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Light Activation for the Versatile and Accurate Kinetic Analysis of Disassembly of Self-Immolative Spacers

Ahmed Alouane , Raphaël Labruère , Thomas Le saux , Isabelle Aujard , Sylvie Dubruille , et al.
Chemistry - A European Journal, 2013, 19 (35), pp.11717-11724. ⟨10.1002/chem.201301298⟩
Article dans une revue istex hal-02137231v1
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Water Residence Time Estimation by 1D Deconvolution in the Form of a l 2 -Regularized Inverse Problem With Smoothness, Positivity and Causality Constraints

Alina G. Meresescu , Matthieu Kowalski , Frédéric Schmidt , François Landais
Computers & Geosciences, 2018, 115, pp.105-121. ⟨10.1016/j.cageo.2018.03.009⟩
Article dans une revue hal-01735678v1

A new delivery system for auristatin in STxB-drug conjugate therapy

Cornélie Batisse , Estelle Dransart , Rafik Ait Sarkouh , Laura Brullé , Siau-Kun Bai , et al.
European Journal of Medicinal Chemistry, 2015, 95, pp.483-491. ⟨10.1016/j.ejmech.2015.03.047⟩
Article dans une revue hal-02137225v1

Application of the ADEPT strategy to the MDR resistance in cancer chemotherapy.

Frédéric Schmidt
Anti-Cancer Drug Design, 1999, 14 (2), pp.93-106
Article dans une revue hal-02137891v1

Glucuronide prodrugs of hydroxy compounds for antibody directed enzyme prodrug therapy (ADEPT) : A phenol nitrogen mustard carbamate

Frédéric Schmidt
Bioorganic and Medicinal Chemistry Letters, 1997, 7 (8), pp.1071-1076. ⟨10.1016/S0960-894X(97)00157-1⟩
Article dans une revue istex hal-02137877v1

Optimizing the formation of biocompatible gold nanorods for cancer research: Functionalization, stabilization and purification

Nicolas Bogliotti , Birgit Oberleitner , Aurelie Di-Cicco , Frédéric Schmidt , Jean-Claude Florent , et al.
Journal of Colloid and Interface Science, 2011, 357 (1), pp.75-81. ⟨10.1016/j.jcis.2011.01.053⟩
Article dans une revue istex hal-02137238v1

Salicylaldehyde derivatives as new protein kinase CK2 inhibitors.

Renaud Prudent , Miriam López-Ramos , Virginie Moucadel , Caroline Barette , David S. Grierson , et al.
Biochimica et Biophysica Acta (BBA) - General Subjects, 2008, 1780 (12), pp.1412-20. ⟨10.1016/j.bbagen.2008.06.010⟩
Article dans une revue istex hal-00345748v1

Synthèse et étude d'une prodrogue de dipyridamole: application de la stratégie ADEPT à la résistance multiple (MDR) en chimiothérapie anticancéreuse

Frédéric Schmidt
Comptes rendus de l’Académie des sciences. Série IIc, Chimie, 1998, 1 (7), pp.421-424. ⟨10.1016/S1387-1609(98)80422-2⟩
Article dans une revue istex hal-02137876v1

A new paclitaxel prodrug for use in ADEPT strategy

Frédéric Schmidt , Emmanuel Bouvier , Sylvie Thirot , Frédéric Schmidt , Claude Monneret
Organic & Biomolecular Chemistry, 2003, 1 (19), pp.3343. ⟨10.1039/b306236h⟩
Article dans une revue hal-02137813v1

Synthesis of Polysubstituted 5-Azaindoles via Palladium-Catalyzed Heteroannulation of Diarylalkynes

Frédéric Schmidt , Géraldine Calvet , Marion Livecchi , Frédéric Schmidt
Journal of Organic Chemistry, 2011, 76 (11), pp.4734-4740. ⟨10.1021/jo200480h⟩
Article dans une revue hal-02137237v1

