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Influence of the Structure of Polyfluorinated Alcohols on Bronsted Acidity/Hydrogen-Bond Donor Ability and Consequences on the Promoter Effect

Daniela Vuluga , Julien Legros , Benoit Crousse , Alexandra M. Z. Slawin , Christian Laurence , et al.
Journal of Organic Chemistry, 2011, 76 (4), pp.1126-1133. ⟨10.1021/jo1023816⟩
Article dans une revue hal-02143178v1

Direct Amination of Arenes with Azodicarboxylates Catalyzed by Bisulfate Salt/HFIP Association

Ren-Jin Tang , Pascal Retailleau , Thierry Milcent , Benoit Crousse
ACS Omega, 2019, 4 (5), pp.8960-8966. ⟨10.1021/acsomega.9b00781⟩
Article dans une revue hal-02347296v1

Hexafluoro-2-propanol Promotes para -Selective C-H Amination of Free Anilines with Azodicarboxylates

Ren-Jin Tang , Thierry Milcent , Benoit Crousse
European Journal of Organic Chemistry, 2017, 2017 (32), pp.4753-4757. ⟨10.1002/ejoc.201700794⟩
Article dans une revue hal-02998179v1

Access to novel amino trifluoromethyl cyclopropane carboxylic acid derivatives

Massaba Keita , Rocco de Bona , Mickaël dos Santos , Olivier Lequin , Sandrine Ongeri , et al.
Tetrahedron, 2013, 69 (15), pp.3308-3315. ⟨10.1016/j.tet.2013.02.012⟩
Article dans une revue istex hal-01366842v1
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5-Fluoro-1,2,3-triazole motif in peptides and its electronic properties

José Laxio Arenas , Pascal Retailleau , Jean-Michel Gillet , Nour-Eddine Ghermani , Sandrine Ongeri , et al.
Organic & Biomolecular Chemistry, 2022, 20 (43), pp.8410-8414. ⟨10.1039/D2OB01716D⟩
Article dans une revue hal-04249450v1

Synthesis of NCF3, NCF2H and NCH2CF3 motifs

Benoit Crousse , Thierry Milcent
merging Fluorinated Motifs. Properties, Synthesis and Applications, 2020
Chapitre d'ouvrage hal-03796648v1

Towards a general synthesis of di-aza-amino acids containing peptides

Faustine Bizet , Nicolo Tonali , Jean-Louis Soulier , Agostino Oliva , Julia Kaffy , et al.
New Journal of Chemistry, 2018, 42 (20), pp.17062-17072. ⟨10.1039/c8nj03635g⟩
Article dans une revue hal-02347605v1

Hexafluoroisopropanol as a Solvent for Halogenation of (Het)aromatics

Ren-Jin Tang , Thierry Milcent , Benoit Crousse
SYNFACTS, 2018, 14 (3), pp.0244. ⟨10.1055/s-0037-1609312⟩
Article dans une revue hal-02347456v1

Regioselective Halogenation of Arenes and Heterocycles in Hexafluoroisopropanol

Ren-Jin Tang , Thierry Milcent , Benoit Crousse
Journal of Organic Chemistry, 2018, 83 (2), pp.930-938. ⟨10.1021/acs.joc.7b02920⟩
Article dans une revue hal-02347571v1

New 10-Trifluoromethyl Monomers, Dimers, and Chimeras of Artemisinin from a Key Allyl Bromide Precursor

Danièle Bonnet-Delpon , Jean-Pierre Bégué , Benoit Crousse , Fabienne Grellepois , Constance Chollet , et al.
Current fluoroorganic chemistry: new synthetic directions, technologies, materials and biological application, ACS Symposium Series, Vol 949, pp.337-351, 2007, ⟨10.1021/bk-2007-0949.ch020⟩
Chapitre d'ouvrage mnhn-02867458v1

Benefits of a Dual Chemical and Physical Activation: Direct aza-Michael Addition of Anilines Promoted by Solvent Effect under High Pressure

