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A palladium-catalyzed coupling of 3-chloroquinoxalinones with various nitrogen-containing nucleophiles

Etienne Brachet , Jean-François Peyrat , Jean-Daniel Brion , Samir Messaoudi , Mouâd Alami
Organic & Biomolecular Chemistry, 2013, 11 (23), pp.3808. ⟨10.1039/c3ob40338f⟩
Article dans une revue hal-03073852v1

Synthesis, biological evaluation, and structure–activity relationships of tri- and tetrasubstituted olefins related to isocombretastatin A-4 as new tubulin inhibitors

Jessy Aziz , Etienne Brachet , Abdallah Hamze , Jean-François Peyrat , Guillaume Bernadat , et al.
Organic & Biomolecular Chemistry, 2013, 11 (3), pp.430-442. ⟨10.1039/c2ob26253c⟩
Article dans une revue hal-03073854v1
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Synthesis of axially chiral biaryl thioglycosides through thiosugar-directed Pd-catalyzed asymmetric C–H activation

Maha Fatthalla , Nicolas Grimblat , Etienne Brachet , Mouad Alami , Vincent Gandon , et al.
Chemical Communications, 2021, 57 (80), pp.10355-10358. ⟨10.1039/d1cc03971g⟩
Article dans une revue hal-03425421v1
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Visible light amination/Smiles cascade: access to phthalazine derivatives

Etienne Brachet , Leyre Marzo , Mohamed Selkti , Burkhard König , Philippe Belmont
Chemical Science, 2016, 7 (8), pp.5002-5006. ⟨10.1039/C6SC01095D⟩
Article dans une revue hal-02384218v1

Palladium-Catalyzed Regioselective Alkynylation of Pyrroles and Azoles under Mild Conditions: Application to the Synthesis of a Dopamine D-4 Receptor Agonist

Etienne Brachet , Philippe Belmont
Journal of Organic Chemistry, 2015, 80 (15), pp.7519-7529. ⟨10.1021/acs.joc.5b01093⟩
Article dans une revue hal-03073838v1

Light on Unsaturated Hydrocarbons - “Gotta Heterofunctionalize Them All”

Doriane Menigaux , Philippe Belmont , Etienne Brachet
European Journal of Organic Chemistry, 2017, 2017 (15), pp.2008-2055. ⟨10.1002/ejoc.201601626⟩
Article dans une revue hal-03073829v1

Visible Light-Induced Regioselective Cycloaddition of Benzoyl Azides and Alkenes To Yield Oxazolines

Peter Bellotti , Julien Brocus , Fatima El Orf , Mohamed Selkti , Burkhard König , et al.
Journal of Organic Chemistry, 2015, 84 (10), pp.6278-6285. ⟨10.1021/acs.joc.9b00568⟩
Article dans une revue hal-02384322v1

Phosphine-Triggered Selectivity Switch in Silver-Catalyzed o-Alkynylbenzohydroxamic Acid Cycloisomerizations

Etienne Brachet , Xavier Bantreil , Aurélie Bourderioux , Pierre Mateo , Caroline Hagerman , et al.
Organic Letters, 2016, 18 (19), pp.4814-4817. ⟨10.1021/acs.orglett.6b02235⟩
Article dans une revue hal-02418682v1

Phosphoramidates as Transient Precursors of Nitrogen‐Centered Radical Under Visible‐Light Irradiation: Application to the Synthesis of Phthalazine Derivatives

Maxime de Abreu , Mohamed Selkti , Philippe Belmont , Etienne Brachet
Advanced Synthesis and Catalysis, 2020, 362 (11), pp.2216-2222. ⟨10.1002/adsc.202000018⟩
Article dans une revue hal-03073822v1

Light-Enabled Radical 1,4-Aryl Migration Via a Phospho-Smiles Rearrangement

Maxime de Abreu , Philippe Belmont , Etienne Brachet
Journal of Organic Chemistry, 2021, ⟨10.1021/acs.joc.0c02540⟩
Article dans une revue hal-03132343v1

Visible light amination/Smiles cascade: access to phthalazine derivatives

Etienne Brachet , Leyre Marzo , Mohamed Selkti , Burkhard König , Philippe Belmont
Chemical Science, 2016, 7 (8), pp.5002-5006. ⟨10.1039/c6sc01095d⟩
Article dans une revue hal-03073836v1

Synergistic Photoredox/Transition-Metal Catalysis for Carbon-Carbon Bond Formation Reactions

Maxime de Abreu , Philippe Belmont , Etienne Brachet
European Journal of Organic Chemistry, 2020, 2020 (10), pp.1327-1378. ⟨10.1002/ejoc.201901146⟩
Article dans une revue hal-03073824v1

Phosphine-Triggered Selectivity Switch in Silver-Catalyzed o -Alkynylbenzohydroxamic Acid Cycloisomerizations

Xavier Bantreil , Aurélie Bourderioux , Pierre Mateo , Caroline Hagerman , Mohamed Selkti , et al.
Organic Letters, 2016, 18 (19), pp.4814-4817. ⟨10.1021/acs.orglett.6b02235⟩
Article dans une revue hal-03534140v1

Palladium-Catalyzed Coupling of N -Amino­azoles with 3-Halo-Substituted ­Quinolin-2(1 H )-ones, Coumarins, Quin­oxalin-2(1 H )-ones, and Chromenes

Thi Thanh Huyen Luong , Etienne Brachet , Jean-Daniel Brion , Samir Messaoudi , Mouâd Alami
European Journal of Organic Chemistry, 2015, 2015 (8), pp.1771-1780. ⟨10.1002/ejoc.201403501⟩
Article dans une revue istex hal-03073839v1

Palladium-Catalyzed Cross-Coupling Reaction of Thioglycosides with (Hetero)aryl Halides

Etienne Brachet , Jean-Daniel Brion , Samir Messaoudi , Mouad Alami
Advanced Synthesis and Catalysis, 2013, pp.n/a-n/a. ⟨10.1002/adsc.201200695⟩
Article dans une revue istex hal-03073850v1

Synergistic Photoredox/Transition-Metal Catalysis for Carbon-Carbon Bond Formation Reactions

Maxime de Abreu , Philippe Belmont , Etienne Brachet
European Journal of Organic Chemistry, 2017, 2017 (15), pp.2008-2055. ⟨10.1002/ejoc.201901146⟩
Article dans une revue hal-02384360v1

Spotlight on Photo‐Induced Aryl Migration Reactions.

