Recherche - Archive ouverte HAL

24 résultats

	Pour les 24 documents Envoyer sur ORCID RSS ATOM Exporter BibTeX XML-TEI CSV RTF EndNote PDF HTML Export avancé	Page :	triés par Pertinence Auteur A→Z Auteur Z→A Titre A→Z Titre Z→A Date de publication croissante Date de publication décroissante Date de dépôt croissante Date de dépôt décroissante

		Zika Virus Methyltransferase: Structure and Functions for Drug Design Perspectives Bruno Coutard , Karine Barral , Julie Lichiere , Barbara Selisko , Baptiste Martin , et al. Journal of Virology, 2017, 91 (5), pp.2202-2218. ⟨10.1128/JVI.02202-16⟩ Article dans une revue hal-01802793v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Assessment of Dengue virus helicase and methyltransferase as targets for fragment-based drug discovery Bruno Coutard , Etienne Decroly , Changqing Li , Andrew Sharff , Julien Lescar , et al. Antiviral Research, 2014, 106, pp.61-70. ⟨10.1016/j.antiviral.2014.03.013⟩ Article dans une revue hal-02061701v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and Antiviral Evaluation of Cis-Substituted Cyclohexenyl and Cyclohexanyl Nucleosides Karine Barral , Jérôme Courcambeck , Gérard Pèpe , Jan Balzarini , Johan Neyts , et al. Journal of Medicinal Chemistry, 2005, 48 (2), pp.450-456. ⟨10.1021/jm0493966⟩ Article dans une revue istex hal-02061654v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		In vitro screening of a FDA approved chemical library reveals potential inhibitors of SARS-CoV-2 replication Franck Touret , Magali Gilles , Karine Barral , Antoine Nougairède , Jacques van Helden , et al. Scientific Reports, 2020, 10 (1), pp.13093. ⟨10.1038/s41598-020-70143-6⟩ Article dans une revue inserm-02944556v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and antiviral evaluation of 3-hydroxy-2-methylpyridin-4-one dideoxynucleoside derivatives Karine Barral , Robert Hider , Jan Balzarini , Johan Neyts , Erik de Clercq , et al. Bioorganic and Medicinal Chemistry Letters, 2003, 13 (24), pp.4371-4374. ⟨10.1016/j.bmcl.2003.09.033⟩ Article dans une revue istex hal-02061650v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Pharmacological inhibition of syntenin PDZ2 domain impairs breast cancer cell activities and exosome loading with syndecan and EpCAM cargo R. Leblanc , R. Kashyap , K. Barral , A.L. Egea‐jimenez , D. Kovalskyy , et al. Journal of Extracellular Vesicles, 2020, 10 (2), ⟨10.1002/jev2.12039⟩ Article dans une revue hal-03152593v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Preparation of thiophenepropenamide derivatives as flavivirus inhibitors in treatment of viral infections Karine Barral , Jean Claude Guillemot , Bruno Canard , Gilles Quérat , Karine Alvarez , et al. France, Patent n° : WO 2017102014. 2017 Brevet hal-02063286v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Discovery of novel dengue virus NS5 methyltransferase non-nucleoside inhibitors by fragment-based drug design Fatiha Benmansour , Iuni Trist , Bruno Coutard , Etienne Decroly , Gilles Querat , et al. European Journal of Medicinal Chemistry, 2017, 125, pp.865-880. ⟨10.1016/j.ejmech.2016.10.007⟩ Article dans une revue hal-02061703v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Acyclic phosphonate nucleotides and human adenylate kinases: impact of a borano group on alpha-P position. D. Topalis , K. Alvarez , K. Barral , Hélène Munier-Lehmann , B. Schneider , et al. Nucleosides, Nucleotides and Nucleic Acids, 2008, 27 (4), pp.319-31. ⟨10.1080/15257770801941952⟩ Article dans une revue pasteur-00316017v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Preparation of purine and pyrimidine acyclic nucleotide analogs as antiviral agents Karine Barral , Bruno Canard , Karine Alvarez , Jean-Louis Romette , Johan Neyts , et al. France, Patent n° : WO 2007-IB4233. 2007 Brevet hal-02063281v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Optimization of a fragment linking hit toward Dengue and Zika virus NS5 methyltransferases inhibitors Jessica Hernandez , Laurent Hoffer , Bruno Coutard , Gilles Quérat , Philippe Roche , et al. European Journal of Medicinal Chemistry, 2019, 161 (4), pp.323-333. ⟨10.1016/j.ejmech.2018.09.056⟩ Article dans une revue inserm-02378768v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis of (±) cis-substituted cyclohexenyl and cyclohexanyl nucleosides via a double Mitsunobu-type reaction Karine Barral , Philippe Halfon , Gérard Pèpe , Michel Camplo Tetrahedron Letters, 2002, 43 (1), pp.81-84. ⟨10.1016/S0040-4039(01)02107-4⟩ Article dans une revue istex hal-02061647v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		In Vitro