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Identification of a non-canonical G3BP-binding sequence in a Mayaro virus nsP3 hypervariable domain

Aymeric Neyret , Eric Bernard , Olivier Aïqui-Reboul-Paviet , William Bakhache , Patrick Eldin , et al.
Frontiers in Cellular and Infection Microbiology, 2022, 12, ⟨10.3389/fcimb.2022.958176⟩
Article dans une revue hal-03796491v1
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Synthesis of Substituted 5′‐Aminoadenosine Derivatives and Evaluation of Their Inhibitory Potential toward CD73

Rayane Ghoteimi , van Tai Nguyen , Rahila Rahimova , Felix Grosjean , Emeline Cros‐perrial , et al.
ChemMedChem, 2019, 14 (15), pp.1431-1443. ⟨10.1002/cmdc.201900348⟩
Article dans une revue hal-02335429v1

Structure-activity relationships of β-hydroxyphosphonate nucleoside analogues as cytosolic 5′-nucleotidase II potential inhibitors: Synthesis, in vitro evaluation and molecular modeling studies.

Maïa Meurillon , Zsuzsanna Marton , Audrey Hospital , Lars Petter Jordheim , Jérôme Béjaud , et al.
European Journal of Medicinal Chemistry, 2014, 77 (April 2014), pp.18-37. ⟨10.1016/j.ejmech.2014.02.055⟩
Article dans une revue hal-00956313v1
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The Glutaminase-Dependent System Confers Extreme Acid Resistance to New Species and Atypical Strains of Brucella

Luca Freddi , Maria Damiano , Laurent Chaloin , Eugenia Pennacchietti , Sascha Al Dahouk , et al.
Frontiers in Microbiology, 2017, 8, pp.2236. ⟨10.3389/fmicb.2017.02236⟩
Article dans une revue hal-01868348v1

Identification and characterization of inhibitors of cytoplasmic 5′-nucleotidase cN-II issued from virtual screening

Lars Petter Jordheim , Zsuzsanna Marton , Moez Rhimi , Emeline Cros-Perrial , Corinne Lionne , et al.
Biochemical Pharmacology, 2013, 85 (4), pp.497-506. ⟨10.1016/j.bcp.2012.11.024⟩
Article dans une revue istex hal-03371022v1

Identification and characterization of inhibitors of cytoplasmic 5′-nucleotidase cN-II issued from virtual screening

Lars Petter Jordheim , Zsuzsanna Marton , Moez Rhimi , Emeline Cros-Perrial , Corinne Lionne , et al.
Biochemical Pharmacology, 2013, 85 (4), pp.497-506. ⟨10.1016/j.bcp.2012.11.024⟩
Article dans une revue istex hal-03370997v1

Design of Carrier Peptide-Oligonucleotide Conjugates with Rapid Membrane Translocation and Nuclear Localization Properties

L. Chaloin , P. Vidal , Philippe Lory , J. Mery , N. Lautredou , et al.
Biochemical and Biophysical Research Communications, 1998, 243 (2), pp.601-608. ⟨10.1006/bbrc.1997.8050⟩
Article dans une revue istex hal-02088286v1

Coarse-Grained Simulations of the HIV-1 Matrix Protein Anchoring: Revisiting Its Assembly on Membrane Domains.

Landry Charlier , Maxime Louet , Laurent Chaloin , Patrick Fuchs , Jean Martinez , et al.
Biophysical Journal, 2014, 106 (3), pp.577-585. ⟨10.1016/j.bpj.2013.12.019⟩
Article dans une revue hal-01105330v1

Synthesis of (R)- and (S)-ßhydroxyphosphonate acyclonucleosides: structural analogues of Adefovir (PMEA)

Mahesh Kasthuri , Laurent Chaloin , Christian Perigaud , Suzanne Peyrottes
Tetrahedron: Asymmetry, 2011, 22, pp.1505-1511. ⟨10.1016/j.tetasy.2011.08.010⟩
Article dans une revue hal-00637860v1
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An evolutionarily conserved N-terminal leucine is essential for MX1 GTPase antiviral activity against different families of RNA viruses

Joe Mckellar , Mary Arnaud-Arnould , Laurent Chaloin , Marine Tauziet , Charlotte Arpin-André , et al.
Journal of Biological Chemistry, 2023, 299 (1), pp.102747. ⟨10.1016/j.jbc.2022.102747⟩
Article dans une revue hal-03937465v1
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Molecular basis for the lack of enantioselectivity of human 3-phosphoglycerate kinase.

