CV Kevin Cariou

Laure Peilleron, Kevin Cariou. Synthetic approaches towards avibactam and other diazabicyclooctane β-lactamase inhibitors. Organic and Biomolecular Chemistry, Royal Society of Chemistry, 2020, ⟨10.1039/C9OB02605C⟩. ⟨hal-02466833⟩

Capucine Mahe, Kevin Cariou. Ynamides in Free Radical Reactions. Advanced Synthesis and Catalysis, Wiley-VCH Verlag, In press, ⟨10.1002/adsc.202000849⟩. ⟨hal-02962628⟩

Yan Lin, Yih Ong, Sarah Keller, Rafika Bouchene, Eric Manoury, et al.. Synthesis, Characterization and Antiparasitic Activity of Organometallic Derivatives of the Anthelmintic Drug Albendazole. Dalton Transactions, Royal Society of Chemistry, 2020, 49 (20), pp.6616-6626. ⟨10.1039/d0dt01107j⟩. ⟨hal-02555378⟩

Sarah Keller, Yih Ching Ong, Yan Lin, Kevin Cariou, Gilles Gasser. A tutorial for the assessment of the stability of organometallic complexes in biological media. Journal of Organometallic Chemistry, Elsevier, 2019, pp.121059. ⟨10.1016/j.jorganchem.2019.121059⟩. ⟨hal-02393969⟩

Laure Peilleron, Pascal Retailleau, Kevin Cariou. Synthesis of cyclic N-hydroxylated ureas and oxazolidinone oximes enabled by chemoselective iodine(III)-mediated radical or cationic cyclizations of unsaturated N-alkoxyureas. Advanced Synthesis and Catalysis, Wiley-VCH Verlag, 2019, 361 (22), pp.5160-5169. ⟨10.1002/adsc.201901135⟩. ⟨hal-02403999⟩

Agathe D’hollander, Laure Peilleron, Tatyana Grayfer, Kevin Cariou. Halonium-Induced Polyene Cyclizations. SYNTHESIS, Georg Thieme Verlag, 2019, 51 (08), pp.1753-1769. ⟨10.1055/s-0037-1612254⟩. ⟨hal-02307164⟩

Fernanda Neumann, Stéphanie Gourdain, Christelle Albac, Alain Dekker, Linh Chi Bui, et al.. DYRK1A inhibition and cognitive rescue in a Down syndrome mouse model are induced by new fluoro-DANDY derivatives. Scientific Reports, Nature Publishing Group, 2018, 8, pp.2859. ⟨10.1038/s41598-018-20984-z⟩. ⟨hal-02292094⟩

Robert Dodd, Kevin Cariou. Ketenimines Generated from Ynamides: Versatile Building Blocks for Nitrogen-Containing Scaffolds. Chemistry - A European Journal, Wiley-VCH Verlag, 2018, 24 (10), pp.2297-2304. ⟨10.1002/chem.201704689⟩. ⟨hal-02307203⟩

Laure Peilleron, Tatyana Grayfer, Joëlle Dubois, Robert Dodd, Kevin Cariou, et al.. Iodine(III)-mediated halogenations of acyclic monoterpenoids. Beilstein Journal of Organic Chemistry, Beilstein-Institut, 2018, 14, pp.1103-1111. ⟨10.3762/bjoc.14.96⟩. ⟨hal-02307167⟩

Tatyana Grayfer, Pascal Retailleau, Robert Dodd, Joëlle Dubois, Kevin Cariou. Chemodivergent, Tunable, and Selective Iodine(III)-Mediated Bromo-Functionalizations of Polyprenoids. Organic Letters, American Chemical Society, 2017, 19 (18), pp.4766-4769. ⟨10.1021/acs.orglett.7b02125⟩. ⟨hal-02307207⟩

Diego Silva, Edmilson Maria, Rosa Suárez Ordóñez, Josiane Thierry, Kevin Cariou, et al.. Synthesis of Orthogonally N-Protected, C-4 Functionalized Cyclic Guanidines from L-Serine. SYNLETT, Georg Thieme Verlag, 2017, 28 (07), pp.815-818. ⟨10.1055/s-0036-1589935⟩. ⟨hal-02307213⟩

Eugénie Romero, Corinne Minard, Mohamed Benchekroun, Sandrine Ventre, Pascal Retailleau, et al.. Base-Mediated Generation of Ketenimines from Ynamides: Direct Access to Azetidinimines by an Imino Staudinger Synthesis. Chemistry - A European Journal, Wiley-VCH Verlag, 2017, 23 (53), pp.12991-12994. ⟨10.1002/chem.201702545⟩. ⟨hal-02307210⟩

Tatyana D. Grayfer, Philippe Grellier, Elisabeth Mouray, Robert H Dodd, Joëlle Dubois, et al.. Mallotojaponins B and C: Total Synthesis, Antiparasitic Evaluation, and Preliminary SAR Studies. Organic Letters, American Chemical Society, 2016, 18 (4), pp.708-711. ⟨mnhn-02047323⟩

R. Beltran, S. Nocquet-Thibault, F. Blanchard, R. Dodd, K. Cariou. PIFA-mediated ethoxyiodination of enamides with potassium iodide. Organic and Biomolecular Chemistry, Royal Society of Chemistry, 2016, 14 (36), pp.8448-8451. ⟨10.1039/C6OB01673A⟩. ⟨hal-02307217⟩

