Evaluation of borinic acids as new, fast hydrogen peroxide–responsive triggers
Blaise Gatin-Fraudet
,
Roxane Ottenwelter
,
Thomas Le Saux
,
Stéphanie Norsikian
,
Mathilde Pucher
,
et al.
Proceedings of the National Academy of Sciences of the United States of America , 2021, 118 (50), pp.e2107503118.
⟨10.1073/pnas.2107503118⟩
Article dans une revue
hal-03542546v1
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2′-Modified thymidines with bioorthogonal cyclopropene or sydnone as building blocks for copper-free postsynthetic functionalization of chemically synthesized oligonucleotides
Alexandra Bristiel
,
Manon Cadinot
,
Mathieu Pizzonero
,
Frédéric Taran
,
Dominique Urban
,
et al.
Article dans une revue
hal-04281606v1
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Synthesis of chemical tools to label the mycomembrane of corynebacteria using modified iron( iii ) chloride-mediated protection of trehalose
Mathieu Carlier
,
Emilie Lesur
,
Aurélie Baron
,
Aurélie Lemétais
,
Karine Guitot
,
et al.
Article dans une revue
hal-03801948v1
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Mechanistic insights on the inhibition of c5 DNA methyltransferases by zebularine.
Christine Champion
,
Dominique Guianvarc'H
,
Catherine Sénamaud-Beaufort
,
Renata Z Jurkowska
,
Albert Jeltsch
,
et al.
Article dans une revue
hal-00627422v1
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Structure-Guided Optimization of DNA Methyltransferase Inhibitors
Alexandre Erdmann
,
Paola B. Arimondo
,
Dominique Guianvarc'H
MedinaFranco, JL.
EPI-INFORMATICS: DISCOVERY AND DEVELOPMENT OF SMALL MOLECULE EPIGENETIC DRUGS AND PROBES , ELSEVIER ACADEMIC PRESS INC, pp.53-73, 2016, 978-0-12-802808-7.
⟨10.1016/B978-0-12-802808-7.00003-4⟩
Chapitre d'ouvrage
hal-01365334v1
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Sequence-specific base pair mimics are efficient topoisomerase IB inhibitors.
Pierre Vekhoff
,
Maria Duca
,
Dominique Guianvarc'H
,
Rachid Benhida
,
Paola B Arimondo
Article dans une revue
hal-00683339v1
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Combined analysis of DNA methylation and cell cycle in cancer cells
Cecile Desjobert
,
Mounir El Mai
,
Tom Gerard-Hirne
,
Dominique Guianvarc'H
,
Arnaud Carrier
,
et al.
Article dans une revue
hal-01365337v1
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An active site mutant of Escherichia coli cyclopropane fatty acid synthase forms new non-natural fatty acids providing insights on the mechanism of the enzymatic reaction
Guangqi E
,
Thierry Drujon
,
Isabelle Correia
,
Olivier Ploux
,
Dominique Guianvarc'H
Article dans une revue
istex
hal-02467802v1
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Label-free measurement of histone lysine methyltransferases activity by MALDI-TOF mass spectrometry.
Karine Guitot
,
Silvia Scarabelli
,
Thierry Drujon
,
Gérard Bolbach
,
Mehdi Amoura
,
et al.
Article dans une revue
hal-00982533v1
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Identification of Novel Inhibitors of DNA Methylation by Screening of a Chemical Library.
Alexandre Ceccaldi
,
Arumugam Rajavelu
,
Sergey Ragozin
,
Catherine Sénamaud-Beaufort
,
Pavel Bashtrykov
,
et al.
Article dans une revue
hal-00777786v1
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Rapid synthesis of new DNMT inhibitors derivatives of procainamide.
Ludovic Halby
,
Christine Champion
,
Catherine Sénamaud-Beaufort
,
Sophie Ajjan
,
Thierry Drujon
,
et al.
Article dans une revue
istex
hal-00680950v1
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Improving the Selectivity of the Phosphoric Acid β-Elimination on a Biotinylated Phosphopeptide.
Lucrèce Matheron
,
Séverine Clavier
,
Oumar Diebate
,
Philippe Karoyan
,
Gérard Bolbach
,
et al.
Article dans une revue
hal-00730383v1
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Fast Access to 5-Hydroxymethyl Derivatives of 2′-Deoxyuridine Promoted by Acidic Amberlyst 15 Resin
D. Liu
,
O. Monfret
,
Y. Bourdreux
,
D. Urban
,
D. Guianvarc’h
,
et al.
Article dans une revue
hal-04047031v1
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β-Amino acids containing peptides and click-cyclized peptide as β-turn mimics: a comparative study with 'conventional' lactam- and disulfide-bridged hexapeptides.