Chemical Biology: Contribution to Molecular Therapeutic Innovation – A New Role for Chemistry? Report from the Thematic Symposium Organized by the SCT (French Medicinal Chemistry Society), November 26th, 2013

Frédéric Schmidt , Pascal George , Janos Sapi
ACS Chemical Biology, 2014, 9 (4), pp.849-852. ⟨10.1021/cb500173s⟩
Article dans une revue hal-02137230v1

New Taxol® (paclitaxel) prodrugs designed for ADEPT and PMT strategies in cancer chemotherapy

Abdessamad El Alaoui , Nabendu Saha , Frédéric Schmidt , Claude Monneret , Claude Florent
Bioorganic and Medicinal Chemistry, 2006, 14 (14), pp.5012-5019. ⟨10.1016/j.bmc.2006.03.002⟩
Article dans une revue istex hal-02137811v1

Cyclointercalands.- Incorporation of the phenazine group and of metal binding subunits into macrocyclic receptor molecules.

Frédéric Schmidt
Tetrahedron Letters, 1988, 29 (41), pp.5255-5258. ⟨10.1016/S0040-4039(00)80730-3⟩
Article dans une revue istex hal-02137881v1

A chemically encoded timer for dual molecular delivery at tailored ranges and concentrations

Silvia Serra , Ahmed Alouane , Thomas Le Saux , Steve Huvelle , Raphaël Plasson , et al.
Chemical Communications, 2018, 54 (49), pp.6396-6399. ⟨10.1039/C8CC03253J⟩
Article dans une revue hal-03028566v1
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Planetary Data in the Virtual Observatory: VESPA (Virtual European Solar and Planetary Access)

Stéphane Erard , Baptiste Cecconi , Pierre Le Sidaner , A. P. Rossi , L. Tomasik , et al.
5th Planetary Data Workshop (PDW) and 2nd Planetary Science Informatics & Data Analytics (PSIDA) meeting, Jun 2021, Virtual Meeting, United States
Communication dans un congrès insu-03443277v1

“Self-Immolative” Spacer for Uncaging with Fluorescence Reporting

Raphaël Labruère , Ahmed Alouane , Thomas Le saux , Isabelle Aujard , Philippe Pelupessy , et al.
Angewandte Chemie International Edition, 2012, 51 (37), pp.9344-9347. ⟨10.1002/anie.201204032⟩
Article dans une revue istex hal-02137233v1

[Glucuronyl paclitaxel (Taxol) derivatives as tumor activated prodrugs].

Frédéric Schmidt
Annales Pharmaceutiques Françaises, 2005, 63 (1), pp.53-62
Article dans une revue hal-02137884v1

Prodrug Mono therapy: synthesis and biological evaluation of an etoposide glucuronide-prodrug

Frédéric Schmidt , Claude Monneret
Bioorganic and Medicinal Chemistry, 2003, 11 (10), pp.2277-2283. ⟨10.1016/s0968-0896(03)00108-1⟩
Article dans une revue istex hal-02137819v1

Effective antitumor therapy based on a novel antibody-drug conjugate targeting the Tn carbohydrate antigen

Frédéric Schmidt
OncoImmunology, 2016, 5 (7), pp.e1171434. ⟨10.1080/2162402X.2016.1171434⟩
Article dans une revue hal-02137864v1
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Implementation strategies for hyperspectral unmixing using Bayesian source separation.

Frédéric Schmidt , Albrecht Schmidt , Erwan Tréguier , Maël Guiheneuf , Saïd Moussaoui , et al.
IEEE Transactions on Geoscience and Remote Sensing, 2010, 48 (11), pp.4003-4013. ⟨10.1109/TGRS.2010.2062190⟩
Article dans une revue hal-03556769v1

Cancer Chemotherapy: A Paclitaxel Prodrug for ADEPT (Antibody-Directed Enzyme Prodrug Therapy)

Frédéric Schmidt
European Journal of Organic Chemistry, 2001, 2001 (11), pp.2129-2134. ⟨10.1002/1099-0690(200106)2001:11<2129::AID-EJOC2129>3.0.CO;2-#⟩
Article dans une revue istex hal-02137899v1

Targeted Shiga toxin-drug conjugates prepared via Cu-free click chemistry.

