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Reversing HIV latency via sphingosine-1-phosphate receptor 1 signaling

 Charline Duquenne , Sandrine Gimenez , Adeline Guigues , Benjamin Viala , Caroline Boulouis , et al.
AIDS. Official journal of the international AIDS Society, 2017, 31 (18), pp.2443 - 2454. ⟨10.1097/QAD.0000000000001649⟩
Article dans une revue hal-01635726v1
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Oligomerization of a G protein-coupled receptor in neurons controlled by its structural dynamics

 Thor C Møller , Jérôme Hottin , Caroline Clerté , Jurriaan M. Zwier , Thierry Durroux , et al.
Scientific Reports, 2018, 8 (1), ⟨10.1038/s41598-018-28682-6⟩
Article dans une revue hal-02398134v1

Agonist-independent activation of metabotropic glutamate receptors by the intracellular protein Homer.

 Fabrice Ango , Laurent Prézeau , Thomas Muller , Jian C. Tu , Bo Xiao , et al.
Nature, 2001, 411 (6840), pp.962-5. ⟨10.1038/35082096⟩
Article dans une revue inserm-00318959v1

Time-Resolved Förster Resonance Energy Transfer-Based Technologies to Investigate G Protein-Coupled Receptor Machinery

 Pauline Scholler , Jurriaan Zwier , Eric Trinquet , Philippe Rondard , Jean-Philippe Pin , et al.
Fluorescence-Based Biosensors - From Concepts to Applications, 113, Elsevier, pp.275-312, 2013, Progress in Molecular Biology and Translational Science, ⟨10.1016/B978-0-12-386932-6.00007-7⟩
Chapitre d'ouvrage hal-03363917v1
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Different EGF ‐induced receptor dimer conformations for signaling and internalization

 Jordi Haubrich , Jurriaan Zwier , Fabienne Charrier-Savournin , Laurent Prézeau , Jean‐philippe Pin
FASEB Journal, 2024, 38 (1), pp.e23356. ⟨10.1096/fj.202301209R⟩
Article dans une revue hal-04472295v1
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Real-time analysis of agonist-induced activation of protease-activated receptor 1/Galphai1 protein complex measured by bioluminescence resonance energy transfer in living cells.

 Mohammed Akli Ayoub , Damien Maurel , Virginie Binet , Michel Fink , Laurent Prézeau , et al.
Molecular Pharmacology, 2007, 71 (5), pp.1329-40. ⟨10.1124/mol.106.030304⟩
Article dans une revue hal-00318930v1

Synthesis and pharmacological characterization of conformationally restricted 2-amino-Adipic acid analogs and carboxycyclopropyl glycines as selective metabotropic glutamate 2 receptor agonists

 Markus Staudt , Na Liu , Fanny Malhaire , Yasaman Doroudian , Laurent Prézeau , et al.
European Journal of Medicinal Chemistry, 2024, 266, pp.116157. ⟨10.1016/j.ejmech.2024.116157⟩
Article dans une revue hal-04415292v1

Re-expression of the neurodevelopmental protein filamin A in glioblastoma via signaling switch of the urotensin II vasoactive peptide receptor

 Alexandre Mutel , Céline Lecointre , Kleouforo Paul Dembele , Pierre-Olivier Guichet , L Mouchard , et al.
22nd International Symposium on Regulatory Peptides, Sep 2018, Acapulco, Mexico
Communication dans un congrès hal-02296705v1
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GPCR interaction as a possible way for allosteric control between receptors

 Jean-Philippe Pin , Julie Kniazeff , Laurent Prézeau , Jiang-Feng Liu , Philippe Rondard
Molecular and Cellular Endocrinology, 2019, ⟨10.1016/j.mce.2019.02.019⟩
Article dans une revue hal-02396289v1
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BAY36-7620: a potent non-competitive mGlu1 receptor antagonist with inverse agonist activity.

