Kevin Cariou

Documents

Publications

	N-Metallocenyl Ynamides: Preparation, Reactivity and Synthesis of ansa[3]-Ferrocenylamides Capucine Mahe , Olivier Blacque , Gilles Gasser , Vincent Gandon , Kevin Cariou Organic Letters, 2023, ⟨10.1021/acs.orglett.2c04169⟩ Article dans une revue hal-03966748v1
	Phototherapeutic anticancer strategies with first-row transition metal complexes: a critical review Lisa Gourdon , Kevin Cariou , Gilles Gasser Chemical Society Reviews, 2022, ⟨10.1039/D1CS00609F⟩ Article dans une revue hal-03542713v1
	Base‐Mediated Generation of Ketenimines from Ynamides: Addition of Hydrazones to Give Acetimidohydrazides** Capucine Mahe , Agathe C A d'Hollander , Kevin Cariou European Journal of Organic Chemistry, 2022, 2022 (18), pp.e202200028. ⟨10.1002/ejoc.202200028⟩ Article dans une revue hal-03721985v1
	Base-Mediated Generation of Ketenimines from Ynamides: [3+2] Annulation with Azaallyl Anions Agathe C A d'Hollander , Eugénie Romero , Kamsana Vijayakumar , Camille Le Houérou , Pascal Retailleau Advanced Synthesis and Catalysis, 2021, 363 (11), pp.2903-2908. ⟨10.1002/adsc.202100047⟩ Article dans une revue hal-03227971v1
	Azetidinimines as a novel series of non-covalent broad-spectrum inhibitors of β-lactamases with submicromolar activities against carbapenemases KPC-2 (class A), NDM-1 (class B) and OXA-48 (class D) Eugénie Romero , Saoussen Oueslati , Mohamed Benchekroun , Agathe C.A. D’hollander , Sandrine Ventre European Journal of Medicinal Chemistry, 2021, 219, pp.113418. ⟨10.1016/j.ejmech.2021.113418⟩ Article dans une revue hal-04433352v1
	Photoinduced Aerobic Iodoarene-Catalyzed Spirocyclization of N-Oxy-Amides to N-Fused Spirolactams Loïc Habert , Kevin Cariou Angewandte Chemie International Edition, 2021, 60 (1), pp.171-175. ⟨10.1002/anie.202009175⟩ Article dans une revue hal-03367856v1
	Ynamides in Free Radical Reactions Capucine Mahe , Kevin Cariou Advanced Synthesis and Catalysis, inPress, ⟨10.1002/adsc.202000849⟩ Article dans une revue hal-02962628v1
	Synthetic approaches towards avibactam and other diazabicyclooctane β-lactamase inhibitors Laure Peilleron , Kevin Cariou Organic & Biomolecular Chemistry, 2020, ⟨10.1039/C9OB02605C⟩ Article dans une revue hal-02466833v1
	Synthesis, Characterization and Antiparasitic Activity of Organometallic Derivatives of the Anthelmintic Drug Albendazole Yan Lin , Yih Ching Ong , Sarah Keller , Rafika Bouchene , Eric Manoury Dalton Transactions, 2020, 49 (20), pp.6616-6626. ⟨10.1039/d0dt01107j⟩ Article dans une revue hal-02555378v1
	A tutorial for the assessment of the stability of organometallic complexes in biological media Sarah Keller , Yih Ching Ong , Yan Lin , Kevin Cariou , Gilles Gasser Journal of Organometallic Chemistry, 2019, pp.121059. ⟨10.1016/j.jorganchem.2019.121059⟩ Article dans une revue hal-02393969v1
