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David Bénimélis

37
Documents

Publications

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Synergistic effect of tryptamine-urea derivatives to overcome the chromosomally-mediated colistin resistance in Klebsiella pneumoniae

Chaimae Majdi , Jean Dessolin , David Bénimélis , Catherine Dunyach-Rémy , Alix Pantel
Bioorganic and Medicinal Chemistry, 2024, 100, pp.117604. ⟨10.1016/j.bmc.2024.117604⟩
Article dans une revue hal-04419733v1
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Antibacterial Activity and Untargeted Metabolomics Profiling of Acalypha arvensis Poepp

V. Thesnor , Roland Molinié , Ryland Giebelhaus , A. Paulina de la Mata Espinosa , James Harynuk
Molecules, 2023, 28 (23), pp.7882. ⟨10.3390/molecules28237882⟩
Article dans une revue hal-04419754v1
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Microwave-assisted synthesis of new environmentally friendly biodegradable and antibacterial heterocycles

Miyanou Rosales-Hurtado , Valentin Duvauchelle , David Bénimélis , Maya Ogawa-Okada , Naofumi Yamamoto
Environmental Chemistry Letters, 2022, ⟨10.1007/s10311-022-01522-w⟩
Article dans une revue hal-03805578v1
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Isolation and Identification of Flavones Responsible for the Antibacterial Activities of Tillandsia Bergeri Extracts.

Mame-Marietou Lo , Zohra Benfodda , Catherine Dunyach-Rémy , David Bénimélis , Romain Roulard
ACS Omega, 2022, 7 (40), pp.35851--35862. ⟨10.1021/acsomega.2c04195⟩
Article dans une revue hal-03823329v1
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Catalyst-Free Site Selective Hydroxyalkylation of 5-Phenylthiophen-2-amine with α-Trifluoromethyl Ketones through Electrophilic Aromatic Substitution

Valentin Duvauchelle , David Bénimélis , Patrick Meffre , Zohra Benfodda
Molecules, 2022, 27 (3), pp.925. ⟨10.3390/molecules27030925⟩
Article dans une revue hal-03550954v1
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Extraction and Identification of Volatile Organic Compounds in Scentless Flowers of 14 Tillandsia Species Using HS-SPME/GC-MS

Alexandre Gonzalez , Zohra Benfodda , David Bénimélis , Jean-Xavier Fontaine , Roland Molinié
Metabolites, 2022, 12 (9), pp.628. ⟨10.3390/metabo12070628⟩
Article dans une revue hal-03725030v1
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Development of a HS-SPME/GC-MS Method for the Extraction and Identification of the Volatile Compounds Emitted by Flowers of Tillandsia xiphioides

Mame-Marietou Lo , Zohra Benfodda , David Bénimélis , Jean-Xavier J.-X. Fontaine , Roland Molinié
ACS Omega, 2021, 6 (19), pp.12691-12698. ⟨10.1021/acsomega.1c00917⟩
Article dans une revue hal-03243914v1
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Synthesis, Structure Elucidation, Antibacterial Activities, and Synergistic Effects of Novel Juglone and Naphthazarin Derivatives Against Clinical Methicillin-Resistant Staphylococcus aureus Strains

Valentin Duvauchelle , Chaimae Majdi , David Bénimélis , Catherine Dunyach-Remy , Patrick Meffre
Frontiers in Chemistry, 2021, 9, ⟨10.3389/fchem.2021.773981⟩
Article dans une revue hal-03446358v1
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Extraction and Identification of Volatile Organic Compounds Emitted by Fragrant Flowers of Three Tillandsia Species by HS-SPME/GC-MS

Mame-Marietou Lo , Zohra Benfodda , David Bénimélis , Jean-Xavier Fontaine , Roland Molinié
Metabolites, 2021, 11 (9), pp.594. ⟨10.3390/metabo11090594⟩
Article dans une revue hal-03334373v1
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Critical parameters in surface plasmon resonance biosensor development the interaction between estrogen receptor and estrogen response element as model

Sandrine Bayle , David Bénimèlis , Joel Chopineau , Benoit Roig , Denis Habauzit
Biochimie, 2020, 171-172, pp.12-20. ⟨10.1016/j.biochi.2020.01.015⟩
Article dans une revue hal-02470894v1
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Ethynylglycine synthon, a useful precursor for the synthesis of biologically active compounds: an update. Part II: synthetic uses of ethynylglycine synthon

Zohra Benfodda , David Bénimélis , Gianna Reginato , Patrick Meffre
Amino Acids, 2018, 50 (10), pp.1307-1328. ⟨10.1007/s00726-018-2628-1⟩
Article dans une revue hal-01859944v1
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Synthesis of 1,4-disubstituted 1,2,3-triazole Derivatives Using Click Chemistry and their Src Kinase Activities

