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New N4-substituted piperazine naphthamide derivatives as BACE1 inhibitors

Y. Laras , C. Garino , J. Dessolin , C. Wecq , A. Rolland , et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2008, 24 (1), pp.181-87
Article dans une revue hal-00428703v1

Direct C-H Arylation of Quinones with Anilines

Marc Lamblin , Guillaume Naturale , Jean Dessolin , Francois-Xavier Felpin
SYNLETT, 2012, 11, pp.1621-1624. ⟨10.1055/s-0031-1291163⟩
Article dans une revue hal-02142691v1
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Molecular Determinants for OMF Selectivity in Tripartite RND Multidrug Efflux Systems

Esther Boyer , Jean Dessolin , Margaux Lustig , Marion Decossas , Gilles Phan , et al.
Antibiotics, 2022, 11 (2), pp.126. ⟨10.3390/antibiotics11020126⟩
Article dans une revue hal-03815594v1

Double-drug development against antioxidant enzymes from Plasmodium falciparum

Christophe Biot , Jean Dessolin , Philippe Grellier , Elisabeth Davioud-Charvet
Redox Report, 2013, 8 (5), pp.280-283. ⟨10.1179/135100003225002916⟩
Article dans une revue mnhn-02867482v1

Novel phenyl(thio)ureas bearing (thio)oxothiazoline group as potential BACE-1 inhibitors: synthesis and biological evaluation

Federico Andreoli , Abdallah Larbi Doukara , Mohammed Amine Mehdid , Nicolas Vanthuyne , Christian Roussel , et al.
Journal of Enzyme Inhibition and Medicinal Chemistry, 2011, 28 (1), pp.153-162. ⟨10.3109/14756366.2011.642375⟩
Article dans une revue hal-02527926v1

Direct C-H Alkylation of Naphthoquinones with Amino Acids Through a Revisited Kochi-Anderson Radical Decarboxylation: Trends in Reactivity and Applications

Guillaume Naturale , Marc Lamblin , Claude Commandeur , Francois-Xavier Felpin , Jean Dessolin
European Journal of Organic Chemistry, 2012, 29, pp.5774-5788. ⟨10.1002/ejoc.201200722⟩
Article dans une revue istex hal-02142684v1

Impact of lipid polyunsaturation on dopamine D2 receptor activation and signaling

Véronique de Smedt-Peyrusse , Marie-Lise Jobin , R. Baccouch , M. Wang , J. Heuninck , et al.
12. EBSA European Biophysics Congress, Jul 2019, Madrid, Spain. European Biophysics Journal, 48 (Supplement: 1), 2019
Poster de conférence hal-02734710v1

Synthesis and biological activity of phosphonate analogues and geometric isomers of the highly potent phosphoantigen (E)-1-hydroxy-2-methylbut-2-enyl 4-diphosphate

A. Boedec , H. Sicard , J. Dessolin , G. Herbette , S. Ingoure , et al.
Journal of Medicinal Chemistry, 2008, 51, pp.1747-1754
Article dans une revue hal-00305902v1

Practical Pd/C-Catalysed Suzuki-Miyaura Reactions for the Preparation of 3-Aryl-4-oxypyridin-2(1H)-ones, 3-Aryl-2,4-oxypyridines and 3-Aryl-2,4-oxyquinolines as Useful Intermediates for the Synthesis of Biologically Active Compounds

Marc Lamblin , Hugo Bares , Jean Dessolin , Christel Marty , Nathalie Bourgougnon , et al.
European Journal of Organic Chemistry, 2012, 28, pp.5525-5533. ⟨10.1002/ejoc.201200721⟩
Article dans une revue istex hal-02142685v1
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Cholesterol impacts chemokine CCR5 receptor ligand binding activity

Pierre Calmet , Christophe Cullin , Sandra Cortès , Maylou Vang , Nada Lepejova Caudy , et al.
FEBS Journal, 2019, ⟨10.1111/febs.15145⟩
Article dans une revue hal-03101449v1
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A Complex Interplay of Anionic Phospholipid Binding Regulates 3′-Phosphoinositide-Dependent-Kinase-1 Homodimer Activation

Gloria De las Heras-Martínez , Véronique Calleja , Rémy Bailly , Jean Dessolin , Banafshé Larijani , et al.
Scientific Reports, 2019, 9 (1), ⟨10.1038/s41598-019-50742-8⟩
Article dans une revue hal-02327975v1

Bis-8-hydroxy quinoline and Bis-8-hydroxy-quinaldine N-susbtituted amines: A single methyl group structural difference between the two heterocycles, which modulates the antiproliferative effects

S. Madonna , A. Marcowycz , D. Lamoral-Theys , G.Van Goietsenoven , J. Dessolin , et al.
Journal of Heterocyclic Chemistry, 2010, 47, pp.719-723. ⟨10.1002/jet.304⟩
Article dans une revue hal-00563200v1

Design, synthesis and biological evaluation of Pontin ATPase inhibitors through a molecular docking approach.

Judith Elkaim , Marc Lamblin , Michel Laguerre , Jean Rosenbaum , Patrick Lestienne , et al.
Bioorganic and Medicinal Chemistry Letters, 2014, 24 (11), pp.2512-2516. ⟨10.1016/j.bmcl.2014.04.003⟩
Article dans une revue hal-01001838v1
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Synergistic effect of tryptamine-urea derivatives to overcome the chromosomally-mediated colistin resistance in Klebsiella pneumoniae

Chaimae Majdi , Jean Dessolin , David Bénimélis , Catherine Dunyach-Rémy , Alix Pantel , et al.
Bioorganic and Medicinal Chemistry, 2024, 100, pp.117604. ⟨10.1016/j.bmc.2024.117604⟩
Article dans une revue hal-04419733v1

JOINT 12th EBSA congress and 10th ICBP – IUPAP congress, July 20-24, 2019, Madrid, Spain – Abstracts

Jean Dessolin
European Biophysics Journal, 2019, 48 (JOINT 12th EBSA congress and 10th ICBP – IUPAP congress, July 20-24, 2019, Madrid, Spain – Abstracts), pp.S1-264. ⟨10.1007/s00249-019-01373-4⟩
Article dans une revue hal-02394826v1

Synthesis and biological evaluation of hydrophilic embelin derivatives

Marc Lamblin , Antoine Sallustrau , Claude Commandeur , Thierry Cresteil , François-Xavier Felpin , et al.
Tetrahedron, 2012, 68 (24), pp.4655-4663. ⟨10.1016/j.tet.2012.04.024⟩
Article dans une revue istex hal-00740998v1