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Pyridine-3,4-dicarboximide as starting material for the total synthesis of the natural product eupolauramine and its isomer iso-eupolauramine endowed with anti-tubercular activities

 Gildas Perdigao , Céline Deraeve , Georgia Mori , Maria Rosalia Pasca , G. Pratviel , et al.
Tetrahedron, 2015, 71 (10), pp.1555-1559. ⟨10.1016/j.tet.2015.01.034⟩
Article dans une revue hal-01920329v1

Synthesis, oxidation potential and anti–mycobacterial activity of isoniazid and analogues: Insights into the molecular isoniazid activation mechanism

 Julie Laborde , Céline Deraeve , Léa Lecoq , Alix Sournia-Saquet , Jean-Luc Stigliani , et al.
ChemistrySelect, 2016, 1 (2), pp.172-179. ⟨10.1002/slct.201600040⟩
Article dans une revue hal-01929903v1

Synthesis and mechanistic investigation of iron(II) complexes of isoniazid and derivatives as a redox-mediated activation strategy for anti-tuberculosis therapy

 Julie Laborde , Céline Deraeve , Francisca Gilmara De Mesquita Vieira , Alix Sournia-Saquet , Lionel Rechignat , et al.
Journal of Inorganic Biochemistry, 2018, 179, pp.71-81. ⟨10.1016/j.jinorgbio.2017.11.013⟩
Article dans une revue hal-01952877v1

Preparation and study of new poly-8-hydroxyquinoline chelators for an anti-alzheimer strategy

 Christophe Boldron , Céline Deraeve , Heinz Gornitzka , B. Meunier , Marguerite Pitie , et al.
Chemistry - A European Journal, 2008, pp.682-696
Article dans une revue hal-00371845v1

Terpyridine-Based Heteroditopic Ligand for Ru(II)Ln(3)(III) Metallostar Architectures (Ln = Gd, Eu, Nd, Yb) with MRI/Optical or Dual-Optical Responses

 Alexandre Boulay , Céline Deraeve , Luce Vander Elst , Nadine Leygue , Olivier Maury , et al.
Inorganic Chemistry, 2015, 54 (4), pp.1414-1425. ⟨10.1021/ic502342x⟩
Article dans une revue hal-01234063v1
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Pd-catalyzed C–C and C–N cross-coupling reactions in 2-aminothieno[3,2- d ]pyrimidin-4(3 H )-one series for antiplasmodial pharmacomodulation

 Romain Mustière , Prisca Lagardère , Sébastien Hutter , Céline Deraeve , Florian Schwalen , et al.
RSC Advances, 2022, 12 (31), pp.20004-20021. ⟨10.1039/D2RA01687G⟩
Article dans une revue hal-03726141v1
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Synthèse et évaluation biologique de dérivés polyquinoléine chélateurs d'ions métalliques en relation avec la maladie d'Alzheimer

 Céline Deraeve
Autre. Université Paul Sabatier - Toulouse III, 2006. Français. ⟨NNT : ⟩
Thèse tel-00142741v1
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N-heterocyclic carbene-iridium complexes as photosensitizers for in vitro photodynamic therapy to trigger non-apoptotic cell death in cancer cells

 Xing Wang , Chen Zhang , Ryma Madji , Camille Voros , Serge Mazères , et al.
Molecules, 2023, 28 (2), pp.691. ⟨10.3390/molecules28020691⟩
Article dans une revue hal-03870710v2
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Novel molecule combinations and corresponding hybrids targeting artemisinin-resistant Plasmodium falciparum parasites

 Manel Ouji , Michel Nguyen , Romain Mustière , Tony Jimenez , Jean-Michel Augereau , et al.
Bioorganic and Medicinal Chemistry Letters, 2021, 39, pp.127884. ⟨10.1016/j.bmcl.2021.127884⟩
Article dans une revue hal-03170976v1

Isoniazid: an update on the multiple mechanisms for a singular action

 Vania Bernardes-Génisson , Céline Deraeve , Aurélien Chollet , Jean Bernadou , G. Pratviel
Current Medicinal Chemistry, 2013, 20 (35), pp.4370-85. ⟨10.2174/15672050113109990203⟩
Article dans une revue hal-00993170v1

Psoromic Acid is a Selective and Covalent Rab-Prenylation Inhibitor Targeting Autoinhibited RabGGTase

 Céline Deraeve , Zhong Guo , Robin Bon , Wulf Blankenfeldt , Raffaella Dilucrezia , et al.
Journal of the American Chemical Society, 2012, 134 (17), pp.7384-7391. ⟨10.1021/ja211305j⟩
Article dans une revue hal-02909744v1

Ethionamide biomimetic activation and an unprecedented mechanism for its conversion into active and non-active metabolites

 Julie Laborde , Céline Deraeve , Carine Guyard-Duhayon , G. Pratviel , Vania Bernardes-Génisson
Organic & Biomolecular Chemistry, 2016, 14 (37), pp.8848-8858. ⟨10.1039/C6OB01561A⟩
Article dans une revue hal-01929907v1

Preparation of Cyclo-Phen-Type Ligands : Chelators of Metal ions as potential therapeutic agents in the treatment of neurodegenerative diseases

 B. Meunier , Christophe Boldron , Marguerite Pitie , Céline Deraeve , Ingrid van Der Auwera , et al.
ChemBioChem, 2005, 6, pp.1976-1980
Article dans une revue hal-00361604v1
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Synthesis, Characterization, and Antileishmanial Activity of Neutral Gold(I) Complexes with N-heterocyclic Carbene Ligands Bearing Sulfur-Containing Side Arms

 Soumia Ftouh , Sandra Bourgeade-Delmas , Mohamed Belkadi , Céline Deraeve , Catherine Hemmert , et al.
Organometallics, 2021, 40 (10), pp.1466-1473. ⟨10.1021/acs.organomet.1c00113⟩
Article dans une revue hal-03233814v1
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New 8-Nitroquinolinone Derivative Displaying Submicromolar in Vitro Activities against Both Trypanosoma brucei and cruzi

 Julien Pedron , Clotilde Boudot , Jean-Yves Brossas , Emilie Pinault , Sandra Bourgeade-Delmas , et al.
ACS Medicinal Chemistry Letters, 2020, 11 (4), pp.464-472. ⟨10.1021/acsmedchemlett.9b00566⟩
Article dans une revue hal-02476867v1

Insights into the cholecystokinin 2 receptor binding site and processes of activation.

 Michaël Paillasse , Céline Deraeve , Philippe de Médina , Loubna Mhamdi , Gilles Favre , et al.
Molecular Pharmacology, 2006, 70 (6), pp.1935-45. ⟨10.1124/mol.106.029967⟩
Article dans une revue inserm-00519168v1

Update of antitubercular prodrugs from a molecular perspective: Mechanisms of action, bioactivation pathways, and associated resistance

 Julie Laborde , Céline Deraeve , Vania Bernardes-Génisson
ChemMedChem, 2017, 12 (20), pp.1657-1676. ⟨10.1002/cmdc.201700424⟩
Article dans une revue hal-01939397v1
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