Marie Huynh , Maxime de Abreu , Philippe Belmont , Etienne Brachet
Chemistry - A European Journal, 2020, ⟨10.1002/chem.202003507⟩
Article dans une revue hal-03073199v1

Synthesis, biological evaluation, and structure-activity relationships of tri- and tetrasubstituted olefins related to isocombretastatin A-4 as new tubulin inhibitors.

Jessy Aziz , Etienne Brachet , Abdallah Hamze , Jean-François Peyrat , Guillaume Bernadat , et al.
Organic & Biomolecular Chemistry, 2013, 11 (3), pp.430-42. ⟨10.1039/c2ob26253c⟩
Article dans une revue hal-00798259v1
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Nouvelles réactions métallocatalyées pour la création de liaisons C-N et C-S : applications à la synthèse d'inhibiteurs de la Hsp90

Etienne Brachet
Sciences agricoles. Université Paris Sud - Paris XI, 2013. Français. ⟨NNT : 2013PA114836⟩
Thèse tel-01232125v1
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Synthesis, 3D-structure and stability analyses of NRPa-308, a new promising anti-cancer agent

Etienne Brachet , Aurore Dumond , Wang-Qing Liu , Marie Fabre , Mohamed Selkti , et al.
Bioorganic and Medicinal Chemistry Letters, 2019, 29 (24), pp.126710. ⟨10.1016/j.bmcl.2019.126710⟩
Article dans une revue hal-02418648v1

Stereoselective Palladium-Catalyzed Alkenylation and Alkynylation of Thioglycosides

Etienne Brachet , Jean-Daniel Brion , Mouad Alami , Samir Messaoudi
Advanced Synthesis and Catalysis, 2013, 355 (13), pp.2627-2636. ⟨10.1002/adsc.201300419⟩
Article dans une revue istex hal-03073842v1

Visible-Light Heterofunctionalization Light on Unsaturated Hydrocarbons -"Gotta Heterofunctionalize Them All

Etienne Brachet
European Journal of Organic Chemistry, 2017, 2017 (15), pp.2008-2055. ⟨10.1002/ejoc.201601626⟩
Article dans une revue hal-02418679v1

Silver-catalyzed tandem cycloisomerization/hydroarylation reactions and mechanistic investigations for an efficient access to 1,2-dihydroisoquinolines

Maxime de Abreu , Yue Tang , Etienne Brachet , Mohamed Selkti , Véronique Michelet , et al.
Organic & Biomolecular Chemistry, 2021, ⟨10.1039/D0OB02197K⟩
Article dans une revue hal-03132346v1

Palladium-Catalyzed Cross-Coupling of 1-Aminoazoles with Aryl Chlorides: Application to the Synthesis of Unsymmetrical N,N′ -Diaryl-1-aminoindoles

Etienne Brachet , Samir Messaoudi , Jean-François Peyrat , Jean-Daniel Brion , Mouad Alami
Advanced Synthesis and Catalysis, 2012, 354 (14-15), pp.2829-2839. ⟨10.1002/adsc.201200440⟩
Article dans une revue istex hal-03073855v1

Palladium-Catalyzed Regioselective Alkynylation of Pyrroles and Azoles under Mild Conditions: Application to the Synthesis of a Dopamine D-4 Receptor Agonist

Etienne Brachet , Philippe Belmont
Journal of Organic Chemistry, 2015, 80 (15), pp.7519-7529. ⟨10.1021/acs.joc.5b01093⟩
Article dans une revue hal-02384634v1
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Neuropilin 1 and Neuropilin 2 gene invalidation or pharmacological inhibition reveals their relevance for the treatment of metastatic renal cell carcinoma

Aurore Dumond , Etienne Brachet , Jérôme Durivault , Valérie Vial , Anna Puszko , et al.
Journal of experimental & clinical cancer research, 2021, 40, pp.33. ⟨10.1186/s13046-021-01832-x⟩
Article dans une revue hal-03132345v1

Pd-Catalyzed Reaction of Sterically Hindered Hydrazones with Aryl Halides: Synthesis of Tetra-Substituted Olefins Related to iso -Combretastatin A4

Etienne Brachet , Abdallah Hamze , Jean-François Peyrat , Jean-Daniel Brion , Mouad Alami
Organic Letters, 2010, 12 (18), pp.4042-4045. ⟨10.1021/ol101639g⟩
Article dans une revue hal-03073857v1
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Visible light C-H amidation of heteroarenes with benzoyl azides

Etienne Brachet , T. Ghosh , I. Ghosh , B König
Chemical Science, 2015, 6 (2), pp.987-992. ⟨10.1039/c4sc02365j⟩
Article dans une revue hal-02418685v1

Nickel-Catalyzed Arylation, Alkenylation, and Alkynylation of Unprotected Thioglycosides at Room Temperature

Etienne Brachet , Jean-Daniel Brion , Mouad Alami , Samir Messaoudi
Chemistry - A European Journal, 2013, 19 (45), pp.15276-15280. ⟨10.1002/chem.201302999⟩
Article dans une revue istex hal-03073844v1