Christophe Mallet

Documents

Publications

	GPER involvement in inflammatory pain Baptiste Jouffre , Alexandre Acramel , Yves Jacquot , Laurence Daulhac , Christophe Mallet Steroids, 2023, 200, pp.109311. ⟨10.1016/j.steroids.2023.109311⟩ Article dans une revue hal-04337675v1
	An Updated Review on the Metabolite (AM404)-Mediated Central Mechanism of Action of Paracetamol (Acetaminophen): Experimental Evidence and Potential Clinical Impact Christophe Mallet , Jules Desmeules , Rassa Pegahi , Alain Eschalier Journal of Pain Research, 2023, 16, pp.1081 - 1094. ⟨10.2147/jpr.s393809⟩ Article dans une revue hal-04337681v1
	Identification of a human estrogen receptor α tetrapeptidic fragment with dual antiproliferative and anti-nociceptive action Baptiste Jouffre , Alexandre Acramel , Mathilde Belnou , Maria Francesca Santolla , Marianna Talia Scientific Reports, 2023, 13 (1), pp.1326. ⟨10.1038/s41598-023-28062-9⟩ Article dans une revue hal-04087799v1
	Role of T CD4+ cells, macrophages, C-low threshold mechanoreceptors and spinal Cav3.2 channels in inflammation and related pain-like symptoms in murine inflammatory models Elodie Picard , Nicolas Kerckhove , Amaury François , Ludivine Boudieu , Elisabeth Billard British Journal of Pharmacology, 2023, 180 (4), pp.385-400. ⟨10.1111/bph.15956⟩ Article dans une revue hal-03790651v1
	Design, synthesis and biological evaluation of conformationnally-restricted analogues of E7010 as inhibitors of tubulin assembly (ITA) and vascular disrupting agents (VDA) Vassili Prudhomme , Mélissa Cucca , Lionel Nauton , Elsa Andrieu , Mathilde Fereyrolles European Journal of Medicinal Chemistry, 2022, 244, pp.114809. ⟨10.1016/j.ejmech.2022.114809⟩ Article dans une revue hal-03959739v1
	Centrally expressed Cav3.2 T-type calcium channel is critical for the initiation and maintenance of neuropathic pain Sophie L Fayad , Guillaume Ourties , Benjamin Le Gac , Baptiste Jouffre , Sylvain Lamoine eLife, 2022, 11, pp.e79018. ⟨10.7554/elife.79018⟩ Article dans une revue hal-03942925v1
	Centrally expressed Cav3.2 T-type calcium channel is critical for the initiation and maintenance of neuropathic pain Sophie Fayad , Guillaume Ourties , Benjamin Le Gac , Baptiste Jouffre , Sylvain Lamoine eLife, 2022, 11, ⟨10.7554/eLife.79018⟩ Article dans une revue hal-04256569v1
	L’évaluation de la douleur chez l’animal de laboratoire Christine Courteix , Alain Eschalier , Christophe Mallet Douleur et Analgésie, 2021, 34 (2), pp.114-122. ⟨10.3166/dea-2021-0145⟩ Article dans une revue hal-03418812v1
	Paracetamol analogues conjugated by FAAH induce TRPV1-mediated antinociception without causing acute liver toxicity Johan Å.Nilsson , Christophe Mallet , Kiseko Shionoya , Anders Blomgren , Anders Sundin European Journal of Medicinal Chemistry, 2021, 213, pp.113042. ⟨10.1016/j.ejmech.2020.113042⟩ Article dans une revue hal-04256629v1
	The Antitumor Peptide ERα17p Exerts Anti-Hyperalgesic and Anti-Inflammatory Actions Through GPER in Mice Christophe Mallet , Ludivine Boudieu , Sylvain Lamoine , Catherine Coudert , Yves Jacquot Frontiers in Endocrinology, 2021, 12, ⟨10.3389/fendo.2021.578250⟩ Article dans une revue hal-04256623v1
