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23

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Journal articles23 documents

  • Matúš Hlaváč, Lucia Kováčiková, Marta Šoltésová Prnová, Gabriela Addová, Gilles Hanquet, et al.. Novel substituted N-benzyl(oxotriazinoindole) inhibitors of aldose reductase exploiting ALR2 unoccupied interactive pocket. Bioorganic and Medicinal Chemistry, Elsevier, 2021, 29, pp.115885. ⟨10.1016/j.bmc.2020.115885⟩. ⟨hal-03052028⟩
  • Gilles Hanquet, Matúš Hlaváč, Lucia Kováčiková, Marta Šoltésová Prnová, Peter Šramel, et al.. Development of Novel Oxotriazinoindole Inhibitors of Aldose Reductase: Isosteric Sulfur/Oxygen Replacement in the Thioxotriazinoindole Cemtirestat Markedly Improved Inhibition Selectivity. Journal of Medicinal Chemistry, American Chemical Society, 2020, 63 (1), pp.369-381. ⟨10.1021/acs.jmedchem.9b01747⟩. ⟨hal-03052056⟩
  • Matúš Hlaváč, Lucia Kováčiková, Marta Prnová, Gabriela Addová, Gilles Hanquet, et al.. Novel substituted N-benzyl(oxotriazinoindole) inhibitors of aldose reductase exploiting ALR2 unoccupied interactive pocket. Bioorganic and Medicinal Chemistry, Elsevier, 2020. ⟨hal-03070904⟩
  • Anna Santarsiero, Antonella Bochicchio, Maria Funicello, Paolo Lupattelli, Sabine Choppin, et al.. New synthesized polyoxygenated diarylheptanoids suppress lipopolysaccharide-induced neuroinflammation. Biochemical and Biophysical Research Communications, Elsevier, 2020. ⟨hal-03077267⟩
  • Anna Santarsiero, Antonella Bochicchio, Maria Funicello, Paolo Lupattelli, Sabine Choppin, et al.. New synthesized polyoxygenated diarylheptanoids suppress lipopolysaccharide-induced neuroinflammation. Biochemical and Biophysical Research Communications, Elsevier, 2020, 529 (4), pp.1117-1123. ⟨10.1016/j.bbrc.2020.06.122⟩. ⟨hal-03076397⟩
  • Frédéric R. Leroux, Thomas Guérin, Nadiia Pikun, Ryutaro Morioka, Armen Panossian, et al.. Synthesis and Use of Trifluoromethylthiolated Ketenimines. Chemistry - A European Journal, Wiley-VCH Verlag, 2020, ⟨10.1002/chem.202002723⟩. ⟨hal-02990038⟩
  • Yangyi Qiu, Shu Ting Chan, Lin Lin, Tsun Lam Shek, Tsz Fung Tsang, et al.. Design, synthesis and biological evaluation of antimicrobial diarylimine and –amine compounds targeting the interaction between the bacterial NusB and NusE proteins. European Journal of Medicinal Chemistry, Elsevier, 2019, 178, pp.214-231. ⟨10.1016/j.ejmech.2019.05.090⟩. ⟨hal-03054499⟩
  • Yangyi Qiu, Shu Ting Chan, Lin Lin, Tsun Lam Shek, Tsz Fung Tsang, et al.. Nusbiarylins, a new class of antimicrobial agents: Rational design of bacterial transcription inhibitors targeting the interaction between the NusB and NusE proteins. Bioorganic Chemistry, Elsevier, 2019, 92, pp.103203. ⟨10.1016/j.bioorg.2019.103203⟩. ⟨hal-03054418⟩
  • Yangyi Qiu, Shu Chan, Lin Lin, Tsun Shek, Tsz Tsang, et al.. Design, Synthesis and Biological Evaluation of Antimicrobial Diarylimine and -amine Compounds Targeting the Interaction between the Bacterial NusB and NusE Proteins. European Journal of Medicinal Chemistry, Elsevier, 2019. ⟨hal-03079069⟩
  • Yangyi Qiu, Shu Chan, Lin Lin, Tsun Shek, Tsz Tsang, et al.. Nusbiarylins, a New Class of Antimicrobial Agents: Rational Design of Bacterial Transcription Inhibitors Targeting the Interaction between the NusB and NusE Proteins. Bioorganic Chemistry, Elsevier, 2019. ⟨hal-03079075⟩
  • Paul Massé, Sabine Choppin, Lucia Chiummiento, Gilles Hanquet, Francoise Colobert. Unintended Formation of a 26-Membered Cycle in the Course of a Novel Approach to Myricanol, a Strained [7,0]-metacyclophane. SYNLETT, Georg Thieme Verlag, 2019. ⟨hal-03075499⟩