	Halonium-Induced Polyene Cyclizations Agathe D’hollander , Laure Peilleron , Tatyana Grayfer , Kevin Cariou Synthesis: Journal of Synthetic Organic Chemistry, 2019, 51 (08), pp.1753-1769. ⟨10.1055/s-0037-1612254⟩ Article dans une revue hal-02307164v1
	Synthesis of cyclic N-hydroxylated ureas and oxazolidinone oximes enabled by chemoselective iodine(III)-mediated radical or cationic cyclizations of unsaturated N-alkoxyureas Laure Peilleron , Pascal Retailleau , Kevin Cariou Advanced Synthesis and Catalysis, 2019, 361 (22), pp.5160-5169. ⟨10.1002/adsc.201901135⟩ Article dans une revue hal-02403999v1
	Iodine(III)-mediated halogenations of acyclic monoterpenoids Laure Peilleron , Tatyana Grayfer , Joëlle Dubois , Robert H Dodd , Kevin Cariou Beilstein Journal of Organic Chemistry, 2018, 14, pp.1103-1111. ⟨10.3762/bjoc.14.96⟩ Article dans une revue hal-02307167v1
	Ketenimines Generated from Ynamides: Versatile Building Blocks for Nitrogen-Containing Scaffolds Robert H Dodd , Kevin Cariou Chemistry - A European Journal, 2018, 24 (10), pp.2297-2304. ⟨10.1002/chem.201704689⟩ Article dans une revue hal-02307203v1
	DYRK1A inhibition and cognitive rescue in a Down syndrome mouse model are induced by new fluoro-DANDY derivatives Fernanda Neumann , Stéphanie Gourdain , Christelle Albac , Alain D Dekker , Linh Chi Bui Scientific Reports, 2018, 8, pp.2859. ⟨10.1038/s41598-018-20984-z⟩ Article dans une revue hal-02292094v1
	Synthesis of Orthogonally N-Protected, C-4 Functionalized Cyclic Guanidines from L-Serine Diego Silva , Edmilson Maria , Rosa Suárez Ordóñez , Josiane Thierry , Kevin Cariou SYNLETT, 2017, 28 (07), pp.815-818. ⟨10.1055/s-0036-1589935⟩ Article dans une revue hal-02307213v1
	Chemodivergent, Tunable, and Selective Iodine(III)-Mediated Bromo-Functionalizations of Polyprenoids Tatyana Grayfer , Pascal ́ Retailleau , Robert H Dodd , Joëlle Dubois , Kevin Cariou Organic Letters, 2017, 19 (18), pp.4766-4769. ⟨10.1021/acs.orglett.7b02125⟩ Article dans une revue hal-02307207v1
	Base-Mediated Generation of Ketenimines from Ynamides: Direct Access to Azetidinimines by an Imino Staudinger Synthesis Eugénie Romero , Corinne Minard , Mohamed Benchekroun , Sandrine Ventre , Pascal ́ Retailleau Chemistry - A European Journal, 2017, 23 (53), pp.12991-12994. ⟨10.1002/chem.201702545⟩ Article dans une revue hal-02307210v1
	Assessing Ligand and Counterion Effects in the Noble Metal Catalyzed Cycloisomerization Reactions of 1,6-Allenynes: a Combined Experimental and Theoretical Approach Florian Jaroschik , Antoine Simonneau , Gilles Lemiere , Kevin Cariou , Nicolas Agenet ACS Catalysis, 2016, 6 (8), pp.5146-5160. ⟨10.1021/acscatal.5b02696⟩ Article dans une revue hal-01397955v1
	Mallotojaponins B and C: Total Synthesis, Antiparasitic Evaluation and Preliminary SAR Studies Tatyana Grayfer , Philippe Grellier , Elisabeth Mouray , Robert H Dodd , Joëlle Dubois Organic Letters, 2016, 18 (4), pp.708-711. ⟨10.1021/acs.orglett.5b03676⟩ Article dans une revue hal-02420932v1