Alena Fedotova , Benoît Crousse , Isabelle Chataigner , Jacques Maddaluno , Alexander Yu. Rulev , et al.
Journal of Organic Chemistry, 2015, 80 (20), pp.10375-10379. ⟨10.1021/acs.joc.5b01756⟩
Article dans une revue hal-02019190v1

Fluorous 4- N , N -Dimethylaminopyridine (DMAP) Salts as Simple Recyclable Acylation Catalysts

Daniela Vuluga , Julien Legros , Benoit Crousse , Danièle Bonnet-Delpon
Chemistry - A European Journal, 2010, 16 (6), pp.1776-1779. ⟨10.1002/chem.200902982⟩
Article dans une revue istex hal-02326126v1

Orally Active Antimalarials: Hydrolytically Stable Derivatives of 10-Trifluoromethyl Anhydrodihydroartemisinin †

Fabienne Grellepois , Fatima Chorki , Michèle Ourévitch , Sébastien Charneau , Philippe Grellier , et al.
Journal of Medicinal Chemistry, 2004, 47 (6), pp.1423-1433. ⟨10.1021/jm030947m⟩
Article dans une revue istex mnhn-02867479v1

Facile Access to Fluorinated Aryl and Vinyl Ethers through Copper-Catalysed Reaction of Fluoro Alcohols

Daniela Vuluga , Julien Legros , Benoit Crousse , Danièle Bonnet-Delpon
European Journal of Organic Chemistry, 2009, 2009 (21), pp.3513-3518. ⟨10.1002/ejoc.200900303⟩
Article dans une revue istex hal-02326135v1

Aminocyclopropanes as precursors of endoperoxides with antimalarial activity

Claire Madelaine , Olivier Buriez , Benoit Crousse , Isabelle Florent , Philippe Grellier , et al.
Organic & Biomolecular Chemistry, 2010, 8 (24), pp.5591. ⟨10.1039/c0ob00308e⟩
Article dans une revue istex mnhn-02047403v1

Bisulfate Salt-Catalyzed Friedel–Crafts Benzylation of Arenes with Benzylic Alcohols

Ren-Jin Tang , Thierry Milcent , Benoit Crousse
Journal of Organic Chemistry, 2018, 83 (22), pp.14001-14009. ⟨10.1021/acs.joc.8b02361⟩
Article dans une revue hal-02347577v1
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β-chlorovinylaldehydes as intermediates in the synthesis of new substituted β–fluoroalkoxyvinyl aldehydes and corresponding alcohols

Sondes Ghrairi , Khaled Essalah , Benoit Crousse , Thouraya Barhoumi-Slimi
Journal of Fluorine Chemistry, 2021, 248, ⟨10.1016/j.jfluchem.2021.109837⟩
Article dans une revue hal-03796609v1
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Difluoroalanine: Synthesis, Incorporation in Peptides, and Hydrophobic Contribution Assessment

Yazid Boutahri , Khoubaib Ben Haj Salah , Nicolas Tisserand , Nathalie Lensen , Benoit Crousse , et al.
2023
Pré-publication, Document de travail hal-04249424v1

The main and recent syntheses of the N-CF3 motif

Thierry Milcent , Benoit Crousse
Comptes Rendus. Chimie, 2018, 21 (8), pp.771-781. ⟨10.1016/j.crci.2017.09.003⟩
Article dans une revue hal-02347644v1

Synthesis of α-CF3 azanorbornene and azetidines by aza Diels–Alder or iodine-mediated cyclizations: application in ROMP and ligand design

Gilles Berger , Luca Fusaro , Michel Luhmer , Arie van Der Lee , Benoît Crousse , et al.
Tetrahedron Letters, 2014, 55 (46), pp.6339 - 6342. ⟨10.1016/j.tetlet.2014.09.105⟩
Article dans une revue hal-01687576v1
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Designed Glycopeptidomimetics Disrupt Protein–Protein Interactions Mediating Amyloid β-Peptide Aggregation and Restore Neuroblastoma Cell Viability