  • Chloé Batisse, Maria Cespedes Davila, Marco Castello, Amélia Messara, Bertrand Vivet, et al.. Efficient asymmetric synthesis of aryl difluoromethyl sulfoxides and their use to access enantiopure α-difluoromethyl alcohols. Tetrahedron, Elsevier, 2019, 75 (23), pp.3063-3079. ⟨10.1016/j.tet.2019.04.037⟩. ⟨hal-02400108⟩
  • Lucie Schiavo, L Lebedel, P Massé, Sabine Choppin, Gilles Hanquet. Access to Wieland–Miescher Diketone-Derived Building Blocks by Stereoselective Construction of the C-9 Quaternary Carbon Center Using the Mukaiyama Aldol Reaction. Journal of Organic Chemistry, American Chemical Society, 2018, 83 (12), pp.6247-6258. ⟨10.1021/acs.joc.7b02862⟩. ⟨hal-02150059⟩
  • Antonella Bochicchio, Lucie Schiavo, L Chiummiento, P Lupattelli, M Funicello, et al.. Convergent total synthesis of (±) myricanol, a cyclic natural diarylheptanoid. Organic and Biomolecular Chemistry, Royal Society of Chemistry, 2018, 16, pp.8859-8869. ⟨10.1039/C8OB02052C⟩. ⟨hal-02158253⟩
  • H Norouzi-Arasi, X Salom-Roig, S Lanners, Gilles Hanquet. First Total Synthesis of Pamamycin-621D. Current Organic Synthesis, 2018, 15, pp.105-109. ⟨10.2174/1570179414666170525103947⟩. ⟨hal-02167613⟩
  • ChloÉ Batisse, Armen Panossian, Gilles Hanquet, Frédéric Leroux. Access towards enantiopure α,α-difluoromethyl alcohols by means of sulfoxides as traceless chiral auxiliaries. Chemical Communications, Royal Society of Chemistry, 2018, 54 (74), pp.10423-10426. ⟨10.1039/C8CC05571H⟩. ⟨hal-02150060⟩
  • Giorgio Della Sala, Marina Sicignano, Rosaria Schettini, Francesco de Riccardis, Luigi Cavallo, et al.. Switchable Diastereoselectivity in the Fluoride-Promoted Vinylogous Mukaiyama–Michael Reaction of 2-[(Trimethylsilyl)oxy]furan Catalyzed by Crown Ethers. Journal of Organic Chemistry, American Chemical Society, 2017, 82 (13), pp.6629-6637. ⟨10.1021/acs.joc.7b00743⟩. ⟨hal-03054554⟩
  • E Evain-Bana, Lucie Schiavo, C Bour, Don Antoine Lanfranchi, S Berardozzi, et al.. Synthesis, biological evaluation and molecular modeling studies on novel quinonoid inhibitors of CDC25 phosphatases. Journal of Enzyme Inhibition and Medicinal Chemistry, 2017, 32, pp.113-118. ⟨10.1080/14756366.2016.1238364⟩. ⟨hal-02161666⟩
  • M Murár, J Dobiaš, P Šramel, G Addová, Gilles Hanquet, et al.. Novel CLK1 inhibitors based on N-aryloxazol-2-amine skeleton - A possible way to dual VEGFR2 TK/CLK ligands. European Journal of Medicinal Chemistry, Elsevier, 2017, 126, pp.754-761. ⟨10.1016/j.ejmech.2016.11.003⟩. ⟨hal-02170487⟩
  • D Kahraman, Gilles Hanquet, L Jeanmart, S Lanners, Peter Sramel, et al.. Quinoides and VEGFR2 TKIs influence the fate of hepatocellular carcinoma and its cancer stem cells. MedChemComm, 2017, 8, pp.81-87. ⟨10.1039/C6MD00392C⟩. ⟨hal-02177405⟩
  • Lucie Schiavo, L Jeanmart, S Lanners, Sabine Choppin, Gilles Hanquet. FeCl3.6H2O/acetaldehyde, a versatile system for the deprotection of ketals and acetals via a transacetalization process. New Journal of Chemistry, Royal Society of Chemistry, 2017, 41, pp.1421-1424. ⟨10.1039/C6NJ03439J⟩. ⟨hal-02167611⟩
  • Gilles Hanquet, Xavier Salom-Roig, Steve Lanners. New Insights into the Synthesis and Biological Activity of the Pamamycin Macrodiolides. CHIMIA, Schweizerische Chemische Gesellschaft, 2016, 70 (1), pp.20-28. ⟨10.2533/chimia.2016.20⟩. ⟨hal-03054586⟩
  • Antonella Bochicchio, Rossella Cefola, Sabine Choppin, Françoise Colobert, Maria Antonietta Di Noia, et al.. Selective Claisen rearrangement and iodination for the synthesis of polyoxygenated allyl phenol derivatives. Tetrahedron Letters, Elsevier, 2016, 57 (36), pp.4053-4055. ⟨10.1016/j.tetlet.2016.07.079⟩. ⟨hal-03054575⟩