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Radiosynthesis and Radiotracer Properties of a 7-(2-[18F]Fluoroethoxy)-6-methoxypyrrolidinylquinazoline for Imaging of Phosphodiesterase 10A with PET

Aurélie Maisonial-Besset , Uta Funke , Winnie Deuther-Conrad , Gregor Schwan , Aurélie Maisonial , et al.
Pharmaceuticals Policy and Law, 2012, 5 (12), pp.169 - 188. ⟨10.3390/ph5020169⟩
Article dans une revue hal-01677646v1
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Synthesis and In Vitro Comparison of DOTA, NODAGA and 15-5 Macrocycles as Chelators for the 64Cu-Labelling of Immunoconjugates

Aurélie Maisonial-Besset , Tiffany Witkowski , Mercedes Quintana , Sophie Besse , Vincent Gaumet , et al.
Molecules, 2022, 28 (1), pp.75. ⟨10.3390/molecules28010075⟩
Article dans une revue hal-03911093v1

Is tetraspanin 8 a target for radioimmunotherapy in syngeneic APC/min colorectal cancer model ?

Mathilde Bonnet , Aurelie Maisonial-Besset , T Witkowski , Gwenaëlle Roche , A Briat , et al.
9th European Conference on Tetraspanins, Sep 2019, Budenheim, Germany
Communication dans un congrès hal-02524663v1
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[18F]ML-10 PET imaging fails to assess early response to neoadjuvant chemotherapy in a preclinical model of triple negative breast cancer

Elodie Jouberton , Sébastien Schmitt , Emmanuel Chautard , Aurélie Maisonial-Besset , Marie Roy , et al.
EJNMMI Research, 2020, 10 (1), pp.2. ⟨10.1186/s13550-019-0587-5⟩
Article dans une revue hal-02489788v1
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Automation of the radiosynthesis and purification procedures for [18F]Fluspidine preparation, a new radiotracer for clinical investigations in PET imaging of σ1 receptors in brain

Aurélie Maisonial-Besset , Uta Funke , Barbara Wenzel , Steffen Fischer , Katharina Holl , et al.
Applied Radiation and Isotopes, 2014, 84, pp.1-7. ⟨10.1016/j.apradiso.2013.10.015⟩
Article dans une revue hal-01677559v1

Simple and convenient conversion of acridones into 9-unsubstituted acridines via acridanes using borane tetrahydrofuran complex

Nicolas Desbois , Anna Szollosi , Aurélie Maisonial , Valérie Weber , Emmanuel Moreau , et al.
Tetrahedron Letters, 2009, 50 (49), pp.6894 - 6896. ⟨10.1016/j.tetlet.2009.09.141⟩
Article dans une revue istex hal-01677641v1

Design, synthesis and preliminary biological evaluation of acridine compounds as potential agents for a combined targeted chemo-radionuclide therapy approach to melanoma

Nicolas Desbois , Maryline Gardette , Janine Papon , Pierre Labarre , Aurélie Maisonial , et al.
Bioorganic and Medicinal Chemistry, 2008, 16 (16), pp.7671-7690. ⟨10.1016/j.bmc.2008.07.015⟩
Article dans une revue istex hal-01494523v1

Novel Radioiodinated and Radiofluorinated Analogues of FT-2102 for SPECT or PET Imaging of mIDH1 Mutant Tumours

Valérie Weber , Lucie Arnaud , Sladjana Dukic-Stefanovic , Barbara Wenzel , Valérie Roux , et al.
Molecules, 2022, 27 (12), pp.3766. ⟨10.3390/molecules27123766⟩
Article dans une revue hal-03868150v1
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Targeting cyclic nucleotide phosphodiesterase 5 (PDE5) in brain: Toward the development of a PET radioligand labeled with fluorine-18

Barbara Wenzel , Jianrong Liu , Sladjana Dukic-Stefanovic , Winnie Deuther-Conrad , Rodrigo Teodoro , et al.
Bioorganic Chemistry, 2019, 86, pp.346-362. ⟨10.1016/j.bioorg.2019.01.037⟩
Article dans une revue hal-02090315v1

Nouveaux Complexes de Platine à Visée Antitumorale

David J Aitken , Isabelle Canet , Arnaud Gautier , Marlène Goubert , J. Kozelka , et al.
1ères Journées Scientifiques du CLARA (Canceropôle Lyon Auvergne Rhône Alpes), 2006, Vulcania, Saint Ours les Roches, France
Communication dans un congrès hal-00021192v1
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Base/cryptand/metal-free automated nucleophilic radiofluorination of [ 18 F]FDOPA from iodonium salts: importance of hydrogen carbonate counter ion