	Paracetamol is a centrally acting analgesic using mechanisms located in the periaqueductal grey David André Barrière , Fawzi Boumezbeur , Romain Dalman , Roberto Cadeddu , Damien Richard Richard British Journal of Pharmacology, 2020, 177 (8), pp.1773-1792. ⟨10.1111/bph.14934⟩ Article dans une revue hal-02380187v1
	Ethosuximide improves chronic pain-induced anxiety- and depression-like behaviors Nicolas Kerckhove , Ludivine Boudieu , Guillaume Ourties , Justine Bourdier , Laurence Daulhac European Neuropsychopharmacology, 2019, 29, pp.1419 - 1432. ⟨10.1016/j.euroneuro.2019.10.012⟩ Article dans une revue hal-03488870v1
	Inhibition of Cav3.2 calcium channels: A new target for colonic hypersensitivity associated with low‐grade inflammation Elodie Picard , Frédéric Antonio Carvalho , Francina Agosti , Emmanuel Bourinet , Denis Ardid British Journal of Pharmacology, 2019, 176 (7), pp.950-963. ⟨10.1111/bph.14608⟩ Article dans une revue hal-04317223v1
	The Peptide ERα17p Is a GPER Inverse Agonist that Exerts Antiproliferative Effects in Breast Cancer Cells Rosamaria Lappano , Christophe Mallet , Bruno Rizzuti , Fedora Grande , Giulia Raffaella Galli Cells, 2019, Molecular and Cellular Mechanisms of Cancers: Breast Cancer, 8 (6), pp.590. ⟨10.3390/cells8060590⟩ Article dans une revue hal-02273130v1
	A tetrapeptide class of biased analgesics from an Australian fungus targets the µ-opioid receptor Zoltan Dekan , Setareh Sianati , Arsalan Yousuf , Katy Sutcliffe , Alexander Gillis Proceedings of the National Academy of Sciences of the United States of America, 2019, 116 (44), pp.22353-22358. ⟨10.1073/pnas.1908662116⟩ Article dans une revue hal-04257287v1
	Optimization of the synthesis of a key intermediate for the preparation of glucocorticoids Romain Jouve , Vincent Thery , Sylvie Ducki , Julie Helfenbein , Christophe Thiery Steroids, 2018, 137, pp.14 - 21. ⟨10.1016/j.steroids.2018.06.007⟩ Article dans une revue hal-01875170v1
	Assessment of the effectiveness and safety of Ethosuximide in the Treatment of non-Diabetic Peripheral Neuropathic Pain: EDONOT—protocol of a randomised, parallel, controlled, double-blinded and multicentre clinical trial Nicolas Kerckhove , Christophe Mallet , Bruno Pereira , Chouki Chenaf , Christian Duale BMJ Open, 2016, 6 (12), pp.e013530. ⟨10.1136/bmjopen-2016-013530⟩ Article dans une revue hal-04337204v1
	FAAH inhibitors in the limelight, but regrettably Christophe Mallet , Claude Dubray , Christian Dualé International Journal of Clinical Pharmacology and Therapeutics, 2016, 54 (07), pp.498 - 501. ⟨10.5414/cp202687⟩ Article dans une revue hal-04337687v1
	Colonic overexpression of the T‐type calcium channel Cav 3.2 in a mouse model of visceral hypersensitivity and in irritable bowel syndrome patients J. Scanzi , A. Accarie , E. Muller , Bruno Pereira , Y. Aissouni Neurogastroenterology & Motility, 2016, 28 (11), pp.1632-1640. ⟨10.1111/nmo.12860⟩ Article dans une revue hal-04317301v1
	Supra-spinal FAAH is required for the analgesic action of paracetamol in an inflammatory context Romain Dalmann , Laurence Daulhac , Myriam Antri , Alain Eschalier , Christophe Mallet Neuropharmacology, 2015, 91, pp.63-70. ⟨10.1016/j.neuropharm.2014.11.006⟩ Article dans une revue hal-04326283v1