Florian Jaroschik, Antoine Simonneau, Gilles Lemiere, Kevin Cariou, Nicolas Agenet, et al.. Assessing Ligand and Counterion Effects in the Noble Metal Catalyzed Cycloisomerization Reactions of 1,6-Allenynes: a Combined Experimental and Theoretical Approach. ACS Catalysis, American Chemical Society, 2016, 6 (8), pp.5146-5160. ⟨10.1021/acscatal.5b02696⟩. ⟨hal-01397955⟩

Tatyana Grayfer, Philippe Grellier, Elisabeth Mouray, Robert Dodd, Joëlle Dubois, et al.. Mallotojaponins B and C: Total Synthesis, Antiparasitic Evaluation and Preliminary SAR Studies. Organic Letters, American Chemical Society, 2016, 18 (4), pp.708-711. ⟨10.1021/acs.orglett.5b03676⟩. ⟨hal-02420932⟩

Marion Daniel, Florent Blanchard, Sophie Nocquet-Thibault, Kevin Cariou, Robert Dodd. Halocyclization of Unsaturated Guanidines Mediated by Koser's Reagent and Lithium Halides.. Journal of Organic Chemistry, American Chemical Society, 2015, 80 (21), pp.10624-33. ⟨10.1021/acs.joc.5b01750⟩. ⟨hal-03023458⟩

S. Nocquet-Thibault, Anita Marie Rayar, Pascal Retailleau, Kevin Cariou, Robert Dodd. Iodine(III)-mediated diazidation and azido-oxyamination of enamides. Chemistry - A European Journal, Wiley-VCH Verlag, 2015, 21 (40), pp.14205-14210. ⟨10.1002/chem.201501782⟩. ⟨hal-03026966⟩

Sophie Nocquet-Thibault, Corinne Minard, Pascal Retailleau, Kevin Cariou, Robert H. Dodd. Iodine(III)-mediated ethoxychlorination of enamides with iron(III) chloride. Tetrahedron, Elsevier, 2014, 70 (38), pp.6769-6775. ⟨10.1016/j.tet.2014.07.066⟩. ⟨hal-01067773⟩

C. Minard, C. Palacio, K. Cariou, Robert H Dodd. Selective Suzuki-Miyaura monocouplings with symmetrical dibromoarenes and aryl ditriflates for the one-pot synthesis of unsymmetrical triaryls. European Journal of Organic Chemistry, Wiley-VCH Verlag, 2014, 2014 (14), pp.2942-2955. ⟨10.1002/ejoc.201400090⟩. ⟨hal-00994366⟩

Alexandre Hentz, Pascal Retailleau, Vincent Gandon, Kevin Cariou, Robert H Dodd. Transition-metal-free tunable chemoselective N functionalization of indoles with ynamides.. Angewandte Chemie International Edition, Wiley-VCH Verlag, 2014, 53 (32), pp.8333-8337. ⟨10.1002/anie.201402767⟩. ⟨hal-01065687⟩

Sophie Nocquet-Thibault, Pascal Retailleau, Kevin Cariou, Robert H Dodd. Iodine(III)-Mediated Umpolung of Bromide Salts for the Ethoxybromination of Enamides.. Organic Letters, American Chemical Society, 2013, 15 (8), pp.1842-5. ⟨10.1021/ol400453b⟩. ⟨hal-00827755⟩

Stéphanie Gourdain, Julien Dairou, Clément Denhez, Linh Chi Bui, Fernando Rodrigues-Lima, et al.. Development of DANDYs, New 3,5-Diaryl-7-azaindoles Demonstrating Potent DYRK1A Kinase Inhibitory Activity.. Journal of Medicinal Chemistry, American Chemical Society, 2013, 56 (23), pp.9569-9585. ⟨10.1021/jm401049v⟩. ⟨hal-00933939⟩

Masafumi Nakanishi, Corinne Minard, Pascal Retailleau, Kevin Cariou, Robert H Dodd. Copper(I) catalyzed regioselective asymmetric alkoxyamination of aryl enamide derivatives.. Organic Letters, American Chemical Society, 2011, 13 (21), pp.5792-5. ⟨10.1021/ol202367d⟩. ⟨hal-00647697⟩

Gianna Reginato, Alessandro Mordini, Patrick Meffre, Alice Tenti, Michela Valacchi, et al.. New unsaturated amino acids containing an allylsilane moiety on the lateral chain. Tetrahedron: Asymmetry, Elsevier, 2006, 17 (6), pp.922-926. ⟨10.1016/j.tetasy.2006.02.017⟩. ⟨hal-02002619⟩

Agathe D’hollander, Eugénie Romero, Kamsana Vijayakumar, Camille Le Houérou, Pascal Retailleau, et al.. Base-Mediated Generation of Ketenimines from Ynamides: [3+2] Annulation with Azaallyl Anions. 2020. ⟨hal-02998846⟩

Eugénie Romero, Saoussen Oueslati, Mohamed Benchekroun, Agathe D’hollander, Sandrine Ventre, et al.. Azetidinimines as a novel series of non-covalent broad-spectrum inhibitors of β-lactamases with submicromolar activities against carbapenemases of classes A, B and D. 2020. ⟨hal-02998861⟩