Aurélie Maisonial-Besset , Audrey Serre , Ali Ouadi , Sébastien Schmitt , Damien Canitrot , et al.
European Journal of Organic Chemistry, 2018, 2018 (48), pp.7058-7065. ⟨10.1002/ejoc.201801608⟩
Article dans une revue hal-02343361v1

Radiosynthesis and biological evaluation of [18F]AG-120 for PET imaging of the mutant isocitrate dehydrogenase 1 in glioma

Thu Hang Lai , Barbara Wenzel , Sladjana Dukić-Stefanović , Rodrigo Teodoro , Lucie Arnaud , et al.
European Journal of Nuclear Medicine and Molecular Imaging, 2023, ⟨10.1007/s00259-023-06515-7⟩
Article dans une revue hal-04298024v1

Synthesis, radiofluorination and pharmacological evaluation of a fluoromethyl spirocyclic PET tracer for central σ1 receptors and comparison with fluoroalkyl homologs

Aurélie Maisonial-Besset , Aurélie Maisonial , Eva Grosse Maestrup , Christian Wiese , Achim Hiller , et al.
Bioorganic and Medicinal Chemistry, 2012, 20 (1), pp.257 - 269. ⟨10.1016/j.bmc.2011.11.002⟩
Article dans une revue istex hal-01677635v1
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Control of the Platinum(II) ligating properties of rigid 1,2-diamines: the case of trans-2,3-diaminonorbornane.

Aurélie Maisonial , Mounir Traïkia , Arnaud Gautier , David J Aitken
Tetrahedron Letters, 2006, 47 (46), pp.8091-8093. ⟨10.1016/jtetlet.2006.09.054⟩
Article dans une revue hal-00118388v1
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Development of a new radiofluorinated quinoline analog for PET imaging of phosphodiesterase 5 (PDE5) in brain

Jianrong Liu , Barbara Wenzel , Sladjana Dukic-Stefanovic , Rodrigo Teodoro , Friedrich-Alexander Ludwig , et al.
Pharmaceuticals, 2016, 9 (2), pp.22. ⟨10.3390/ph9020022⟩
Article dans une revue hal-01677542v1

Synthesis, radiolabeling and preliminary in vivo evaluation of multimodal radiotracers for PET imaging and targeted radionuclide therapy of pigmented melanoma

Aurélie Maisonial-Besset , Emilie M.F. Billaud , Aurélie Besse , Latifa Vidal , Aurélien Vidal , et al.
European Journal of Medicinal Chemistry, 2015, 92, pp.818 - 838. ⟨10.1016/j.ejmech.2015.01.034⟩
Article dans une revue hal-01677566v1
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Targeting the Tetraspanins with Monoclonal Antibodies in Oncology: Focus on Tspan8/Co-029

Mathilde Bonnet , Aurélie Maisonial-Besset , Yingying Zhu , Tiffany Witkowski , Gwenaelle Roche , et al.
Cancers, 2019, 11 (2), pp.179. ⟨10.3390/cancers11020179⟩
Article dans une revue hal-02343370v1

Préparation de nouveaux complexes de platine à visée antitumorale

David J Aitken , Isabelle Canet , Arnaud Gautier , Marlène Goubert , Jiri Kozelka , et al.
Bulletin du Cancer, 2006, 93, pp.137-138
Article dans une revue hal-00362020v1

Click Chelators – The Behavior of Platinum and Palladium Complexes in the Presence of Guanosine and DNA

Aurélien Chevry , Marie-Laure Teyssot , Aurélie Maisonial , Pascale Lemoine , Bernard Viossat , et al.
European Journal of Inorganic Chemistry, 2010, 22, pp.3513-3519. ⟨10.1002/ejic.201000183⟩
Article dans une revue istex hal-00530546v1

Synthesis, radioiodination and in vivo screening of novel potent iodinated and fluorinated radiotracers as melanoma imaging and therapeutic probes

Aurélie Maisonial-Besset , Emilie M.F. Billaud , Sophie Besse , Latifa Rbah-Vidal , Janine Papon , et al.
European Journal of Medicinal Chemistry, 2013, 63, pp.840 - 853. ⟨10.1016/j.ejmech.2012.11.047⟩
Article dans une revue istex hal-01677574v1