Maud Larregola
,
Olivier Lequin
,
Philippe Karoyan
,
Dominique Guianvarc'H
,
Solange Lavielle
Article dans une revue
istex
hal-00642781v1
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Hijacking DNA methyltransferase transition state analogues to produce chemical scaffolds for PRMT inhibitors
Ludovic Halby
,
Nils Marechal
,
Dany Pechalrieu
,
Vincent Cura
,
Don-Marc Franchini
,
et al.
Philosophical Transactions of the Royal Society B: Biological Sciences , 2018, 373 (1748), pp.20170072.
⟨10.1098/rstb.2017.0072⟩
Article dans une revue
hal-02094589v1
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Peptidoglycan potentiates the membrane disrupting effect of the carboxyamidated form of DMS-DA6, a Gram-positive selective antimicrobial peptide isolated from Pachymedusa dacnicolor skin
Sébastien Cardon
,
Emmanuelle Sachon
,
Ludovic Carlier
,
Thierry Drujon
,
Astrid Walrant
,
et al.
Article dans une revue
hal-02346622v1
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Synthesis and Evaluation of Analogues of N-Phthaloyl-L-tryptophan (RG108) as Inhibitors of DNA Methyltransferase 1.
Saâdia Asgatay
,
Christine Champion
,
Gaël Marloie
,
Thierry Drujon
,
Catherine Senamaud-Beaufort
,
et al.
Article dans une revue
hal-00920710v1
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PSL Chemical Biology Symposia Third Edition: A Branch of Science in its Explosive Phase
Leeroy Baron
,
Justine Hadjerci
,
Leishemba Thoidingjam
,
Marina Plays
,
Romain Bucci
,
et al.
Article dans une revue
hal-04092530v1
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Challenges in developing novel DNA methyltransferase inhibitors for cancer therapy
Dominique Guianvarc'H
,
Paola B Arimondo
Article dans une revue
hal-01365345v1
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A direct label-free MALDI-TOF mass spectrometry based assay for the characterization of inhibitors of protein lysine methyltransferases
Karine Guitot
,
Thierry Drujon
,
Fabienne Burlina
,
Sandrine Sagan
,
Sandra Beaupierre
,
et al.
Article dans une revue
hal-01536705v1
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First access to a mycolic acid-based bioorthogonal reporter for the study of the mycomembrane and mycoloyltransferases in Corynebacteria
Emilie Lesur
,
Aurélie Baron
,
Christiane Dietrich
,
Marie Buchotte
,
Gilles Doisneau
,
et al.
Article dans une revue
hal-04388218v1
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Probing the in-air growth of large area of 3D functional structures into a 2D supramolecular nanoporous network
Romain Brisse
,
Dominique Guianvarc'H
,
Christelle Mansuy
,
Sandrine Sagan
,
David Kreher
,
et al.
Article dans une revue
hal-01969600v1
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Identification of inhibitors of the E. coli cyclopropane fatty acid synthase from the screening of a chemical library: In vitro and in vivo studies.
Dominique Guianvarc'H
,
Guangqi E
,
Thierry Drujon
,
Camille Rey
,
Qian Wang
,
et al.
Article dans une revue
istex
hal-00294830v1
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Photoactivatable oligonucleotide probes to trap single-stranded DNA binding proteins: Updating the potential of 4-thiothymidine from a comparative study
Tom Gérard-Hirne
,
Frédéric Thiebaut
,
Emmanuelle Sachon
,
Alexandre Désert
,
Thierry Drujon
,
et al.
Article dans une revue
hal-03970700v1
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Preparation of 5‐Hydroxymethyl‐pyrimidine Based Nucleosides: A Reinvestigation
Océane Monfret
,
Dan Liu
,
Paulin Rollando
,
Yann Bourdreux
,
Dominique Urban
,
et al.
Article dans une revue
hal-04281656v1
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An active site mutant of Escherichia coli cyclopropane fatty acid synthase forms new non-natural fatty acids providing insights on the mechanism of the enzymatic reaction.
E. Guangqi
,
Thierry Drujon
,
Isabelle Correia
,
Olivier Ploux
,
Dominique Guianvarc'H
Article dans une revue
istex
hal-00860261v1
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C5-DNA methyltransferase inhibitors: from screening to effects on zebrafish embryo development.
Alexandre Ceccaldi
,
Arumugam Rajavelu
,
Christine Champion
,
Christine Rampon
,
Renata Z. Jurkowska
,
et al.
Article dans une revue
istex
hal-00632453v1
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