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Crosslinking photosensitized by a ruthenium chelate as a tool for labeling and topographical studies of G-protein-coupled receptors

I. Duroux-Richard , P. Vassault , G. Subra , J.-F. Guichou , E. Richard , et al.
Chemistry and Biology, 2005, 12, pp.15-24. ⟨10.1016/j.chembiol.2004.10.008⟩
Article dans une revue hal-00017005v1
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Vasopressin receptors and pharmacological chaperones: From functional rescue to promising therapeutic strategies.

Bernard Mouillac , Christiane Mendre
Pharmacological Research, 2014, 83, pp.74-8. ⟨10.1016/j.phrs.2013.10.007⟩
Article dans une revue inserm-00909101v1
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Biased agonist pharmacochaperones of the AVP V2 receptor may treat congenital nephrogenic diabetes insipidus.

Frédéric Jean-Alphonse , Sanja Perkovska , Marie-Céline Frantz , Thierry Durroux , Catherine Méjean , et al.
Journal of the American Society of Nephrology, 2009, 20 (10), pp.2190-203. ⟨10.1681/ASN.2008121289⟩
Article dans une revue inserm-00421838v1
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Heterodimerization with Its Splice Variant Blocks the Ghrelin Receptor 1a in a Non-signaling Conformation

Sophie Mary , Jean-Alain Fehrentz , Marjorie Damian , Gérald Gaibelet , Hélène Orcel , et al.
Journal of Biological Chemistry, 2013, 288 (34), pp.24656-24665. ⟨10.1074/jbc.M113.453423⟩
Article dans une revue hal-02871944v1

Crosslinking photosensitized by a ruthenium chelate as a tool for labeling and topographical studies of G-protein-coupled receptors.

Isabelle Duroux-Richard , Philippe Vassault , Guy Subra , Jean-François Guichou , Eric Richard , et al.
Chemistry and Biology, 2005, 12 (1), pp.15-24. ⟨10.1016/j.chembiol.2004.10.008⟩
Article dans une revue inserm-00145329v1

Design, synthesis and biological studies of a library of NK1-Receptor Ligands Based on a 5-arylthiosubstituted 2-amino-4,6-diaryl-3-cyano-4 H -pyran core: Switch from antagonist to agonist effect by chemical modification

Rocío Recio , Empar Vengut-Climent , Bernard Mouillac , Hélène Orcel , Miguel López-Lázaro , et al.
European Journal of Medicinal Chemistry, 2017, 138, pp.644-660. ⟨10.1016/j.ejmech.2017.06.056⟩
Article dans une revue hal-02075064v1
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Carbohydrate-Based NK1R Antagonists with Broad-Spectrum Anticancer Activity

Rocío Recio , Patricia Lerena , Esther Pozo , José Manuel Calderón-Montaño , Estefanía Burgos-Morón , et al.
Journal of Medicinal Chemistry, 2021, 64 (14), pp.10350-10370. ⟨10.1021/acs.jmedchem.1c00793⟩
Article dans une revue hal-03287315v1
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Differential coupling of the vasopressin V1b receptor through compartmentalization within the plasma membrane.

Hélène Orcel , Laura Albizu , Sanja Perkovska , Thierry Durroux , Christiane Mendre , et al.
Molecular Pharmacology, 2009, 75 (3), pp.637-47. ⟨10.1124/mol.108.049031⟩
Article dans une revue inserm-00362611v1
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Cryo–electron microscopy structure of the antidiuretic hormone arginine-vasopressin V2 receptor signaling complex

Julien Bous , Hélène Orcel , Nicolas Floquet , Cedric Leyrat , Joséphine Lai-Kee-Him , et al.
Science Advances , 2021, 7 (21), pp.eabg5628. ⟨10.1126/sciadv.abg5628⟩
Article dans une revue hal-03240488v1
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New advances in production and functional folding of G-protein-coupled receptors.