C. Gondeau , L. Chaloin , P. Lallemand , B. Roy , C. Périgaud , et al.
Nucleic Acids Research, 2008, 36 (11), pp.3620-9. ⟨10.1093/nar/gkn212⟩
Article dans une revue hal-00311704v1

CD73 inhibition by purine cytotoxic nucleoside analogue-based diphosphonates

Charles Dumontet , Suzanne Peyrottes , Céline Rabeson , Emeline Cros-Perrial , Pierre Yves Géant , et al.
European Journal of Medicinal Chemistry, 2018, 157, pp.1051-1055. ⟨10.1016/j.ejmech.2018.08.035⟩
Article dans une revue hal-02335419v1
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A new peptide vector for efficient delivery of oligonucleotides into mammalian cells

May C Morris , Pierre Vidal , Laurent Chaloin , Frédéric Heitz , Gilles Divita
Nucleic Acids Research, 1997, 25 (14), pp.2730-2736. ⟨10.1093/nar/25.14.2730⟩
Article dans une revue hal-03149766v1

Solid-phase Synthesis and Cellular Localization of a C- and/or N-terminal Labelled Peptide

P. Vidal , L. Chaloin , J. Mery , N. Lamb , N. Lautredou , et al.
Journal of Peptide Science, 1996, 2 (2), pp.125-133. ⟨10.1002/psc.58⟩
Article dans une revue istex hal-02088307v1
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Synthesis and Studies of Potential Inhibitors of CD73 Based on a Triazole Scaffold

Félix Grosjean , Emeline Cros-Perrial , Abdenour Braka , Jean‐pierre Uttaro , Laurent Chaloin , et al.
European Journal of Organic Chemistry, 2022, 2022 (21), ⟨10.1002/ejoc.202101175⟩
Article dans une revue hal-03842146v1
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Potent inhibition of HIV-1 replication by backbone cyclic peptides bearing the Rev arginine rich motif

Laurent Chaloin , Fatima Smagulova , Elana Hariton-Gazal , Laurence Briant , Abraham Loyter , et al.
Journal of Biomedical Science, 2007, 14 (5), pp.565-584. ⟨10.1007/s11373-007-9180-4⟩
Article dans une revue hal-00257424v1

Identification of noncompetitive inhibitors of cytosolic 5′-nucleotidase II using a fragment-based approach

Zsuzsanna Marton , Rémi Guillon , Isabelle Krimm , Rahila Rahimova , David Egron , et al.
Journal of Medicinal Chemistry, 2015, 58 (24), pp.9680-9696. ⟨10.1021/acs.jmedchem.5b01616⟩
Article dans une revue hal-01251800v1

Direct kinetic evidence that lysine 215 is involved in the phospho-transfer step of human 3-phosphoglycerate kinase.

Andrea Varga , Corinne Lionne , Perrine Lallemand , Judit Szabó , Nancy Adamek , et al.
Biochemistry, 2009, 48 (29), pp.6998-7008. ⟨10.1021/bi900396h⟩
Article dans une revue hal-00420536v1
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Cytotoxic and Antitumoral Activity of N-(9H-purin-6-yl) Benzamide Derivatives and Related Water-soluble Prodrugs

Emeline Cros-Perrial , Steve Saulnier , Muhammad Zawwad Raza , Rémi Charmelot , David Egron , et al.
Current Molecular Pharmacology, 2022, 15 (6), pp.883-894. ⟨10.2174/1874467214666211014164406⟩
Article dans une revue hal-03809743v1
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Identification of allosteric inhibitors of the ecto-5'-nucleotidase (CD73) targeting the dimer interface

Rahila Rahimova , Simon Fontanel , Corinne Lionne , Lars Peter Jordheim , Suzanne Peyrottes , et al.
PLoS Computational Biology, 2018, 14 (1), pp.e1005943. ⟨10.1371/journal.pcbi.1005943⟩
Article dans une revue hal-01838257v1