Suppression of K65R Reverse Transcriptase-Mediated Tenofovir- and Adefovir-5'-Diphosphate Resistance Conferred by the Boranophosphonate Derivatives A. Frangeul , Karine Barral , K. Alvarez , B. Canard Antimicrobial Agents and Chemotherapy, 2007, 51 (9), pp.3162-3167. ⟨10.1128/AAC.00145-07⟩ Article dans une revue hal-02061675v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Gln151 of HIV-1 reverse transcriptase acts as a steric gate towards clinically relevant acyclic phosphonate nucleotide analogues. Antoine Frangeul , Cécile Bussetta , Jérôme Deval , Karine Barral , Karine Alvarez , et al. Antiviral Therapy, 2019, 13 (1), pp.115-24 Article dans une revue hal-02061712v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Efficient Conversion of Aromatic Amines into Azides: A One-Pot Synthesis of Triazole Linkages Karine Barral , Adam Moorhouse , John Moses Organic Letters, 2007, 9 (9), pp.1809-1811. ⟨10.1021/ol070527h⟩ Article dans une revue hal-02061672v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Protéine 2C d’Entérovirus : protéine clé de la réplication virale et cible antivirale Priscila El Kazzi , Carole Yaacoub , Ziad Fajloun , Patrice Vanelle , Etienne Decroly , et al. Virologie, 2023, 27 (3), pp.173-188. ⟨10.1684/vir.2023.1001⟩ Article dans une revue hal-04504110v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and Antiviral Evaluation of Cyclic and Acyclic 2-Methyl-3-hydroxy-4-pyridinone Nucleoside Derivatives Karine Barral , Jan Balzarini , Johan Neyts , Erik de Clercq , Robert Hider , et al. Journal of Medicinal Chemistry, 2006, 49 (1), pp.43-50. ⟨10.1021/jm0504306⟩ Article dans une revue istex hal-02061660v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Novel 2-phenyl-5-[(E)-2-(thiophen-2-yl)ethenyl]-1,3,4-oxadiazole and 3-phenyl-5-[(E)-2-(thiophen-2-yl)ethenyl]-1,2,4-oxadiazole derivatives as dengue virus inhibitors targeting NS5 polymerase Fatiha Benmansour , Cecilia Eydoux , Gilles Querat , Xavier de Lamballerie , Bruno Canard , et al. European Journal of Medicinal Chemistry, 2016, 109, pp.146-156. ⟨10.1016/j.ejmech.2015.12.046⟩ Article dans une revue hal-02061730v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis, in Vitro Antiviral Evaluation, and Stability Studies of Novel α-Borano-Nucleotide Analogues of 9-[2-(Phosphonomethoxy)ethyl]adenine and ( R )-9-[2-(Phosphonomethoxy)propyl]adenine Karine Barral , Stephane Priet , Joséphine Sire , Johan Neyts , Jan Balzarini , et al. Journal of Medicinal Chemistry, 2006, 49 (26), pp.7799-7806. ⟨10.1021/jm060030y⟩ Article dans une revue istex hal-02061667v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Discovery of a PDZ Domain Inhibitor Targeting the Syndecan/Syntenin Protein–Protein Interaction: A Semi-Automated “Hit Identification-to-Optimization” Approach Laurent Hoffer , Manon Garcia , Raphael Leblanc , Mikael Feracci , Stéphane Betzi , et al. Journal of Medicinal Chemistry, 2023, ⟨10.1021/acs.jmedchem.2c01569⟩ Article dans une revue hal-04048842v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Borano-nucleotides: new analogues to circumvent HIV-1 RT-mediated nucleoside drug-resistance Karine Alvarez , Jérôme Deval , Boulbaba Selmi , Karine Barral , Joelle Boretto , et al. Nucleosides, Nucleotides and Nucleic Acids, 2005, 24 (5-7), pp.419-422. ⟨10.1081/NCN-200059951⟩ Article dans une revue hal-02061659v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Synthesis and antiviral activity of boranophosphonate isosteres of AZT and d4T monophosphates Karine Barral , Stephane Priet , Céline de Michelis , Joséphine Sire , Johan Neyts , et al. European Journal of Medicinal Chemistry, 2010, 45 (2), pp.849-856. ⟨10.1016/j.ejmech.2009.11.012⟩ Article dans une revue istex hal-02061692v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Acyclic nucleoside thiophosphonates as potent inhibitors of HIV and HBV replication Karine Barral , Clément Weck , Nadine Payrot , Loic Roux , Céline Durafour , et al. European Journal of Medicinal Chemistry, 2011, 46 (9), pp.4281-4288. ⟨10.1016/j.ejmech.2011.06.034⟩ Article dans une revue hal-02061721v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More
		Development of specific dengue virus 2'-O- and N7-methyltransferase assays for antiviral drug screening. Karine Barral , Corinne Sallamand , Christiane Petzold , Bruno Coutard , Axelle Collet , et al. Antiviral Research, 2013, 99 (3), pp.292-300. ⟨10.1016/j.antiviral.2013.06.001⟩ Article dans une revue istex hal-00874640v1	Envoyer sur ORCID Exporter BibTeX XML-TEI Dublin Core DC Terms EndNote DataCite Export avancé Partager Gmail Facebook X LinkedIn More