	PIFA-mediated ethoxyiodination of enamides with potassium iodide R. Beltran , S. Nocquet-Thibault , Fabian Blanchard , R. Dodd , K. Cariou Organic & Biomolecular Chemistry, 2016, 14 (36), pp.8448-8451. ⟨10.1039/C6OB01673A⟩ Article dans une revue hal-02307217v1
	Iodine(III)-mediated diazidation and azido-oxyamination of enamides S. Nocquet-Thibault , Anita Marie Rayar , Pascal ́ Retailleau , Kevin Cariou , Robert Dodd Chemistry - A European Journal, 2015, 21 (40), pp.14205-14210. ⟨10.1002/chem.201501782⟩ Article dans une revue hal-03026966v1
	Halocyclization of Unsaturated Guanidines Mediated by Koser's Reagent and Lithium Halides. Marion Daniel , Florent Blanchard , Sophie Nocquet-Thibault , Kevin Cariou , Robert H Dodd Journal of Organic Chemistry, 2015, 80 (21), pp.10624-33. ⟨10.1021/acs.joc.5b01750⟩ Article dans une revue hal-03023458v1
	Iodine(III)-mediated ethoxychlorination of enamides with iron(III) chloride Sophie Nocquet-Thibault , Corinne Minard , Pascal Retailleau , Kevin Cariou , Robert H. Dodd Tetrahedron, 2014, 70 (38), pp.6769-6775. ⟨10.1016/j.tet.2014.07.066⟩ Article dans une revue hal-01067773v1
	Selective Suzuki-Miyaura monocouplings with symmetrical dibromoarenes and aryl ditriflates for the one-pot synthesis of unsymmetrical triaryls C. Minard , C. Palacio , K. Cariou , Robert H Dodd European Journal of Organic Chemistry, 2014, 2014 (14), pp.2942-2955. ⟨10.1002/ejoc.201400090⟩ Article dans une revue hal-00994366v1
	Transition-metal-free tunable chemoselective N functionalization of indoles with ynamides. Alexandre Hentz , Pascal Retailleau , Vincent Gandon , Kevin Cariou , Robert H Dodd Angewandte Chemie International Edition, 2014, 53 (32), pp.8333-8337. ⟨10.1002/anie.201402767⟩ Article dans une revue hal-01065687v1
	Development of DANDYs, New 3,5-Diaryl-7-azaindoles Demonstrating Potent DYRK1A Kinase Inhibitory Activity. Stéphanie Gourdain , Julien Dairou , Clément Denhez , Linh Chi Bui , Fernando Rodrigues-Lima Journal of Medicinal Chemistry, 2013, 56 (23), pp.9569-9585. ⟨10.1021/jm401049v⟩ Article dans une revue hal-00933939v1
	Iodine(III)-Mediated Umpolung of Bromide Salts for the Ethoxybromination of Enamides. Sophie Nocquet-Thibault , Pascal Retailleau , Kevin Cariou , Robert H Dodd Organic Letters, 2013, 15 (8), pp.1842-5. ⟨10.1021/ol400453b⟩ Article dans une revue hal-00827755v1
	Copper(I) catalyzed regioselective asymmetric alkoxyamination of aryl enamide derivatives. Masafumi Nakanishi , Corinne Minard , Pascal Retailleau , Kevin Cariou , Robert H Dodd Organic Letters, 2011, 13 (21), pp.5792-5. ⟨10.1021/ol202367d⟩ Article dans une revue hal-00647697v1
	New unsaturated amino acids containing an allylsilane moiety on the lateral chain Gianna Reginato , Alessandro Mordini , Patrick Meffre , Alice Tenti , Michela Valacchi Tetrahedron: Asymmetry, 2006, 17 (6), pp.922-926. ⟨10.1016/j.tetasy.2006.02.017⟩ Article dans une revue hal-02002619v1

