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Beef conjugated linoleic acid isomers reduce human cancer cell growth even when associated with other beef fatty acids

Anne de La Torre , Eric Debiton , Pierre Juaneda , Denis Durand , Jean-Michel Chardigny , et al.
British Journal of Nutrition, 2006, 95 (2), pp.346-352
Article dans une revue hal-01056754v1

Synthèse et évaluation biologique d'inhibiteurs potentiels de tyrosines kinases utilisables en imagerie.

Mathieu Sassatelli , Fadoua Bouchikhi , Samir Messaoudi , Bettina Aboab , Eric Debiton , et al.
1ères Journées Scientifiques du CLARA (Canceropôle Lyon Auvergne Rhône Alpes), 2006, Saint Ours les Roches, France
Communication dans un congrès hal-00019222v1

Synthesis and antiproliferative activities of indolin-2-one derivatives bearing amino-acid moieties

Fabrice Anizon , Mathieu Sassatelli , Eric Debiton , Bettina Aboab , Pascale Moreau , et al.
Organic Chemistry-Present and Future, Apr 2007, Louvain-la-Neuve, Belgium
Communication dans un congrès hal-00150120v1

Design, synthesis and preliminary biological evaluation of acridine compounds as potential agents for a combined targeted chemo-radionuclide therapy approach to melanoma

Nicolas Desbois , Maryline Gardette , Janine Papon , Pierre Labarre , Aurélie Maisonial , et al.
Bioorganic and Medicinal Chemistry, 2008, 16 (16), pp.7671-7690. ⟨10.1016/j.bmc.2008.07.015⟩
Article dans une revue istex hal-01494523v1

Synthesis and biological evaluation of a new scaffold for Pim kinase inhibitors

Laurent Gavara , Emmanuelle Saugues , Georges Alves , Eric Debiton , Fabrice Anizon , et al.
1er colloque Franco-Roumain de Chimie Médicinale COFr-RoCM, Oct 2010, Iasi, Romania
Communication dans un congrès hal-00531747v1
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Determination of eumelanin and pheomelanin in melanomas using solid-phase extraction and high performance liquid chromatography -diode array detection (HPLC-DAD) analysis

Benjamin Rioux , Jacques Rouanet , Hussein Akil , Sophie Besse , Eric Debiton , et al.
Journal of Chromatography B Biomedical Sciences and Applications, 2019, 1113, pp.60-68. ⟨10.1016/j.jchromb.2019.03.010⟩
Article dans une revue hal-02346260v1

Synthesis and kinases inhibitory potencies of aminopyrimidyl-indole derivatives

Rufine Akué-Gédu , Eric Debiton , Y. Ferandin , L. Meijer , Michelle Prudhomme , et al.
Drug Discovery and Selection, Jul 2009, Orléans, France
Communication dans un congrès hal-00389425v1

Novel imidazo[1,2-a]naphthyridinic systems (part 1): Synthesis, antiproliferative and DNA-intercalating activities

Emmanuel Moreau , Mounir Andaloussi , Nicolas Masurier , Jacques Lacroix , René C Gaudreault , et al.
European Journal of Medicinal Chemistry, 2008, 43 (11), pp.2505 - 2517. ⟨10.1016/j.ejmech.2008.02.017⟩
Article dans une revue istex hal-01677576v1
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Synthesis and antiproliferative activities of diversely substituted glycosyl-isoindigo derivatives.

Mathieu Sassatelli , Fadoua Bouchikhi , Samir Messaoudi , Fabrice Anizon , Eric Debiton , et al.
European Journal of Medicinal Chemistry, 2006, 41, pp.88-100. ⟨10.1016/j.ejmech.2005.10.004⟩
Article dans une revue hal-00020445v1

A Convenient Route to New (Radio)Fluorinated and (Radio)Iodinated Cyclic Tyrosine Analogs

Maria Chao , Jean-Michel Chezal , Eric Debiton , Damien Canitrot , Tiffany Witkowski , et al.
Pharmaceuticals, 2022, 15 (2), pp.162. ⟨10.3390/ph15020162⟩
Article dans une revue hal-03867865v1

Conjugated linoleic acid isomers and their conjugated derivatives inhibit growth of human cancer cell lines

Anne de La Torre , Eric Debiton , Denys Durand , Jean-Michel Chardigny , Olivier Berdeaux , et al.
Anticancer Research, 2005, 25 (6B), pp.3943-3949
Article dans une revue hal-02679711v1

Imidazonaphthyridine systems (part 2): Functionalization of the phenyl ring linked to the pyridine pharmacophore and its replacement by a pyridinone ring produces intriguing differences in cytocidal activity

Emmanuel Moreau , Nicolas Masurier , Eric Debiton , Alicia Jacquemet , Antoine Bussière , et al.
European Journal of Medicinal Chemistry, 2012, 52, pp.137 - 150. ⟨10.1016/j.ejmech.2012.03.011⟩
Article dans une revue istex hal-01677549v1

Synthesis and antiproliferative activities of diversely substituted glycosyl-isoindigo derivatives.