	Cav3.2 calcium channels: the key protagonist of the supraspinal effect of paracetamol Nicolas Kerckhove , Christophe Mallet , Amaury François , Mathieu Boudes , Jean Chemin Pain, 2014, 155 (4), pp.764-772. ⟨10.1016/j.pain.2014.01.015⟩ Article dans une revue hal-02356344v1
	Prise en charge médicamenteuse de la douleur Christophe Mallet , Chouki Chenaf Cerveau & psycho. L'essentiel, 2014, 17 Article dans une revue hal-04273988v1
	Fatty Acid Amide Hydrolase-Dependent Generation of Antinociceptive Drug Metabolites Acting on TRPV1 in the Brain David A Barrière , Christophe Mallet , Anders Blomgren , Charlotte Simonsen , Laurence Daulhac PLoS ONE, 2013, 8 (8), pp.e70690. ⟨10.1371/journal.pone.0070690⟩ Article dans une revue hal-04337223v1
	Monoacylglycerols Activate TRPV1 – A Link between Phospholipase C and TRPV1 Peter M Zygmunt , Anna Ermund , Pouya Movahed , David A Andersson , Charlotte Simonsen PLoS ONE, 2013, 8 (12), pp.e81618. ⟨10.1371/journal.pone.0081618⟩ Article dans une revue hal-04337227v1
	Le paracétamol : un ancêtre plein d’avenir Christophe Mallet , David Barrière , Alain Eschalier Therapies, 2012, 67 (4), pp.277-281. ⟨10.2515/therapie/2012039⟩ Article dans une revue hal-04337690v1
	Mise au point sur les mécanismes de l'action antalgique du paracétamol Christophe Mallet , Alain Eschalier Urgence Pratique, 2012, 115, pp.29-31 Article dans une revue hal-04273935v1
	Drug-induced GABA transporter currents enhance GABA release to induce opioid withdrawal behaviors Elena Bagley , Jennifer Hacker , Vladimir Chefer , Christophe Mallet , Gavan Mcnally Nature Neuroscience, 2011, 14 (12), pp.1548-1554. ⟨10.1038/nn.2940⟩ Article dans une revue hal-04337230v1
	Le paracétamol, de nouvelles cibles pour un vieux médicament David André Barrière , Christophe Mallet , Alain Eschalier La Lettre de l’Institut UPSA de la Douleur, 2010, 33 Article dans une revue hal-04273458v1
	TRPV1 in Brain Is Involved in Acetaminophen-Induced Antinociception Christophe Mallet , David Barrière , Anna Ermund , Bo Jönsson , Alain Eschalier PLoS ONE, 2010, 5 (9), pp.e12748. ⟨10.1371/journal.pone.0012748⟩ Article dans une revue hal-04326308v1
	Endocannabinoids Can Open the Pain Gate Macdonald Christie , Christophe Mallet Science Signaling, 2009, 2 (88), ⟨10.1126/scisignal.288pe57⟩ Article dans une revue hal-04337579v1
	Endocannabinoid and serotonergic systems are needed for acetaminophen-induced analgesia Christophe Mallet , Laurence Daulhac , Jérôme Bonnefont , Catherine Ledent , Monique Etienne Pain, 2008, 139 (1), pp.190-200. ⟨10.1016/j.pain.2008.03.030⟩ Article dans une revue hal-04326295v1
	Acetaminophen recruits spinal p42/p44 mAPKs and GH/IGF-1 receptors to produce analgesia via the serotonergic system Jérôme Bonnefont , Laurence Daulhac , Monique Etienne , Eric Chapuy , Christophe Mallet Molecular Pharmacology, 2007, 71 (2), pp.407-415. ⟨10.1124/mol.106.025775⟩ Article dans une revue hal-02659399v1
	Diabetes-Induced Mechanical Hyperalgesia Involves Spinal Mitogen-Activated Protein Kinase Activation in Neurons and Microglia via N -Methyl-D-aspartate-Dependent Mechanisms Laurence Daulhac , Christophe Mallet , Christine Courteix , Monique Etienne , Eliane Duroux Molecular Pharmacology, 2006, 70 (4), pp.1246-1254. ⟨10.1124/mol.106.025478⟩ Article dans une revue hal-04326273v1