	Base-Mediated Generation of Ketenimines from Ynamides: [3+2] Annulation with Azaallyl Anions Agathe D’hollander , Eugénie Romero , Kamsana Vijayakumar , Camille Le Houérou , Pascal Retailleau 2020 Pré-publication, Document de travail hal-02998846v1
	Azetidinimines as a novel series of non-covalent broad-spectrum inhibitors of β-lactamases with submicromolar activities against carbapenemases of classes A, B and D Eugénie Romero , Saoussen Oueslati , Mohamed Benchekroun , Agathe D’hollander , Sandrine Ventre 2020 Pré-publication, Document de travail hal-02998861v1

Kevin Cariou

Publications

N-Metallocenyl Ynamides: Preparation, Reactivity and Synthesis of ansa[3]-Ferrocenylamides

Phototherapeutic anticancer strategies with first-row transition metal complexes: a critical review

Base‐Mediated Generation of Ketenimines from Ynamides: Addition of Hydrazones to Give Acetimidohydrazides**

Base-Mediated Generation of Ketenimines from Ynamides: [3+2] Annulation with Azaallyl Anions

Azetidinimines as a novel series of non-covalent broad-spectrum inhibitors of β-lactamases with submicromolar activities against carbapenemases KPC-2 (class A), NDM-1 (class B) and OXA-48 (class D)

Photoinduced Aerobic Iodoarene-Catalyzed Spirocyclization of N-Oxy-Amides to N-Fused Spirolactams

Ynamides in Free Radical Reactions

Synthetic approaches towards avibactam and other diazabicyclooctane β-lactamase inhibitors

Synthesis, Characterization and Antiparasitic Activity of Organometallic Derivatives of the Anthelmintic Drug Albendazole

A tutorial for the assessment of the stability of organometallic complexes in biological media

Halonium-Induced Polyene Cyclizations

Synthesis of cyclic N-hydroxylated ureas and oxazolidinone oximes enabled by chemoselective iodine(III)-mediated radical or cationic cyclizations of unsaturated N-alkoxyureas

Iodine(III)-mediated halogenations of acyclic monoterpenoids

Ketenimines Generated from Ynamides: Versatile Building Blocks for Nitrogen-Containing Scaffolds

DYRK1A inhibition and cognitive rescue in a Down syndrome mouse model are induced by new fluoro-DANDY derivatives

Synthesis of Orthogonally N-Protected, C-4 Functionalized Cyclic Guanidines from L-Serine

Chemodivergent, Tunable, and Selective Iodine(III)-Mediated Bromo-Functionalizations of Polyprenoids

Base-Mediated Generation of Ketenimines from Ynamides: Direct Access to Azetidinimines by an Imino Staudinger Synthesis

Assessing Ligand and Counterion Effects in the Noble Metal Catalyzed Cycloisomerization Reactions of 1,6-Allenynes: a Combined Experimental and Theoretical Approach

Mallotojaponins B and C: Total Synthesis, Antiparasitic Evaluation and Preliminary SAR Studies

PIFA-mediated ethoxyiodination of enamides with potassium iodide

Iodine(III)-mediated diazidation and azido-oxyamination of enamides

Halocyclization of Unsaturated Guanidines Mediated by Koser's Reagent and Lithium Halides.

Iodine(III)-mediated ethoxychlorination of enamides with iron(III) chloride

Selective Suzuki-Miyaura monocouplings with symmetrical dibromoarenes and aryl ditriflates for the one-pot synthesis of unsymmetrical triaryls

Transition-metal-free tunable chemoselective N functionalization of indoles with ynamides.

Development of DANDYs, New 3,5-Diaryl-7-azaindoles Demonstrating Potent DYRK1A Kinase Inhibitory Activity.

Iodine(III)-Mediated Umpolung of Bromide Salts for the Ethoxybromination of Enamides.

Copper(I) catalyzed regioselective asymmetric alkoxyamination of aryl enamide derivatives.

New unsaturated amino acids containing an allylsilane moiety on the lateral chain

Base-Mediated Generation of Ketenimines from Ynamides: [3+2] Annulation with Azaallyl Anions

Azetidinimines as a novel series of non-covalent broad-spectrum inhibitors of β-lactamases with submicromolar activities against carbapenemases of classes A, B and D