Translocating peptides and proteins and their use for gene delivery

May Morris , Laurent Chaloin , Frederic Heitz , Gilles Divita
Current Opinion in Biotechnology, 2000, 11 (5), pp.461-466. ⟨10.1016/s0958-1669(00)00128-2⟩
Article dans une revue istex hal-03130072v1

A novel potent strategy for gene delivery using a single peptide vector as a carrier

M. Morris , L. Chaloin , J. Mery , F. Heitz , G. Divita
Nucleic Acids Research, 1999, 27 (17), pp.3510-3517. ⟨10.1093/nar/27.17.3510⟩
Article dans une revue hal-03130242v1
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HIV-1 viral infectivity factor interacts with microtubule-associated protein light chain 3 and inhibits autophagy

Sophie Borel , Véronique Robert-Hebmann , Jamal Alfaisal , Ashish Jain , Mathias Faure , et al.
AIDS. Official journal of the international AIDS Society, 2015, 29 (3), pp.275-286. ⟨10.1097/QAD.0000000000000554⟩
Article dans une revue hal-02421817v1
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VSV-G pseudotyping rescues HIV-1 CA mutations that impair core assembly or stability

Sonia Brun , Maxime Solignat , Bernard Gay , Eric Bernard , Laurent Chaloin , et al.
Retrovirology, 2008, 5, pp.57. ⟨10.1186/1742-4690-5-57⟩
Article dans une revue hal-02147193v1
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Synthesis of Pyrimidine-Containing Nucleoside β-(R/S)-Hydroxyphosphonate Analogues

Maïa Meurillon , Laurent Chaloin , Christian Perigaud , Suzanne Peyrottes
European Journal of Organic Chemistry, 2011, 20-21, pp.3794-3802. ⟨10.1002/ejoc.201100219⟩
Article dans une revue istex hal-00616845v1

Drug discovery and optimization targeting CD73 to restore anticancer immune response

Braka A. , Rahila Rahimova , Suzanne Peyrottes , Lars Petter Jordheim , C. Caux , et al.
The 18th Symposium (PP19) on Purine and Pyrimidine Metabolism in Man, The Purine and Pyrimidine Society, Jun 2019, Lyon, France
Communication dans un congrès hal-02435174v1
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Dihydropyrimidinase protects from DNA replication stress caused by cytotoxic metabolites

J. Basbous , Antoine Aze , Laurent Chaloin , Rana Lebdy , Dana Hodroj , et al.
Nucleic Acids Research, 2020, 48 (4), pp.1886-1904. ⟨10.1093/nar/gkz1162⟩
Article dans une revue hal-02556387v1
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Beta-hydroxyphosphonate ribonucleoside analogues derived from 4-substituted-1,2,3-triazoles as IMP/GMP mimics: synthesis and biological evaluation

Tai Nguyen Van , Audrey Hospital , Corinne Lionne , Lars P. Jordheim , Charles Dumontet , et al.
Beilstein Journal of Organic Chemistry, 2016, 12, pp.1476--1486. ⟨10.3762/bjoc.12.144⟩
Article dans une revue hal-01812668v1

Regions 1.2 and 3.2 of the RNA Polymerase σ Subunit Promote DNA Melting and Attenuate Action of the Antibiotic Lipiarmycin

Zakia Morichaud , Laurent Chaloin , Konstantin Brodolin
Journal of Molecular Biology, 2016, 428 (2), pp.463 - 476. ⟨10.1016/j.jmb.2015.12.017⟩
Article dans une revue hal-01868357v1

Determination and quantification of intracellular fludarabine triphosphate, cladribine triphosphate and clofarabine triphosphate by LC–MS/MS in human cancer cells

Céline Rabeson , Pierre Yves Géant , Laurent Chaloin , Jean-Yves Puy , Lars Petter Jordheim , et al.
Journal of Chromatography B Biomedical Sciences and Applications, 2017, 1053, pp.101-110. ⟨10.1016/j.jchromb.2017.03.024⟩
Article dans une revue hal-02364216v1