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Could we expect new praziquantel derivatives ? A meta pharmacometrics/pharmacoinformatics analysis of all antischistosomal praziquantel derivatives found in the literature

 V.B. Ribeiro da Silva , B. Boucherle , J. El-Methni , B. Hoffmann , A.L. da Silva , et al.
SAR and QSAR in Environmental Research, 2019, 30 (6), pp.383 - 401. ⟨10.1080/1062936X.2019.1607898⟩
Article dans une revue hal-03928621v1
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Traditional uses, phytochemistry and pharmacological properties of African Nauclea species: A review

 Romain Haudecoeur , Marine Peuchmaur , Basile Pérès , Maxime Rome , Germain Sotoing Taïwe , et al.
Journal of Ethnopharmacology, 2018, 212, pp.106-136. ⟨10.1016/j.jep.2017.10.011⟩
Article dans une revue hal-04019717v1

An expeditious access to 5-pyrimidinol derivatives from cyclic methylglyoxal diadducts, formation of argpyrimidines under physiological conditions and discovery of new CFTR inhibitors.

 Brice-Loïc Renard , Benjamin Boucherle , Bruno Maurin , Marie-Carmen Molina , Caroline Norez , et al.
European Journal of Medicinal Chemistry, 2011, 46 (5), pp.1935-41. ⟨10.1016/j.ejmech.2011.02.037⟩
Article dans une revue istex hal-00582439v1
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Exploring the structure-activity relationship of benzylidene-2,3-dihydro-1H-inden-1-one compared to benzofuran-3(2H)-one derivatives as inhibitors of tau amyloid fibers

 Emeline Boukherrouba , Camille Larosa , Kim-Anh Nguyen , Jérémy Caburet , Laurent Lunven , et al.
European Journal of Medicinal Chemistry, 2022, 231, pp.114139. ⟨10.1016/j.ejmech.2022.114139⟩
Article dans une revue hal-04014492v1
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Investigation of chemical composition and biological activities of $Ajuga\ pyramidalis$—isolation of iridoids and phenylethanoid glycosides

 Anthonin Gori , Benjamin Boucherle , Aurélien Rey , Maxime Rome , Caroline Barette , et al.
Metabolites, 2023, 13, pp.128. ⟨10.3390/metabo13010128⟩
Article dans une revue hal-04014499v1

Structure-Based Design of PDZ Ligands as Inhibitors of 5-HT2A Receptor/PSD-95 PDZ1 Domain Interaction Possessing Anti-hyperalgesic Activity

 Alexandre Vogrig , Liam Dorr , Naoual Bouzidi , Benjamin Boucherle , Anne-Sophie Wattiez , et al.
ACS Chemical Biology, 2013, 8, pp.2209-2216. ⟨10.1021/cb400308u⟩
Article dans une revue hal-00948867v1
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Synthèse et évaluation de modulateurs de la protéine CFTR

 Benjamin Boucherle
Chimie. Université Joseph-Fourier - Grenoble I, 2008. Français. ⟨NNT : ⟩
Thèse tel-00347412v1

Identification of PDZ ligands by docking-based virtual screening for the development of novel analgesic agents

 Naoual Bouzidi , Hemantkumar Deokar , Alexandre Vogrig , Benjamin Boucherle , Isabelle Ripoche , et al.
Bioorganic and Medicinal Chemistry Letters, 2013, 23, pp.2624-2627. ⟨10.1016/j.bmcl.2013.02.100⟩
Article dans une revue istex hal-00846217v1

NMR evaluation of interactions between substituted-indole and PDZ1 domain of PSD-95

 Alexandre Vogrig , Benjamin Boucherle , I. Ripoche , I. Abrunhosa-Thomas , Lu-Yun Lian , et al.
Bioorganic and Medicinal Chemistry Letters, 2011, 21 (11), pp.3349-3353. ⟨10.1016/j.bmcl.2011.04.011⟩
Article dans une revue istex hal-03027170v1
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Development of an innovative maceration technique to optimize extraction and phase partition of natural products

 Anthonin Gori , Benjamin Boucherle , Aurélien Rey , Maxime Rome , Nicola Fuzzati , et al.
Fitoterapia, 2021, 148, pp.104798. ⟨10.1016/j.fitote.2020.104798⟩
Article dans une revue hal-04014497v1
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Arylthiosemicarbazones as antileishmanial agents

 José Ignacio Manzano , Florent Cochet , Benjamin Boucherle , Verónica Gómez-Pérez , Ahcène Boumendjel , et al.
European Journal of Medicinal Chemistry, 2016, 123, pp.161-170. ⟨10.1016/j.ejmech.2016.07.014⟩
Article dans une revue hal-04014490v1

Nauclea latifolia: biological activity and alkaloid phytochemistry of a West African tree

 Benjamin Boucherle , Romain Haudecoeur , Emerson Ferreira Queiroz , Michel de Waard , Jean-Luc Wolfender , et al.
Natural Product Reports, 2016, 33 (9), pp.1034-1043. ⟨10.1039/c6np00039h⟩
Article dans une revue hal-02141583v1
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Aurones and derivatives as promising New Delhi metallo-β-lactamase (NDM-1) inhibitors

 Jérémy Caburet , Federica Verdirosa , Matis Moretti , Brayan Roulier , Giorgia Simoncelli , et al.
Bioorganic and Medicinal Chemistry Letters, 2024, 97, pp.117559. ⟨10.1016/j.bmc.2023.117559⟩
Article dans une revue hal-04429770v1
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Targeting different binding sites in the CFTR structures allows to synergistically potentiate channel activity

 Lionel Froux , Ahmad Elbahnsi , Benjamin Boucherle , Arnaud Billet , Nesrine Baatallah , et al.
European Journal of Medicinal Chemistry, 2020, 190, pp.112116. ⟨10.1016/j.ejmech.2020.112116⟩
Article dans une revue hal-02924784v1
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