Alexandre Lebeau , Cyril Abrioux , David Bénimèlis , Zohra Benfodda , Patrick Meffre
Medicinal Chemistry, 2017, Medicinal Chemistry, 13, pp.40-48. ⟨10.2174/1573406412666160404125718⟩
Article dans une revue hal-01495029v1
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Synthesis of a Novel Rhizobitoxine-Like Triazole-Containing Amino Acid

Thibaut Boibessot , David Bénimélis , Marion Jean , Zohra Benfodda , Patrick Meffre
SYNLETT, 2016, 27 (19), pp.2685-2688. ⟨10.1055/s-0036-1588300⟩
Article dans une revue hal-01404310v1
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The Rational Design, Synthesis, and Antimicrobial Properties of Thiophene Derivatives That Inhibit Bacterial Histidine Kinases

Thibaut Boibessot , Christopher Zschiedrich , Alexandre Lebeau , David Bénimélis , Catherine Dunyach-Remy
Journal of Medicinal Chemistry, 2016, 59, pp.8830-8847. ⟨10.1021/acs.jmedchem.6b00580⟩
Article dans une revue hal-01543599v1
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Advances in the synthesis of α‑quaternary α‑ethynyl α‑amino acids

Thibaut Boibessot , David Bénimélis , Patrick Meffre , Zohra Benfodda
Amino Acids, 2016, 48 (9), pp.2081-2101. ⟨10.1007/s00726-016-2276-2⟩
Article dans une revue hal-01540958v1
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Ethynylglycine synthon, a useful precursor for the synthesis of biologically active compounds: an update

Zohra Benfodda , David Bénimélis , Gianna Reginato , Patrick Meffre
Amino Acids, 2015, 47 (2), pp.271-279. ⟨10.1007/s00726-014-1902-0⟩
Article dans une revue hal-01676812v1
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Synthesis, resolution, and determination of absolute configuration of protected α-ethynylphenylalanine enantiomers

Z Benfodda , David Bénimèlis , Marion Jean , Jean-Valère Naubron , Valerie Rolland
Amino Acids, 2015, 47 (5), pp.899-907. ⟨10.1007/s00726-015-1917-1⟩
Article dans une revue hal-02002634v1
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Impact of biochemical design on estrogen receptor/estrogen response element interaction by surface plasmon resonance technology

Denis Habauzit , Sandrine Bayle , David Benimelis , Joel Chopineau , Benoît Roig
Archives of Biochemistry and Biophysics, 2014, 541, pp.61-66. ⟨10.1016/j.abb.2013.11.006⟩
Article dans une revue hal-00936061v1

Synthesis of cis-5-Trifluoromethylproline from L-Glutamic Acid

Stéphanie Ortial , Rajesh Dave , Zohra Benfodda , David Bénimélis , Patrick Meffre
SYNLETT, 2013, 2014 (25), pp.0569-0573. ⟨10.1055/s-0033-1340553⟩
Article dans une revue hal-00969187v1

Analysis of the Volatile Organic Compounds of Tillandsia flowers by HS-SPME/GC-MS

Alexandre Gonzalez , Zohra Benfodda , David Bénimélis , Jean-Xavier J.-X. Fontaine , Roland Molinié
Analytics 2022, Sep 2022, Nantes, France
Communication dans un congrès hal-03806502v1

Rational design, synthesis and antimicrobial properties of thiophene derivatives that inhibit bacterial histidine kinases

Zohra Benfodda , Miyanou Rosales-Hurtado , Thibaut Boibessot , Christopher Zschiedrich , Alexandre Lebeau
2nd international conference Antimicrobial and antibacterial Istanbul Turkey, Nov 2019, Istanbul, Turkey
Communication dans un congrès hal-02400581v1

Rational design, synthesis and antimicrobial properties of thiophene derivatives that inhibit bacterial histidine kinases

Zohra Benfodda , Thibaut Boibessot , Christopher Zschiedrich , Alexandre Lebeau , David Bénimèlis
24th ISCB international conference-Frontier research in chemistry&biology interface, Jan 2018, JAIPUR, India
Communication dans un congrès hal-01998540v1

Synthesis of 5-trifluoromethylproline from L-glutamic acid

Stéphanie Ortial , Rajesh Dave , Zohra Benfodda , David Bénimèlis , Patrick Meffre
14th International Congress on Amino Acids, Peptides and Proteins, Aug 2015, Wien, Austria. pp.615-636, ⟨10.1007/s00726-015-2160-5⟩
Communication dans un congrès hal-02010135v1

Addendum to Abstracts presented at the 14th International Congress on Amino Acids, Peptides and Proteins

Patrick Meffre , Zohra Benfodda , David Bénimèlis , Stéphanie Ortial , Valerie Rolland
14th International Congress on Amino Acids, Peptides and Proteins, Aug 2015, Vienna, Austria. pp.615-636
Communication dans un congrès hal-02002708v1

Synthesis of acetylenic analogue of phenylalanine.