Vesela Kostova , Michel Azoulay , Laura Brullé , Siau-Kun Bai , Jean-Claude Florent , et al.
Bioorganic and Medicinal Chemistry, 2015, 23 (22), pp.7150-7. ⟨10.1016/j.bmc.2015.10.010⟩
Article dans une revue hal-01298164v1

In vitro fluorine-19 nuclear magnetic resonance study of the liberation of antitumor nitrogen mustard from prodrugs

Frédéric Schmidt
Journal of the Chemical Society, Perkin Transactions 1, 1999, 14 (10), pp.1302-1308. ⟨10.1039/B111549A⟩
Article dans une revue istex hal-02137875v1

Synthese d'ynamines fonctionnalisees en β de la triple liaison et stereoselectivite de l'hydrolyse des cycloadduits formes avec la cyclopentenone et les lactones α-β insaturees

Frédéric Schmidt
Tetrahedron Letters, 1982, 23 (17), pp.1821-1824. ⟨10.1016/S0040-4039(00)86750-7⟩
Article dans une revue istex hal-02137901v1

Absolute Quantification of Drug Vector Delivery to the Cytosol

Marco Lucchino , Anne Billet , Siau‐kun Bai , Estelle Dransart , Justine Hadjerci , et al.
Angewandte Chemie International Edition, 2021, 60 (27), pp.14824-14830. ⟨10.1002/anie.202102332⟩
Article dans une revue hal-04092139v1

Applications in remote sensing—natural landscapes

Touria Bajjouk , Florian de Boissieu , Jocelyn Chanussot , Sylvain Dout , Marie Dumont , et al.
Hyperspectral Imaging, 32, Elsevier Ltd, pp.371-410, 2020, Data Handling in Science and Technology, 978-0-444-63977-6. ⟨10.1016/B978-0-444-63977-6.00016-X⟩
Chapitre d'ouvrage hal-02477896v1

Cancer chemotherapy: A SN-38 (7-Ethyl-10-hydroxycamptothecin) glucuronide prodrug for treatment by a PMT (Prodrug monoTherapy) strategy

Stéphane Angenault , Sylvie Thirot , Frédéric Schmidt , Claude Monneret , Bruno Pfeiffer , et al.
Bioorganic and Medicinal Chemistry Letters, 2003, 13 (5), pp.947-950. ⟨10.1016/s0960-894x(02)01080-6⟩
Article dans une revue istex hal-02137820v1

Palladium-Catalyzed Synthesis of 2,3-Disubstituted 5-Azaindoles via Heteroannulation Reaction and of 2-Substituted 5-Azaindoles through Domino Sila-Sonogashira/5-Endo Cyclization

Marion Livecchi , Géraldine Calvet , Frédéric Schmidt
Journal of Organic Chemistry, 2012, 77 (11), pp.5006-5016. ⟨10.1021/jo300481s⟩
Article dans une revue hal-02137234v1

A double-triggered self-immolative spacer for increased selectivity of molecular release

Steve Huvelle , Thomas Le Saux , Ludovic Jullien , Frédéric Schmidt
Organic & Biomolecular Chemistry, 2021, 20 (1), pp.240-246. ⟨10.1039/D1OB02124A⟩
Article dans une revue hal-04059747v1

Disassembly Kinetics of Quinone-Methide-Based Self-Immolative Spacers that Contain Aromatic Nitrogen Heterocycles

Ahmed Alouane , Raphaël Labruère , Katherine Silvestre , Thomas Le saux , Frédéric Schmidt , et al.
Chemistry - An Asian Journal, 2014, 9 (5), pp.1334-1340. ⟨10.1002/asia.201400051⟩
Article dans une revue istex hal-02137229v1