 8-nitroquinoline series
Lucie Paloque
,
Pierre Verhaeghe
,
Magali Casanova
,
Caroline Castera-Ducros
,
Aurélien Dumètre
,
et al.
European Journal of Medicinal Chemistry, 2012, 54, pp.75-86
Article dans une revue
hal-02049707v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Synthesis, structures, and biological studies of heterobimetallic Au(I)-Ru(II) complexes involving N-heterocyclic carbene-based multidentate ligands
Luca Boselli
,
Maëlle Carraz
,
S. Mazeres
,
Lucie Paloque
,
German Gonzalez-Aspajo
,
et al.
Article dans une revue
hal-01925137v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Evaluation of antiplasmodial and antileishmanial activities of herbal medicine Pseudelephantopus spiralis (Less.) Cronquist and isolated hirsutinolide-type sesquiterpenoids
Cynthia Girardi
,
Nicolas Fabre
,
Lucie Paloque
,
Arba Pramundita Ramadani
,
Françoise Benoit-Vical
,
et al.
Article dans une revue
hal-01925138v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Synthesis, characterization, and antileishmanial activities of gold(I) complexes involving quinoline functionalized N-heterocyclic carbenes
Lucie Paloque
,
Catherine Hemmert
,
Alexis Valentin
,
Heinz Gornitzka
Article dans une revue
hal-01925132v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Endoperoxide-based compounds: cross-resistance with artemisinins and selection of a Plasmodium falciparum lineage with a K13 non-synonymous polymorphism
Lucie Paloque
,
Benoit Witkowski
,
Joël Lelièvre
,
Manel Ouji
,
Tanila Ben Haddou
,
et al.
Article dans une revue
hal-01963522v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Novel 8-nitroquinolin-2(1 H )-ones as NTR-bioactivated antikinetoplastid molecules: Synthesis, electrochemical and SAR study
Julien Pedron
,
Clotilde Boudot
,
Sébastien Hutter
,
Sandra Bourgeade-Delmas
,
Jean-Luc Stigliani
,
et al.
Article dans une revue
hal-01888465v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Hybrid Peptide-Alkoxyamine Drugs: A Strategy for the Development of a New Family of Antiplasmodial Drugs
Ange W Embo-Ibouanga
,
Michel Nguyen
,
Lucie Paloque
,
Mathilde Coustets
,
Jean-Patrick Joly
,
et al.
Article dans une revue
hal-04515160v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Polyunsaturated fatty acid metabolites: biosynthesis in Leishmania and role in parasite/host interaction
Lucie Paloque
,
Teresa Pérez-Berezo
,
Anne Abot
,
Jessica Dalloux-Chioccioli
,
Sandra Bourgeade-Delmas
,
et al.
Article dans une revue
hal-02140502v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Antitrypanosomatid Pharmacomodulation at Position 3 of the 8-Nitroquinolin-2(1 H)-one Scaffold Using Palladium-Catalysed Cross-Coupling Reactions
Julien Pedron
,
Clotilde Boudot
,
Sandra Bourgeade-Delmas
,
Alix Sournia-Saquet
,
Lucie Paloque
,
et al.
Article dans une revue
hal-01888530v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Identification of compounds active against quiescent artemisinin-resistant Plasmodium falciparum parasites via the quiescent-stage survival assay (QSA)
Thibaud Reyser
,
Lucie Paloque
,
Manel Ouji
,
Michel Nguyen
,
Sandie Ménard
,
et al.
Article dans une revue
hal-02948398v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Plasmodium falciparum resistance to artemisinin-based combination therapies (ACTs): Fears of widespread drug resistance
Françoise Benoit-Vical
,
Lucie Paloque
,
Jean-Michel Augereau
Bulletin de l'Académie Nationale de Médecine, 2016, 200 (3), pp.477-489
Article dans une revue
hal-01937598v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Antileishmanial pharmacomodulation in 8-nitroquinolin-2(1H)-one series
Charline Kieffer
,
Anita Cohen
,
Pierre Verhaeghe
,
Lucie Paloque
,
Sébastien Hutter
,
et al.
Article dans une revue
hal-01460646v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Antiprotozoal properties of Indonesian medicinal plant extracts
Arba Pramundita Ramadani
,
Lucie Paloque
,
Hugo Belda
,
Hady Anshory Tamhid
,
Jumina Masriani
,
et al.
Article dans une revue
hal-01963518v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Zebiriosides A-L, oleanane saponins from the roots of Dendrobangia boliviana
Ilhem Zebiri
,
Mohamed Haddad
,
Laurent Duca
,
Dominique Harakat
,
Billy Cabanillas
,
et al.