Filtrer vos résultats

Zika Virus Methyltransferase: Structure and Functions for Drug Design Perspectives

Assessment of Dengue virus helicase and methyltransferase as targets for fragment-based drug discovery

Synthesis and Antiviral Evaluation of Cis-Substituted Cyclohexenyl and Cyclohexanyl Nucleosides

In vitro screening of a FDA approved chemical library reveals potential inhibitors of SARS-CoV-2 replication

Synthesis and antiviral evaluation of 3-hydroxy-2-methylpyridin-4-one dideoxynucleoside derivatives

Pharmacological inhibition of syntenin PDZ2 domain impairs breast cancer cell activities and exosome loading with syndecan and EpCAM cargo

Preparation of thiophenepropenamide derivatives as flavivirus inhibitors in treatment of viral infections

Discovery of novel dengue virus NS5 methyltransferase non-nucleoside inhibitors by fragment-based drug design

Acyclic phosphonate nucleotides and human adenylate kinases: impact of a borano group on alpha-P position.

Preparation of purine and pyrimidine acyclic nucleotide analogs as antiviral agents

Optimization of a fragment linking hit toward Dengue and Zika virus NS5 methyltransferases inhibitors

Synthesis of (±) cis-substituted cyclohexenyl and cyclohexanyl nucleosides via a double Mitsunobu-type reaction

In Vitro Suppression of K65R Reverse Transcriptase-Mediated Tenofovir- and Adefovir-5'-Diphosphate Resistance Conferred by the Boranophosphonate Derivatives

Gln151 of HIV-1 reverse transcriptase acts as a steric gate towards clinically relevant acyclic phosphonate nucleotide analogues.

Efficient Conversion of Aromatic Amines into Azides: A One-Pot Synthesis of Triazole Linkages

Protéine 2C d’Entérovirus : protéine clé de la réplication virale et cible antivirale

Synthesis and Antiviral Evaluation of Cyclic and Acyclic 2-Methyl-3-hydroxy-4-pyridinone Nucleoside Derivatives

Novel 2-phenyl-5-[(E)-2-(thiophen-2-yl)ethenyl]-1,3,4-oxadiazole and 3-phenyl-5-[(E)-2-(thiophen-2-yl)ethenyl]-1,2,4-oxadiazole derivatives as dengue virus inhibitors targeting NS5 polymerase

Synthesis, in Vitro Antiviral Evaluation, and Stability Studies of Novel α-Borano-Nucleotide Analogues of 9-[2-(Phosphonomethoxy)ethyl]adenine and ( R )-9-[2-(Phosphonomethoxy)propyl]adenine

Discovery of a PDZ Domain Inhibitor Targeting the Syndecan/Syntenin Protein–Protein Interaction: A Semi-Automated “Hit Identification-to-Optimization” Approach

Borano-nucleotides: new analogues to circumvent HIV-1 RT-mediated nucleoside drug-resistance

Synthesis and antiviral activity of boranophosphonate isosteres of AZT and d4T monophosphates

Acyclic nucleoside thiophosphonates as potent inhibitors of HIV and HBV replication

Development of specific dengue virus 2'-O- and N7-methyltransferase assays for antiviral drug screening.