 Fiona Y. Carroll , Andreas Stolle , Philip M. Beart , Arnd Voerste , Isabelle Brabet , et al.
Molecular Pharmacology, 2001, 59 (5), pp.965-73. ⟨10.1124/mol.59.5.965⟩
Article dans une revue inserm-00319007v1

The chemokine CXC4 and CC2 receptors form homo- and heterooligomers that can engage their signaling G-protein effectors and betaarrestin

 Sylvain Armando , Julie Quoyer , Viktorya Lukashova , Arhamatoulaye Maiga , Yann Percherancier , et al.
FASEB Journal, 2014, 28 (10), pp.4509--23. ⟨10.1096/fj.13-242446⟩
Article dans une revue hal-01950128v1
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Asymmetric functioning of dimeric metabotropic glutamate receptors disclosed by positive allosteric modulators.

 Cyril Goudet , Julie Kniazeff , Veronika Hlavackova , Fanny Malhaire , Damien Maurel , et al.
Journal of Biological Chemistry, 2005, 280 (26), pp.24380-5. ⟨10.1074/jbc.M502642200⟩
Article dans une revue inserm-00318925v1
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Cell surface protein-protein interaction analysis with combined time-resolved FRET and snap-tag technologies: application to GPCR oligomerization

 Damien Maurel , Laetitia Comps-Agrar , Carsten Brock , Marie-Laure Rives , Emmanuel Bourrier , et al.
Nature Methods, 2008, 5 (6), pp.561. ⟨10.1038/nmeth.1213⟩
Article dans une revue hal-00318856v1
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The G Protein-Coupled Receptor UT of the Neuropeptide Urotensin II Displays Structural and Functional Chemokine Features

 Hélène Castel , Laurence Desrues , Jane-Eileen Joubert , Marie-Christine Tonon , Laurent Prézeau , et al.
Frontiers in Endocrinology, 2017, 8, pp.76. ⟨10.3389/fendo.2017.00076⟩
Article dans une revue hal-02280590v1

The vasoactive peptide urotensin II as a new chemokine exhibits migration/adhesion mesenchymal properties accompanying angiogenesis during glioma development

 Hélène Castel , Pierre-Olivier Guichet , Céline Lecointre , Vadim Lejoncour , Eileen Joubert Jane , et al.
4ème Journée Scientifique de l’IRIB, Jun 2015, Rouen, France
Poster de conférence hal-02352398v1
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Among the twenty classical L-amino acids, only glutamate directly activates metabotropic glutamate receptors.

 Mélanie Frauli , Pascal Neuville , Claire Vol , Jean-Philippe Pin , Laurent Prézeau
Neuropharmacology, 2006, 50 (2), pp.245-53. ⟨10.1016/j.neuropharm.2005.09.016⟩
Article dans une revue inserm-00318879v1
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HTRF® total and phospho-YAP(Ser127) cellular assays

 Diana Zindel , Claire Vol , Odile Lecha , Isabelle Bourquignon , Merve Bilgic , et al.
The Hippo pathway: Methods and Protocols, 1893, pp.153-166, 2019, Methods in Molecular Biology, ⟨10.1007/978-1-4939-8910-2_13⟩
Chapitre d'ouvrage hal-02396286v1
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Amino-pyrrolidine tricarboxylic acids give new insight into group III metabotropic glutamate receptor activation mechanism.

 Mélanie Frauli , Nadia Hubert , Stephan Schann , Nicolas Triballeau , Hugues-Olivier Bertrand , et al.
Molecular Pharmacology, 2007, 71 (3), pp.704-12. ⟨10.1124/mol.106.030254⟩
Article dans une revue inserm-00318866v1

Impact of a key ancestral deletion in chemokine and vasoactive peptide receptors on G protein couplings and chemotaxis

 Jane Eilen Joubert , Laurence Desrues , Nicolas Perzo , B Taddese , Céline Lecointre , et al.
GPCRs: Beyond Structure Towards Therapy, Sep 2015, Prato, Italy
Communication dans un congrès hal-02296948v1

Signaling switch of the urotensin II vasosactive peptide GPCR: prototypic chemotaxic mechanism in glioma