Zohra Benfodda , Stéphanie Ortial , David Bénimélis , Valerie Rolland , Patrick Meffre
13th International Congress on Amino acids, peptides and proteins, Oct 2013, Galvestion (Texas), United States. pp.611, ⟨10.1007/s00726-013-1540-y⟩
Communication dans un congrès hal-00993416v1

New developments in the synthesis of acetylenic analogues of glutamate

Patrick Meffre , Zohra Benfodda , David Bénimélis , Valérie Rolland , Francine C. Acher
12 th International Congress on Amino Acids, Peptides and Proteins, Aug 2011, Beijing, China. pp.S79, ⟨10.1007/s00726-011-0955-6⟩
Communication dans un congrès hal-00621161v1

Synthesis of acetylenic analogues of glutamate

Zohra Benfodda , David Bénimèlis , Patrick Meffre , Francine C. Acher
10th International Congress on amino acids and proteins, Aug 2007, Kallithea, Greece
Communication dans un congrès hal-01998510v1

Synthesis of acetylenic analogues of glutamate

Patrick Meffre , Zohra Benfodda , David Bénimèlis , Guillaume Vierling , Francine C. Acher
10th International Congress on Amino Acids and Proteins (ICAAP), Aug 2007, Kalithea, Chalkidiki, Greece. pp.I-LXX, ⟨10.1007/s00726-007-0578-0⟩
Communication dans un congrès hal-02010124v1
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Synergistic Effects of Novel Naphthoquinone Derivatives Against Clinical Methicilin-Resistant Staphylococcus aureus Strain

Valentin Duvauchelle , Chaimae Majdi , David Bénimélis , Catherine Dunyach-Rémy , Patrick Meffre
REncontres en Chimie Organique Biologique 18 (RECOB18), Mar 2022, Aussois, France.
Poster de conférence hal-03700525v1
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Synthesis and biological evaluations of new families of histidine kinases inhibitors

Valentin Duvauchelle , Miyanou Rosales-Hurtado , Thibaut Boibessot , David Bénimèlis , Catherine Dunyach-Remy
GSO-JMJC-JED2019, Oct 2019, Montpellier, France.
Poster de conférence hal-02333120v1

Design and synthesis of novel HLM 006474 derivatives.

Zohra Benfodda , Gerardo Cebrian Cebrian-Torrejon , Bourguet Romane , Sciortino Giuseppe , Jean-Didier Maréchal
24th ISCB international conference-Frontier research in chemistry&biology interface., Jan 2018, JAIPUR, India
Poster de conférence hal-01998366v1
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Synthesis of thiophene derivatives: Potential new inhibitors of histidine kinases

Miyanou Rosales-Hurtado , Thibaut Boibessot , Christopher Zschiedrich , Alexandre Lebeau , David Bénimélis
Rencontres en Chimie Organique Biologique (Recob 17), Mar 2018, Aussois, France.
Poster de conférence hal-01997587v1

Synthesis of Novel Triazole Amino Acids Analogues of Natural Amino Acids

Patrick Meffre , Thibaut Boibessot , David Bénimèlis , Zohra Benfodda
20th European symposium on Organic Chemistry (ESOC), Jul 2017, Cologne, Germany
Poster de conférence hal-02011261v1

Synthesis of triazole amino acids

Zohra Benfodda , Thibaut Boibessot , Alexandre Lebeau , David Bénimèlis , Patrick Meffre
14th International Congress on Amino Acids, Peptides and Proteins, Aug 2015, Vienne, Austria
Poster de conférence hal-01998273v1

Design and synthesis of 1,4-disubstituted 1,2,3-triazole derivatives as Histidine Kinase inhibitor.

Zohra Benfodda , Alexandre Lebeau , David Bénimèlis , Hendrik Szurmant , Patrick Meffre
77th Harden Conference: Two Component Signalling in Bacteria: Integrating Approaches and Science, Aug 2015, Warwickshire, United Kingdom
Poster de conférence hal-01998338v1

Synthesis of ethynyl phenylalanine

Zohra Benfodda , David Bénimèlis , Valérie Rolland , Patrick Meffre
The 5th European Chemistry Congress, Aug 2014, Istanbul, Turkey
Poster de conférence hal-01998193v1

Synthesis of ethynyl phenylalanine

Zohra Benfodda , David Benimelis , Valerie Rolland , Thibaut Boibessot , Patrick Meffre
21ème journée de l’Institut de Recherche Pierre Fabre (IRPF) de chimie. Chambre de commerce et d’industrie de Castres, Sep 2014, Castres, France
Poster de conférence hal-01998205v1