A 18F-Labeled Fluorobutyl-Substituted Spirocyclic Piperidine Derivative as a Selective Radioligand for PET Imaging of Sigma1 Receptors

Aurélie Maisonial-Besset , Aurélie Maisonial , Eva Grosse maestrup , Steffen Fischer , Achim Hiller , et al.
ChemMedChem, 2011, 6 (8), pp.1401 - 1410. ⟨10.1002/cmdc.201100108⟩
Article dans une revue istex hal-01677661v1

Single Photon Emission Computed Tomography/Positron Emission Tomography Imaging and Targeted Radionuclide Therapy of Melanoma: New Multimodal Fluorinated and Iodinated Radiotracers

Aurélie Maisonial-Besset , Aurélie Maisonial , Bertrand Kuhnast , Janine Papon , Raphaël Boisgard , et al.
Journal of Medicinal Chemistry, 2011, 54 (8), pp.2745 - 2766. ⟨10.1021/jm101574q⟩
Article dans une revue hal-01677589v1

The Use of [ 125 I] Scintigraphic In Vivo Imaging in Melanoma-Bearing Mice for a Rapid Prescreening of Vectors to Melanoma Tissue

Aurélie Maisonial-Besset , Elisabeth Miot-Noirault , Janine Papon , Marilyne Gardette , Mathilde Bonnet-Duquennoy , et al.
Cancer Biotherapy and Radiopharmaceuticals, 2009, 24 (5), pp.629 - 636. ⟨10.1089/cbr.2008.0608⟩
Article dans une revue hal-01677683v1

Use of 3-[ 18 F]fluoropropanesulfonyl chloride as a prosthetic agent for the radiolabelling of amines: Investigation of precursor molecules, labelling conditions and enzymatic stability of the corresponding sulfonamides

Aurélie Maisonial-Besset , Reik Löser , Steffen Fischer , Achim Hiller , Martin Köckerling , et al.
Beilstein Journal of Organic Chemistry, 2013, 9, pp.1002 - 1011. ⟨10.3762/bjoc.9.115⟩
Article dans une revue hal-01677632v1

Synthesis, Radiofluorination, and in Vivo Evaluation of Novel Fluorinated and Iodinated Radiotracers for PET Imaging and Targeted Radionuclide Therapy of Melanoma

Aurélie Maisonial-Besset , Emilie M F Billaud , Latifa Vidal , Aurélie Vidal , Sophie Besse , et al.
Journal of Medicinal Chemistry, 2013, 56 (21), pp.8455 - 8467. ⟨10.1021/jm400877v⟩
Article dans une revue hal-01677595v1
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Tetraspanin 8 (TSPAN 8) as a potential target for radio-immunotherapy of colorectal cancer

Aurelie Maisonial-Besset , Tiffany Witkowski , Isabelle Navarro-Teulon , Odile Berthier-Vergnes , Giovanna Fois , et al.
Oncotarget, 2017, 8, pp.22034-22047. ⟨10.18632/oncotarget.15787⟩
Article dans une revue hal-01611133v1

click chelators for platinum-based anticancer drugs

Aurélie Maisonial , Patrycja Serafin , Mounir Traïkia , Eric Debiton , Vincent Thery , et al.
European Journal of Organic Chemistry, 2008, 2008 (2), pp.298-305. ⟨10.1002/ejic.200700849⟩
Article dans une revue istex hal-00204439v1

Synthesis and antiviral activity of an imidazo[1,2-a]pyrrolo[2,3-c]pyridine series against the bovine viral diarrhea virus

Emmanuel Moreau , Jean-Michel J.-M. Chezal , Jan Paeshuyse , Vincent Gaumet , Damien Canitrot , et al.
European Journal of Medicinal Chemistry, 2010, 45 (5), pp.2044 - 2047. ⟨10.1016/j.ejmech.2010.01.023⟩
Article dans une revue istex hal-01677567v1
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Synthesis and in vitro evaluation of new fluorinated quinoline derivatives with high affinity for PDE5: Towards the development of new PET neuroimaging probes

Jianrong Liu , Aurelie Maisonial-Besset , Barbara Wenzel , Damien Canitrot , Ariane Baufond , et al.
European Journal of Medicinal Chemistry, 2017, 136, pp.548 - 560. ⟨10.1016/j.ejmech.2017.03.091⟩
Article dans une revue hal-01671041v1