 Céline Lecointre , Laurence Desrues , Jane Eileen Joubert , Nicolas Perzo , Pierre-Olivier Guichet , et al.
Oncogene, 2015, 34 (39), pp.5080-5094. ⟨10.1038/onc.2014.433⟩
Article dans une revue hal-02367872v1
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Identification of key phosphorylation sites in PTH1R that determine arrestin3 binding and fine-tune receptor signaling

 Diana Zindel , S. Engel , A. R. Bottrill , Jean-Philippe Pin , Laurent Prézeau , et al.
Biochemical Journal, 2016, 473 (22), pp.4173--4192. ⟨10.1042/BCJ20160740⟩
Article dans une revue hal-01940960v1
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Common structural requirements for heptahelical domain function in class A and class C G protein-coupled receptors.

 Virginie Binet , Béatrice Duthey , Jennifer Lecaillon , Claire Vol , Julie Quoyer , et al.
Journal of Biological Chemistry, 2007, 282 (16), pp.12154-63. ⟨10.1074/jbc.M611071200⟩
Article dans une revue inserm-00318820v1
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Non-classical ligand-independent regulation of Go protein by an orphan Class C GPCR

 Mariana Hajj , Teresa de Vita , Claire Vol , Charlotte Renassia , Jean-Charles Bologna , et al.
Molecular Pharmacology, 2019, 96 (2), pp.233-246. ⟨10.1124/mol.118.113019⟩
Article dans une revue hal-02396282v1
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Pharmacological evidence for a metabotropic glutamate receptor heterodimer in neuronal cells

 David Moreno-Delgado , Thor C Møller , Jeanne Ster , Jesús Giraldo , Damien Maurel , et al.
eLife, 2017, 6, ⟨10.7554/eLife.25233⟩
Article dans une revue hal-02073201v1
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The heptahelical domain of GABA(B2) is activated directly by CGP7930, a positive allosteric modulator of the GABA(B) receptor.

 Virginie Binet , Carole Brajon , Laurent Le Corre , Francine Acher , Jean-Philippe Pin , et al.
Journal of Biological Chemistry, 2004, 279 (28), pp.29085-91. ⟨10.1074/jbc.M400930200⟩
Article dans une revue inserm-00318926v1

Allosteric functioning of dimeric class C G-protein-coupled receptors.

 Jean-Philippe Pin , Julie Kniazeff , Jianfeng Liu , Virginie Binet , Cyril Goudet , et al.
FEBS Journal, 2005, 272, pp.2947-55. ⟨10.1111/j.1742-4658.2005.04728.x⟩
Article dans une revue inserm-00094959v1
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A single subunit (GB2) is required for G-protein activation by the heterodimeric GABA(B) receptor.

 Béatrice Duthey , Sara Caudron , Julie Perroy , Bernhard Bettler , Laurent Fagni , et al.
Journal of Biological Chemistry, 2002, 277 (5), pp.3236-41. ⟨10.1074/jbc.M108900200⟩
Article dans une revue inserm-00318936v1
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Targeting the Brain with Single-Domain Antibodies: Greater Potential Than Stated So Far?

 Mireille Elodie Tsitokana , Pierre-André Lafon , Laurent Prézeau , Jean-Philippe Pin , Philippe Rondard
International Journal of Molecular Sciences, 2023, 24 (3), pp.2632. ⟨10.3390/ijms24032632⟩
Article dans une revue hal-03991195v1
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SGIP1 modulates kinetics and interactions of the cannabinoid receptor 1 and G protein‐coupled receptor kinase 3 signalosome

 Matej Gazdarica , Judith Noda , Oleh Durydivka , Vendula Novosadova , Ken Mackie , et al.
Journal of Neurochemistry, 2022, 160 (6), pp.625-642. ⟨10.1111/jnc.15569⟩
Article dans une revue hal-03761588v1

Functional characterization of eel dopamine D2 receptors and involvement in the direct inhibition of pituitary gonadotropins

 Cécile Jolly , Karine Rousseau , Laurent Prézeau , Claire Vol , Jonna Tomkiewicz , et al.
Journal of Neuroendocrinology, 2016, 28 (9), ⟨10.1111/jne.12411⟩
Article dans une revue istex hal-01366809v1
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