	Paracetamol is a centrally acting analgesic using mechanisms located in the periaqueductal grey Christophe Mallet , David André Barrière , Fouad Boumezbeur , Romain Dalmann , Roberto Cadeddu Annual Meeting of French Society of Pharmacology and Therapeutics, Jun 2021, Online, France Communication dans un congrès hal-03745618v1

	Involvment of Cav3.2 calcium channels in oesteoarthritis pain Guillaume Ourties , Laurence Daulhac , Alain Eschalier , Christophe Mallet EFIC pain school, Jun 2019, cracovie, Poland Poster de conférence hal-02363984v1

	Traitements de la douleur, Approche pharmacologique Nicolas Authier , Bénédicte Eschalier , Chouki Chenaf , Marie Zenut , Christophe Mallet Traité de Médecine (5ème édition), TDM, pp.S10-P01-C11, 2018, 9782901094012 Chapitre d'ouvrage hal-04273871v1
	Pharmacology and Mechanism of Action of Acetaminophen Christophe Mallet , Alain Eschalier Pharmacology of Pain, IASP press, 2015, 0931092787 Chapitre d'ouvrage hal-04337640v1

	Centrally expressed Cav3.2 T-type calcium channel is critical for the initiation and maintenance of neuropathic pain Sophie L Fayad , Guillaume Ourties , Benjamin Le Gac , Baptiste Jouffre , Sylvain Lamoine 2022 Pré-publication, Document de travail hal-03746638v1

Christophe Mallet

Publications

GPER involvement in inflammatory pain

An Updated Review on the Metabolite (AM404)-Mediated Central Mechanism of Action of Paracetamol (Acetaminophen): Experimental Evidence and Potential Clinical Impact

Identification of a human estrogen receptor α tetrapeptidic fragment with dual antiproliferative and anti-nociceptive action

Role of T CD4+ cells, macrophages, C-low threshold mechanoreceptors and spinal Cav3.2 channels in inflammation and related pain-like symptoms in murine inflammatory models

Design, synthesis and biological evaluation of conformationnally-restricted analogues of E7010 as inhibitors of tubulin assembly (ITA) and vascular disrupting agents (VDA)

Centrally expressed Cav3.2 T-type calcium channel is critical for the initiation and maintenance of neuropathic pain

Centrally expressed Cav3.2 T-type calcium channel is critical for the initiation and maintenance of neuropathic pain

L’évaluation de la douleur chez l’animal de laboratoire

Paracetamol analogues conjugated by FAAH induce TRPV1-mediated antinociception without causing acute liver toxicity

The Antitumor Peptide ERα17p Exerts Anti-Hyperalgesic and Anti-Inflammatory Actions Through GPER in Mice

Paracetamol is a centrally acting analgesic using mechanisms located in the periaqueductal grey

Ethosuximide improves chronic pain-induced anxiety- and depression-like behaviors

Inhibition of Cav3.2 calcium channels: A new target for colonic hypersensitivity associated with low‐grade inflammation

The Peptide ERα17p Is a GPER Inverse Agonist that Exerts Antiproliferative Effects in Breast Cancer Cells

A tetrapeptide class of biased analgesics from an Australian fungus targets the µ-opioid receptor

Optimization of the synthesis of a key intermediate for the preparation of glucocorticoids

Assessment of the effectiveness and safety of Ethosuximide in the Treatment of non-Diabetic Peripheral Neuropathic Pain: EDONOT—protocol of a randomised, parallel, controlled, double-blinded and multicentre clinical trial

FAAH inhibitors in the limelight, but regrettably

Colonic overexpression of the T‐type calcium channel Cav 3.2 in a mouse model of visceral hypersensitivity and in irritable bowel syndrome patients

Supra-spinal FAAH is required for the analgesic action of paracetamol in an inflammatory context

Cav3.2 calcium channels: the key protagonist of the supraspinal effect of paracetamol

Prise en charge médicamenteuse de la douleur

Fatty Acid Amide Hydrolase-Dependent Generation of Antinociceptive Drug Metabolites Acting on TRPV1 in the Brain

Monoacylglycerols Activate TRPV1 – A Link between Phospholipase C and TRPV1

Le paracétamol : un ancêtre plein d’avenir

Mise au point sur les mécanismes de l'action antalgique du paracétamol

Drug-induced GABA transporter currents enhance GABA release to induce opioid withdrawal behaviors

Le paracétamol, de nouvelles cibles pour un vieux médicament

TRPV1 in Brain Is Involved in Acetaminophen-Induced Antinociception

Endocannabinoids Can Open the Pain Gate

Endocannabinoid and serotonergic systems are needed for acetaminophen-induced analgesia

Acetaminophen recruits spinal p42/p44 mAPKs and GH/IGF-1 receptors to produce analgesia via the serotonergic system

Diabetes-Induced Mechanical Hyperalgesia Involves Spinal Mitogen-Activated Protein Kinase Activation in Neurons and Microglia via N -Methyl-D-aspartate-Dependent Mechanisms

Paracetamol is a centrally acting analgesic using mechanisms located in the periaqueductal grey

Involvment of Cav3.2 calcium channels in oesteoarthritis pain

Traitements de la douleur, Approche pharmacologique

Pharmacology and Mechanism of Action of Acetaminophen

Centrally expressed Cav3.2 T-type calcium channel is critical for the initiation and maintenance of neuropathic pain