Article dans une revue
hal-01937592v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
A New Thienopyrimidinone Chemotype Shows Multistage Activity against Plasmodium falciparum, Including Artemisinin-Resistant Parasites
Henriette Bosson-Vanga
,
Nicolas Primas
,
Jean-François Franetich
,
Catherine Lavazec
,
Lina Gomez
,
et al.
Article dans une revue
hal-03363796v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Multiple phenotypic and genotypic artemisinin sensitivity evaluation of Malian Plasmodium falciparum isolates
Karamoko Niare
,
Lucie Paloque
,
Sandie Ménard
,
Pety Tor
,
Arba Pramundita Ramadani
,
et al.
Article dans une revue
hal-01963527v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Plasmodium falciparum: multifaceted resistance to artemisinins
Lucie Paloque
,
Arba Pramundita Ramadani
,
Odile Mercereau-Puijalon
,
Jean-Michel Augereau
,
Françoise Benoit-Vical
Article dans une revue
inserm-01322524v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium
Anita Cohen
,
Peggy Suzanne
,
Jean-Charles Lancelot
,
Pierre Verhaeghe
,
Aurélien Lesnard
,
et al.
Article dans une revue
hal-01460555v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
2-Phenoxy-3-Trichloromethylquinoxalines Are Antiplasmodial Derivatives with Activity against the Apicoplast of Plasmodium falciparum
Dyhia Amrane
,
Christophe-Sébastien Arnold
,
Sébastien Hutter
,
Julen Sanz-Serrano
,
Miguel Collia
,
et al.
Article dans une revue
hal-03323862v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Plasmodium falciparum resistance to artemisinin-based combination therapies: A sword of Damocles in the path toward malaria elimination
Manel Ouji
,
Jean-Michel Augereau
,
Lucie Paloque
,
Françoise Benoit-Vical
Article dans une revue
hal-01963526v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Résistance de l'agent du paludisme, Plasmodium falciparum aux combinaisons thérapeutiques à base d'artémisinine (ACTs) : Craintes d'une chimiorésistance généralisée
Françoise Benoit-Vical
,
Lucie Paloque
,
Jean-Michel Augereau
Bulletin de l'Académie Nationale de Médecine, 2016, 200 (3), pp.477-490
Article dans une revue
hal-03232081v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Synthesis and evaluation of monoamidoxime derivatives: Toward new antileishmanial compounds
Lucie Paloque
,
Ahlem Bouhlel
,
Christophe Curti
,
Aurélien Dumètre
,
Pierre Verhaeghe
,
et al.
Article dans une revue
istex
hal-01460338v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
A new, rapid and sensitive bioluminescence assay for drug screening on Leishmania
Lucie Paloque
,
Nicolas Nvidal@mnhn.Fr Vidal
,
Magali Casanova
,
Aurélien Dumètre
,
Pierre Verhaeghe
,
et al.
Article dans une revue
hal-01460476v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Targeting the human parasite Leishmania donovani: Discovery of a new promising anti-infectious pharmacophore in 3-nitroimidazo[1,2-a]pyridine series
Caroline Castera-Ducros
,
Lucie Paloque
,
Pierre Verhaeghe
,
Magali Casanova
,
Christophe Cantelli
,
et al.
Article dans une revue
istex
hal-01460446v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Epigenetic regulation as a therapeutic target in the malaria parasite Plasmodium falciparum
Thibaud Reyser
,
Lucie Paloque
,
Jean-Michel Augereau
,
Luisa Di Stefano
,
Françoise Benoit-Vical
Article dans une revue
hal-04502290v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Antiplasmodial activities of gold(I) complexes involving functionalized N-heterocyclic carbenes
Catherine Hemmert
,
Arba Pramundita Ramadani
,
Luca Boselli
,
Alvaro Fernandez Alvarez
,
Lucie Paloque
,
et al.
Article dans une revue
hal-01937596v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
Synthèse et évaluations biologiques de nouvelles 8-nitroquinoléin-2(1H)-ones antiparisitaires.
Julien Pedron
,
Clotilde Boudot
,
Sebastien Hutter
,
Sandra Bourgeade-Delmas
,
Lucie Paloque
,
et al.
8èmes Journées du Consortium anti-Parasitaires et anti-Fongique (CaPF), Mar 2018, Lyon, France
Communication dans un congrès
hal-01939612v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|
|
|
A new phthalide derivative from Peperomia nivalis
Pedro Vásquez-Ocmín
,
Mohamed Haddad
,
Alice Gadea
,
Valérie Jullian
,
Denis Castillo
,
et al.
Article dans une revue
ird-01381569v1
|
Partager
Gmail
Facebook
X
LinkedIn
More
|