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Chemo- versus immuno-precipitation of G-quadruplex-DNA (G4DNA): a direct comparison of the efficiency of the antibody BG4 versus the small-molecule ligands TASQs for G4 affinity capture

 Yilong Feng , Zhenyu Luo , Francesco Rota Sperti , Ibai Valverde , Wenli Zhang , et al.
2022
Pré-publication, Document de travail hal-03836040v1

Amide-to-triazole switch vs. in vivo NEP-inhibition approaches to promote radiopeptide targeting of GRPR-positive tumors

 Theodosia Maina , Aikaterini Kaloudi , Ibai E. Valverde , Thomas L. Mindt , Berthold A. Nock
Nuclear Medicine and Biology, 2017, 52, pp.57 - 62. ⟨10.1016/j.nucmedbio.2017.06.001⟩
Article dans une revue hal-01562008v1
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Synthesis, stability and spectral behavior of fluorogenic sulfone-pyronin and sulfone-rosamine dyes

 Garance Dejouy , Myriam Laly , Ibai Valverde , Anthony Romieu
Dyes and Pigments, 2018, 159, pp.262-274. ⟨10.1016/j.dyepig.2018.06.026⟩
Article dans une revue hal-02168863v1
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Biomimetic, smart and multivalent ligands for G-quadruplex isolation and bioorthogonal imaging

 Francesco Rota Sperti , Thibaut Charbonnier , Pauline Lejault , Joanna Zell , Claire Bernhard , et al.
2020
Pré-publication, Document de travail hal-03086822v1
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Quest for novel fluorogenic xanthene dyes: Synthesis, spectral properties and stability of 3-imino-3H-xanthen-6-amine (pyronin) and its silicon analog

 Anthony Romieu , Garance Dejouy , Ibai Valverde
Tetrahedron Letters, 2018, 59 (52), pp.4574-4581. ⟨10.1016/j.tetlet.2018.11.031⟩
Article dans une revue hal-02168864v1
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The multivalent G-quadruplex (G4)-ligands MultiTASQs allow for versatile click chemistry-based investigations

 Francesco Rota Sperti , Jérémie Mitteaux , Joanna Zell , Angélique Pipier , Ibai E Valverde , et al.
RSC Chemical Biology, 2023, 4 (7), pp.456-465. ⟨10.1039/D3CB00009E⟩
Article dans une revue hal-04154672v1

Synthesis of a biologically active triazole-containing analogue of cystatin A through successive peptidomimetic alkyne-azide ligations.

 Ibai E Valverde , Fabien Lecaille , Gilles Lalmanach , Vincent Aucagne , Agnès F Delmas
Angewandte Chemie International Edition, 2012, 51 (3), pp.718-22. ⟨10.1002/anie.201107222⟩
Article dans une revue istex hal-00726293v1
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La multi-ligation triazole : Développement de nouveaux outils pour la synthèse de mimes de protéines par cycloadditions successives

 Ibai Valverde
Chimie. Universite d'Orléans, 2010. Français. ⟨NNT : ⟩
Thèse tel-01157275v1

Biomimetic G-quartet compounds

 David Monchaud , Pauline Lejault , Ibai E. Valverde , Francesco Rota Sperti
France, Patent n° : EP3889155A1. 2021
Brevet hal-03372659v1
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A Modular One-Pot Strategy for the Synthesis of Heterobivalent Tracers

 Thibaud Bailly , Sacha Bodin , Victor Goncalves , Franck Denat , Clément Morgat , et al.
ACS Medicinal Chemistry Letters, In press, ⟨10.1021/acsmedchemlett.3c00057⟩
Article dans une revue hal-04087376v1
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Fluorogenic Enzyme-Triggered Domino Reactions Producing Quinoxalin-2(1H)-one-based Heterocycles

 Garance Dejouy , Kévin Renault , Quentin Bonnin , Arnaud Chevalier , Cédric Michaudet , et al.
Organic Letters, 2020, 22 (16), pp.6494-6499. ⟨10.1021/acs.orglett.0c02287⟩
Article dans une revue hal-03006821v1
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Fluorogenic Enzyme-Triggered Domino Reactions Producing Quinoxalin-2(1 H)-one-based Heterocycles