Jean-Louis Banères , Jean-Luc Popot , Bernard Mouillac
Trends in Biotechnology, 2011, 29 (7), pp.314-22. ⟨10.1016/j.tibtech.2011.03.002⟩
Article dans une revue inserm-00590416v1
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Fluorescent agonists and antagonists for vasopressin/oxytocin g protein-coupled receptors: usefulness in ligand screening assays and receptor studies.

Bernard Mouillac , Maurice Manning , Thierry Durroux
Mini-Reviews in Medicinal Chemistry, 2008, 8 (10), pp.996-1005. ⟨10.2174/138955708785740607⟩
Article dans une revue inserm-00323511v1
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Misfolding of vasopressin receptors: biased agonist pharmacochaperones as potential therapeutics

Christiane Mendre , Bernard Mouillac
Advances in Protein Chemistry and Structural Biology,, 118, pp.249-272, 2019, ⟨10.1016/bs.apcsb.2019.07.002⟩
Chapitre d'ouvrage hal-03444654v1
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Structure of the vasopressin hormone–V2 receptor–β-arrestin1 ternary complex

Julien Bous , Aurélien Fouillen , Hélène Orcel , Stefano Trapani , Xiaojing Cong , et al.
Science Advances , 2022, 8 (35), pp.eabo7761. ⟨10.1126/sciadv.abo7761⟩
Article dans une revue hal-03790728v1
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The ligand-bound state of a G protein-coupled receptor stabilizes the interaction of functional cholesterol molecules

Laura Lemel , Katarzyna Nieścierowicz , M. Dolores García-Fernández , Leonardo Darré , Thierry Durroux , et al.
Journal of Lipid Research, 2021, 62, pp.100059. ⟨10.1016/j.jlr.2021.100059⟩
Article dans une revue hal-03180171v1
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Leukotriene BLT2 receptor monomers activate the G(i2) GTP-binding protein more efficiently than dimers.

Laure Arcemisbehere , Tuhinadri Sen , Laure Boudier , Marie-Noëlle Balestre , Gérald Gaibelet , et al.
Journal of Biological Chemistry, 2010, 285 (9), pp.6337-47. ⟨10.1074/jbc.M109.083477⟩
Article dans une revue inserm-00457594v1

Quantitative MALDI‐MS Binding Assays: An Alternative to Radiolabeling

Maxime Rossato , Guillaume Miralles , Céline M'Kadmi , Mathieu Maingot , Muriel Amblard , et al.
ChemMedChem, 2016, 11 (23), pp.2582-2587. ⟨10.1002/cmdc.201600447⟩
Article dans une revue istex hal-03562144v1

Structures of the arginine-vasopressin and oxytocin receptor signaling complexes

Julien Bous , Aurélien Fouillen , Hélène Orcel , Sébastien Granier , Patrick Bron , et al.
Vitamins and hormones, 2023, Vitamins and Hormones, 123, pp.67-107. ⟨10.1016/bs.vh.2022.12.003⟩
Article dans une revue hal-04213123v1
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A snake toxin as a theranostic agent for the type 2 vasopressin receptor

Laura Droctové , Manon Lancien , Vu Long Tran , Michaël Susset , Benoit Jego , et al.
Theranostics, 2020
Article dans une revue hal-03070378v1

Ghrelin receptor conformational dynamics regulate the transition from a preassembled to an active receptor:Gq complex.

Marjorie Damian , Sophie Mary , Mathieu Maingot , Céline M'Kadmi , Didier Gagne , et al.
Proceedings of the National Academy of Sciences of the United States of America, 2015, 112 (5), pp.1601-1606. ⟨10.1073/pnas.1414618112⟩
Article dans une revue hal-01115392v1

The multifunctional protein GC1q-R interacts specifically with the i3 loop arginine cluster of the vasopressin V-2 receptor

