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Antibody-Hapten Recognition at the Surface of Functionalized Liposomes Studied by SPR: Steric Hindrance of Pegylated Phospholipids in Stealth Liposomes Prepared for Targeted Radionuclide Delivery

 Eliot Botosoa , Mike Maillasson , Marie Mougin-Degraef , Patricia Remaud-Le Saec , Jean-François Gestin , et al.
Journal of Drug Delivery, 2011, 2011, pp.368535. ⟨10.1155/2011/368535⟩
Article dans une revue inserm-02417966v1
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O-66 - Preparation of 211At-labeled aromatic compounds from thioarylprecursors

 Clémence Maingueneau , Romain Eychenne , Jean-François Gestin , François Guérard
International Symposium of radiopharmaceutical sciences, May 2022, Nantes, France
Communication dans un congrès inserm-03842544v1
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Investigation on the reactivity of nucleophilic radiohalogens with arylboronic acids in water: access to an efficient single-step method for the radioiodination and astatination of antibodies

 Marion Berdal , Sébastien Gouard , Romain Eychenne , Séverine Marionneau-Lambot , Mikaël Croyal , et al.
Chemical Science, 2021, 12 (4), pp.1458-1468. ⟨10.1039/D0SC05191H⟩
Article dans une revue inserm-03024891v1

Synthesis of polyaminocarboxylic acids for applications in nuclear medicine

 Jean-Claude Meslin , Sébastien Gouin , Jean-François Gestin , Jean-Claude Meslin , David Deniaud
SFC Eurochem, 2002, Toulouse, France
Communication dans un congrès hal-00021340v1

Method for synthesizing iodo- or astatoarenes using Diaryliodonium Salts

 François Guérard , Jean-François Gestin , Martin W. Brechbiel , Yong-Sok Lee
France, Patent n° : WO 2017/089492 A1. 2017
Brevet inserm-02545737v1
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Unexpected Behavior of the Heaviest Halogen Astatine in the Nucleophilic Substitution of Aryliodonium Salts

 François Guérard , Yong-Sok Lee , Kwamena Baidoo , Jean-François Gestin , Martin W Brechbiel
Chemistry - A European Journal, 2016, 22 (35), pp.12332-9. ⟨10.1002/chem.201600922⟩
Article dans une revue inserm-01387016v1
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Investigation of the complexation of nat Zr(IV) and 89 Zr(IV) by hydroxypyridinones for the development of chelators for PET imaging applications

 François Guérard , Maryline Beyler , Y.-S Lee , Raphaël Tripier , Jean-François Gestin , et al.
Dalton Transactions, 2017, 46, pp.4749-4758. ⟨10.1039/c6dt04625h⟩
Article dans une revue inserm-01496515v1
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Synthesis of C-functionalized TE1PA and comparison with its analogues. An example of bioconjugation on 9E7.4 mAb for multiple myeloma 64 Cu-PET imaging

 Thomas Le Bihan , Anne-Sophie Navarro , Nathalie Le Bris , Patricia Le Saec , Sébastien Gouard , et al.
Organic & Biomolecular Chemistry, 2018, Epub ahead of print. ⟨10.1039/c8ob00499d⟩
Article dans une revue inserm-01804657v1

Efficient Synthesis of a New Potential Chelating Agent for Radioimmunotherapy.

 Sebastien G. Gouin , Jean-Claude Meslin , Sébastien Gouin , Jean-François Gestin , Gérald Remaud , et al.
SYNLETT, 2002, 12, pp.2080-2082
Article dans une revue hal-00015616v1
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Biodistribution, Imaging and Metabolism Studies of 64-Copper Radiolabelled Monoclonal Antibody : Comparison of DOTA and TE1PA Chelating Agents in a Murine Model of Multiple Myeloma

 A. Navarro , T. Le Bihan , Patricia Remaud-Le Saëc , Sébastien Gouard , N. Le Bris , et al.
European Journal of Nuclear Medicine and Molecular Imaging, 2018, 45 (1), pp.S119-S120
Article dans une revue inserm-02344286v1
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Direct nucleophilic radioiodination and astatination of antibodies via pre-conjugated arylboronic acids

 Marion Berdal , Laurent Navarro , Cyrille Alliot , Michel Chérel , Alain Faivre-Chauvet , et al.
Journal of Labelled Compounds and Radiopharmaceuticals, 2019
Article dans une revue inserm-02340736v1
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Targeted alpha-therapy with 211At-anti-mCD138 mAb in a syngeneic murine Multiple Myeloma model : can repeated doses or fractionation protocol overpass single dose efficiency?