 Garance Dejouy , Kévin Renault , Quentin Bonnin , Arnaud Chevalier , Cédric Michaudet , et al.
Organic Letters, 2020, 22 (16), pp.6494-6499. ⟨10.26434/chemrxiv.12613862.v1⟩
Article dans une revue hal-03016953v1
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Theranostics of Primary Prostate Cancer: Beyond PSMA and GRP-R

 Romain Schollhammer , Marie-Laure Quintyn Ranty , Henri de Clermont Gallerande , Florine Cavelier , Ibai E Valverde , et al.
Cancers, 2023, 15 (8), pp.2345. ⟨10.3390/cancers15082345⟩
Article dans une revue hal-04075693v1
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Synthetic routes to novel fluorogenic pyronins and silicon analogs with far-red spectral properties and enhanced aqueous stability

 Garance Dejouy , Kevin Renault , Ibai E. Valverde , Anthony Romieu
Dyes and Pigments, 2020, 180, pp.108496. ⟨10.1016/j.dyepig.2020.108496⟩
Article dans une revue hal-03006830v1
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Synthesis and evaluation of zirconium-89 labelled and long-lived GLP-1 receptor agonists for PET imaging

 Christian Borch Jacobsen , René Raavé , Marie Østergaard Pedersen , Pierre Adumeau , Mathieu Moreau , et al.
Nuclear Medicine and Biology, 2020, 82-83, pp.49-56. ⟨10.1016/j.nucmedbio.2019.11.006⟩
Article dans une revue hal-03004102v1

Towards the simplification of protein synthesis: iterative solid-supported ligations with concomitant purifications.

 Vincent Aucagne , Ibai E Valverde , Philippe Marceau , Mathieu Galibert , Nabil Dendane , et al.
Angewandte Chemie International Edition, 2012, 51 (45), pp.11320-4. ⟨10.1002/anie.201206428⟩
Article dans une revue istex hal-00748170v1
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The multivalent G-quadruplex (G4)-ligands MultiTASQs allow for versatile click chemistry-based investigations

 Francesco Rota Sperti , Jeremie Mitteaux , Joanna Zell , Angelique Pipier , Ibai Valverde , et al.
2022
Pré-publication, Document de travail hal-03836044v1
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1,5-Disubstituted 1,2,3-Triazoles as Amide Bond Isosteres Yield Novel Tumor-Targeting Minigastrin Analogs

 Nathalie M. Grob , Roger Schibli , Martin Béhé , Ibai Valverde , Thomas L. Mindt
ACS Medicinal Chemistry Letters, In press, ⟨10.1021/acsmedchemlett.0c00636⟩
Article dans une revue hal-03178434v1
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The scope of application of macrocyclic polyamines beyond metal chelation

 Pauline Lejault , Katerina Duskova , Claire Bernhard , Ibai E. Valverde , Anthony Romieu , et al.
European Journal of Organic Chemistry, 2019, 2019 (36), pp.6146-6157. ⟨10.1002/ejoc.201900870⟩
Article dans une revue hal-02268694v2
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Synthetic routes to novel fluorogenic pyronins and silicon analogs with far-red spectral properties and enhanced aqueous stability

 Garance Dejouy , Kévin Renault , Ibai E. Valverde , Anthony Romieu
2020
Pré-publication, Document de travail hal-03007352v1
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Biomimetic, Smart, and Multivalent Ligands for G-Quadruplex Isolation and Bioorthogonal Imaging

 Francesco Rota Sperti , Thibaut Charbonnier , Pauline Lejault , Joanna Zell , Claire Bernhard , et al.
ACS Chemical Biology, 2021, 16 (5), pp.905 - 914. ⟨10.1021/acschembio.1c00111⟩
Article dans une revue hal-03321466v1
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Single Peptide Backbone Surrogate Mutations to Regulate Angiotensin GPCR Subtype Selectivity

 Eirinaios Vrettos , Ibai E. Valverde , Alba Mascarin , Patrick Pallier , Linda Cerofolini , et al.
Chemistry - A European Journal, 2020, 26 (47), pp.10690-10694. ⟨10.1002/chem.202000924⟩
Article dans une revue hal-03007010v1

Click a la carte: robust semi-orthogonal alkyne protecting groups for multiple successive azide/alkyne cycloadditions

 Ibai E. Valverde , Agnès F. Delmas , Vincent Aucagne
Tetrahedron, 2009, 65 (36), pp.7597-7602. ⟨10.1016/j.tet.2009.06.093⟩
Article dans une revue istex hal-00525398v1
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