Julia Kaffy , Dimitri Brinet , Jean-Louis Soulier , Isabelle Correia , Nicolo Tonali , et al.
Journal of Medicinal Chemistry, 2016, 59 (5), pp.2025-2040. ⟨10.1021/acs.jmedchem.5b01629⟩
Article dans une revue hal-02467871v1

Direct Access to Substituted 4-CF3 β-Lactams at the C-3 Position

Monika Skibińska , Marcin Kaźmierczak , Thierry Milcent , Tomasz Cytlak , Henryk Koroniak , et al.
Frontiers in Chemistry, 2019, 7, pp.526. ⟨10.3389/fchem.2019.00526⟩
Article dans une revue hal-02347612v1

Solubility switch of gold nanoparticles through hydrogen bond association

Daniela Vuluga , Julien Legros , Benoit Crousse , Danièle Bonnet-Delpon
Chemical Communications, 2008, 40, pp.4954. ⟨10.1039/b810932j⟩
Article dans une revue istex hal-02326146v1
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The use of 4,4,4-trifluorothreonine to stabilize extended peptide structures and mimic β-strands

Yaochun Xu , Isabelle Correia , Tap Ha-Duong , Nadjib Kihal , Jean-Louis Soulier , et al.
Beilstein Journal of Organic Chemistry, 2017, 13, pp.2842 - 2853. ⟨10.3762/bjoc.13.276⟩
Article dans une revue hal-01700974v1

Structure-activity relationships of sugar-based peptidomimetics as modulators of amyloid β-peptide early oligomerization and fibrillization.

Julia Kaffy , Dimitri Brinet , Jean-Louis Soulier , Lucie Khemtémourian , Olivier Lequin , et al.
European Journal of Medicinal Chemistry, 2014, 86C, pp.752-758. ⟨10.1016/j.ejmech.2014.09.031⟩
Article dans une revue hal-01067196v1

Polyfluorinated mercaptoalcohol as a H-bond modifier of poly(2,3,4,5,6-pentafluorostyrene) (PPFS) enhancing miscibility of hydroxylated-PPFS with various acceptor polymers

Jing Chen , Daniela Vuluga , Benoit Crousse , Julien Legros , Jannick Duchet-Rumeau , et al.
Polymer, 2013, 54 (15), pp.3757-3766. ⟨10.1016/j.polymer.2013.05.027⟩
Article dans une revue istex hal-02326099v1
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A one-pot synthesis and X-Ray structural characterization of new highly substituted-allyl carbamates

Sondes Ghrairi , Pascal Retailleau , Benoit Crousse , Thouraya Barhoumi-Slimi
Journal of Molecular Structure, 2022, 1258, pp.132548. ⟨10.1016/j.molstruc.2022.132548⟩
Article dans une revue hal-03796662v1
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Direct access to fluorinated sulfonylhydrazides and study of their reactivity in thiolation reaction on indoles

Benoit Crousse , Tingting Cao
Helvetica Chimica Acta, 2022, 105 (3), ⟨10.1002/hlca.202100196⟩
Article dans une revue hal-04249482v1

Synthesis of Trifluoromethylated Pyrrolidine and Piperidine Amino Acids

Benoît Crousse , Pascal Retailleau , Thierry Milcent , Sandrine Ongeri , Vadim A. Soloshonok
SYNFACTS, 2018, 14 (10), pp.1015. ⟨10.1055/s-0037-1610969⟩
Article dans une revue hal-02347510v1

Straightforward synthesis of 2-propylquinolines under multicomponent conditions in fluorinated alcohols

Ch Venkateswarlu , Pv Balaji , De Kavita , Benoît Crousse , Bruno Figadère , et al.
Journal of Fluorine Chemistry, 2013, pp.94-98. ⟨10.1016/j.jfluchem.2012.12.006⟩
Article dans une revue istex hal-01015813v1