Sebastien Granier , Frederic Jean-Alphonse , Daniel Bacqueville , Arnaud Monteil , Robert Pascal , et al.
Regulatory Peptides, 2008, 148, pp.76-87. ⟨10.1016/j.regpep.2008.01.007⟩
Article dans une revue istex hal-00493436v1

Pharmacological Chaperones as Potential Therapeutic Strategies for Misfolded Mutant Vasopressin Receptors

Bernard Mouillac , Christiane Mendre
Handbook of Experimental Pharmacology, 2018, 245, pp.63-83. ⟨10.1007/164_2017_50⟩
Article dans une revue hal-02073190v1
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THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: G protein‐coupled receptors

Stephen Alexander , Arthur Christopoulos , Anthony P Davenport , Eamonn Kelly , Alistair Mathie , et al.
British Journal of Pharmacology, 2019, 176 (S1), pp.S21-S141. ⟨10.1111/bph.14748⟩
Article dans une revue hal-02388696v1
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[Pharmacological chaperones: a potential therapeutic treatment for conformational diseases]

Christiane Mendre , Bernard Mouillac
Médecine/Sciences, 2010, 26 (6-7), pp.627-35. ⟨10.1051/medsci/2010266-7627⟩
Article dans une revue inserm-00516358v1

Fluorescent-Based Strategies to Investigate G Protein-Coupled Receptors: Evolution of the Techniques to a Better Understanding

Orestis Faklaris , Joyce Heuninck , Amandine Falco , Elise Goyet , Jurriaan M. Zwier , et al.
Structure and Function of GPCRs, pp.217-252, 2017, ⟨10.1007/7355_2017_2⟩
Chapitre d'ouvrage hal-02391215v1
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Structural insights into biased G protein-coupled receptor signaling revealed by fluorescence spectroscopy.

Rita Rahmeh , Marjorie Damian , Martin Cottet , Hélène Orcel , Christiane Mendre , et al.
Proceedings of the National Academy of Sciences of the United States of America, 2012, 109 (17), pp.6733-8. ⟨10.1073/pnas.1201093109⟩
Article dans une revue inserm-00713711v1
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Structure of the antidiuretic hormone vasopressin receptor signalling complex.

Julien Bous , Hélène Orcel , Nicolas Floquet , Cedric Leyrat , Josephine Lai-Kee-Him , et al.
2020
Pré-publication, Document de travail hal-03088027v1
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A new Kunitz‐type snake toxin family associated with an original mode of interaction with the vasopressin 2 receptor

Laura Droctové , Justyna Ciolek , Christiane Mendre , Amélia Chorfa , Paola Huerta , et al.
British Journal of Pharmacology, 2022, Emerging Fields for Therapeutic Targeting of the Aldosterone-Mineralocorticoid Receptor Signaling Pathway, 179 (13), pp.3470-3481. ⟨10.1111/bph.15814⟩
Article dans une revue hal-03629151v1

Cloning, expression and pharmacological characterization of a vasopressin-related receptor in an annelid, the leech Theromyzon tessulatum

A. Levoye , Bernard Mouillac , G. Riviere , D. Vieau , M. Salzet , et al.
Journal of Endocrinology, 2005, 184, pp.277-289. ⟨10.1677/joe.1.05833⟩
Article dans une revue hal-00017042v1
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Bringing GPCR Structural Biology to Medical Applications: Insights from Both V2 Vasopressin and Mu-Opioid Receptors

Aurélien Fouillen , Julien Bous , Sébastien Granier , Bernard Mouillac , Remy Sounier
Membranes, 2023, 13 (6), pp.606. ⟨10.3390/membranes13060606⟩
Article dans une revue hal-04135972v1

Amphipols in G Protein-Coupled Receptor Pharmacology: What Are They Good For?

Sophie Mary , Marjorie Damian , Rita Rahmeh , Bernard Mouillac , Jacky Marie , et al.
Journal of Membrane Biology, 2014, 247 (9-10), pp.853-860. ⟨10.1007/s00232-014-9665-9⟩
Article dans une revue hal-03574639v1