Mathieu Sassatelli , Fadoua Bouchikhi , Samir Messaoudi , Fabrice Anizon , C. Bartomeuf , et al.
Indirubin, the red shade of indigo, 2006, Les Eyzies de Tayac, France
Communication dans un congrès hal-00019219v1

Synthesis, protein kinase inhibitory potencies and in vitro antiproliferative activities of meridianin derivatives

Pascale Moreau , Francis Giraud , Elisabeth Pereira , Fabrice Anizon , Georges Alves , et al.
17th European Symposium on Organic Chemistry, Jul 2011, Hersonissos, Greece
Communication dans un congrès hal-00609975v1

Design, synthesis and in vitro drug release investigation of new potential 5-FU prodrugs

Pierre Daumar , Caroline Decombat , Jean-Michel Chezal , Eric Debiton , Michel Madesclaire , et al.
European Journal of Medicinal Chemistry, 2011, 46 (7), pp.2867-2879. ⟨10.1016/j.ejmech.2011.04.010⟩
Article dans une revue istex hal-03121824v1

Total structure and inhibition of tumor cell proliferation of Laxa phycins

Isabelle Bonnard , Marc Rolland , Jean-Marie Salmon , Eric Debiton , Chantal Barthomeuf , et al.
Journal of Medicinal Chemistry, 2007, 50, pp.1266-1279. ⟨10.1021/jm061307x⟩
Article dans une revue istex hal-00164464v1

Linker structure-activity relationships in fluorodeoxyglucose chlorambucil conjugates for tumor-targeted chemotherapy

Valérie Weber , Mostafa El Hilali , Bastien Reux , Eric Debiton , Fernand Leal , et al.
Bioorganic and Medicinal Chemistry, 2017, 25 (20), pp.5692 - 5708. ⟨10.1016/j.bmc.2017.08.043⟩
Article dans une revue hal-01677115v1
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In vitro biological effects of two anti-diabetic medicinal plants used in Benin as folk medicine.

Fifa Td Bothon , Eric Debiton , Felicien Avlessi , Christiane Forestier , Jean-Claude Teulade , et al.
BMC Complementary and Alternative Medicine, 2013, 13 (1), pp.51. ⟨10.1186/1472-6882-13-51⟩
Article dans une revue inserm-00798331v1
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Synthesis and antiproliferative activities of indolin-2-one derivatives bearing amino acid moieties.

Mathieu Sassatelli , Eric Debiton , Bettina Aboab , Michelle Prudhomme , Pascale Moreau
European Journal of Medicinal Chemistry, 2006, 41, pp.709-716. ⟨10.1016/j.ejmech.2006.03.021⟩
Article dans une revue hal-00119556v1

Kinase inhibitory potencies and in vitro antiproliferative activities of N-10 substituted pyrrolo[2,3-a] carbazole derivatives

Rufine Akué-Gédu , Boris Letribot , Emmanuelle Saugues , Eric Debiton , Fabrice Anizon , et al.
Bioorganic and Medicinal Chemistry Letters, 2012, 22, pp.3807-3809
Article dans une revue hal-00711767v1

Synthesis, protein kinase inhibitory potencies and in vitro antiproliferative activities of meridianin derivatives.

Francis Giraud , Georges Alves , Eric Debiton , Lionel Nauton , Vincent Thery , et al.
Journal of Medicinal Chemistry, 2011, 54, pp.4474-4489
Article dans une revue hal-00609607v1

Chemotherapy inhibits skeletal muscle ubiquitin-proteasome-dependent proteolysis.

Thomas Tilignac , Sandrine Temparis , Lydie Combaret , Daniel Taillandier , Marie-Noëlle Pouch , et al.
Cancer Research, 2002, pp.2771-7
Article dans une revue hal-01919675v1

Synthesis and biological activities of 4-substituted pyrrolo[2,3-a]carbazole Pim kinase inhibitors.

Francis Giraud , Rufine Akué-Gédu , Lionel Nauton , Nicolas Candelon , Eric Debiton , et al.
European Journal of Medicinal Chemistry, 2012, 56, pp.225-236
Article dans une revue hal-00786353v1

Synthesis and biological activities of pyrazolo[3,4-g]quinoxaline derivatives

Laurent Gavara , Emmanuelle Saugues , Georges Alves , Eric Debiton , Fabrice Anizon , et al.
European Journal of Medicinal Chemistry, 2010, 45, pp.5520-5526
Article dans une revue hal-00530614v1

Synthèse et activités biologiques des pyrazolo[3,4-g]quinoxalines

Emmanuelle Saugues , Laurent Gavara , Georges Alves , Eric Debiton , Fabrice Anizon , et al.
SYmposium de Chimie Organique en Centre-Auvergne-Limousin VII, Sep 2010, Beaumont-du-Lac, France
Communication dans un congrès hal-00531716v1
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Synthesis and biological activities of aminopyrimidyl-indoles structurally related to meridianins

Rufine Akué-Gédu , Eric Debiton , Yoan Ferandin , Laurent Meijer , Michelle Prudhomme , et al.
Bioorganic and Medicinal Chemistry, 2009, 17, pp.4420-4424
Article dans une revue hal-00392799v1

click chelators for platinum-based anticancer drugs

Aurélie Maisonial , Patrycja Serafin , Mounir Traïkia , Eric Debiton , Vincent Thery , et al.
European Journal of Organic Chemistry, 2008, 2008 (2), pp.298-305. ⟨10.1002/ejic.200700849⟩
Article dans une revue istex hal-00204439v1