 Sébastien Gouard , Séverine Marionneau-Lambot , Joëlle Gaschet , Sébastien Chouin , F. Haddad , et al.
33rd Annual Congress of the European-Association-of-Nuclear-Medicine (EANM), European-Association-of-Nuclear-Medicine (EANM), Oct 2020, Virtuel, France. pp.S410-S411, ⟨10.1158/1078-0432.CCR-18-⟩
Communication dans un congrès inserm-03500243v1
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Prosthetic groups for radioiodination and astatination of peptides and proteins: a comparative study of five potential bioorthogonal labeling strategies

 Laurent Navarro , Marion Berdal , Michel Chérel , Frédéric Pecorari , Jean-François Gestin , et al.
Bioorganic and Medicinal Chemistry, In press, pp.167-174. ⟨10.1016/j.bmc.2018.11.034⟩
Article dans une revue inserm-01939636v1
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Synthesis of precursors for 211At-labelling of anti-PSMA HuJ591 mAb and stability comparison after in vitro cellular internalization

 Aurélia Roumesy , Sebastien Gouard , Laurent Navarro , Faustine Lelan , Ferid Haddad , et al.
ISRS 2019, May 2019, PEKIN, China. pp.S69-S70
Communication dans un congrès inserm-02340836v1
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Ionic liquid supported organotin reagents to prepare molecular imaging and therapy agents †

 Holisoa Rajerison , Djibril Faye , Aurélia Roumesy , Nicolas Louaisil , Fabien Boeda , et al.
Organic & Biomolecular Chemistry, 2016, 14, pp.2121-2126. ⟨10.1039/c5ob02459e⟩
Article dans une revue inserm-01280171v1
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New synthesis of phenyl-isothiocyanate C-functionalised cyclams. Bioconjugation and 64 Cu phenotypic PET imaging studies of multiple myeloma with the te2a derivative †

 Zakaria Halime , Mathieu Frindel , Nathalie Camus , Pierre-Yves Orain , Marie Lacombe , et al.
Organic & Biomolecular Chemistry, 2015, 13 (46), pp.11302-14. ⟨10.1039/c5ob01618e⟩
Article dans une revue inserm-02418040v1

Synthesis and metal complexation properties of Ph-DTPA and Ph-TTHA: novel radionuclide chelating agents for use in nuclear medicine

 Sebastien Gouin , Jean-François Gestin , Laurent Monrandeau , Fabienne Ségat-Dioury , Jean-Claude Meslin , et al.
Organic & Biomolecular Chemistry, 2005, 3, pp.454-461
Article dans une revue hal-00014703v1

La chimie des agents chélatants bifonctionnels : tout est fait ou reste à faire?

 Sebastien G. Gouin , David Deniaud , Jean-Claude Meslin , Jean-François Gestin
Séminaire du club national des radiopharmaceutiques, Jan 2002, Nantes, France
Communication dans un congrès hal-00022470v1

Method for Radioioidination OR Radioastatination of a Biomolecule

 Marion Berdal , Alain Faivre-Chauvet , Jean-François Gestin , François Guérard
France, Patent n° : 19305563.9 - 1 109. 2019
Brevet inserm-02547459v1
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Bifunctional aryliodonium salts for highly efficient radioiodination and astatination of antibodies

 François Guérard , Laurent Navarro , Y.-S. Lee , Aurélia Roumesy , Cyrille Alliot , et al.
Bioorganic and Medicinal Chemistry, 2017, Epub ahead of print. ⟨10.1016/j.bmc.2017.09.022⟩
Article dans une revue inserm-01592684v1
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Efficacy of Astatine-211 radioimmunotherapy of Multiple Myeloma using an anti-mCD138 monoclonal antibody in a syngeneic murine model

 Sébastien Gouard , Benjamin Chalopin , Catherine Saï-Maurel , François Guérard , Laurent Navarro , et al.
European Journal of Nuclear Medicine and Molecular Imaging, 2018, 45 (1), pp.S166-S167
Article dans une revue inserm-02341491v1

Monopicolinate-dipicolyl Derivative of Triazacyclononane for Stable Complexation of Cu 2+ and 64 Cu 2+

 Melissa Roger , Luis M. P. Lima , Mathieu Frindel , Carlos Platas-Iglesias , Jean-François Gestin , et al.
Inorganic Chemistry, 2013, 52 (9), pp.5246 - 5259. ⟨10.1021/ic400174r⟩
Article dans une revue hal-01555830v1
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Production of [211 At]-Astatinated Radiopharmaceuticals and Applications in Targeted alpha-Particle Therapy

 François Guérard , Jean-François Gestin , Martin W Brechbiel
Cancer Biotherapy and Radiopharmaceuticals, 2013, 28 (1), pp.1-20. ⟨10.1089/cbr.2012.1292⟩
Article dans une revue inserm-02496646v1

Method for Radioiodination or Radioastatination of a biomolecule

 Marion Berdal , François Guérard , Jean-François Gestin , Alain Faivre-Chauvet
France, Patent n° : WO 2020/221744 A1. 2020
Brevet inserm-03013584v1
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An Efficient Route for the Synthesis of New Analogues of Polyaminocarboxylic Acid Incorporating O, N, and S Atoms

 Sebastien Gouin , Eric Benoist , Jean-François Gestin , Jean-Claude Meslin , Sebastien G. Gouin
European Journal of Organic Chemistry, 2004, pp.878-885. ⟨10.1002/ejoc.200300459⟩
Article dans une revue inserm-02418095v1

Radiolabeling and targeting of lipidic nanocapsules for applications in radioimmunotherapy.

 Emmanuelle Jestin , Marie Mougin-Degraef , Alain Faivre-Chauvet , P. Remaud-Le Saec , François Hindré , et al.
The quarterly journal of nuclear medicine and molecular imaging, 2007, 51 (1), pp.51-60
Article dans une revue inserm-00258368v1
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Advances in the Radiolabeling of Antibodies with Astatine-211 : Toward Simplified Procedures and Improved Radiochemical Yields

 François Guérard , Laurent Navarro , Marion Berdal , Ferid Haddad , Michel Chérel , et al.
TAT 11 INTERNATIONAL SYMPOSIUM, Apr 2019, OTTAWA, Canada. pp.S29
Communication dans un congrès inserm-02340810v1

Ionic liquid supported organotin reagents for the manufacturing of radiopharmaceuticals compounds

 Stéphanie Legoupy , Djibril Faye , Jean-François Gestin , Holisoa Rajerison , Alain Faivre-Chauvet , et al.
France, Patent n° : Non spécifié. 2015
Brevet hal-02564078v1
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Cyclam te1pa for 64 Cu PET imaging. Bioconjugation to antibody, radiolabeling and preclinical application in xenografted colorectal cancer

 Mathieu Frindel , Patricia Le Saec , Maryline Beyler , Anne-Sophie Navarro , Catherine Sai-Maurel , et al.
RSC Advances, 2017, 7, pp.9272-9283. ⟨10.1039/c6ra26003a⟩
Article dans une revue inserm-01463724v1

Radiolabeling of HTE1PA: A new monopicolinate cyclam derivative for Cu-64 phenotypic imaging. In vitro and in vivo stability studies in mice

 Mathieu Frindel , Nathalie Camus , Aurore Rauscher , Mickaël Bourgeois , Cyrille Alliot , et al.
Nuclear Medicine and Biology, 2014, 41, pp.e49 - e57. ⟨10.1016/j.nucmedbio.2013.12.009⟩
Article dans une revue hal-01529578v1
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